V. Kartsev

发表

3-Amino-5-(indol-3-yl)methylene-4-oxo-2-thioxothiazolidine Derivatives as Antimicrobial Agents: Synthesis, Computational and Biological Evaluation

V. Poroikov, A. Geronikaki, P. Eleftheriou, 2020, Pharmaceuticals.

Synthesis of Benzoannelated Canthin-6-One Analogs

M. Garazd, V. Kartsev, O. A. Sen’ko, 2017, Chemistry of Natural Compounds.

Antibacterial Activity of Noscapine Analogs.

O. Dontsova, L. Zainullina, Y. Ivanenkov, 2021, Bioorganic & medicinal chemistry letters.

New method for the synthesis of the 1,3-thiazine system. 2-phenylamino-5,6-dihydro-4H-1,3-thiazin-5-ones

N. Sepetov, V. Kartsev, A. M. Sipyagin, 1980 .

Kinetics of hydrolysis of antitumor bisdiazoketones

V. Kartsev, N. M. Emanuel, A. M. Sipyagin, 1984, Pharmaceutical Chemistry Journal.

Kinetic isotope effect in hydrolysis of bisdiazoketones

V. Kartsev, A. M. Sipyagin, L. I. Kirkovskii, 1984 .

Molecular docking, design, synthesis and biological evaluation of novel 2,3-aryl-thiazolidin-4-ones as potent NNRTIs

G. Maga, A. Geronikaki, A. Petrou, 2019, SAR and QSAR in environmental research.

Synthesis of thieno[3,2-d]pyrimidin-4-ones and alkylation thereof

K. Shikhaliev, V. Kartsev, A. S. Shestakov, 2014 .

Disruption of the Complex between GAPDH and Hsp70 Sensitizes C6 Glioblastoma Cells to Hypoxic Stress

V. Kartsev, I. Guzhova, B. Margulis, 2021, International journal of molecular sciences.

Reactions of Indole and Its Derivatives with Cotarnine. Rearrangement of 5-(1-Indolyl)-4-methoxy-6-methyl- 5,6,7,8-tetrahydro[1,3]dioxolo[4,5-g]isoquinolines

V. Kartsev, K. Krasnov, 2002 .

Thermal decomposition of benzoyl azide and diazoacetone in the gas phase

V. G. Prokudin, V. Kartsev, S. A. Vozchikova, 1988 .

Griseofulvin derivatives: Synthesis, molecular docking and biological evaluation.

A. Geronikaki, A. Petrou, M. Soković, 2019, Current topics in medicinal chemistry.

Synthesis, Biological Evaluation and Molecular Docking Studies of 5-Indolylmethylen-4-oxo-2-thioxothiazolidine Derivatives

V. Poroikov, A. Geronikaki, A. Petrou, 2022, Molecules.

REACTION OF 2-CHLORO-1-ALKYL-1H-INDOLE-3-CARBALDEHYDES WITH BARBITURIC ACIDS AND 5-METHYL-2-PHENYL-2,4-DIHYDROPYRAZOL-3-ONE : FORMATION OF COMPOUND WITH EXTREMELY SHORT INTRAMOLECULAR HYDROGEN BOND IN EIGHT-MEMBERED PSEUDOCYCLE

V. Kartsev, K. Suzdalev, M. N. Babakova, 2015 .

Imidazole Derivative As a Novel Translation Inhibitor

P. Sergiev, Y. Ivanenkov, I. Osterman, 2022, Acta naturae.

New Rearrangement in the o-Methoxycarbonyl-ω-diazoacetophenone Series

S. Chapyshev, V. Kartsev, 1992 .

Antibacterial activity of griseofulvin analogs as example of drug repurposing.

