N. Blaton

发表

Synthesis and structure-activity relationships of analogs of 2'-deoxy-2'-(3-methoxybenzamido)adenosine, a selective inhibitor of trypanosomal glycosomal glyceraldehyde-3-phosphate dehydrogenase.

P. Herdewijn, S. van Calenbergh, J. Rozenski, 1995, Journal of medicinal chemistry.

Mechanism of increased dissolution of diazepam and temazepam from polyethylene glycol 6000 solid dispersions.

G. Van den Mooter, N. Blaton, R Kinget, 2002, International journal of pharmaceutics.

Evaluation of Inutec SP1 as a new carrier in the formulation of solid dispersions for poorly soluble drugs.

G. Van den Mooter, N. Blaton, I. Weuts, 2006, International journal of pharmaceutics.

Physicochemical characterization of solid dispersions of the antiviral agent UC-781 with polyethylene glycol 6000 and Gelucire 44/14.

L. Naesens, J. Balzarini, P. Augustijns, 2000, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

Vibrational characterization of the peptide bond.

W. Herrebout, N. Blaton, H. Desseyn, 2003, Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy.

Pyridazine derivatives. Part 40: Reactivity of 5-alkynylpyridazin-3(2H)-ones toward hydrochloric acid

E. Sotelo, Alberto Coelho, N. Blaton, 2005 .

Pyridazine derivatives. Part 38: Efficient Heck alkenylation at position 5 of the 6-phenyl-3(2H)-pyridazinone system ☆

E. Sotelo, Alberto Coelho, N. Blaton, 2004 .

3-Deoxy-1,2-O-isopropylidene-3-C-methyl-5-O-(p-tolylsulfonyl)-d-ribofuranose

P. Herdewijn, N. Blaton, B. Doboszewski, 2007 .

(+)-cis-1-Acetyl-4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy}phenyl)piperazine [(2R,4S)-(+)-ketoconazole]

J. Gerber, N. Blaton, O. Peeters, 2004 .

(+)-1-{(2S)-2-(2,4-Dichlorophenyl)-2-[(2,4-dichlorophenyl)methoxy]ethyl}-1H-imidazole mononitrate [(+)-(S)-miconazole nitrate]

N. Blaton, O. Peeters, J. Gal, 2004 .

4‐(4‐Bromophenyl)‐2,5‐diethoxycarbonyl‐6‐methylthieno[2,3‐b]pyridine

Esperanza Salfrán Solano, N. Blaton, O. Peeters, 2003 .

Copper(II) complexes of pentadentate 17-membered macrocyclic diamidodiamines with N, O or S as additional donors.

N. Blaton, G. Herman, W. Lippens, 2003, Acta crystallographica. Section C, Crystal structure communications.

(+)‐(3S,4R)‐Norcisapride hydrogen (2R,3R)‐tartrate monohydrate

N. Blaton, O. Peeters, 2002 .

p-Formamidobenzoic acid.

N. Blaton, O. Peeters, C. D. De Ranter, 2001, Acta crystallographica. Section C, Crystal structure communications.

9β,11β-Epoxy-3β-hydroxy-5α-androstan-17-one

N. Blaton, O. Peeters, C. J. Ranter, 2001 .

9α-Chloro-3β,11β-dihydroxy-5α-androstan-17-one

N. Blaton, O. Peeters, C. J. Ranter, 2001 .

(R)‐1‐{(2‐Oxo‐1,2‐dihydroquinolin‐6‐yl)[3‐(trifluoromethyl)phenyl]methyl}‐1H‐1,2,4‐triazol‐4‐ium bromide

N. Blaton, O. Peeters, C. J. Ranter, 2001 .

Tribenzylphosphine oxide.

N. Blaton, O. Peeters, C. D. De Ranter, 2000, Acta crystallographica. Section C, Crystal structure communications.

20-Hydroxyimino-5α-pregna-9(11),16-dien-3β-yl acetate and 17-oxo-5α-androst-9(11)-en-3β-yl acetate

N. Blaton, O. Peeters, C. J. Ranter, 2000 .

Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25.

