B. Masjost

Structure-based optimization of novel azepane derivatives as PKB inhibitors.

R. Huber, R. Engh, C. Breitenlechner, 2004, Journal of medicinal chemistry.

Bisubstrate inhibitors for the enzyme catechol-O-methyltransferase (COMT): influence of inhibitor preorganisation and linker length between the two substrate moieties on binding affinity.

F. Diederich, C. Lerner, A. Ruf, 2003, Organic & biomolecular chemistry.

X-ray Crystal Structure of a Bisubstrate Inhibitor Bound to the Enzyme Catechol-O-methyltransferase: A Dramatic Effect of Inhibitor Preorganization on Binding Affinity.

F. Diederich, C. Lerner, A. Ruf, 2001, Angewandte Chemie.

Structure-based design, synthesis, and in vitro evaluation of bisubstrate inhibitors for catechol O-methyltransferase (COMT).

F. Diederich, F. Winkler, E. Borroni, 2000, Chemistry.

Cobalt-mediated [2+2+2] cycloaddition versus C-H and N-H activation of pyridones and pyrazinones with alkynes: an experimental study.

K. Vollhardt, M. J. Eichberg, V. Gandon, 2007, Chemistry.

Design and crystal structures of protein kinase B-selective inhibitors in complex with protein kinase A and mutants.

R. Huber, R. Engh, D. Bossemeyer, 2005, Journal of medicinal chemistry.