V. Poroikov, A. Geronikaki, A. Petrou, 2020, International journal of antimicrobial agents.

Inter-ring long-range spin-spin proton coupling in some 8-hydroxyquinoline derivatives

V. Kartsev, I. Vystorop, A. Fomichov, 1993 .

Application of Docking Analysis in the Prediction and Biological Evaluation of the Lipoxygenase Inhibitory Action of Thiazolyl Derivatives of Mycophenolic Acid

A. Saxena, A. Geronikaki, P. Eleftheriou, 2018, Molecules.

Halogenated pyridines 5. Structure of the products of cyclization of chlorine-containingδ-oxonitriles

Z. G. Aliev, K. I. Kobrakov, V. K. Korolev, 1995 .

Scope and limitations of the T-reaction employing some functionalized C-H-acids and naturally occurring secondary amines

C. Hametner, Constantin Rabong, U. Jordis, 2008 .

4-(Indol-3-yl)thiazole-2-amines and 4-ιndol-3-yl)thiazole Acylamines as Νovel Antimicrobial Agents: Synthesis, In Silico and In Vitro Evaluation

A. Geronikaki, A. Petrou, I. Vizirianakis, 2021, Pharmaceuticals.

Experimental and In Silico Evaluation of New Heteroaryl Benzothiazole Derivatives as Antimicrobial Agents

A. Geronikaki, A. Petrou, J. Glamočlija, 2022, Antibiotics.

Carbonic Anhydrase Inhibition with Sulfonamides Incorporating Pyrazole- and Pyridazinecarboxamide Moieties Provides Examples of Isoform-Selective Inhibitors

C. Supuran, M. Pinteala, A. Angeli, 2021, Molecules.

NATURAL COMPOUNDS IN DRUG DISCOVERY. BIOLOGICAL ACTIVITY AND NEW TRENDS IN THE CHEMISTRY OF ISOQUINOLINE ALKALOIDS

V. Kartsev, 2004, Medicinal Chemistry Research.

Chromene-Containing Aromatic Sulfonamides with Carbonic Anhydrase Inhibitory Properties

C. Supuran, M. Pinteala, A. Angeli, 2021, International journal of molecular sciences.

Synthesis and Antimicrobial Activity of New Heteroaryl(aryl) Thiazole Derivatives Molecular Docking Studies

A. Geronikaki, A. Petrou, J. Glamočlija, 2022, Antibiotics.

1-Nicotinoylbenzotriazole: A Convenient Tool for Site-Selective Protection of 5,7-Dihydroxycoumarins

V. Kartsev, O. Chupakhin, V. Charushin, 2019, Synthesis.

Direct Modification of Quercetin by 6-Nitroazolo[1,5-a]Pyrimidines

V. Kartsev, O. Chupakhin, V. Rusinov, 2016, Chemistry of Natural Compounds.

Chemical Modification of Plant Alkaloids. 4. Reaction of Cotarnine with Bifunctional NH- and CH-Acids

V. Kartsev, S. F. Vasilevskii, K. Krasnov, 2005, Chemistry of Natural Compounds.

Benzothiazole and Chromone Derivatives as Potential ATR Kinase Inhibitors and Anticancer Agents

D. Spinelli, A. Geronikaki, A. Petrou, 2022, Molecules.

Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation

C. Supuran, A. Kazaks, K. Tārs, 2019, Molecules.

5-(1H-Indol-3-ylmethylene)-4-oxo-2-thioxothiazolidin-3-yl)alkancarboxylic Acids as Antimicrobial Agents: Synthesis, Biological Evaluation, and Molecular Docking Studies

A. Geronikaki, A. Petrou, A. Ćirić, 2020, Molecules.

Synthesis of 1-Amino-3-oxo-2,7-naphthyridines via Smiles Rearrangement: A New Approach in the Field of Chemistry of Heterocyclic Compounds

D. Spinelli, A. Geronikaki, S. Sirakanyan, 2022, International journal of molecular sciences.

Pyrazolo[4,3-c]pyridine Sulfonamides as Carbonic Anhydrase Inhibitors: Synthesis, Biological and In Silico Studies