P Augustijns, R. Busson, P. Augustijns, 2001, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

Improvement of the dissolution rate of artemisinin by means of supercritical fluid technology and solid dispersions.

P. Augustijns, G. Van den Mooter, N. Blaton, 2003, International journal of pharmaceutics.

Conformational analysis of C3′-substituted pyrimidine nucleosides by X-ray diffraction

N. Blaton, O. Peeters, C. J. Ranter, 1993 .

Synthesis and Structure of 2′,3′-Dideoxy-3′-fluoro-5-cyanouridine

P. Herdewijn, A. Aerschot, N. Blaton, 1990 .

2,5‐Diethoxycarbonyl‐6‐methyl‐4‐phenylthieno[2,3‐b]pyridine

N. Blaton, O. Peeters, C. J. Ranter, 2003 .

Ethyl 5‐ethoxymethylene‐2‐methyl‐6‐oxo‐4‐phenyl‐1,4,5,6‐tetrahydropyridine‐3‐carboxylate

N. Blaton, O. Peeters, C. J. Ranter, 2003 .

2-(4-Methoxyphenyl)aminobenzoic acid

N. Blaton, O. Peeters, C. J. Ranter, 2001 .

2-[(4-Carboxyphenyl)amino]-4-chlorobenzoic acid monohydrate

N. Blaton, O. Peeters, C. J. Ranter, 2001 .

Synthesis of homo-N-nucleosides, a series of C1' branched-chain nucleosides

P. Herdewijn, J. Rozenski, N. Blaton, 1996 .

Use of Cyclohexene Epoxides in the Preparation of Carbocyclic Nucleosides

P. Herdewijn, J. Rozenski, J. Balzarini, 1996 .

Pyridazine derivatives. Part 39: Reactivity of 5-iodopyridazin-3(2H)-ones in palladium-catalysed reactions

E. Sotelo, Alberto Coelho, N. Blaton, 2004 .

Design and molecular modelling of antisense pyranosyl oligonucleotides

N. Blaton, O. Peeters, C. J. Ranter, 1993 .

Structure of 1-(2-deoxy-β-D-ribopyranosyl)-5-iodouracil

P. Herdewijn, A. Aerschot, N. Blaton, 1991 .

Pharmaceutical performance of solid dispersions containing poly(ethylene glycol) 6000 and diazepam or temazepam

S. Verheyen, G. Van den Mooter, N. Blaton, 2004 .

Pharmaceutical performance of solid dispersions containing poly(ethylene) glycol 6000 and diazepam or temazepamInfluence of grinding

S. Verheyen, G. Van den Mooter, N. Blaton, 2003 .

Axial-equatorial interactions in chelates of β-diones. Crystal and molecular structure of bis(3-nitro-2,4-pentanedionato) copper(II)

N. Blaton, A. Stergiou, C. Tsiamis, 1998 .

A new method of synthesis of boltwoodite and of formation of sodium boltwoodite, uranophane, sklodowskite and kasolite from boltwoodite

N. Blaton, R. Vochten, L. Haverbeke, 1997 .

The structure and physicochemical characteristics of a synthetic phase compositionally intermediate between liebigite and andersonite

N. Blaton, R. Vochten, L. Haverbeke, 1994 .

Pyridazine Derivatives. Part 21: Synthesis and Structural Study of Novel 4-Aryl-2,5-dioxo-8-phenylpyrido[2,3-d]pyridazines

E. Sotelo, M. Suárez, N. Blaton, 2000 .

Synthesis, crystal structure and molecular modeling (AM1) of two 5-arylidene derivatives of Meldrum's acid

M. Suárez, N. Blaton, O. Peeters, 2000 .

Structure of the antiviral drug ethyl 4-{2-[1-(6-methyl-3-pyridazinyl)-4-piperidinyl]ethoxy}benzoate

N. Blaton, O. Peeters, C. J. Ranter, 1991 .

Synthesis and structural study of novel 1,4,5,6,7,8-hexahydroquinolines†

N. Martín, M. Suárez, N. Blaton, 2000 .

A joint experimental and theoretical structural study of novel substituted 2,5-dioxo-1,2,3,4,5,6,7,8-octahydroquinolines

N. Martín, M. Suárez, N. Blaton, 1999 .

X-Ray and theoretical structural study of novel 5,6,7,8-tetrahydrobenzo-4H-pyrans

N. Martín, M. Suárez, N. Blaton, 2002 .

5-amino-6-phenyl-1,6-dihydropyridazin-3(2H)-one.

