Laura De Luca

Synthesis and biological evaluation of novel antiviral agents as protein–protein interaction inhibitors

Zeger Debyser, Alba Chimirri, Rosaria Gitto, 2014, Journal of enzyme inhibition and medicinal chemistry.

A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series.

Myriam Witvrouw, Zeger Debyser, Alba Chimirri, 2008, Bioorganic & medicinal chemistry letters.

Analysis of the full-length integrase-DNA complex by a modified approach for DNA docking.

Pietro Monforte, Alba Chimirri, Alessandro Pedretti, 2003, Biochemical and biophysical research communications.

4-[1-(4-Fluorobenzyl)-4-hydroxy-1H-indol-3-yl]-2-hydroxy-4-oxobut-2-enoic acid as a prototype to develop dual inhibitors of HIV-1 integration process.

Zeger Debyser, Alba Chimirri, Rosaria Gitto, 2011, Antiviral research.

Pharmacophore-based design of HIV-1 integrase strand-transfer inhibitors.

Myriam Witvrouw, Zeger Debyser, Angela Rao, 2005, Journal of medicinal chemistry.

Computational strategies in discovering novel non-nucleoside inhibitors of HIV-1 RT.

Jan Balzarini, Angela Rao, Maria Zappalà, 2005, Journal of medicinal chemistry.

Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor.

Zeger Debyser, Alba Chimirri, Rosaria Gitto, 2010, Bioorganic & medicinal chemistry.

Discovery of a novel and highly potent noncompetitive AMPA receptor antagonist.

Alba Chimirri, Rosaria Gitto, Silvana Quartarone, 2003, Journal of medicinal chemistry.

QSAR study of anticonvulsant negative allosteric modulators of the AMPA receptor.

Alba Chimirri, Gabriele Costantino, Antonio Macchiarulo, 2004, Journal of medicinal chemistry.