E. Mouray

发表

Detection, characterization, and screening of heme-binding molecules by mass spectrometry for malaria drug discovery.

A. Maciuk, P. Grellier, Katalina Muñoz-Durango, 2012, Analytical chemistry.

One-pot microwave-assisted synthesis and antimalarial activity of ferrocenyl benzodiazepines

Till Bousquet, P. Grellier, E. Mouray, 2011 .

Targeted Isolation of Hemitheion from Mostuea brunonis, a Proposed Biosynthetic Intermediate of Theionbrunonines.

M. Beniddir, P. Grellier, E. Mouray, 2021, Journal of natural products.

Streamlined targeting of Amaryllidaceae alkaloids from the bulbs of Crinum scillifolium using spectrometric and taxonomically-informed scoring metabolite annotations.

J. Gallard, M. Beniddir, P. Grellier, 2020, Phytochemistry.

Sesquiterpene lactones from the endemic Cape Verdean Artemisia gorgonum.

O. Thomas, Soizic Prado, E. Mouray, 2008, Phytochemistry.

Antiplasmodial Biodereplication Based on Highly Efficient Methods

A. Maciuk, J. Gallard, P. Grellier, 2020 .

Synthesis of Novel G Factor or Chloroquine-Artemisinin Hybrids and Conjugates with Potent Antiplasmodial Activity.

P. Grellier, E. Mouray, C. André-Barrès, 2020, ACS medicinal chemistry letters.

Antiplasmodial activity and cytotoxicity of bis-, tris-, and tetraquinolines with linear or cyclic amino linkers.

E. Davioud‐Charvet, C. Sergheraert, L. Maes, 2001, Journal of Medicinal Chemistry.

Characterization of PfDYN2, a dynamin-like protein of Plasmodium falciparum expressed in schizonts.

Sébastien Charneau, P. Grellier, I. Florent, 2007, Microbes and infection.

Highly improved antiparasitic activity after introduction of an N-benzylimidazole moiety on protein farnesyltransferase inhibitors.

P. Grellier, S. Cojean, P. Loiseau, 2016, European journal of medicinal chemistry.

Introduction of methionine mimics on 3-arylthiophene: influence on protein farnesyltransferase inhibition and on antiparasitic activity

P. Grellier, S. Cojean, P. Loiseau, 2013 .

Improvement of the trypanocidal activity of 3-arylthiophene farnesyltransferase inhibitors by modulation of their 3-aryl group

P. Grellier, E. Mouray, J. Dubois, 2012 .

Involvement of calyculin A-sensitive phosphatase(s) in the differentiation of Trypanosoma cruzi trypomastigotes to amastigotes.

J. Blum, V. Sinou, A. Teixeira, 1999, Molecular and biochemical parasitology.

Biodereplication of Antiplasmodial Extracts: Application of the Amazonian Medicinal Plant Piper coruscans Kunth

A. Maciuk, J. Gallard, M. Beniddir, 2022, Molecules.

New protein farnesyltransferase inhibitors in the 3-arylthiophene 2-carboxylic acid series: diversification of the aryl moiety by solid-phase synthesis

P. Grellier, E. Mouray, J. Dubois, 2013, Journal of enzyme inhibition and medicinal chemistry.

New ferrocenic pyrrolo[1,2-a]quinoxaline derivatives: synthesis, and in vitro antimalarial activity--Part II.

G. Déléris, J. Leger, C. Jarry, 2011, European journal of medicinal chemistry.

Eumitrins C-E: Structurally diverse xanthone dimers from the vietnamese lichen Usnea baileyi.

G. Genta‐Jouve, J. Gallard, M. Beniddir, 2019, Fitoterapia.

Synthesis and antimalarial evaluation of new N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives.

C. Sergheraert, P. Melnyk, P. Grellier, 2005, Bioorganic & medicinal chemistry letters.

Programmed Multiple C-H Bond Functionalization of the Privileged 4-hydroxyquinoline Template.

I. Florent, Wei Zhang, E. Mouray, 2021, Chemistry.

Synthesis and in vitro and in vivo antimalarial activity of N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives.

C. Sergheraert, L. Maes, P. Grellier, 2003, Journal of medicinal chemistry.

New ferrocenic pyrrolo[1,2-a]quinoxaline derivatives: synthesis, and in vitro antimalarial activity.

V. Sinou, D. Parzy, C. Jarry, 2008, Bioorganic & medicinal chemistry.

Antimalarial, antitrypanosomal, and antileishmanial activities and cytotoxicity of bis(9-amino-6-chloro-2-methoxyacridines): influence of the linker.

E. Davioud‐Charvet, C. Sergheraert, L. Maes, 2000, Journal of medicinal chemistry.

Synthesis and antimalarial activity of new analogues of amodiaquine.

Philippe Grellier, C. Sergheraert, L. Maes, 2008, European journal of medicinal chemistry.