E. Sotelo, M. Suárez, N. Blaton, 2000, Acta crystallographica. Section C, Crystal structure communications.

Isolation, purification, and stereochemistry of simmondsin

N. Blaton, P. Daenens, M. Cokelaere, 1993 .

Methyl [(1E)-(4-methoxyphenyl)methyleneamino]acetate

Héctor Novoa de Armas, Norbert Blaton, Margarita Suárez Navarro, 2007 .

N6-cyclopentyl-3'-substituted-xylofuranosyladenosines: a new class of non-xanthine adenosine A1 receptor antagonists.

A. IJzerman, J. K. von Frijtag Drabbe Künzel, P. Herdewijn, 1997, Journal of medicinal chemistry.

A straightforward synthesis and structure of unprecedented iminium salts of dihydropyrido[3,2-e][1,3]thiazines

N. Martín, Dolores Molero, R. Martínez‐Álvarez, 2006 .

Synthesis and Structural Study of 3,4‐Dihydro‐2(1H)‐pyridones and Isoxazolo[5,4‐b]pyridin‐6(7H)‐ones

N. Martín, M. Suárez, N. Blaton, 2000 .

Dichloro [1,5‐diphenylcarbazonato‐N,N′]dimercury (II), C13H10N4OHg2Cl2

N. Blaton, O. Peeters, C. J. Ranter, 2010 .

Synthesis and Conformational Study of 3-Hydroxy-4-(Hydroxymethyl)-1-Cyclohexanyl Purines and Pyrimidines.

E. De Clercq, P. Herdewijn, R. Busson, 1997, The Journal of organic chemistry.

Synthesis and structural study of new highly lipophilic 1,4-dihydropyridines

N. Martín, Dolores Molero, R. Martínez‐Álvarez, 2005 .

Structural study of highly halogenated dihydropyridine derivatives as potential calcium channel modulators

N. Martín, R. Martínez‐Álvarez, M. Suárez, 2003 .

Synthesis, crystal structure, and molecular modeling (AM1) of Methyl 6-chloro-4-(2-chlorophenyl)-5-formyl-2-methyl-1, 4-dihydropyridine-3-carboxylate

M. Suárez, N. Blaton, O. Peeters, 2000 .

Access to a new type of homo-C-nucleosides with a ''split'' 8-deazapurine via a 1,3-dipolar cycloaddition reaction

P. Herdewijn, N. Blaton, O. Peeters, 1997 .

3′-Deoxy-3′-hydroxymethyl-aldopentopyranosyl nucleoside synthesis. Part I

P. Herdewijn, J. Rozenski, N. Blaton, 1995 .

Synthesis of β configured 2′,3′-unsaturated pentopyranosyl nucleosides

P. Herdewijn, N. Blaton, B. Doboszewski, 1995 .

Salt formation in solid dispersions consisting of polyacrylic acid as a carrier and three basic model compounds resulting in very high glass transition temperatures and constant dissolution properties upon storage.

G. Verreck, J. Peeters, M. Brewster, 2005, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

Structure of 4(5)-nitroimidazole at 100 K

N. Blaton, O. Peeters, H. D. Bondt, 1993 .

Crystal structure of carnidazole form II from synchrotron X-ray powder diffraction: structural comparison with form I, the hydrated form and the low energy conformations in vacuo.

