M. Díaz-Gavilán

发表

Synthesis of unprecedented scaffold diversity.

David R Spring, Warren R J D Galloway, D. Spring, 2009, Angewandte Chemie.

Diversity-oriented synthesis of bicyclic and tricyclic alkaloids.

Kieron M. G. O'Connell, D. Spring, W. R. Galloway, 2010, Chemical communications.

Synthesis of Unprecedented Scaffold Diversity

D. Spring, W. R. Galloway, Albert Isidro-Llobet, 2009 .

An Introduction to Diversity‐Oriented Synthesis

Kieron M. G. O'Connell, D. Spring, R. J. Spandl, 2009 .

Diversity‐Oriented Synthesis

Kieron M. G. O'Connell, D. Spring, R. J. Spandl, 2009 .

The selective cytotoxic activity in breast cancer cells by an anthranilic alcohol-derived acyclic 5-fluorouracil O,N-acetal is mediated by endoplasmic reticulum stress-induced apoptosis.

A. Martínez-Amat, P. Álvarez, J. Marchal, 2012, European journal of medicinal chemistry.

Oligonucleotide-polyamine conjugates: influence of length and position of 2'-attached polyamines on duplex stability and antisense effect.

C. Noe, M. Díaz-Gavilán, J. Winkler, 2009, European journal of medicinal chemistry.

Salicylic Acid Derivatives Inhibit Oxalate Production in Mouse Hepatocytes with Primary Hyperoxaluria Type 1.

E. Salido, J. A. Gómez-Vidal, M. Díaz-Gavilán, 2018, Journal of medicinal chemistry.

Synthesis of tetrahydrobenzoxazepine acetals with electron-withdrawing groups on the nitrogen atom. Novel scaffolds endowed with anticancer activity against breast cancer cells

J. Marchal, A. Aránega, J. Campos, 2004 .

Lactate dehydrogenase A inhibitors with a 2,8-dioxabicyclo[3.3.1]nonane scaffold: A contribution to molecular therapies for primary hyperoxalurias.

E. Salido, M. Díaz-Gavilán, A. Alejo-Armijo, 2022, Bioorganic chemistry.

Substituent effects on the reaction mode between 2-hydroxybenzyl alcohol derivatives and MEM chloride: synthesis and mechanistic aspects of seven- and ten-membered benzo-fused O,O-acetals

J. Campos, M. Díaz-Gavilán, M. Gallo, 2004 .

Two-directional synthesis as a tool for diversity-oriented synthesis: Synthesis of alkaloid scaffolds

David R Spring, Kieron M. G. O'Connell, Warren R J D Galloway, 2012, Beilstein journal of organic chemistry.

Diversity-oriented synthesis.

David R Spring, Kieron M. G. O'Connell, D. Spring, 2009, Chemical record.

Anticancer activity of (1,2,3,5-tetrahydro-4,1-benzoxazepine-3-yl)-pyrimidines and -purines against the MCF-7 cell line: Preliminary cDNA microarray studies.

J. Marchal, A. Aránega, J. Campos, 2008, Bioorganic & medicinal chemistry letters.

Synthesis of l-Octaarginine through Microencapsulated Palladium-Catalyzed Allyl Ester Deprotection

Ana M. Pérez-López, J. A. Gómez-Vidal, M. Díaz-Gavilán, 2014 .

Synthesis and anticancer activity studies of novel 1-(2,3-dihydro-5H-1,4 -benzodioxepin -3 -yl )uracil and (6'-substituted)-7-or 9 -(2,3 -dihydro -5H-1,4 -benzodioxepin -3 -yl ) -7H-or 9H-purines

J. Marchal, A. Aránega, J. Campos, 2006 .

Structure of Anisakis simplex s.l. populations in a region sympatric for A. pegreffii and A. simplex s.s. Absence of reproductive isolation between both species.

M. Díaz-Gavilán, J. Martín‐Sánchez, A. Valero-López, 2005, Molecular and biochemical parasitology.

Small Molecule-Based Enzyme Inhibitors in the Treatment of Primary Hyperoxalurias

E. Salido, J. A. Gómez-Vidal, M. Díaz-Gavilán, 2021, Journal of personalized medicine.

Synthesis and Anticancer Activity of (R,S)‐9‐(2,3‐Dihydro‐1,4‐Benzoxathiin‐3‐ylmethyl)‐9H‐Purines

J. Marchal, A. Aránega, J. Campos, 2008, ChemMedChem.

From 5-fluorouracil acyclonucleosides to benzo-fused six- and seven-membered rings linked to pyrimidine and purine bases: the shift from differentiating anticancer agents to apoptotic inducers

J. Campos, A. Conejo-García, O. Cruz-López, 2008, Expert opinion on drug discovery.

Synthesis and reactivity of (RS)-6-chloro-7-or 9-(1,2,3,5-tetrahydro -4,1-benzoxazepin-3-yl )-7H-or 9H-purines bearing a nitrobenzenesulfonyl group on the nitrogen atom

J. Campos, D. Choquesillo-Lazarte, M. Díaz-Gavilán, 2007 .

New salicylic acid derivatives, double inhibitors of glycolate oxidase and lactate dehydrogenase, as effective agents decreasing oxalate production.

E. Salido, A. Pey, M. Díaz-Gavilán, 2022, European journal of medicinal chemistry.

A synthetic uracil derivative with antitumor activity through decreasing cyclin D1 and Cdk1, and increasing p21 and p27 in MCF-7 cells

H. Boulaiz, J. Marchal, A. Aránega, 2007, Breast Cancer Research and Treatment.

A nanodelivered Vorinostat derivative is a promising oral compound for the treatment of visceral leishmaniasis

N. de Pedro, E. Belmonte-Reche, M. Díaz-Gavilán, 2019, Pharmacological research.

Effectiveness of an O-Alkyl Hydroxamate in Dogs with Naturally Acquired Canine Leishmaniosis: An Exploratory Clinical Trial

M. Díaz-Gavilán, J. Martín‐Sánchez, J. López-Viota, 2022, Animals : an open access journal from MDPI.

O-alkyl hydroxamates display potent and selective antileishmanial activity.

J. Correa-Basurto, N. de Pedro, Y. Sixto-López, 2020, Journal of medicinal chemistry.

Anticancer activity and cDNA microarray studies of a (RS)-1,2,3,5-tetrahydro-4,1-benzoxazepine-3-yl]-6-chloro-9H-purine, and an acyclic (RS)-O,N-acetalic 6-chloro-7H-purine.

H. Boulaiz, J. Marchal, A. Aránega, 2011, European journal of medicinal chemistry.

(2,3-Dihydro-1,4-benzodioxin-2-yl)methanol

D. Choquesillo-Lazarte, M. Díaz-Gavilán, J. M. C. Rosa, 2007 .

Design, synthesis and anticancer activity against the MCF-7 cell line of benzo-fused 1,4-dihetero seven- and six-membered tethered pyrimidines and purines.

J. Campos, A. Conejo-García, O. Cruz-López, 2008, Current medicinal chemistry.

Study of the factors that control the ratio of the products between 5-fluorouracil, uracil, and tetrahydrobenzoxazepine O,O-acetals bearing electron-withdrawing groups on the nitrogen atom.

J. Campos, M. Díaz-Gavilán, M. Gallo, 2006, The Journal of organic chemistry.