Design, synthesis and antimalarial activity of a glyoxylylhydrazone library.

C. Sergheraert, O. Melnyk, P. Melnyk, 2004, Bioorganic & medicinal chemistry letters.

Synthesis and antimalarial evaluation of new 1,4-bis(3-aminopropyl)piperazine derivatives.

C. Sergheraert, P. Grellier, R. Deprez-Poulain, 2003, Bioorganic & medicinal chemistry letters.

Synthesis of 1-indolyl substituted β-carboline natural products and discovery of antimalarial and cytotoxic activities

M. Bourguet-Kondracki, B. Copp, I. Florent, 2014 .

Mallotojaponins B and C: Total Synthesis, Antiparasitic Evaluation, and Preliminary SAR Studies.

P. Grellier, E. Mouray, J. Dubois, 2016, Organic letters.

In vitro antiparasitic activity of microbial pigments and their combination with phytosynthesized metal nanoparticles.

P. Grellier, E. Mouray, P. Satish, 2015, Parasitology international.

Pleiokomenines A and B: Dimeric Aspidofractinine Alkaloids Tethered with a Methylene Group.

G. Genta‐Jouve, J. Gallard, M. Beniddir, 2017, Organic letters.

Antiplasmodial and cytotoxic activities of medicinal plants traditionally used in the village of Kiohima, Uganda.

Soizic Prado, B. Bodo, V. Dumontet, 2011, Journal of ethnopharmacology.

Synthesis of novel guttiferone A derivatives: in-vitro evaluation toward Plasmodium falciparum, Trypanosoma brucei and Leishmania donovani.

J. Wansi, Marie-Christine Lallemand, N. Gaboriaud-Kolar, 2013, European journal of medicinal chemistry.

Hydroperoxy-cycloartane triterpenoids from the leaves of Markhamia lutea, a plant ingested by wild chimpanzees.

Soizic Prado, B. Bodo, V. Dumontet, 2009, Phytochemistry.

Activity of Ocimum basilicum, Ocimum canum, and Cymbopogon citratus essential oils against Plasmodium falciparum and mature-stage larvae of Anopheles funestus s.s.

P. Grellier, E. Mouray, Philippe Belong, 2014, Parasite.

Replacement of the 4′‐Hydroxy Group of Amodiaquine and Amopyroquine by Aromatic and Aliphatic Substituents: Synthesis and Antimalarial Activity

E. Pǎunescu, P. Melnyk, P. Grellier, 2009, ChemMedChem.

Theionbrunonines A and B: Dimeric Vobasine Alkaloids Tethered by a Thioether Bridge from Mostuea brunonis.

Pierre Champy, Erwan Poupon, Mehdi A Beniddir, 2018, Organic letters.

The Traditional Medicine Spilanthes acmella, and the Alkylamides Spilanthol and Undeca‐2E‐ene‐8,10‐diynoic Acid Isobutylamide, Demonstrate In Vitro and In Vivo Antimalarial Activity

P. Grellier, Kevin Spelman, E. Mouray, 2011, Phytotherapy research : PTR.

Unexpected talaroenamine derivatives and an undescribed polyester from the fungus Talaromyces stipitatus ATCC10500.

A. Escargueil, G. Genta‐Jouve, Soizic Prado, 2015, Phytochemistry.

Biochemical properties and cellular localization of Plasmodium falciparum protein disulfide isomerase.

C. Sergheraert, P. Grellier, M. Moutiez, 2007, Biochimie.

Towards the synthesis of bisubstrate inhibitors of protein farnesyltransferase: Synthesis and biological evaluation of new farnesylpyrophosphate analogues.

Philippe Grellier, P. Grellier, E. Mouray, 2010, Bioorganic & medicinal chemistry.

Corynanthean-Epicatechin Flavoalkaloids from Corynanthe pachyceras

J. Gallard, M. Beniddir, P. Grellier, 2020, Molecules.

Photosensitized Inactivation of Plasmodium falciparum‐ and Babesia divergens‐Infected Erythrocytes in Whole Blood by Lipophilic Pheophorbide Derivatives

V. Agmon, R. Santus, S. Gatt, 1997, Vox sanguinis.

Selective inhibition of PfA-M1, over PfA-M17, by an amino-benzosuberone derivative blocks malaria parasites development in vitro and in vivo

C. Tarnus, I. Florent, E. Mouray, 2017, Malaria Journal.

Plasmodium Telomeric Sequences: Structure, Stability and Quadruplex Targeting by Small Compounds

Patrizia Alberti, Philippe Grellier, J. Mergny, 2008, Chembiochem : a European journal of chemical biology.

The Escherichia coli ribosomal protein S16 is an endonuclease

O. Pellegrini, E. Bonnefoy, J. Oberto, 1996, Molecular microbiology.

An imbalance of HU synthesis induces mucoidy in Escherichia coli.

