E. Kelly

发表

Agonist‐selective mechanisms of GPCR desensitization

E. Kelly, C. P. Bailey, G. Henderson, 2008, British journal of pharmacology.

Octimibate, a potent non‐prostanoid inhibitor of platelet aggregation, acts via the prostacyclin receptor

T. Rink, J. Macdermot, T. Hallam, 1991, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Catalytic receptors

Stephen P. H. Alexander, C. Southan, D. Fabbro, 2021, British journal of pharmacology.

Agonist‐independent internalization of metabotropic glutamate receptor 1a is arrestin‐ and clathrin‐dependent and is suppressed by receptor inverse agonists

S. Mundell, P. Roberts, E. Kelly, 2004, Journal of neurochemistry.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Nuclear hormone receptors

Adam J Pawson, Stephen P. H. Alexander, C. Southan, 2017, British journal of pharmacology.

The Concise Guide to PHARMACOLOGY 2015/16: Transporters

Adam J Pawson, Stephen P. H. Alexander, C. Southan, 2015, British journal of pharmacology.

The Concise Guide to PHARMACOLOGY 2015/16: Enzymes

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2015, British journal of pharmacology.

Effect of Tamoxifen and Brain-Penetrant Protein Kinase C and c-Jun N-Terminal Kinase Inhibitors on Tolerance to Opioid-Induced Respiratory Depression in Mice

Sarah L. Withey, W. Dewey, E. Kelly, 2017, The Journal of Pharmacology and Experimental Therapeutics.

Effect of tamoxifen and brain penetrant PKC and JNK inhibitors on tolerance to opioid-induced respiratory depression in mice

Sarah L. Withey, W. Dewey, E. Kelly, 2017 .

Elucidating agonist-selective mechanisms of G protein-coupled receptor desensitization

E. Kelly, C. Bailey, 2011 .

A Novel G Protein–Biased Agonist at the δ Opioid Receptor with Analgesic Efficacy in Models of Chronic Pain

V. Tékus, Z. Helyes, E. Kelly, 2019, The Journal of Pharmacology and Experimental Therapeutics.

A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor

Andrew M. Piggott, R. Sessions, A-M Wang, 2019, Proceedings of the National Academy of Sciences.

Desensitization of endogenously expressed delta-opioid receptors: no evidence for involvement of G protein-coupled receptor kinase 2.

E. Kelly, J. Willets, 2001, European journal of pharmacology.

Agonist-Selective Mechanisms of μ-Opioid Receptor Desensitization in Human Embryonic Kidney 293 Cells

S. Mundell, S. Oldfield, E. Kelly, 2006, Molecular Pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Enzymes

Adam J Pawson, Stephen P. H. Alexander, C. Southan, 2017, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Transporters

Adam J Pawson, Stephen P. H. Alexander, C. Southan, 2017, British journal of pharmacology.

Regulation of P2Y1 Receptor Traffic by Sorting Nexin 1 is Retromer Independent

S. Mundell, P. Cullen, E. Kelly, 2010, Traffic.

The novel μ‐opioid receptor agonist PZM21 depresses respiration and induces tolerance to antinociception

S. Husbands, W. Dewey, E. Kelly, 2018, British journal of pharmacology.

Opioid receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

E. J. Simon, H. Ueda, M. Bruchas, 2019, IUPHAR/BPS Guide to Pharmacology CITE.

Morphine‐induced internalization of the L83I mutant of the rat μ‐opioid receptor

S. Mundell, S. Oldfield, C. Krasel, 2015, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: G protein‐coupled receptors

Arthur Christopoulos, Christopher Southan, Stephen PH Alexander, 2017, British journal of pharmacology.

Fentanyl depression of respiration: comparison with heroin and morphine

W. Dewey, E. Kelly, G. Henderson, 2019, bioRxiv.

Oxycodone‐induced tolerance to respiratory depression: reversal by ethanol, pregabalin and protein kinase C inhibition

W. Dewey, E. Kelly, G. Henderson, 2018, British journal of pharmacology.

Adenosine receptor desensitization and trafficking.