H. Schenk, G. Van den Mooter, N. Blaton, 2006, Journal of pharmaceutical sciences.

The Crystal Structure of 1‐{2,4‐Dichloro‐β‐ [(2,4‐Dichloro‐Benzyl)Oxy] Phenethyl} Imidazole Hemihydrate: Miconazole. 1/2 H2O

N. Blaton, O. Peeters, C. J. Ranter, 2010 .

cis-1-Acetyl-4-(4-{[2-(2,4-dichlorophenyl)-2-(1H-1-imidazolylmethyl)-1,3-dioxolan-4-yl]methoxy}phenyl)piperazine: ketoconazole. A crystal structure with disorder

N. Blaton, O. Peeters, C. J. Ranter, 1979 .

cis-2-sec-Butyl-4-{4-[4-(4-{[2-(2,4-dichlorophenyl)-2-(1H-1,2,4-triazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy}phenyl)-1-piperazinyl]phenyl}-2,4-dihydro-3H-1,2,4-triazol-3-one (Itraconazole)

N. Blaton, O. Peeters, C. J. Ranter, 1996 .

The crystal and molecular structure of trans-tetrakis(miconazole)cobalt(II) nitrate, (C18H14Cl4N2O)4Co(NO3)2

N. Blaton, O. Peeters, C. J. Ranter, 1978 .

Thermal Properties of Hot-Stage Extrudates of Itraconazole and Eudragit E100. Phase separation and polymorphism

J. Dressman, G. Verreck, P. Augustijns, 2002 .

Physico-chemical characterization of solid dispersions of temazepam with polyethylene glycol 6000 and PVP K30

Patrick Augustijns, Norbert Blaton, P. Augustijns, 1998 .

Solid state characterization and crystal structure from X-ray powder diffraction of two polymorphic forms of ranitidine base.

J. Martens, G. Van den Mooter, N. Blaton, 2009, Journal of pharmaceutical sciences.

Characterization of physico-chemical properties and pharmaceutical performance of sucrose co-freeze-dried solid nanoparticulate powders of the anti-HIV agent loviride prepared by media milling.

P Augustijns, L. Froyen, M. Brewster, 2007, International journal of pharmaceutics.

Synthesis and anti-HIV evaluation of 2',3'-dideoxyribo-5-chloropyrimidine analogues: reduced toxicity of 5-chlorinated 2',3'-dideoxynucleosides.

E. De Clercq, G. Janssen, J. Balzarini, 1990, Journal of medicinal chemistry.

Conformational Analysis of Substituent Effects on the Sugar Puckering Mode and the anti-HIV Activity of 2′,3′-Dideoxypyrimidine Nucleosides

P. Herdewijn, A. Aerschot, A. Van Aerschot, 1993 .

Unexpected Shift to a 4-Imino Tautomer Upon N4-Acylation of 5-Methylcytosin-1-yl Nucleoside Analogues

P. Herdewijn, R. Busson, A. Aerschot, 1999 .

ENANTIOSELECTIVE APPROACH TO THE SYNTHESIS OF CYCLOHEXANE CARBOCYCLIC NUCLEOSIDES

P. Herdewijn, R. Busson, J. Rozenski, 1998 .

5'-Deoxy congeners of 9-(3-amido-3-deoxy-beta-D-xylofuranosyl)-N(6)-cyclopentyladenine: new adenosine A(1) receptor antagonists and inverse agonists.

A. IJzerman, V. Vanheusden, P. Herdewijn, 2002, Journal of medicinal chemistry.

Synthesis and Anti-HIV Evaluation of 2′,3′-Dideoxyribo-5-chloropyrimidine Analogues: Reduced Toxicity of 5-Chlorinated 2′,3′-Dideoxynucleosides.

P. Herdewijn, G. Janssen, A. Aerschot, 1990 .

2'-Azido-2',3'-dideoxythymidine: synthesis and crystal structure of a 2'-substituted dideoxynucleoside.

