L. Elster

发表

Bioluminescence Resonance Energy Transfer as a Screening Assay: Focus on Partial and Inverse Agonism

C. Elling, L. Elster, A. Heding, 2007, Journal of biomolecular screening.

Guanylin and uroguanylin mRNA expression is increased following Roux-en-Y gastric bypass, but guanylins do not play a significant role in body weight regulation and glycemic control

Søren L Pedersen, P. J. Larsen, P. Vilmann, 2018, Peptides.

β-Arrestin-Based Bret2 Screening Assay for the “Non”-β-Arrestin Binding CB1 Receptor

M. Vrecl, D. L. Almholt, L. Elster, 2009, Journal of biomolecular screening.

Half-Life Extending Modifications of Peptide YY3-36 Direct Receptor-Mediated Internalization.

Søren L Pedersen, N. Hatzakis, S. Nielsen, 2019, Molecular pharmaceutics.

Lipidated PrRP31 metabolites are long acting dual GPR10 and NPFF2 receptor agonists with potent body weight lowering effect

Søren L Pedersen, J. Jelsing, N. Vrang, 2022, Scientific Reports.

Negative modulation of GABAA α5 receptors by RO4938581 attenuates discrete sub-chronic and early postnatal phencyclidine (PCP)-induced cognitive deficits in rats

C. Bundgaard, M. Didriksen, P. Larsen, 2012, Psychopharmacology.

Effects of gamma-aminobutyric acid (GABA) on synaptogenesis and synaptic function.

A. Schousboe, G. Hansen, L. Elster, 1998, Perspectives on developmental neurobiology.

Role of GABAA and GABAB Receptors in Ca++ Homeostasis and Transmitter Release in Cerebellar Granule Neurons

A. Schousboe, P. Krogsgaard‐Larsen, J. Kardos, 1996 .

Differential distribution of GABAA receptor subunits in soma and processes of cerebellar granule cells: Effects of maturation and a GABA agonist

A. Schousboe, G. Hansen, J. Fritschy, 1995, International Journal of Developmental Neuroscience.

Role of GABAB receptors in intracellular Ca2+ homeostasis and possible interaction between GABAA and GABAB receptors in regulation of transmitter release in cerebellar granule neurons

A. Schousboe, P. Krogsgaard‐Larsen, J. Kardos, 1994, Journal of neuroscience research.

ω‐Contoxin binding sites and regulation of transmitter release in cerebellar granule neurons

A. Schousboe, L. Elster, R. Squires, 1994, Journal of neuroscience research.

Expression of the GABAA receptor α6 subunit in cultured cerebellar granule cells is developmentally regulated by activation of GABAA receptors

Bo Belhage, Arne Schousboe, B. X. Carlson, 1997 .

The identification of GPR3 inverse agonist AF64394; the first small molecule inhibitor of GPR3 receptor function.

S. Poda, F. Loechel, C. Volbracht, 2014, Bioorganic & medicinal chemistry letters.

Optimisation of in silico derived 2-aminobenzimidazole hits as unprecedented selective kappa opioid receptor agonists.

T. Frimurer, I. Khanna, T. Högberg, 2015, Bioorganic & medicinal chemistry letters.

Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists.

T. Frimurer, I. Khanna, T. Högberg, 2012, Bioorganic & medicinal chemistry letters.

Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: part 2.

T. Frimurer, I. Khanna, T. Högberg, 2012, Bioorganic & medicinal chemistry letters.

Structural basis for constitutive activity and agonist‐induced activation of the enteroendocrine fat sensor GPR119

T. Frimurer, M. S. Engelstoft, C. Norn, 2014, British journal of pharmacology.

Discovery of novel, orally available benzimidazoles as melanin concentrating hormone receptor 1 (MCHR1) antagonists.

T. Frimurer, I. Khanna, T. Högberg, 2010, Bioorganic & medicinal chemistry letters.

Molecular determinants of desensitization and assembly of the chimeric GABAA receptor subunits (α1/γ2) and (γ2/α1) in combinations with β2 and γ2

U. Kristiansen, A. Schousboe, R. Olsen, 2001, Neurochemistry International.

Functional properties of glycine receptors expressed in primary cultures of mouse cerebellar granule cells

U. Kristiansen, A. Schousboe, P. Wahl, 1998, Neuroscience.

Identification and Function of Glycine Receptors in Cultured Cerebellar Granule Cells

A. Schousboe, P. Wahl, L. Elster, 1994, Journal of neurochemistry.

Pharmacological and functional implications of developmentally-regulated changes in GABA(A) receptor subunit expression in the cerebellum.

B. X. Carlson, A. Schousboe, L. Elster, 1998, European journal of pharmacology.

Stable GABAA receptor intermediates in SF‐9 cells expressing α1, β2 and γ2 subunits

A. Schousboe, R. Olsen, L. Elster, 2000 .

Uncovering CNS access of lipidated exendin-4 analogues by quantitative whole-brain 3D light sheet imaging

J. Hecksher-Sørensen, C. Clemmensen, J. Skytte, 2023, Neuropharmacology.

Structural basis for constitutive activity and agonist‐induced activation of the enteroendocrine fat sensor GPR119

T. Frimurer, M. S. Engelstoft, L. Elster, 2014, British journal of pharmacology.

Negative modulation of GABAA α5 receptors by RO4938581 attenuates discrete sub-chronic and early postnatal phencyclidine (PCP)-induced cognitive deficits in rats

C. Bundgaard, M. Didriksen, P. Larsen, 2011, Psychopharmacology.

Synthesis and SAR studies of benzimidazole derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: Focus to detune hERG inhibition

T. Frimurer, I. Khanna, T. Högberg, 2011 .