Jeewoo Lee

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Discovery of an Orally Bioavailable Benzofuran Analogue That Serves as a β-Amyloid Aggregation Inhibitor for the Potential Treatment of Alzheimer's Disease.

Jiyoun Lee, D. Jo, H. Hong, 2018, Journal of medicinal chemistry.

Novel Hypoxia-Inducible Factor 1α (HIF-1α) Inhibitors for Angiogenesis-Related Ocular Diseases: Discovery of a Novel Scaffold via Ring-Truncation Strategy.

Chang Sik Cho, Jeeyeon Lee, Sang -Geon Kim, 2018, Journal of medicinal chemistry.

Differential Regulation of Gene Expression in Lung Cancer Cells by Diacyglycerol-Lactones and a Phorbol Ester Via Selective Activation of Protein Kinase C Isozymes

M. Kazanietz, P. Blumberg, M. Abba, 2019, Scientific Reports.

Characterization of AJH-836, a diacylglycerol-lactone with selectivity for novel PKC isozymes

M. Kazanietz, P. Blumberg, R. Garg, 2018, Journal of Biological Chemistry.

Beyond the affinity for protein kinase C: exploring 2-phenyl-3-hydroxypropyl pivalate analogues as C1 domain-targeting ligands

D. Rossi, S. Collina, A. Pascale, 2015 .

α-Arylidene Diacylglycerol-Lactones (DAG-Lactones) as Selective Ras Guanine-Releasing Protein 3 (RasGRP3) Ligands.

P. Blumberg, M. Peach, N. Lewin, 2018, Journal of medicinal chemistry.

Design and synthesis of protein kinase C epsilon selective diacylglycerol lactones (DAG-lactones).

P. Blumberg, D. H. Kim, N. Lewin, 2015, European journal of medicinal chemistry.

In vitro and in silico determination of glutaminyl cyclase inhibitors

Son Tung Ngo, N. T. Tung, Jeewoo Lee, 2019, RSC advances.

Discovery of a Simplified Deguelin Analog as an HSP90 C-terminal Inhibitor for HER2-positive Breast Cancer.

Hyun-Ju Park, Jihyae Ann, Jeewoo Lee, 2021, Bioorganic & medicinal chemistry letters.

A novel HSP90 inhibitor targeting the C-terminal domain attenuates trastuzumab resistance in HER2-positive breast cancer

Ji Young Kim, Hyun-Ju Park, J. Seo, 2020, Molecular Cancer.

Transient receptor potential vanilloid type 1 antagonists: a patent review (2011 – 2014)

M. Cui, Sun Choi, P. K. Sharma, 2015, Expert opinion on therapeutic patents.

Contributions of TRPV1, endovanilloids, and endoplasmic reticulum stress in lung cell death in vitro and lung injury.

C. Reilly, Jeewoo Lee, G. Yost, 2012, American journal of physiology. Lung cellular and molecular physiology.

Deguelin Analogue SH-1242 Inhibits Hsp90 Activity and Exerts Potent Anticancer Efficacy with Limited Neurotoxicity.

So-Jung Park, Jeeyeon Lee, Sonia J. Park, 2016, Cancer research.

Lovastatin enhances Aβ production and senile plaque deposition in female Tg2576 mice

J. H. Boo, I. Mook‐Jung, Seung U. Kim, 2003, Neurobiology of Aging.

A novel HSP90 inhibitor SL-145 suppresses metastatic triple-negative breast cancer without triggering the heat shock response

J. Seo, Jihyae Ann, Jeewoo Lee, 2022, Oncogene.

Dorsal root ganglion neurons innervating skeletal muscle respond to physiological combinations of protons, ATP, and lactate mediated by ASIC, P2X, and TRPV1.

A. Light, J. Rainier, R. Hughen, 2008, Journal of neurophysiology.

Synthesis of 7'-[123I]iodo-D-luciferin for in vivo studies of firefly luciferase gene expression.

Kyung-Han Lee, Y. Choe, Jeewoo Lee, 2004, Bioorganic & medicinal chemistry letters.

6-Phenoxy-2-phenylbenzoxazoles, novel inhibitors of receptor for advanced glycation end products (RAGE).

