Giovanni Muncipinto

发表

Short synthesis of skeletally and stereochemically diverse small molecules by coupling petasis condensation reactions to cyclization reactions.

Giovanni Muncipinto, Stuart L Schreiber, Naoya Kumagai, 2006, Angewandte Chemie.

Impact of Stereospecific Intramolecular Hydrogen Bonding on Cell Permeability and Physicochemical Properties

Richard Svensson, Giovanni Muncipinto, Fabrizio Giordanetto, 2014, Journal of medicinal chemistry.

Cycloaddition reactions in Diversity‐Oriented Synthesis

Giovanni Muncipinto, 2013 .

Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and Cholinesterases.

P. Carrupt, Alessandra Nurisso, N. Denora, 2015, Journal of medicinal chemistry.

Solid-phase synthesis and insights into structure-activity relationships of safinamide analogues as potent and selective inhibitors of type B monoamine oxidase.

C. Caccia, F. Leonetti, O. Nicolotti, 2007, Journal of medicinal chemistry.

Diversity-Oriented Synthesis-Facilitated Medicinal Chemistry: Toward the Development of Novel Antimalarial Agents

Carol A. Mulrooney, Jeremy R. Duvall, S. Schreiber, 2014, Journal of medicinal chemistry.

Labeling Preferences of Diazirines with Protein Biomolecules.

Hung-Yi Wu, Giovanni Muncipinto, L. Jones, 2020, Journal of the American Chemical Society.

Identification of Highly Specific Diversity-Oriented Synthesis-Derived Inhibitors of Clostridium difficile.

Joshua A. Bittker, Jeremy R. Duvall, M. Foley, 2017, ACS infectious diseases.

Catalytic diastereoselective petasis reactions.

S. Schreiber, S. Schaus, Giovanni Muncipinto, 2011, Angewandte Chemie.

Expanding Stereochemical and Skeletal Diversity Using Petasis Reactions and 1,3-Dipolar Cycloadditions

P. Clemons, S. Schreiber, N. Kumagai, 2010, Organic letters.

Diversity-oriented synthesis yields a new drug lead for treatment of chagas disease.

Jeremy R. Duvall, S. Schreiber, Ana Rodriguez, 2014, ACS medicinal chemistry letters.

A twenty-year journey exploring coumarin-based derivatives as bioactive molecules

F. Leonetti, O. Nicolotti, M. Catto, 2022, Frontiers in Chemistry.

Toward a fragment-based approach to MMPs inhibitors: an expedite and efficient synthesis of N-hydroxylactams

F. Leonetti, O. Nicolotti, M. Catto, 2012 .

Synthesis and profiling of a diverse collection of azetidine-based scaffolds for the development of CNS-focused lead-like libraries.

Giovanni Muncipinto, Lakshmi B. Akella, Byung-Chul Suh, 2012, The Journal of organic chemistry.

Discovery of a novel class of potent coumarin monoamine oxidase B inhibitors: development and biopharmacological profiling of 7-[(3-chlorobenzyl)oxy]-4-[(methylamino)methyl]-2H-chromen-2-one methanesulfonate (NW-1772) as a highly potent, selective, reversible, and orally active monoamine oxidase B i

C. Caccia, F. Leonetti, O. Nicolotti, 2009, Journal of medicinal chemistry.

Screening of Matrix Metalloproteinases Available from the Protein Data Bank: Insights into Biological Functions, Domain Organization, and Zinc Binding Groups

Angelo Carotti, Francesco Leonetti, Orazio Nicolotti, 2007, J. Chem. Inf. Model..

Structural and conformational determinants of macrocycle cell permeability.

Ulf Norinder, Christian Tyrchan, Giovanni Muncipinto, 2016, Nature chemical biology.

Modulators of Hepatic Lipoprotein Metabolism Identified in a Search for Small-Molecule Inducers of Tribbles Pseudokinase 1 Expression

Jeremy R. Duvall, A. Subramanian, M. Foley, 2015, PloS one.

Modulators of Hepatic Lipoprotein Metabolism Identified in a Search for Small-Molecule Inducers of Tribbles Pseudokinase 1 Expression

Jeremy R. Duvall, A. Subramanian, M. Foley, 2015, PloS one.

Synthesis and profiling of a diverse collection of azetidine-based scaffolds for the development of CNS-focused lead-like libraries.

Carol A. Mulrooney, Jeremy R. Duvall, M. Foley, 2012, The Journal of organic chemistry.