S. Mundell, E. Kelly, 2011, Biochimica et biophysica acta.

Evidence for co-expression and desensitization of A2a and A2b adenosine receptors in NG108-15 cells.

S. Mundell, E. Kelly, 1998, Biochemical pharmacology.

Ligand bias at the μ-opioid receptor.

E. Kelly, 2013, Biochemical Society transactions.

The Effect of Protein Kinase C and G Protein-coupled Receptor Kinase Inhibition on Tolerance Induced by ␮-opioid Agonists of Different Efficacy

W. Dewey, E. Kelly, G. Henderson, 2022 .

Pre-treatment with a PKC or PKA inhibitor prevents the development of morphine tolerance but not physical dependence in mice

W. Dewey, E. Kelly, G. Henderson, 2008, Brain Research.

Evidence for an important role of protein phosphatases in the mechanism of morphine tolerance

W. Dewey, E. Kelly, G. Henderson, 2007, Brain Research.

Pathways for internalization and recycling of the chemokine receptor CCR5.

P. Strange, E. Kelly, A. Mueller, 2002, Blood.

Internalization and desensitization of the oxytocin receptor is inhibited by Dynamin and clathrin mutants in human embryonic kidney 293 cells.

S. Mundell, C. McArdle, E. Kelly, 2006, Molecular endocrinology.

Signaling and antiproliferative effects of type I and II gonadotropin-releasing hormone receptors in breast cancer cells.

C. McArdle, E. Kelly, A. R. Finch, 2004 .

Identification of phosphorylation sites in the COOH‐terminal tail of the μ‐opioid receptor

S. Oldfield, A. Tobin, J. Benovic, 2013, Journal of neurochemistry.

Chronic ethanol promotes the neuronal differentiation of NG108-15 cells independently of toxin-sensitive G-proteins.

M. Connor, P. K. Harrison, E. Kelly, 1997, Environmental toxicology and pharmacology.

Enhanced expression of G protein‐coupled receptor kinase 2 selectively increases the sensitivity of A2A adenosine receptors to agonist‐induced desensitization

S. Mundell, J. Benovic, J. Luty, 1998, British journal of pharmacology.

A dominant negative mutant of the G protein-coupled receptor kinase 2 selectively attenuates adenosine A2 receptor desensitization.

S. Mundell, J. Benovic, E. Kelly, 1997, Molecular pharmacology.

Arrestin isoforms dictate differential kinetics of A2B adenosine receptor trafficking.

S. Mundell, J. Benovic, E. Kelly, 2000, Biochemistry.

The effect of inhibitors of receptor internalization on the desensitization and resensitization of three Gs‐coupled receptor responses

S. Mundell, E. Kelly, 1998, British journal of pharmacology.

G protein‐coupled receptor kinase 6 (GRK6) selectively regulates endogenous secretin receptor responsiveness in NG108‐15 cells

E. Kelly, J. Willets, R. Ghadessy, 2003, British journal of pharmacology.

Gsα-dependent and -independent desensitisation of prostanoid IP receptor-activated adenylyl cyclase in NG108-15 cells

Robert J. Williams, E. Kelly, 1994 .

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Introduction and Other Protein Targets

Stephen P. H. Alexander, C. Southan, D. Fabbro, 2021, British journal of pharmacology.

Agonist‐induced internalization of the metabotropic glutamate receptor 1a is arrestin‐ and dynamin‐dependent

S. Mundell, E. Kelly, G. Pula, 2001, Journal of neurochemistry.

Efficacy and ligand bias at the μ‐opioid receptor

E. Kelly, 2013, British journal of pharmacology.

Morphine‐induced respiratory depression is independent of β‐arrestin2 signalling

S. Schulz, E. Kelly, G. Henderson, 2020, British journal of pharmacology.

The subtleties of µ‐opioid receptor phosphorylation

E. Kelly, 2011, British journal of pharmacology.

Regulation of gonadotropin-releasing hormone receptors by protein kinase C: inside out signalling and evidence for multiple active conformations.