Jiyoun Lee, Y. Suh, H. Hong, 2015, Bioorganic & medicinal chemistry.

Discovery of a Small Molecule that Enhances Astrocytogenesis by Activation of STAT3, SMAD1/5/8, and ERK1/2 via Induction of Cytokines in Neural Stem Cells.

Jiyoun Lee, Hyun-Jung Kim, S. Kong, 2016, ACS chemical neuroscience.

Discovery of novel anti-breast cancer agents derived from deguelin as inhibitors of heat shock protein 90 (HSP90).

Ji Young Kim, Hyun-Ju Park, Raghaba Sahu, 2020, Bioorganic & medicinal chemistry letters.

Discovery of Novel Dual Adenosine A2A and A1 Receptor Antagonists with 1H-Pyrazolo[3,4-d]pyrimidin-6-amine Core Scaffold as Anti-Parkinson’s Disease Agents

Jihyae Ann, Jeewoo Lee, Juyoung Jung, 2022, Pharmaceuticals.

Inhibition of glutaminyl cyclase ameliorates amyloid pathology in an animal model of Alzheimer's disease via the modulation of γ-secretase activity.

Hyundong Song, I. Mook‐Jung, Jeewoo Lee, 2014, Journal of Alzheimer's disease : JAD.

Synthesis and biological evaluation of 3-(2-aminoethyl) uracil derivatives as gonadotropin-releasing hormone (GnRH) receptor antagonists.

Jiyoun Lee, So young Lee, Jihyae Ann, 2018, European journal of medicinal chemistry.

Structural anatomy of Protein Kinase C C1 domain interactions with diacylglycerol and other agonists

J. Sacchettini, T. Igumenova, I. Krieger, 2022, Nature Communications.

2-Sulfonamidopyridine C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists.

Sun Choi, Jeewoo Lee, P. Blumberg, 2016, Bioorganic & medicinal chemistry.

Migration of neutrophils targeting amyloid plaques in Alzheimer's disease mouse model

Sung Hoon Baik, D. Irimia, I. Mook‐Jung, 2014, Neurobiology of Aging.

Fine tuning of 4,6-bisphenyl-2-(3-alkoxyanilino)pyrimidine focusing on the activity-sensitive aminoalkoxy moiety for a therapeutically useful inhibitor of receptor for advanced glycation end products (RAGE).

Jeeyeon Lee, Hyun-Ju Park, Y. Suh, 2015, Bioorganic & medicinal chemistry.

Discovery of potent indazole-based human glutaminyl cyclase (QC) inhibitors as Anti-Alzheimer's disease agents.

Heejin Ha, Jihyae Ann, Young-Ho Kim, 2022, European journal of medicinal chemistry.

Discovery of Conformationally Restricted Human Glutaminyl Cyclase Inhibitors as Potent Anti-Alzheimer's Agents by Structure-Based Design.

S. J. Y. Macalino, M. Cui, Sun Choi, 2019, Journal of medicinal chemistry.

Potent human glutaminyl cyclase inhibitors as potential anti-Alzheimer's agents: Structure-activity relationship study of Arg-mimetic region.

M. Cui, Sun Choi, Jiyoun Lee, 2018, Bioorganic & medicinal chemistry.

Combination of a Rapidly Penetrating Agonist and a Slowly Penetrating Antagonist Affords Agonist Action of Limited Duration at the Cellular Level

P. Blumberg, L. Pearce, Jihyae Ann, 2019, Biomolecules & therapeutics.

Discovery of highly potent human glutaminyl cyclase (QC) inhibitors as anti-Alzheimer's agents by the combination of pharmacophore-based and structure-based design.

Jiyoun Lee, Heejin Ha, Jihyae Ann, 2021, European journal of medicinal chemistry.

6,6-Fused heterocyclic ureas as highly potent TRPV1 antagonists.

K. Schiene, Sun Choi, Jeewoo Lee, 2015, Bioorganic & medicinal chemistry letters.

Discovery of dual-acting opioid ligand and TRPV1 antagonists as novel therapeutic agents for pain.

