G. Luisi

发表

Anti-Oxidant and Tyrosinase Inhibitory In Vitro Activity of Amino Acids and Small Peptides: New Hints for the Multifaceted Treatment of Neurologic and Metabolic Disfunctions

A. Mollica, G. Zengin, A. Stefanucci, 2018, Antioxidants.

Nitrobenzoxadiazole-based GSTP1-1 inhibitors containing the full peptidyl moiety of (pseudo)glutathione

S. Carradori, A. Mollica, A. Caccuri, 2016, Journal of enzyme inhibition and medicinal chemistry.

Synthesis and activity of novel glutathione analogues containing an urethane backbone linkage.

A. Caccuri, G. Luisi, A. Di Stefano, 2003, Farmaco.

ψ(SO2-NH) transition state isosteres of peptides. Synthesis of the glutathione disulfide analogue

G. Luisi, F. Pinnen, A. Calcagni, 1993 .

Biochemical and pharmacological investigation of novel nociceptin/OFQ analogues and N/OFQ-RYYRIK hybrid peptides

A. Mollica, A. Magyar, A. Stefanucci, 2019, Peptides.

New Compounds for the Management of Trypanosoma brucei Infection

S. Carradori, G. Luisi, 2021, Topics in Medicinal Chemistry.

Potent isozyme-selective inhibition of human glutathione S-transferase A1-1 by a novel glutathione S-conjugate

A. Caccuri, G. Luisi, A. Di Stefano, 2005, Amino Acids.

Human caspase-3 inhibition by Z-tLeu-Asp-H: tLeu(P2) counterbalances Asp(P4) and Glu(P3) specific inhibitor truncation.

P. Ascenzi, M. Marino, G. Luisi, 2008, Biochemical and biophysical research communications.

Synthesis and biological evaluation of a novel pyroglutamyl-modified TRH analogue.

G. Orlando, L. Brunetti, L. Recinella, 2002, Farmaco.

psi(SO2NH) transition state isosteres of peptides. Synthesis and bioactivity of sulfonamido pseudopeptides related to carnosine.

G. Luisi, A. Di Stefano, S. Dupré, 1999, Farmaco.

Synthesis and preliminary pharmacological evaluation of trans-2-amino-5(6)-chloro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes as dopamine receptor ligands.

C. Martini, A. Lucacchini, B. Costa, 2002, Farmaco.

Synthesis and preliminary pharmacological evaluation of 5-hydroxy- and 5,6-dihydroxy-1,2,3,7,12,12a-hexahydrobenzo[5,6]cyclohepta[1,2,3-ij]isoquinoline derivatives as dopamine receptor ligands.

C. Martini, A. Lucacchini, B. Costa, 2001, Bioorganic & medicinal chemistry.

Antioxidant properties of different products and additives in white wine.

G. Luisi, R. Zironi, F. Battistutta, 2015, Food chemistry.

Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (Pseudo)-Dipeptidyl Appendages: In Vitro and Computational Studies

S. Carradori, C. Supuran, Mariangela Agamennone, 2022, Molecules.

Design and synthesis of glutathione analogues.

G. Luisi, F. Pinnen, G. Lucente, 1998, Farmaco.

Synthesis and activity of the glutathione analogue γ‐(L‐γ‐azaglutamyl)‐L‐cysteinyl‐glycine

G. Luisi, S. Dupré, F. Pinnen, 2009 .

Synthesis and Activity of the Glutathione Analogue γ‐(L‐γ‐Oxaglutamyl)‐L‐cysteinyl‐glycine

G. Luisi, S. Dupré, F. Pinnen, 1996 .

Antimalarial Agents from Medicinal Plant and Fungal Sources

S. Carradori, R. Grande, D. Secci, 2020 .

Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents

S. Parapini, C. De Monte, S. Carradori, 2015, Journal of enzyme inhibition and medicinal chemistry.

Chemical composition and biological activity of Capparis spinosa L. from Lipari Island

E. Novellino, A. Mollica, G. Zengin, 2019, South African Journal of Botany.

Peptides containing the sulfonamide junction: Synthesis, structure, and conformation of Z-Tau-Pro-Phe-NHiPr

M. Paci, G. Luisi, G. Pochetti, 1997 .

Approaches to pseudopeptidic ergopeptines. Part 3.1 Consequences of the incorporation of an α-azaphenylalanine residue into the ergotamine oxa-cyclolic system

G. Luisi, F. Pinnen, A. Calcagni, 1997 .

Approaches to pseudopeptidic ergopeptines. Synthesis and molecular structure of an α-aza-phenylalanine-containing oxa-cyclol

G. Luisi, F. Pinnen, G. Lucente, 1993 .

APPROACHES TO PSEUDOPEPTIDIC ERGOPEPTINES. PART 3. CONSEQUENCES OF THE INCORPORATION OF AN ALPHA -AZAPHENYLALANINE RESIDUE INTO THE ERGOTAMINE OXA-CYC LOLIC SYSTEM

G. Luisi, F. Pinnen, A. Calcagni, 1997 .

Cyclization under mild conditions of salicyloyl-dipeptides.