C. McArdle, C. Caunt, E. Kelly, 2004, Endocrinology.

Inhibition of ADP-ribosyltransferase increases synthesis of Gs alpha in neuroblastoma x glioma hybrid cells and reverses iloprost-dependent heterologous loss of fluoride-sensitive adenylate cyclase.

L. Donnelly, R. Boyd, J. Macdermot, 1995, Biochemical pharmacology.

NaF and guanine nucleotides modulate adenylate cyclase activity in NG108‐15 cells by interacting with both Gs and Gi

J. Macdermot, E. Kelly, M. Keen, 1990, British journal of pharmacology.

Critical Assessment of G Protein-Biased Agonism at the μ-Opioid Receptor.

S. Schulz, M. Canals, E. Kelly, 2020, Trends in pharmacological sciences.

Rapid Agonist-induced Desensitization and Internalization of the A2B Adenosine Receptor Is Mediated by a Serine Residue Close to the COOH Terminus*

S. Mundell, J. Benovic, E. Kelly, 2001, The Journal of Biological Chemistry.

Effects of acute and chronic ethanol on cyclic AMP accumulation in NG108‐15 cells: differential dependence of changes on extracellular adenosine

P. K. Harrison, E. Kelly, Rj Williams, 1995, British journal of pharmacology.

Measurement of adenylyl cyclase activity in cell membranes.

E. Kelly, R. Williams, 1995, Methods in molecular biology.

The Concise Guide to PHARMACOLOGY 2015/16: G protein‐coupled receptors

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2015, British journal of pharmacology.

Agonist‐induced internalization of metabotropic glutamate receptor 1A: structural determinants for protein kinase C‐ and G protein‐coupled receptor kinase‐mediated internalization

S. Mundell, P. Roberts, E. Kelly, 2003, Journal of neurochemistry.

Metabotropic glutamate receptor 1 internalization induced by muscarinic acetylcholine receptor activation: differential dependency of internalization of splice variants on nonvisual arrestins.

S. Mundell, D. Holman, P. Roberts, 2002, Molecular pharmacology.

G protein-coupled receptor kinases 3 and 6 use different pathways to desensitize the endogenous M3 muscarinic acetylcholine receptor in human SH-SY5Y cells.

R. Challiss, E. Kelly, S. Nahorski, 2001, Molecular pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Catalytic receptors

Christopher Southan, John A Peters, Elena Faccenda, 2019, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Transporters

Christopher Southan, John A Peters, Elena Faccenda, 2019, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Ion channels

Christopher Southan, Jörg Striessnig, John A Peters, 2019, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: G protein‐coupled receptors

Arthur Christopoulos, Christopher Southan, John A Peters, 2019, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Enzymes

Christopher Southan, John A Peters, Elena Faccenda, 2019, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Overview

Arthur Christopoulos, Christopher Southan, Stephen PH Alexander, 2017, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Other ion channels

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2017, British journal of pharmacology.

Involvement of PKCα and G‐protein‐coupled receptor kinase 2 in agonist‐selective desensitization of µ‐opioid receptors in mature brain neurons

S. Oldfield, E. Kelly, G. Henderson, 2009, British journal of pharmacology.

THEMED ISSUE: GPCR RESEARCH PAPER Involvement of PKCa and G-protein-coupled receptor kinase 2 in agonist-selective desensitization of m-opioid receptors in mature brain neurons

S. Oldfield, A. Teschemacher, C. McArdle, 2009 .

Endomorphin-2: A Biased Agonist at the μ-Opioid Receptor

S. Mundell, C. McArdle, S. Charlton, 2012, Molecular Pharmacology.

Cyclic AMP produces desensitization of prostacyclin and adenosine A2 receptors in hybrid cell lines but does not affect Gs function.

K. Docherty, J. Macdermot, E. Kelly, 1992, Biochimica et biophysica acta.

Primate vascular responses to octimibate, a non‐prostanoid agonist at the prostacyclin receptor

E. F. Smith, T. Rink, A. Heagerty, 1991, British journal of pharmacology.

Segregation of discrete Gsα‐mediated responses that accompany homologous or heterologous desensitization in two related somatic hybrids

J. Macdermot, E. Kelly, M. Keen, 1990, British journal of pharmacology.

A selective binding site for 3H-NECA that is not an adenosine A2 receptor.