E. De Clercq, P. Herdewijn, J. Balzarini, 1990, Antiviral Research.

Solid state properties of pure UC‐781 and solid dispersions with polyvinylpyrrolidone (PVP K30)

L. Naesens, J. Balzarini, P. Augustijns, 2001, The Journal of pharmacy and pharmacology.

Easy Synthesis and Different Conformational Behavior of Purine and Pyrimidine .beta.-D-glycero-Pent-2'-enopyranosyl Nucleosides

P. Herdewijn, N. Blaton, B. Doboszewski, 1995 .

The effect of pressure and temperature on the vibrational spectra of different hydrogen bonded systems.

R. Miao, N. Blaton, N Blaton, 2001, Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy.

Physical stability of solid dispersions of the antiviral agent UC-781 with PEG 6000, Gelucire 44/14 and PVP K30.

G. Van den Mooter, N. Blaton, R Kinget, 2002, International journal of pharmaceutics.

The interaction of chromium(VI), chromium(III) and chromium(II) with diphenylcarbazide, diphenylcarbazone and diphenylcarbadiazone

N. Blaton, O. Peeters, C. J. Ranter, 1977 .

Phase characterization of indomethacin in binary solid dispersions with PVP VA64 or Myrj 52.

G. Van den Mooter, N. Blaton, Héctor Novoa de Armas, 2007, International journal of pharmaceutics.

Polymorphism of Alprazolam (Xanax): a review of its crystalline phases and identification, crystallographic characterization, and crystal structure of a new polymorph (form III).

G. Van den Mooter, N. Blaton, O. Peeters, 2007, Journal of pharmaceutical sciences.

Contribution to the Complex-Formation of Diphenylcarbazone with cations. Complexes of Zinc, Nickel, and Cobalt

N. Blaton, O. Peeters, C. J. Ranter, 2010 .

Hydrogen-bonding patterns in rac-1-acetyl-5-methyl-2-thioxoimidazolidin-4-one.

N. Blaton, A. Bahsas, G. Delgado, 2007, Acta crystallographica. Section C, Crystal structure communications.

Mössbauer effect study of anapaite, Ca2Fe2+(PO4)2 · 4H2O, and of its oxidation products

N. Blaton, S. Eeckhout, E. De Grave, 1999 .

Structure of 3-{2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)piperidino]ethyl}-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one (risperidone)

N. Blaton, O. Peeters, C. J. Ranter, 1993 .

Crystal and molecular structure ofN-[1-(2-phenylethyl)-4-piperidinylium]-N-phenylpropanamide (fentanyl) citrate-toluene solvate

Oswald M. Peeters, Norbert Blaton, K. Goubitz, 1979 .

Structure of 1‐(2‐deoxy‐2‐fluoro‐α‐d‐arabinopyranosyl)‐5‐iodouracil

P. Herdewijn, A. Aerschot, N. Blaton, 1991 .

Structural studies of substituted 6,7-benzomorphan compounds. VI. (−)-(1R,5R,9R,13R)-2'-Hydroxy-5,9α-dimethyl-2-(tetrahydrofurfuryl)-6,7-benzomorphan and (−)-(1R,5R,9R,13S)-2'-hydroxy-5,9-dimethyl-2-(tetrahydrofurfuryl)-6,7-benzomorphan tartrate monohydrate

N. Blaton, O. Peeters, C. J. Ranter, 1982 .

A new synthetic method for proline diphenyl phosphonates

A. Lambeir, A. Haemers, K. Augustyns, 1995 .

A joint theoretical and experimental structural study of 5-carboxyethyl-3-(2 '-furfurylmethyl) tetrahydro-2H-1,3,5-thiadiazine-2-thione

N. Martín, M. Suárez, N. Blaton, 2001 .

Ethyl methyl 1,4-dihydro-4-(3-nitrophenyl)-2, 6-bis(1-piperidylmethyl)pyridine-3,5-dicarboxylate.