Ji-Young Hwang, Larry V. Pearce, Peter M. Blumberg, 2019, European journal of medicinal chemistry.

Pyrazole-5-carboxamides, novel inhibitors of receptor for advanced glycation end products (RAGE).

Hyun-Ju Park, Y. Suh, Kyeojin Kim, 2014, European journal of medicinal chemistry.

Discovery of 1-(1H-Indazol-4-yl)-3-((1-Phenyl-1H-Pyrazol-5-yl)methyl) Ureas as Potent and Thermoneutral TRPV1 Antagonists.

G. Bahrenberg, P. Blumberg, Sun-Ok Kwon, 2020, Bioorganic & medicinal chemistry letters.

Discovery of indane propanamides as potent and selective TRPV1 antagonists.

G. Bahrenberg, P. Blumberg, Y. H. Kim, 2019, Bioorganic & medicinal chemistry letters.

Discovery of 2-(3,5-difluoro-4-methylsulfonaminophenyl)propanamides as potent TRPV1 antagonists.

G. Bahrenberg, P. Blumberg, Changhoon Kim, 2018, Bioorganic & medicinal chemistry letters.

t-Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Sun Choi, G. Bahrenberg, P. Blumberg, 2017, Bioorganic & medicinal chemistry.

Discovery of N-(3-fluoro-4-methylsulfonamidomethylphenyl)urea as a potent TRPV1 antagonistic template.

Sun Choi, P. Blumberg, Changhoon Kim, 2016, Bioorganic & medicinal chemistry letters.

Structure activity relationships of benzyl C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists.

M. Cui, Sun Choi, G. Bahrenberg, 2015, Bioorganic & medicinal chemistry.

α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists.

M. Cui, Sun Choi, G. Bahrenberg, 2015, Bioorganic & medicinal chemistry letters.

Pyridine C-region analogs of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

HyungChul Ryu, Suyoung Yoon, K. Schiene, 2015, European journal of medicinal chemistry.

Aminopropyl carbazole analogues as potent enhancers of neurogenesis.

Jiyoun Lee, Jeewoo Lee, Hyun-Jung Kim, 2013, Bioorganic & medicinal chemistry.

Ligand-based design, synthesis, and biological evaluation of 2-aminopyrimidines, a novel series of receptor for advanced glycation end products (RAGE) inhibitors.

Hyun-Ju Park, Y. Suh, H. Hong, 2012, Journal of medicinal chemistry.

Curcumin interacts directly with the Cysteine 259 residue of STAT3 and induces apoptosis in H-Ras transformed human mammary epithelial cells

Do-Hee Kim, Y. Surh, H. Na, 2018, Scientific Reports.

Conformationally constrained analogues of diacylglycerol (DAG). Part 19: Asymmetric syntheses of (3R)- and (3S)-3-hydroxy-4,4-disubstituted heptono-1,4-lactones as protein kinase C (PK-C) ligands with increased hydrophilicity

P. Blumberg, V. Marquez, K. Nacro, 2002 .

Discovery of an Orally Bioavailable Gonadotropin-Releasing Hormone Receptor Antagonist.

Jiyoun Lee, So young Lee, Jihyae Ann, 2016, Journal of medicinal chemistry.

Development of a novel Hsp90 inhibitor NCT-50 as a potential anticancer agent for the treatment of non-small cell lung cancer

Hyun-Ju Park, Ho Jin Lee, Jihyae Ann, 2018, Scientific Reports.

A novel C-terminal heat shock protein 90 inhibitor that overcomes STAT3-Wnt-β-catenin signaling-mediated drug resistance and adverse effects

Hyun-Ju Park, Ho Jin Lee, Jihyae Ann, 2022, Theranostics.

C-terminal HSP90 inhibitor L80 elicits anti-metastatic effects in triple-negative breast cancer via STAT3 inhibition.

Ji Young Kim, J. Seo, Jihyae Ann, 2019, Cancer letters.

Synthesis and Evaluation of a Novel Deguelin Derivative, L80, which Disrupts ATP Binding to the C-terminal Domain of Heat Shock Protein 90

So-Jung Park, Hyun-Ju Park, Ho-Yyoung Lee, 2015, Molecular Pharmacology.

