Peter M Blumberg

发表

Screening TRPV1 antagonists for the treatment of pain: lessons learned over a decade

P. Blumberg, A. Szallasi, József Lázár, 2009, Expert opinion on drug discovery.

2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent transient receptor potential vanilloid 1 (TRPV1) antagonists: structure-activity relationships of 2-amino derivatives in the N-(6-trifluoromethylpyridin-3-ylmethyl) C-region.

Dong Wook Kang, Sun Choi, Mi-Yeon Kim, 2012, Journal of medicinal chemistry.

Crystal structure of the Cys2 activator-binding domain of protein kinase Cδ in complex with phorbol ester

J. Hurley, Gongyi Zhang, M. Kazanietz, 1995, Cell.

Stereospecific high-affinity TRPV1 antagonists: chiral N-(2-benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide analogues.

Dong Wook Kang, Attila Toth, HyungChul Ryu, 2008, Journal of medicinal chemistry.

Role of phorbol ester localization in determining protein kinase C or RasGRP3 translocation: real-time analysis using fluorescent ligands and proteins.

Shaomeng Wang, P. Blumberg, G. Hur, 2005, Molecular cancer therapeutics.

N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues: novel potent and high affinity antagonists and partial antagonists of the vanilloid receptor.

Ji-Min Kim, Attila Toth, Jiyoun Lee, 2003, Journal of medicinal chemistry.

Pyridine C-region analogs of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

HyungChul Ryu, Suyoung Yoon, K. Schiene, 2015, European journal of medicinal chemistry.

Absolute quantitation of endogenous proteins with precision and accuracy using a capillary Western system.

P. Blumberg, P. Goldsmith, Peter M Blumberg, 2013, Analytical biochemistry.

Synthesis and biological evaluation of [¹¹C]SB366791: a new PET-radioligand for in vivo imaging of the TRPV1 receptor.

Koen Van Laere, Guy Bormans, Alfons Verbruggen, 2013, Nuclear medicine and biology.

2-(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists: structure activity relationships of the 2-oxy pyridine C-region.

Dong Wook Kang, Sun Choi, HyungChul Ryu, 2013, European journal of medicinal chemistry.

Molecular Determinants of Vanilloid Sensitivity in TRPV1*

Attila Toth, Vellarkad N Viswanadhan, J. Treanor, 2004, Journal of Biological Chemistry.