Rasmus P Clausen

Pharmacological Characterization and Modeling of the Binding Sites of Novel 1,3-Bis(pyridinylethynyl)benzenes as Metabotropic Glutamate Receptor 5-Selective Negative Allosteric Modulators

Christina Mølck, David E. Gloriam, Hans Bräuner-Osborne, 2012, Molecular Pharmacology.

First Demonstration of a Functional Role for Central Nervous System Betaine/γ-Aminobutyric Acid Transporter (mGAT2) Based on Synergistic Anticonvulsant Action among Inhibitors of mGAT1 and mGAT2

Scott Slough, Arne Schousboe, A. Schousboe, 2005, Journal of Pharmacology and Experimental Therapeutics.

Structure-activity relationships of selective GABA uptake inhibitors.

Arne Schousboe, A. Schousboe, J. Greenwood, 2006, Current topics in medicinal chemistry.

Selective mGAT2 (BGT-1) GABA uptake inhibitors: design, synthesis, and pharmacological characterization.

Arne Schousboe, A. Schousboe, P. Krogsgaard‐Larsen, 2013, Journal of medicinal chemistry.

The glutamate receptor GluR5 agonist (S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid and the 8-methyl analogue: synthesis, molecular pharmacology, and biostructural characterization.

Peter Naur, Hans Bräuner-Osborne, P. Naur, 2009, Journal of medicinal chemistry.

Novel high-affinity and selective biaromatic 4-substituted gamma-hydroxybutyric acid (GHB) analogues as GHB ligands: design, synthesis, and binding studies.

Hans Bräuner-Osborne, P. Wellendorph, B. Frølund, 2008, Journal of medicinal chemistry.

Structure–Activity Relationships for Negative Allosteric mGluR5 Modulators

Christina Mølck, Hans Bräuner-Osborne, Kasper Harpsøe, 2012, ChemMedChem.

Selective inhibitors of GABA uptake: synthesis and molecular pharmacology of 4-N-methylamino-4,5,6,7-tetrahydrobenzo[d]isoxazol-3-ol analogues.

Arne Schousboe, A. Schousboe, P. Krogsgaard‐Larsen, 2005, Bioorganic & medicinal chemistry.