J. Macdermot, E. Kelly, M. Keen, 1989, Biochemical pharmacology.

Assay of G protein-coupled receptor kinase activity by rhodopsin phosphorylation.

E. Kelly, A. Gagnon, 1997, Methods in molecular biology.

Prolonged ethanol administration prevents the development of tolerance to morphine-induced respiratory depression.

Joanne Roberts, W. Dewey, E. Kelly, 2019, Drug and alcohol dependence.

Ethanol Reversal of Tolerance to the Respiratory Depressant Effects of Morphine

Sarah L. Withey, A. Lingford-Hughes, M. Hickman, 2015, Neuropsychopharmacology.

Role of protein kinase C and μ-opioid receptor (MOPr) desensitization in tolerance to morphine in rat locus coeruleus neurons

W. Dewey, E. Kelly, G. Henderson, 2009, The European journal of neuroscience.

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Nuclear hormone receptors

Stephen P. H. Alexander, C. Southan, K. Korach, 2021, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Introduction and Other Protein Targets

Arthur Christopoulos, Adam J. Pawson, Michael Spedding, 2019, British Journal of Pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein‐coupled receptors

Stephen P. H. Alexander, Leigh A. Stoddart, Kalyan C. Tirupula, 2021, British journal of pharmacology.

Deletion of the distal COOH‐terminus of the A2B adenosine receptor switches internalization to an arrestin‐ and clathrin‐independent pathway and inhibits recycling

S. Mundell, T. Palmer, J. Benovic, 2010, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Enzymes

Stephen P. H. Alexander, C. Southan, D. Fabbro, 2021, British journal of pharmacology.

Agonist-selective mechanisms of μ-opioid receptor ( MOR ) desensitization in HEK 293 cells

S. Mundell, S. Oldfield, E. Kelly, 2006 .

μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization

S. Charlton, C. Krasel, W. Dewey, 2010, Molecular Pharmacology.

Desensitization and internalization of metabotropic glutamate receptor 1a following activation of heterologous Gq/11-coupled receptors.

S. Mundell, P. Roberts, E. Kelly, 2004, Biochemistry.

Pertussis toxin separates two muscarinic receptor-effector mechanisms in the striatum.

E. Kelly, S. Nahorski, T. A. Rooney, 1985, European journal of pharmacology.

How important is protein kinase C in mu-opioid receptor desensitization and morphine tolerance?

W. Dewey, E. Kelly, G. Henderson, 2006, Trends in pharmacological sciences.

Interaction With the Lipid Membrane Influences Fentanyl Pharmacology

R. Sessions, S. Charlton, R. Corey, 2022, Advances in Drug and Alcohol Research.

Protein Kinase C Activation Enhances Morphine-Induced Rapid Desensitization of μ-Opioid Receptors in Mature Rat Locus Ceruleus Neurons

E. Kelly, G. Henderson, C. Bailey, 2004, Molecular Pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Ion channels

Adam J Pawson, Stephen P. H. Alexander, L. Kaczmarek, 2021, British journal of pharmacology.

The anomalous pharmacology of fentanyl

Graeme Henderson, E. Kelly, Katy J Sutcliffe, 2021, British journal of pharmacology.

A Biased View of μ-Opioid Receptors?

E. Kelly, Alexandra E. Conibear, 2019, Molecular Pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Ligand‐gated ion channels

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2017, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Voltage‐gated ion channels

Christopher Southan, Stephen PH Alexander, Jörg Striessnig, 2017, British journal of pharmacology.

The Concise Guide to PHARMACOLOGY 2015/16: Ligand‐gated ion channels

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2015, British journal of pharmacology.

Inverse agonism at the P2Y12 receptor and ENT1 transporter blockade contribute to platelet inhibition by ticagrelor.