Synthesis and Evaluation of a Novel Deguelin Derivative , L 80 , which Disrupts ATP Binding to the C-terminal Domain of Heat Shock Protein 90

So-Jung Park, Hyun-Ju Park, Ho-Yyoung Lee, 2015 .

Discovery of Non-pungent Transient Receptor Potential Vanilloid 1 (TRPV1) Agonist as Strong Topical Analgesic.

S. Hwang, P. Blumberg, L. Pearce, 2019, Journal of medicinal chemistry.

Structure-activity relationship of leucyladenylate sulfamate analogues as leucyl-tRNA synthetase (LRS)-targeting inhibitors of Mammalian target of rapamycin complex 1 (mTORC1).

Jiyoun Lee, Changhoon Kim, Woong Sub Byun, 2019, Bioorganic & medicinal chemistry.

Discovery of novel leucyladenylate sulfamate surrogates as leucyl-tRNA synthetase (LRS)-targeted mammalian target of rapamycin complex 1 (mTORC1) inhibitors.

Won Kyung Kim, Jiyoun Lee, Jihyae Ann, 2018, Bioorganic & medicinal chemistry.

Discovery of simplified leucyladenylate sulfamates as novel leucyl-tRNA synthetase (LRS)-targeted mammalian target of rapamycin complex 1 (mTORC1) inhibitors.

Won Kyung Kim, Sunghoon Kim, Jiyoun Lee, 2016, Bioorganic & medicinal chemistry.

Curcumin suppresses oncogenicity of human colon cancer cells by covalently modifying the cysteine 67 residue of SIRT1.

Do-Hee Kim, Y. Surh, H. Na, 2018, Cancer letters.

Ring-truncated deguelin derivatives as potent Hypoxia Inducible Factor-1α (HIF-1α) inhibitors.

So-Jung Park, D. Oh, Hyun-Ju Park, 2015, European journal of medicinal chemistry.

Uric acid induces endothelial dysfunction by vascular insulin resistance associated with the impairment of nitric oxide synthesis

Byung-Hoon Lee, Moo-Yeol Lee, You-Jin Choi, 2014, FASEB journal : official publication of the Federation of American Societies for Experimental Biology.

Discovery of novel heat shock protein (Hsp90) inhibitors based on luminespib with potent antitumor activity.

Jeewoo Lee, Juyoung Jung, Jinsun Kwon, 2020, Bioorganic & medicinal chemistry letters.

Intracellular amyloid-β accumulation in calcium-binding protein-deficient neurons leads to amyloid-β plaque formation in animal model of Alzheimer's disease.

Sung Hoon Baik, Hyundong Song, I. Mook‐Jung, 2012, Journal of Alzheimer's disease : JAD.

Structure-activity relationship investigation of Phe-Arg mimetic region of human glutaminyl cyclase inhibitors.

M. Cui, Sun Choi, Heejin Ha, 2018, Bioorganic & medicinal chemistry.

Discovery of Potent Human Glutaminyl Cyclase Inhibitors as Anti-Alzheimer's Agents Based on Rational Design.

M. Cui, Sun Choi, Jiyoun Lee, 2017, Journal of medicinal chemistry.

Investigation of B,C-ring truncated deguelin derivatives as heat shock protein 90 (HSP90) inhibitors for use as anti-breast cancer agents.

Ji Young Kim, Hyun-Ju Park, Kyu-Won Kim, 2019, Bioorganic & medicinal chemistry.

Discovery of Benzopyridone-Based Transient Receptor Potential Vanilloid 1 Agonists and Antagonists and the Structural Elucidation of Their Activity Shift.

Sun Choi, Yoonji Lee, P. Blumberg, 2021, Journal of medicinal chemistry.

Inhibition of mouse skin tumor promotion by anti-inflammatory diarylheptanoids derived from Alpinia oxyphylla Miquel (Zingiberaceae).

Y. Surh, Kwang-Kyun Park, K. Chun, 2002, Oncology research.

Comparative Effects of Curcumin and Tetrahydrocurcumin on Dextran Sulfate Sodium-induced Colitis and Inflammatory Signaling in Mice

Do-Hee Kim, Y. Surh, H. Na, 2018, Journal of cancer prevention.