C. Supuran, M. Pinteala, A. Angeli, 2022, Pharmaceuticals.

Synthesis and Neurotropic Activity of New Heterocyclic Systems: Pyridofuro[3,2-d]pyrrolo[1,2-a]pyrimidines, Pyridofuro[3,2-d]pyrido[1,2-a]pyrimidines and Pyridofuro[3′,2′:4,5]pyrimido[1,2-a]azepines

D. Spinelli, A. Geronikaki, A. Petrou, 2021, Molecules.

Complex formation of copper(II) and nickel(II) with N-arylthiopicolinamides

Z. G. Aliev, V. Kartsev, A. P. Ranskii, 1993 .

Diastereoselective synthesis of 1-alkyl-2,4,6-trioxoperhydropyrimidine-5-spiro-3′-(1′,2′,3′,4′-tetrahydroquinolines)

V. Khrustalev, V. Kartsev, K. Krasnov, 2010 .

Stereochemical outcome of the T-reaction employing chiral bicyclic amines

Constantin Rabong, U. Jordis, V. Kartsev, 2007 .

Synthesis of thiazoles and thiadiazoles from 1,2-bis(diazoacetyl)ethane

V. Kartsev, F. A. Medvedev, G. N. Voronina, 1980, Chemistry of Heterocyclic Compounds.

Synthesis of thiazoles and thiadiazoles from 1,2-bis(diazoacetyl)ethane

V. Kartsev, F. A. Medvedev, G. N. Voronina, 1980 .

Synthesis, structure, and spectral characteristics of copper complexes with picolinic acid derivatives

Z. G. Aliev, L. Atovmyan, V. Kartsev, 1988 .

Synthesis of Colchicine C-10-Amino-Acid Derivatives

M. Garazd, V. Kartsev, Y. Garazd, 2015, Chemistry of Natural Compounds.

Complex formation of some pesticides with adenosine triphosphoric acid

V. Kartsev, R. Gvozdev, E. Saratovskikh, 1988 .

Chemical modification of plant alkaloids. 6. T-reactions of anabasine derivatives

V. Kartsev, K. Krasnov, 2011, Chemistry of Natural Compounds.

Crystal structure of ω-diazoacetophenone

Z. G. Aliev, L. Atovmyan, V. Kartsev, 1985 .

Scope and Limitations of the T-Reaction Employing Some Functionalized C—H Acids and Naturally Occurring Secondary Amines.

C. Hametner, Constantin Rabong, U. Jordis, 2008 .

New Sulfanilamide Derivatives Incorporating Heterocyclic Carboxamide Moieties as Carbonic Anhydrase Inhibitors

C. Supuran, V. De Luca, C. Capasso, 2021, Pharmaceuticals.

Synthesis and structure of dimethyl 3-(2-furoyl)pyrazole-4,5-dicarboxylate

Z. G. Aliev, L. Atovmyan, V. Kartsev, 1982 .

Mass-spectrometric study of the cyclization reactions of diazoketones. 8. 1-Diazo-3,4-epoxy-4-arylbutan-2-ones

V. Kartsev, P. Sharbatyan, V. Petrosyan, 1986 .

Diazo carbonyl derivatives of heterocycles. 3. Alternative 1,3-dipolar addition to azidoalkyl α-diazo ketones and synthesis of five-membered heterocycles based on them

T. S. Pokidova, A. Nabatov, V. Kartsev, 1984 .

Synthesis and biological evaluation of potent antifungal agents.

A. Geronikaki, F. Macaev, V. Kartsev, 2013, Current topics in medicinal chemistry.

Collision-induced dissociation study of cyclization of α-diazo-ω-arylsulphonylaminoalkan-2-ones

A. Lebedev, V. Kartsev, V. Petrosyan, 1992 .

Novel isatin-derived molecules activate p53 via interference with Mdm2 to promote apoptosis

G. Melino, O. Demidov, P. Davidovich, 2018, Cell cycle.

Synthesis of Alkaloid Sinomenine Derivatives Containing a Pyrimidine Substituent in Ring A

V. Kartsev, E. Shults, A. O. Finke, 2021, Chemistry of Heterocyclic Compounds.

Structure of Dirithromycin Bound to the Bacterial Ribosome Suggests New Ways for Rational Improvement of Macrolides.