S. Gottesman, E. Mouray, E. Painbeni, 1993, Journal of molecular biology.

Cloning of Plasmodium falciparum protein disulfide isomerase homologue by affinity purification using the antiplasmodial inhibitor 1,4‐bis{3‐[N‐(cyclohexyl methyl)amino]propyl}piperazine 1

C. Sergheraert, H. Drobecq, P. Grellier, 2000, FEBS letters.

High and Low Affinity Receptors for Human Interleukin for DA Cells / Leukemia Inhibitory Factor on Human Cells

I. Anegon, D. Heymann, J. Soulillou, 2001 .

High and low affinity receptors for human interleukin for DA cells/leukemia inhibitory factor on human cells. Molecular characterization and cellular distribution.

I. Anegon, D. Heymann, J. Soulillou, 1992, The Journal of biological chemistry.

Synthesis and Antiplasmodial Activity of Novel Fosmidomycin Derivatives and Conjugates with Artemisinin and Aminochloroquinoline

P. Grellier, E. Mouray, M. Baltas, 2020, Molecules.

Aminobenzosuberone derivatives as PfA-M1 inhibitors: Molecular recognition and antiplasmodial evaluation.

C. Tarnus, E. Salomon, M. Torchy, 2020, Bioorganic chemistry.

Revisiting Previously Investigated Plants: A Molecular Networking-Based Study of Geissospermum laeve.

Marc Litaudon, Pierre Champy, Alexander E Fox Ramos, 2017, Journal of natural products.

Molecular Networking Reveals Serpentinine-Related Bisindole Alkaloids from Picralima nitida, a Previously Well-Investigated Species.

J. Gallard, M. Beniddir, P. Grellier, 2020, Journal of natural products.

Secondary Metabolites from the Culture of the Marine-derived Fungus Paradendryphiella salina PC 362H and Evaluation of the Anticancer Activity of Its Metabolite Hyalodendrin

A. Escargueil, S. Lemaire, S. Chaouch, 2020, Marine drugs.

Diversity and biological activities of the bacterial community associated with the marine sponge Phorbas tenacior (Porifera, Demospongiae)

M. Bourguet-Kondracki, A. Ereskovsky, I. Florent, 2014, Letters in applied microbiology.

Structure-activity relationship and molecular modelling studies of quinazolinedione derivatives MMV665916 as potential antimalarial agent.

M. Spichty, I. Florent, E. Mouray, 2021, Bioorganic & medicinal chemistry.

From the Spectroscopic Reassessment of Authentic Alkaloid Samples to the Molecular Networking-Guided Discovery of Criophylline-Related Analogues from Callichilia inaequalis.

S. Agnandji, P. Retailleau, J. Gallard, 2023, Journal of natural products.

Selective inhibition of PfA-M1, over PfA-M17, by an amino-benzosuberone derivative blocks malaria parasites development in vitro and in vivo

C. Tarnus, I. Florent, E. Mouray, 2017, Malaria Journal.

Access to new endoperoxide derivatives by electrochemical oxidation of substituted 3-azabicyclo[4.1.0]hept-4-enes.

A. Marinetti, I. Florent, E. Mouray, 2015, Chemistry.

Synthesis and in vitro antiplasmodial activity of ferrocenyl aminoquinoline derivatives.

Till Bousquet, P. Grellier, E. Mouray, 2015, European journal of medicinal chemistry.

Antiplasmodial Phenolic compounds from Piptadenia pervillei

P. Rasoanaivo, P. Grellier, D. Ramanitrahasimbola, 2008, Planta medica.

Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline.

C. Sergheraert, L. Maes, P. Melnyk, 2008, European journal of medicinal chemistry.

Synthesis and antimalarial activity of new amino analogues of amodiaquine.

E. Pǎunescu, P. Melnyk, P. Grellier, 2008, Medicinal chemistry (Shariqah (United Arab Emirates)).

Synthesis and antimalarial evaluation of new 1,4-bis(3-aminopropyl)piperazine derivatives.

C. Sergheraert, P. Grellier, R. Deprez-Poulain, 2003, Bioorganic & medicinal chemistry letters.

Facile Formation of Methylenebis(chalcone)s through Unprecedented Methylenation Reaction. Application to Antiparasitic and Natural Product Synthesis

P. Grellier, E. Mouray, J. Dubois, 2014 .

New ferrocenic pyrrolo[1,2-a]quinoxaline derivatives: synthesis, and in vitro antimalarial activity.

V. Sinou, D. Parzy, C. Jarry, 2008, Bioorganic & medicinal chemistry.

Corrigendum to: Cloning of Plasmodium falciparum protein disulfide isomerase homologue by affinity purification using the antiplasmodial inhibitor 1,4‐bis{3‐[N‐(cyclohexyl methyl)amino]propyl}piperazine

C. Sergheraert, H. Drobecq, P. Grellier, 2001 .