2-(4-Methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure-activity relationships in the B and C-regions.

Vladimir A. Pavlyukovets, P. Blumberg, Keliang Liu, 2012, Bioorganic & medicinal chemistry.

In vitro characterization of the thermoneutral transient receptor potential vanilloid-1 (TRPV1) inhibitor GRTE16523.

G. Bahrenberg, N. Damann, Jihyae Ann, 2020, European journal of pharmacology.

Discovery of 5-(N-Hydroxycarbamimidoyl) Benzofuran Derivatives as Novel Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitors.

Jihyae Ann, Jeewoo Lee, Juyoung Jung, 2021, Bioorganic & Medicinal Chemistry Letters.

Differential modulation of agonist and antagonist structure activity relations for rat TRPV1 by cyclosporin A and other protein phosphatase inhibitors

Dong Wook Kang, Attila Toth, HyungChul Ryu, 2008, Naunyn-Schmiedeberg's Archives of Pharmacology.

Physiologically based pharmacokinetic modeling of SNU-0039, an anti-Alzheimer’s agent, in rats

S. Chong, Dae-Duk Kim, C. Shim, 2011, Journal of Pharmacokinetics and Pharmacodynamics.

The carbonate analogues of 5'-halogenated resiniferatoxin as TRPV1 ligands.

Sun Choi, P. Blumberg, L. Pearce, 2013, European journal of medicinal chemistry.

Functional Group-Dependent Induction of Astrocytogenesis and Neurogenesis by Flavone Derivatives

Y. M. Kim, Hyun-Jung Kim, Jin-Mi Kang, 2019, Biomolecules.

Halogenation of 4-hydroxy/amino-3-methoxyphenyl acetamide TRPV1 agonists showed enhanced antagonism to capsaicin.

Vladimir A. Pavlyukovets, P. Blumberg, L. Pearce, 2010, Bioorganic & medicinal chemistry.

Different vanilloid agonists cause different patterns of calcium response in CHO cells heterologously expressing rat TRPV1.

P. Blumberg, Yun Wang, L. Pearce, 2005, Life sciences.

Structural anatomy of C1 domain interactions with DAG and other agonists

J. Sacchettini, T. Igumenova, I. Krieger, 2021, bioRxiv.

A two-photon fluorescent probe for amyloid-β plaques in living mice.

Sung Hoon Baik, Hyung Joong Kim, Hyundong Song, 2013, Chemical communications.

Differential Regulation of Gene Expression in Lung Cancer Cells by Diacyglycerol-Lactones and a Phorbol Ester Via Selective Activation of Protein Kinase C Isozymes

M. Kazanietz, P. Blumberg, M. Abba, 2019, Scientific Reports.

The C-terminal HSP90 inhibitor NCT-58 kills trastuzumab-resistant breast cancer stem-like cells

Ji Young Kim, J. Seo, Jihyae Ann, 2021, Cell death discovery.

Chiral 2-phenyl-3-hydroxypropyl esters as PKC-alpha modulators: HPLC enantioseparation, NMR absolute configuration assignment, and molecular docking studies.

F. Vasile, D. Potenza, D. Rossi, 2021, Chirality.

Transient Receptor Potential Vanilloid-1 (TRPV1) Is a Mediator of Lung Toxicity for Coal Fly Ash Particulate Material

J. Veranth, C. Reilly, Jeewoo Lee, 2012, Molecular Pharmacology.

Structure-Activity Relationship of Capsaicin Analogs and Transient Receptor Potential Vanilloid 1-Mediated Human Lung Epithelial Cell Toxicity

Thomas E Cheatham, Manivannan Ethirajan, Kiumars Shahrokh, 2011, Journal of Pharmacology and Experimental Therapeutics.

4-Aminophenyl acetamides and propanamides as potent transient receptor potential vanilloid 1 (TRPV1) ligands.

Sun Choi, G. Bahrenberg, P. Blumberg, 2018, Bioorganic & medicinal chemistry.