P. Sergiev, O. Dontsova, A. Konevega, 2019 .

Structure of Dirithromycin Bound to the Bacterial Ribosome Suggests New Ways for Rational Improvement of Macrolides

P. Sergiev, O. Dontsova, A. Konevega, 2019, Antimicrobial Agents and Chemotherapy.

Madumycin II inhibits peptide bond formation by forcing the peptidyl transferase center into an inactive state

P. Sergiev, O. Dontsova, A. Konevega, 2017, Nucleic acids research.

Synthesis of 3,3-dimethyl-6-oxopyrano[3,4-c]pyridines and their antiplatelet and vasodilatory activity.

D. Spinelli, P. Mladěnka, J. Pourová, 2021, The Journal of pharmacy and pharmacology.

Diazocarbonyl derivatives of heterocycles. 7. Synthesis, properties, and structure of 2,4-diazido-6-diazoacetylpyrimidine

Z. G. Aliev, L. Atovmyan, V. Kartsev, 1990 .

Transition-Metal-Free С–С Coupling of 5,7-Dihydroxybenzopyrones with Quinoxalones and Pteridinones

V. Kartsev, O. Chupakhin, V. Charushin, 2018, Synthesis.

Transition-Metal-Free Cross-Dehydrogenative Coupling of Triazines with 5,7-Dihydroxycoumarins

V. Kartsev, O. Chupakhin, V. Charushin, 2016 .

Synthesis of Benzoannelated Canthin-6-One Analogs

M. Garazd, V. Kartsev, O. A. Sen’ko, 2017, Chemistry of Natural Compounds.

Photolysis of 2-azido-3,4,6-trichloro-5-cyanopyridine

V. Kartsev, É. M. Gizatullina, 1991 .

New Bicyclic Pyridine-Based Hybrids Linked to the 1,2,3-Triazole Unit: Synthesis via Click Reaction and Evaluation of Neurotropic Activity and Molecular Docking

D. Spinelli, A. Geronikaki, A. Petrou, 2023, Molecules.

Synthesis and antimicrobial activity of new 2‐piperazin‐1‐yl‐N‐1,3‐thiazol‐2‐ylacetamides of cyclopenta[c]pyridines and pyrano[3,4‐c]pyridines

D. Spinelli, A. Geronikaki, A. Petrou, 2020, Archiv der Pharmazie.

Synthesis of new heterocyclic systems fused at pyrazolo[3,4-c]-2,7-naphthyridine core

D. Spinelli, A. Geronikaki, S. Sirakanyan, 2022, Mendeleev Communications.

Synthesis of 2-amino-5,5-dialkyl-4-arylmethylidene-2-oxazolines from 2-alkyl-4-arylbut-3-yn-2-ols and guanidine

D. S. Baranov, V. Kartsev, S. Vasilevsky, 2012 .

5-(1 H -Indol-3-ylmethylene)-4-oxo-2-thioxothiazolidin-3-yl)alkancarboxylic Acids as Antimicrobial Agents: Synthesis, Biological Evaluation, and Molecular Docking Studies

A. Geronikaki, A. Petrou, A. Ćirić, 2020 .

Discovery of Novel EGFR Inhibitor Targeting Wild-Type and Mutant Forms of EGFR: In Silico and In Vitro Study

T. Rungrotmongkol, K. Choowongkomon, A. Geronikaki, 2023, Molecules.

Chemical Modification of Plant Alkaloids. 7. T-Reaction of an Aloperine Derivative

V. Kartsev, T. Timofeeva, V. Khrustalev, 2017, Chemistry of Natural Compounds.

Appendix A. dithioloquinolinethiones as new potential multitargeted antibacterial and antifungal agents: Synthesis, biological evaluation and molecular docking studies.