S. Mundell, A. Mumford, E. Kelly, 2016, Blood.

Dopamine D-2 receptors inhibit D-1 stimulated cyclic AMP accumulation in striatum but not limbic forebrain

E. Kelly, S. Nahorski, 1987, Naunyn-Schmiedeberg's Archives of Pharmacology.

Selective Reduction in A2 Adenosine Receptor Desensitization Following Antisense‐Induced Suppression of G Protein‐Coupled Receptor Kinase 2 Expression

J M Willets, J L Parent, J L Benovic, 1999, Journal of neurochemistry.

Somatostatin Receptor Desensitization in NG108-15 Cells

J. Luty, V. Beaumont, E. Kelly, 1998, The Journal of Biological Chemistry.

The Concise Guide to PHARMACOLOGY 2015/16: Voltage‐gated ion channels

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2015, British journal of pharmacology.

Arrestin Scaffolds NHERF1 to the P2Y12 Receptor to Regulate Receptor Internalization*

S. Mundell, E. Kelly, M. Cunningham, 2012, The Journal of Biological Chemistry.

The Concise Guide to PHARMACOLOGY 2015/16: Catalytic receptors

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2015, British journal of pharmacology.

μ-Opioid receptor desensitization: homologous or heterologous?

J. Lowe, E. Kelly, G. Henderson, 2012, The European journal of neuroscience.

Novel GPCR paradigms at the μ‐opioid receptor

A. Christopoulos, M. Canals, E. Kelly, 2015, British journal of pharmacology.

The opioid receptor pharmacology of GSK1521498 compared to other ligands with differential effects on compulsive reward-related behaviours

E. Bullmore, S. Mundell, P. Nathan, 2014, Psychopharmacology.

Ethanol differentially regulates guanine nucleotide-binding protein alpha subunit expression in NG108-15 cells independently of extracellular adenosine.

E. Kelly, P. Horne, M. A. Veale, 1993, Molecular pharmacology.

A novel G protein‐biased agonist at the μ opioid receptor induces substantial receptor desensitisation through G protein‐coupled receptor kinase

S. Schulz, S. Husbands, L. Toll, 2020, British journal of pharmacology.

G‐protein‐coupled receptor dephosphorylation at the cell surface

Eamonn Kelly, E. Kelly, 2006, British journal of pharmacology.

Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts

N. Marrion, S. Oldfield, A. Randall, 2009, Molecular Pharmacology.

ARF6 Activated by the LHCG Receptor through the Cytohesin Family of Guanine Nucleotide Exchange Factors Mediates the Receptor Internalization and Signaling*

E. Kelly, V. Kanamarlapudi, A. López Bernal, 2012, The Journal of Biological Chemistry.

Endocytosis of G Protein-Coupled Receptors Is Regulated by Clathrin Light Chain Phosphorylation

S. Mundell, E. Smythe, E. Kelly, 2012, Current Biology.

THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Transporters

Stephen P. H. Alexander, C. Southan, P. Dawson, 2021, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Catalytic receptors

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2017, British journal of pharmacology.

Guanine nucleotide sensitivity of [3H]iloprost binding to prostacyclin receptors.

J. Macdermot, E. Kelly, M. Keen, 1991, European journal of pharmacology.

Role of G Protein–Coupled Receptor Kinases 2 and 3 in μ-Opioid Receptor Desensitization and Internalization

Sarah L. Withey, C. Chavkin, S. Husbands, 2015, Molecular Pharmacology.

Biased Agonism: Lessons from Studies of Opioid Receptor Agonists.

Graeme Henderson, E. Kelly, Alexandra E. Conibear, 2022, Annual review of pharmacology and toxicology.

Ethanol Reversal of Cellular Tolerance to Morphine in Rat Locus Coeruleus Neurons

Sarah L. Withey, S. Oldfield, W. Dewey, 2013, Molecular Pharmacology.

μ-Opioid Receptor Desensitization in Mature Rat Neurons: Lack of Interaction between DAMGO and Morphine

E. Kelly, G. Henderson, C. Bailey, 2003, The Journal of Neuroscience.

Role of Acetaldehyde in Ethanol Reversal of Tolerance to Morphine-Induced Respiratory Depression in Mice

Graeme Henderson, W. Dewey, E. Kelly, 2022, Advances in Drug and Alcohol Research.