Pyrazole C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Sun Choi, G. Bahrenberg, P. Blumberg, 2017, Bioorganic & medicinal chemistry letters.

2-Aryl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists.

M. Cui, Sun Choi, P. K. Sharma, 2014, Bioorganic & medicinal chemistry letters.

TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides.

Sun Choi, HyungChul Ryu, Peter M. Blumberg, 2013, Bioorganic & medicinal chemistry.

2-(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists: structure activity relationships of the 2-oxy pyridine C-region.

Dong Wook Kang, Sun Choi, HyungChul Ryu, 2013, European journal of medicinal chemistry.

2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists.

K. Schiene, M. Cui, Sun Choi, 2014, Bioorganic & medicinal chemistry letters.

An Aminopropyl Carbazole Derivative Induces Neurogenesis by Increasing Final Cell Division in Neural Stem Cells

Hyun-Jung Kim, S. Kong, Jihyae Ann, 2015, Biomolecules & therapeutics.

Calcium‐dependent and independent mechanisms of capsaicin receptor (TRPV1)‐mediated cytokine production and cell death in human bronchial epithelial cells

C. Reilly, Jeewoo Lee, G. Yost, 2005, Journal of biochemical and molecular toxicology.

Differential effects of MEK inhibitors on rat neural stem cell differentiation: Repressive roles of MEK2 in neurogenesis and induction of astrocytogenesis by PD98059.

Hyun-Jung Kim, Jeewoo Lee, Ha-Rim Lee, 2019, Pharmacological research.

Hypoxia-mediated retinal neovascularization and vascular leakage in diabetic retina is suppressed by HIF-1α destabilization by SH-1242 and SH-1280, novel hsp90 inhibitors

Chang Sik Cho, Ho-Yyoung Lee, Jin Hyoung Kim, 2014, Journal of Molecular Medicine.

Novel Radiolabeled Vanilloid with Enhanced Specificity for Human Transient Receptor Potential Vanilloid 1 (TRPV1).

P. Blumberg, L. Pearce, Jihyae Ann, 2017, Journal of medicinal chemistry.

Kinetics of Penetration Influence the Apparent Potency of Vanilloids on TRPV1

Vladimir A. Pavlyukovets, P. Blumberg, S. Wincovitch, 2006, Molecular Pharmacology.

Activation of Munc13-1 by Diacylglycerol (DAG)-Lactones.

V. Marquez, Jihyae Ann, Jeewoo Lee, 2023, Biochemistry.

Syntheses and Antitumor Activities of Neorautenol and Shinpterocarpin Analogs

Jihyae Ann, Jeewoo Lee, Van-Hai Hoang, 2023, Bioorganic & Medicinal Chemistry Letters.

Development of a novel Hsp90 inhibitor NCT-50 as a potential anticancer agent for the treatment of non-small cell lung cancer

Hyun-Ju Park, Ho Jin Lee, Jihyae Ann, 2018, Scientific Reports.

The SAR analysis of TRPV1 agonists with the α-methylated B-region.

Vladimir A. Pavlyukovets, P. Blumberg, L. Pearce, 2012, Bioorganic & medicinal chemistry letters.

Discovery of RC-752, a Novel Sigma-1 Receptor Antagonist with Antinociceptive Activity: A Promising Tool for Fighting Neuropathic Pain

U. Laforenza, A. Tesei, D. Rossi, 2023, Pharmaceuticals.

Hypoxia-mediated retinal neovascularization and vascular leakage in diabetic retina is suppressed by HIF-1α destabilization by SH-1242 and SH-1280, novel hsp90 inhibitors

Chang Sik Cho, Sonia J. Park, Ho-Yyoung Lee, 2014, Journal of Molecular Medicine.

The HSP90 inhibitor HVH-2930 exhibits potent efficacy against trastuzumab-resistant HER2-positive breast cancer

Jihyae Ann, Jeewoo Lee, Soeun Park, 2024, Theranostics.

Stereospecific high-affinity TRPV1 antagonists: chiral N-(2-benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide analogues.

Dong Wook Kang, Attila Toth, HyungChul Ryu, 2008, Journal of medicinal chemistry.