K. Shikhaliev, S. Medvedeva, A. Geronikaki, 2019, European journal of medicinal chemistry.

Modified Coumarins. 35. Synthesis of Coumarins Containing a Lupinine Moiety

M. Garazd, V. Kartsev, Y. Garazd, 2016, Chemistry of Natural Compounds.

Modified Coumarins. 33. Synthesis of Furo- and Dihydropyranocoumarins Containing a Lupinine Moiety

M. Garazd, V. Kartsev, Y. Garazd, 2015, Chemistry of Natural Compounds.

Synthesis and Anti-Infective Activity of 2-Heteroaryl(Acyl)-9,10,12,13-Tetramethoxy-3-Methyl-4,5-Dihydro-3H-Phenanthro[1,2-d]Azepines

V. Kartsev, A. Klimenko, L. Fetisov, 2018, Russian journal of bioorganic chemistry.

Stereoselective Modification of Cytisine: T-Reaction for Construction of Benzoannelated Anagyrine Skeleton

V. Kartsev, K. Krasnov, 2007 .

Chemical Modification of Plant Alkaloids. III. X-Ray Diffraction and NMR Studies of the Structure of 1,3-Dimethyl-5-arylmethyl-5-cytisylmethylbarbituric Acids

V. Kartsev, V. Khrustalev, K. Krasnov, 2002, Chemistry of Natural Compounds.

Unusual Reaction of Alkaloid Cotarnine with 1,3-Dimethylbarbituric Acid

V. Kartsev, K. Krasnov, 2002 .

Unconventional recyclization of cotarnine under the action of 1,3-dimethylbarbituric acid

V. G. Kartsev, V. Kartsev, V. Khrustalev, 2007 .

Unusual Reaction of Alkaloid Cotarnine with 1,3-Dimethylbarbituric Acid.

V. Kartsev, K. Krasnov, 2002 .

Synthesis of N-Acylamino-Acid Derivatives of Cytisine

M. Garazd, V. Kartsev, A. V. Yazlovitskii, 2016, Chemistry of Natural Compounds.

Substituted furan sulfonamides as carbonic anhydrase inhibitors: Synthesis, biological and in silico studies.

C. Supuran, A. Angeli, A. Geronikaki, 2023, Bioorganic chemistry.

Chemical modification of plant alkaloids. I. Aminomethylation of barbituric acid derivatives by cytisine

V. Kartsev, K. Krasnov, A. S. Gorovoi, 2000, Chemistry of Natural Compounds.

N-Derivatives of (Z)-Methyl 3-(4-Oxo-2-thioxothiazolidin-5-ylidene)methyl)-1H-indole-2-carboxylates as Antimicrobial Agents—In Silico and In Vitro Evaluation

A. Geronikaki, A. Petrou, I. Vizirianakis, 2023, Pharmaceuticals.

Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors

C. Supuran, C. Capasso, A. Angeli, 2023, International journal of molecular sciences.

The novel structural modification of pyridoxal via its cyclization into 2-acyl- and 2-heteroarylfuro[2,3-c]pyridines

V. Kartsev, A. Klimenko, A. Morkovnik, 2019, Mendeleev Communications.

Direct Modification of Quercetin by 6-Nitroazolo[1,5-a]Pyrimidines

V. Kartsev, O. Chupakhin, V. Rusinov, 2016, Chemistry of Natural Compounds.

Chemical Modification of Plant Alkaloids. 7. T-Reaction of an Aloperine Derivative

V. Kartsev, T. Timofeeva, V. Khrustalev, 2017, Chemistry of Natural Compounds.

Identification of Novel Antibacterials Using Machine Learning Techniques

Alex Zhavoronkov, Yan A. Ivanenkov, Ilya A. Osterman, 2019, Front. Pharmacol..