D. Kalinin

发表

Microscale Parallel Synthesis of Acylated Aminotriazoles Enabling the Development of Factor XIIa and Thrombin Inhibitors

U. Karst, C. Daniliuc, S. Platte, 2021, Chemmedchem.

Acylated 1H-1,2,4-Triazol-5-amines Targeting Human Coagulation Factor XIIa and Thrombin: Conventional and Microscale Synthesis, Anticoagulant Properties, and Mechanism of Action.

A. Poso, U. Karst, H. Humpf, 2020, Journal of medicinal chemistry.

Insights into the Zinc-Dependent Deacetylase LpxC: Biochemical Properties and Inhibitor Design.

D. Kalinin, Ralph Holl, 2016, Current topics in medicinal chemistry.

Novel Potent Proline-Based Metalloproteinase Inhibitors: Design, (Radio)Synthesis, and First in Vivo Evaluation as Radiotracers for Positron Emission Tomography.

S. Rose-John, M. Schäfers, D. Kalinin, 2016, Journal of medicinal chemistry.

Diuretic activity and toxicity of some Verbascum nigrum extracts and fractions

D. Kalinin, S. Kalinina, A. Dolzhenko, 2014, Pharmaceutical biology.

Auranthine, a Benzodiazepinone from Penicillium aurantiogriseum: Refined Structure, Absolute Configuration, and Cytotoxicity.

H. Humpf, C. Mück‐Lichtenfeld, C. Daniliuc, 2018, Journal of natural products.

Semisynthetic Approach toward Biologically Active Derivatives of Phenylspirodrimanes from S. chartarum

H. Humpf, E. Würthwein, D. Kalinin, 2022, ACS omega.

A novel multicomponent microwave-assisted synthesis of 5-aza-adenines

D. Kalinin, S. Kalinina, A. Dolzhenko, 2013 .

A one-pot, three-component, microwave-promoted synthesis of 2-amino-substituted 7-amino-1,2,4-triazolo[1,5-a][1,3,5]triazines

D. Kalinin, S. Kalinina, A. Dolzhenko, 2013 .

Proline-based hydroxamates targeting the zinc-dependent deacetylase LpxC: Synthesis, antibacterial properties, and docking studies.

W. Sippl, M. Schäfers, Jelena Melesina, 2019, Bioorganic & medicinal chemistry.

A new synthesis of amino substituted azolo[1,3,5]triazines via reaction of N1,N1-dimethyl-N2-azolylformamidines with cyanamide

D. Kalinin, S. Kalinina, A. Dolzhenko, 2013 .

Synthesis of novel trichloromethyl substituted azolo[1,3,5]triazines

D. Kalinin, S. Kalinina, A. Dolzhenko, 2012 .

Synthesis, local anaesthetic and antiarrhythmic activities of N-alkyl derivatives of proline anilides.

D. Kalinin, S. Kalinina, A. Dolzhenko, 2013, European journal of medicinal chemistry.

Factor XII(a) inhibitors: a review of the patent literature

D. Kalinin, 2021, Expert opinion on therapeutic patents.

Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors

W. Sippl, C. Romier, M. Jung, 2019, ChemMedChem.

LpxC inhibitors: a patent review (2010-2016)

D. Kalinin, Ralph Holl, 2017, Expert opinion on therapeutic patents.

Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants.

Takayoshi Suzuki, W. Sippl, C. Romier, 2018, Journal of medicinal chemistry.

Development of Novel Quinoxaline-Based κ-Opioid Receptor Agonists for the Treatment of Neuroinflammation.

T. Che, S. Ständer, B. Wünsch, 2018, Journal of medicinal chemistry.

Microwave-Assisted Synthesis, Structure, and Preliminary Biological Evaluation of Novel 6-Methoxy-5,6-dihydro-5-azapurines

L. Heitman, Rongfang Liu, C. Daniliuc, 2023, ACS omega.

Amide-functionalized 1,2,4-Triazol-5-amines as Covalent Inhibitors of Blood Coagulation Factor XIIa and Thrombin.

A. Poso, U. Karst, C. Daniliuc, 2022, ACS pharmacology & translational science.

Microscale Parallel Synthesis of Acylated Aminotriazoles Enabling FXIIa and Thrombin Inhibitors Development.

U. Karst, C. Daniliuc, S. Platte, 2021, ChemMedChem.

Replacement of the Benzylpiperidine Moiety with Fluorinated Phenylalkyl Side Chains for the Development of GluN2B Receptor Ligands

S. Ametamey, B. Wünsch, D. Kalinin, 2018, ChemMedChem.

Platelet functional abnormalities in pediatric patients with kaposiform hemangioendothelioma/Kasabach-Merritt phenomenon

A. Martyanov, M. Panteleev, A. Sveshnikova, 2023, Blood advances.