Yasutaka Hoashi

发表

Enantioselective Michael reaction of malonates to nitroolefins catalyzed by bifunctional organocatalysts.

Y. Takemoto, T. Okino, Yasutaka Hoashi, 2003, Journal of the American Chemical Society.

Bifunctional thiourea-catalyzed enantioselective double Michael reaction of γ,δ-unsaturated β-ketoester to nitroalkene: asymmetric synthesis of (−)-epibatidine

Y. Takemoto, Yasutaka Hoashi, Takaya Yabuta, 2004 .

Enantioselective tandem michael reaction to nitroalkene catalyzed by bifunctional thiourea : total synthesis of (-)-epibatidine

Y. Takemoto, Yasutaka Hoashi, Takaya Yabuta, 2006 .

Discovery of novel 5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridine derivatives as γ-secretase modulators.

Yasutaka Hoashi, Tomoko Igari, T. Takai, 2015, Bioorganic & medicinal chemistry letters.

Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists.

Takahiko Yano, Yasutaka Hoashi, Y. Kosugi, 2018, Bioorganic & medicinal chemistry.

Anti-tumor activity of KNTC2 siRNA in orthotopic tumor model mice of hepatocellular carcinoma.

K. Kikuchi, Y. Kawamata, Mika Teratani, 2017, Biochemical and biophysical research communications.

Enantio- and diastereoselective Michael reaction of 1,3-dicarbonyl compounds to nitroolefins catalyzed by a bifunctional thiourea.

Y. Takemoto, T. Okino, Yasutaka Hoashi, 2005, Journal of the American Chemical Society.

1,6-Dihydro-2H-indeno[5,4-b]furan derivatives: design, synthesis, and pharmacological characterization of a novel class of highly potent MT₂-selective agonists.

Masaharu Nakayama, K. Hirai, Yasutaka Hoashi, 2011, Journal of medicinal chemistry.

Synthesis of 4-aza analog of ramelteon: a novel tricyclic 1,6,7,8-tetrahydro-2H-cyclopenta[d]furo[2,3-b]pyridine derivative as melatonin receptor ligand

Yasutaka Hoashi, O. Uchikawa, T. Takai, 2011 .

Synthesis of a novel series of tricyclic dihydrofuran derivatives: discovery of 8,9-dihydrofuro[3,2-c]pyrazolo[1,5-a]pyridines as melatonin receptor (MT1/MT2) ligands.

Masaharu Nakayama, K. Hirai, Yasutaka Hoashi, 2011, Journal of medicinal chemistry.

Thiourea-catalyzed nucleophilic addition of TMSCN and ketene silyl acetals to nitrones and aldehydes

Y. Takemoto, T. Okino, Yasutaka Hoashi, 2003 .

Enantioselective Michael Addition to α,β‐Unsaturated Imides Catalyzed by a Bifunctional Organocatalyst

Y. Takemoto, T. Okino, Yasutaka Hoashi, 2005 .

Enantio- and diastereoselective Michael reaction of 1,3-dicarbonyl compounds to nitroolefins catalyzed by a bifunctional thiourea.

Y. Takemoto, T. Okino, Yasutaka Hoashi, 2005, Journal of the American Chemical Society.

Synthesis of pyrazolo[1,5-a]pyridines by thermal intramolecular cyclization

Yasutaka Hoashi, T. Takai, T. Koike, 2013 .

Reductively Cleavable Nanocaplets for siRNA Delivery by Template-Assisted Oxidative Polymerization.

T. Aida, P. K. Hashim, Yasutaka Hoashi, 2015, Journal of the American Chemical Society.

Design and synthesis of piperazine derivatives as a novel class of γ-secretase modulators that selectively lower Aβ₄₂ production.

Yasutaka Hoashi, Tomoko Igari, Eiji Honda, 2015, Bioorganic & medicinal chemistry.

Enantioselective Michael addition to alpha,beta-unsaturated imides catalyzed by a bifunctional organocatalyst.

Y. Takemoto, Yasutaka Hoashi, Tomotaka Okino, 2005, Angewandte Chemie.