G. Luisi, F. Pinnen, A. Calcagni, 2009, International journal of peptide and protein research.

Approaches to pseudopeptidic ergopeptines. Part 2. Consequences of the incorporation of an α-azaproline residue into the oxacyclolic system

G. Luisi, F. Pinnen, A. Calcagni, 1994 .

Serine-containing 10-membered cyclodepsipeptides. Synthesis and molecular structure of PhCH2CO-DSer-Pro-Pro- and PhCH2CO-DSer-Pro-DPro-.

G. Luisi, F. Pinnen, E. Gavuzzo, 2009, International journal of peptide and protein research.

Ten-membered cyclotripeptides. III. Synthesis and conformation of cyclo(-Me beta Ala-Phe-Pro-) and cyclo(-Me beta Ala-Phe-DPro-).

G. Luisi, F. Pinnen, G. Lucente, 2009, International journal of peptide and protein research.

Discovery of arginine-containing tripeptides as a new class of pancreatic lipase inhibitors.

E. Novellino, A. Mollica, G. Zengin, 2019, Future medicinal chemistry.

Discovery of novel amide tripeptides as pancreatic lipase inhibitors by virtual screening

E. Novellino, A. Mollica, G. Zengin, 2019, New Journal of Chemistry.

Activation of β- and γ-carbonic anhydrases from pathogenic bacteria with tripeptides

A. Mollica, C. Supuran, C. Capasso, 2018, Journal of enzyme inhibition and medicinal chemistry.

Nitrogen- and Sulfur-Containing Heterocycles as Dual Anti-oxidant and Anti-cancer Agents

S. Carradori, D. Secci, G. Luisi, 2021, Handbook of Oxidative Stress in Cancer: Mechanistic Aspects.

Novel Cyclic Biphalin Analogues by Ruthenium-Catalyzed Ring Closing Metathesis: in Vivo and in Vitro Biological Profile.

E. Novellino, A. Mollica, G. Zengin, 2019, ACS medicinal chemistry letters.

Fluorescent-labeled bioconjugates of the opioid peptides biphalin and DPDPE incorporating fluorescein-maleimide linkers.

V. Hruby, S. Carradori, A. Mollica, 2017, Future medicinal chemistry.

Synthesis and neuromodulatory effects of TRH-related peptides: inhibitory activity on catecholamine release in vitro

M. Vacca, G. Orlando, C. Ferrante, 2013, Pharmacological reports : PR.

Biofilm and Quorum Sensing inhibitors: the road so far

S. Carradori, Cristina Campestre, G. Luisi, 2020, Expert opinion on therapeutic patents.

Pseudopeptides Containing Isothiazolidine‐1,1‐dioxide‐3‐carboxylic Acid: Synthesis and Properties of (S)‐Isothiazolidine‐1,1‐dioxide‐3‐carboxylic Acid, a New γ ‐ Sultam Analogue of Pyroglutamic Acid

G. Luisi, Francesco Pinnen, 1993 .

Nine-membered cyclodepsitripeptides containing the retroisomeric sequence of ergot peptides.

G. Luisi, F. Pinnen, A. Calcagni, 2009, International journal of peptide and protein research.

Hybrid peptides endomorphin-2/DAMGO: design, synthesis and biological evaluation.

A. Mollica, A. Stefanucci, G. Luisi, 2013, European journal of medicinal chemistry.

Ac-tLeu-Asp-H is the minimal and highly effective human caspase-3 inhibitor: biological and in silico studies

A. Di Pizio, P. Ascenzi, M. Marino, 2014, Amino Acids.

Dual targeting of cancer-related human matrix metalloproteinases and carbonic anhydrases by chiral N-(biarylsulfonyl)-phosphonic acids

C. Supuran, Cristina Campestre, Mariangela Agamennone, 2017, Journal of enzyme inhibition and medicinal chemistry.

Virtual screening identification and chemical optimization of substituted 2-arylbenzimidazoles as new non-zinc-binding MMP-2 inhibitors.

A. Di Pizio, Mariangela Agamennone, A. Laghezza, 2019, Bioorganic & medicinal chemistry.

Ac-tLeu-Asp-H is the minimal and highly effective human caspase-3 inhibitor: biological and in silico studies

A. Di Pizio, P. Ascenzi, M. Marino, 2014, Amino Acids.

Synthesis and neuromodulatory effects of TRH-related peptides: inhibitory activity on catecholamine release in vitro.

M. Vacca, G. Orlando, C. Ferrante, 2013, Pharmacological reports : PR.