Ethanol and pregabalin reverse oxycodone tolerance

W. Dewey, E. Kelly, G. Henderson, 2018 .

Fentanyl binds to the μ-opioid receptor via the lipid membrane and transmembrane helices

R. Sessions, S. Charlton, R. Corey, 2021, bioRxiv.

Centaurin-α1, an ADP-Ribosylation Factor 6 GTPase Activating Protein, Inhibits β2-Adrenoceptor Internalization

S. Mundell, K. Venkateswarlu, E. Kelly, 2005, Molecular Pharmacology.

Centaurin-alpha 1, an ADP-ribosylation factor 6 GTPase activating protein, inhibits beta 2-adrenoceptor internalization.

S. Mundell, K. Venkateswarlu, E. Kelly, 2005, Molecular pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Introduction and Other Protein Targets

Arthur Christopoulos, Christopher Southan, Jörg Striessnig, 2019, British journal of pharmacology.

Opioid receptors in GtoPdb v.2023.1 Opioid receptors in GtoPdb v.2023.1

E. J. Simon, H. Ueda, M. Bruchas, 2023 .

Role of protein kinase C and μ-opioid receptor (MOPr) desensitization in tolerance to morphine in rat locus coeruleus neurons

W. Dewey, E. Kelly, G. Henderson, 2009, The European Journal of Neuroscience.

Role of G Protein – Coupled Receptor Kinases 2 and 3 in m-Opioid Receptor Desensitization and Internalization s

Sarah L. Withey, C. Chavkin, S. Husbands, 2015 .

The opioid receptor pharmacology of GSK1521498 compared to other ligands with differential effects on compulsive reward-related behaviours

E. Bullmore, S. Mundell, P. Nathan, 2014, Psychopharmacology.

Neurochemical and behavioural evidence that dopamine D-2 receptors in striatum couple to the Ni regulatory protein and inhibition of cyclic AMP accumulation

E. Kelly, S. Nahorski, A. L. Willcocks, 1987, Naunyn-Schmiedeberg's Archives of Pharmacology.

Attempts to Characterise Dopamine Receptor-Effector Mechanisms in the Brain

E. Kelly, S. Nahorski, 1988 .

Drug Binding Poses Relate Structure with Efficacy in the μ Opioid Receptor

Eamonn Kelly, Graeme Henderson, Richard B. Sessions, 2017, Journal of molecular biology.

THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Nuclear hormone receptors

Christopher Southan, John A Peters, Elena Faccenda, 2019, British journal of pharmacology.

Analysis of mGluR1a constitutive internalization using a pulse-chase enzyme-linked immuno-sorbant assay (ELISA).

S. Mundell, P. Roberts, E. Kelly, 2005, Journal of biochemical and biophysical methods.

Second messenger‐dependent protein kinases and protein synthesis regulate endogenous secretin receptor responsiveness

E. Kelly, R. Ghadessy, 2002, British journal of pharmacology.

Gs alpha-dependent and -independent desensitisation of prostanoid IP receptor-activated adenylyl cyclase in NG108-15 cells.

E. Kelly, R. Williams, 1994, European Journal of Pharmacology.

The Concise Guide to PHARMACOLOGY 2015/16: Nuclear hormone receptors

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2015, British journal of pharmacology.

Chronic Ethanol Reduces Immunologically Detectable Gqα/11α in NG108–15 Cells

E. Kelly, Robert J Williams, 1993 .

Metabotropic glutamate receptor mGlu2 is resistant to homologous agonist-induced desensitization but undergoes protein kinase C-mediated heterologous desensitization.

D. Jane, P. Roberts, P. Howson, 2010, European journal of pharmacology.

The Concise Guide to PHARMACOLOGY 2015/16: Other ion channels

Christopher Southan, Stephen PH Alexander, Eamonn Kelly, 2015, British journal of pharmacology.

Expression and desensitisation of A2 purinoceptors on cultured bovine aortic endothelial cells.

