Raphaël Rahmani

发表

Structural basis for modulation of a G-protein-coupled receptor by allosteric drugs

Albert C. Pan, R. Dror, D. Shaw, 2013, Nature.

3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis.

J. Baell, V. Avery, S. Charman, 2013, European journal of medicinal chemistry.

Structure‐Activity Studies of Truncated Latrunculin Analogues with Antimalarial Activity

Brian J. Smith, J. Baell, J. Baum, 2020, ChemMedChem.

trans-1,2-Disiloxybenzocyclobutene, an adequate partner for the auto-oxidation: EPR/spin trapping and theoretical studies.

Raphaël Rahmani, J. Parrain, L. Commeiras, 2014, Physical chemistry chemical physics : PCCP.

Copper‐Catalyzed Preparation of γ‐Alkylidenebutenolides and Isocoumarins under Mild Palladium‐Free Conditions

Raphaël Rahmani, J. Parrain, L. Commeiras, 2009 .

Dramatic influence of the substitution of alkylidene-5H-furan-2-ones in Diels-Alder cycloadditions with o-quinonedimethide as diene partner: en route to the CDEF polycyclic ring system of lactonamycin.

S. Dubois, Raphaël Rahmani, J. Parrain, 2012, Organic & biomolecular chemistry.

Diels-Alder cycloaddition of o-quinonedimethides and alkylidene-5H-furan-2-ones: new and rapid access to lambertellol cores and arthrinone derivatives.

Raphaël Rahmani, J. Parrain, L. Commeiras, 2010, Organic & biomolecular chemistry.

Copper-Catalyzed Preparation of γ-Alkylidenebutenolides and Isocoumarins under Mild Palladium-Free Conditions.

Raphaël Rahmani, J. Parrain, L. Commeiras, 2009 .

Pyridyl benzamides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei.

Christel A. S. Bergström, J. Baell, V. Avery, 2014, Journal of medicinal chemistry.

Direct-type aldol reactions of fluorenylidene-protected/activated glycine esters with aldehydes for the synthesis of β-hydroxy-α-amino acid derivatives.

Raphaël Rahmani, Y. Yamashita, S. Kobayashi, 2012, Chemistry, an Asian journal.

Hit-to-Lead Optimization of a Novel Class of Potent, Broad-Spectrum Trypanosomacides.

Ana Rodriguez, K. Read, J. Baell, 2016, Journal of medicinal chemistry.

Structural Basis for the Selective Binding of Inhibitors to 6-Hydroxymethyl-7,8-dihydropterin Pyrophosphokinase from Staphylococcus aureus and Escherichia coli.

J. Baell, Zhong-Chang Wang, T. Peat, 2016, Journal of medicinal chemistry.

Metabolomics and lipidomics reveal perturbation of sphingolipid metabolism by a novel anti-trypanosomal 3-(oxazolo[4,5-b]pyridine-2-yl)anilide

K. Read, J. Baell, M. McConville, 2016, Metabolomics.

Truncated Latrunculins as Actin Inhibitors Targeting Plasmodium falciparum Motility and Host Cell Invasion.

Christopher J. Tonkin, Brian J. Smith, J. Baell, 2016, Journal of medicinal chemistry.

6-Arylpyrazine-2-carboxamides: A New Core for Trypanosoma brucei Inhibitors.

J. Baell, V. Avery, S. Charman, 2015, Journal of medicinal chemistry.

Drug discovery and human African trypanosomiasis: a disease less neglected?

J. Baell, Raphaël Rahmani, Lori Ferrins, 2013, Future medicinal chemistry.

Crystal structure of the M5 muscarinic acetylcholine receptor

Alice E. Berizzi, C. Langmead, P. Sexton, 2019, Proceedings of the National Academy of Sciences.

Crystal structure of the M5muscarinic acetylcholine receptor.

Alice E. Berizzi, C. Langmead, P. Sexton, 2019 .

Structure-based design and development of functionalized Mercaptoguanine derivatives as inhibitors of the folate biosynthesis pathway enzyme 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase from Staphylococcus aureus.

J. Baell, Zhong-Chang Wang, J. Newman, 2014, Journal of medicinal chemistry.

Structure of the M5 muscarinic acetylcholine receptor (M5-T4L) bound to tiotropium

Alice E. Berizzi, C. Langmead, P. Sexton, 2019 .

Discovery of Potent N-Ethylurea Pyrazole Derivatives as Dual Inhibitors of Trypanosoma brucei and Trypanosoma cruzi.

Ana Rodriguez, J. Baell, V. Avery, 2019, ACS medicinal chemistry letters.

6-Arylpyrazine-2-carboxamides: A New Core for Trypanosoma brucei Inhibitors.

J. Baell, V. Avery, S. Charman, 2015, Journal of medicinal chemistry.

8-Mercaptoguanine Derivatives as Inhibitors of Dihydropteroate Synthase.

J. Baell, Zhong-Chang Wang, T. Peat, 2018, Chemistry.

Dramatic influence of the substitution of alkylidene-5H-furan-2-ones in Diels-Alder cycloadditions with o-quinonedimethide as diene partner: en route to the CDEF polycyclic ring system of lactonamycin.

S. Dubois, Raphaël Rahmani, J. Parrain, 2012, Organic & biomolecular chemistry.