Justin E. Jones

发表

Design, synthesis, and kinetic characterization of protein N-terminal acetyltransferase inhibitors.

T. Arnesen, J. Varhaug, P. Thompson, 2013, ACS chemical biology.

Suppression of colitis in mice by Cl-amidine: a novel peptidylarginine deiminase inhibitor.

Deepak Poudyal, T. Davis, A. Chumanevich, 2011, American journal of physiology. Gastrointestinal and liver physiology.

Activity-based protein profiling of protein arginine methyltransferase 1.

P. Thompson, Justin E. Jones, Obiamaka Obianyo, 2011, ACS chemical biology.

Synthesis and screening of a haloacetamidine containing library to identify PAD4 selective inhibitors.

P. Thompson, S. Coonrod, V. Subramanian, 2012, ACS chemical biology.

Substrate specificity and kinetic studies of PADs 1, 3, and 4 identify potent and selective inhibitors of protein arginine deiminase 3.

P. Thompson, B. Knuckley, Justin E. Jones, 2010, Biochemistry.

Mechanistic Studies of Protein Arginine Deiminase 2: Evidence for a Substrate-Assisted Mechanism

P. Thompson, Daniel M. Lewallen, B. Knuckley, 2014, Biochemistry.

A Chloroacetamidine‐Based Inactivator of Protein Arginine Methyltransferase 1: Design, Synthesis, and In Vitro and In Vivo Evaluation

M. Stallcup, P. Thompson, Young-Ho Lee, 2010, Chembiochem : a European journal of chemical biology.

Protein arginine deiminase 4 (PAD4): Current understanding and future therapeutic potential.

P. Thompson, B. Knuckley, Justin E. Jones, 2009, Current opinion in drug discovery & development.

Mechanistic studies of agmatine deiminase from multiple bacterial species.

P. Thompson, Justin E. Jones, Corey P. Causey, 2010, Biochemistry.

The development of N-α-(2-carboxyl)benzoyl-N(5)-(2-fluoro-1-iminoethyl)-l-ornithine amide (o-F-amidine) and N-α-(2-carboxyl)benzoyl-N(5)-(2-chloro-1-iminoethyl)-l-ornithine amide (o-Cl-amidine) as second generation protein arginine deiminase (PAD) inhibitors.

Yuan Luo, A. Chumanevich, L. Hofseth, 2011, Journal of medicinal chemistry.

Characterization and inactivation of an agmatine deiminase from Helicobacter pylori.

L. Lebioda, P. Thompson, B. Knuckley, 2010, Bioorganic chemistry.

A fluopol-ABPP HTS assay to identify PAD inhibitors.

Steven J Brown, B. Cravatt, P. Thompson, 2010, Chemical communications.

A fluopol-ABPP HTS assay to identify PAD inhibitors.

Steven J Brown, B. Cravatt, P. Thompson, 2010, Chemical communications.