J. Duque, N. Blaton, O. Peeters, 2000, Acta Crystallographica Section C: Crystal Structure Communications.

Conformational properties of pyranosyl nucleosides by X-ray diffraction and modelling techniques

N. Blaton, O. Peeters, C. J. Ranter, 1993 .

(−)-(R)-N-[(3,4-Dihydro-2H-1-benzopyran-2-yl)methyl]-N'-(1,4,5,6-tetrahydro-2-pyrimidyl)-1,3-propanediaminium Dibromide

N. Blaton, O. Peeters, C. J. Ranter, 1996 .

Structures of 1-(2,3-dideoxy-erythro-α-D-hexopyranosyl)thymine and the 1-(2,3-dideoxy-erythro-β-D-hexopyranosyl)thymine.dioxane complex

P. Herdewijn, A. Aerschot, N. Blaton, 1991 .

Ethyl Methyl 1,4-Dihydro-4-(3-nitrophenyl)-2,6-bis (1-piperidylmethyl)pyridine-3,5-dicarboxylate.

J. Duque, N. Blaton, O. Peeters, 2001 .

Structure and absolute configuration of nebivolol: (±)‐(R*{S*[S*‐(S*)]})‐α,α'‐[iminobis(methylene)]bis(6‐fluoro‐3,4‐dihydro‐2H‐1‐benzopyran‐2‐methanol) (nebivolol) hydrochloride (I) and (+)‐(S{R[R‐(R)]})‐nebivolol hydrobromide dihydrate (II)

N. Blaton, O. Peeters, C. J. Ranter, 1993 .

1-(2,3-Dideoxy-erythro-β-d-hexopyranosyl)cytosine: an example of the conformational and stacking properties of pyranosyl pyrimidine nucleosides. A crystallographic and computational approach

P. Herdewijn, A. Aerschot, N. Blaton, 1992 .

Experimental and theoretical structural study of 2‐pyridyl‐ and 4‐hydroxyphenyl‐1,4‐dihydropyridine derivatives

N. Martín, M. Suárez, N. Blaton, 2000 .

Thermal characterization of the antiviral drug UC-781 and stability of its glass

Lieve Naesens, Jan Balzarini, Patrick Augustijns, 2001 .

2-(2-Methyl-5-nitro-1-imidazolyl)ethanol (metronidazole)

N. Blaton, O. Peeters, C. J. Ranter, 1979 .

Crystal structure of a (25R)-2α,3α-epoxy-5α-spirostan-6, 23-dione hemi-ethyl acetate solvate

N. Blaton, O. Peeters, C. D. De Ranter, 2000 .

Crystal structure of a novel tertiary phosphine coordination complex: dichlorobis(tribenzylphosphine)nickel(II)

J. López, J. Moreno, N. Blaton, 2000 .

Structure of the Neuroleptic Drug N-((1-Allyl-2-pyrrolidinyl)methyl)-6-methoxy-1H-benzotriazole-5-carboxamide Hydrochloride (Alizapride)

N. Blaton, O. Peeters, C. J. Ranter, 1990 .

Structure of the neuroleptic drug N‐[(1‐allyl‐2‐pyrrolidinyl)methyl]‐6‐methoxy‐1H‐benzotriazole‐5‐carboxamide hydrochloride (alizapride)

N. Blaton, O. Peeters, C. J. Ranter, 1990 .

THE CRYSTAL STRUCTURES OF SYNTHETIC POTASSIUM – TRANSITION-METAL ZIPPEITE-GROUP PHASES

N. Blaton, O. Peeters, R. Vochten, 2008 .

The structure and physicochemical characteristics of synthetic zippeite

N. Blaton, O. Peeters, K. Vanspringel, 1995 .

Structure of a nucleoside analogue, 3'-deoxy-2'-fluorothymidine

P. Herdewijn, A. Aerschot, N. Blaton, 1990 .

Structure of a nucleoside analogue, 3'-deoxy-3'-fluorothymidine.

N. Blaton, O. Peeters, C. D. De Ranter, 1990, Acta crystallographica. Section C, Crystal structure communications.

Synthesis of sodium weeksite and its transformation into weeksite

N. Blaton, O. Peeters, R. Vochten, 1997 .