J. Macdermot, E. Kelly, M. Keen, 1989, Cardiovascular research.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Voltage‐gated ion channels

Adam J Pawson, Stephen P. H. Alexander, C. Southan, 2017, British journal of pharmacology.

signalling with ability to activate internalization

S. Charlton, C. Krasel, W. Dewey, 2010 .

Opioid receptors in GtoPdb v.2021.3

E. J. Simon, H. Ueda, M. Bruchas, 2021, IUPHAR/BPS Guide to Pharmacology CITE.

Carfentanil is a β‐arrestin‐biased agonist at the μ opioid receptor

Graeme Henderson, R. Sessions, S. Groom, 2023, British journal of pharmacology.

Methadone: does it really have low efficacy at μ-opioid receptors?

N. Marrion, E. Kelly, G. Henderson, 2008, Neuroreport.

C‐terminal splice variants of the μ‐opioid receptor: existence, distribution and functional characteristics

S. Oldfield, E. Kelly, G. Henderson, 2008, Journal of neurochemistry.

The Concise Guide to PHARMACOLOGY 2015/16: Catalytic receptors

Adam J Pawson, Stephen P. H. Alexander, C. Southan, 2015, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Voltage‐gated ion channels

Adam J Pawson, Stephen P. H. Alexander, C. Southan, 2017, British journal of pharmacology.

THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Ligand‐gated ion channels

Adam J Pawson, Stephen P. H. Alexander, C. Southan, 2017, British journal of pharmacology.

Novel GPCR paradigms at the μ‐opioid receptor

A. Christopoulos, M. Canals, E. Kelly, 2015, British journal of pharmacology.

Adenosine receptor desensitization and trafficking.

S. Mundell, E. Kelly, 2011, Biochimica et biophysica acta.

Drug Binding Poses Relate Structure with Efficacy in the μ Opioid Receptor

R. Sessions, E. Kelly, G. Henderson, 2017, Journal of molecular biology.

ARF6 Activated by the LHCG Receptor through the Cytohesin Family of Guanine Nucleotide Exchange Factors Mediates the Receptor Internalization and Signaling*

E. Kelly, V. Kanamarlapudi, A. López Bernal, 2012, The Journal of Biological Chemistry.

Activation of cyclic AMP-dependent protein kinase inhibits the desensitization and internalization of metabotropic glutamate receptors 1a and 1b.

S. Mundell, D. Jane, P. Roberts, 2004, Molecular pharmacology.

The Concise Guide to PHARMACOLOGY 2023/24: Catalytic receptors

J. Stasch, J. Armstrong, E. Faccenda, 2023, British journal of pharmacology.

Opus: University of Bath Online Publication Store Ethanol Reversal of Tolerance to the Respiratory Depressant Effects of Morphine

Sarah L. Withey, A. Lingford-Hughes, M. Hickman, 2022 .

The Concise Guide to PHARMACOLOGY 2023/24: Introduction and Other Protein Targets

J. Cidlowski, T. Arumugam, C. Sobey, 2023, British journal of pharmacology.

The Effect of Protein Kinase C and G Protein-Coupled Receptor Kinase Inhibition on Tolerance Induced by μ-Opioid Agonists of Different Efficacy

E. Kelly, B. H. Gabra, L. Hull, 2010, Journal of Pharmacology and Experimental Therapeutics.

The Concise Guide to PHARMACOLOGY 2023/24: Ion channels

J. Trimmer, W. Catterall, S. Grissmer, 2023, British journal of pharmacology.

The Concise Guide to PHARMACOLOGY 2023/24: Enzymes

J. Stasch, C. Dessauer, J. Armstrong, 2023, British journal of pharmacology.

Role of G Protein–Coupled Receptor Kinases 2 and 3 in μ-Opioid Receptor Desensitization and Internalization

Sarah L. Withey, C. Chavkin, S. Husbands, 2015, Molecular Pharmacology.

The Concise Guide to PHARMACOLOGY 2023/24: Transporters

D. Thwaites, J. Armstrong, E. Faccenda, 2023, British journal of pharmacology.

The Concise Guide to PHARMACOLOGY 2023/24: Nuclear hormone receptors

J. Cidlowski, J. Armstrong, E. Faccenda, 2023, British journal of pharmacology.