T. Besson

发表

Synthesis of novel 5-substituted indirubins as protein kinases inhibitors.

Olivier Lozach, Laurent Meijer, Thierry Besson, 2006, Bioorganic & medicinal chemistry.

Synthesis and fluorescent properties of some heterobifunctional and rigidized 7‐aminocoumarins

G. Guillaumet, T. Besson, G. Coudert, 1991 .

Erymildbraedin A and B, two novel cytotoxic dimethylpyrano-isoflavones from the stem bark of Erythrina mildbraedii: evaluation of their activity toward endocrine cancer cells

M. Alexis, X. Alexi, A. Skaltsounis, 2010, Journal of enzyme inhibition and medicinal chemistry.

Structure of Pb2+/dCMP and Pb2+/CMP complexes as characterized by tandem mass spectrometry and IRMPD spectroscopy

P. Maître, J. Tortajada, J. Salpin, 2011 .

Room-temperature infrared spectroscopy combined with mass spectrometry distinguishes gas-phase protein isomers.

R. Zubarev, J. Lemaire, P. Maître, 2009, Angewandte Chemie.

Structure of electron-capture dissociation fragments from charge-tagged peptides probed by tunable infrared multiple photon dissociation.

F. Tureček, J. Chamot-Rooke, J. Lemaire, 2008, Journal of the American Chemical Society.

Microwave-Assisted Sequential One-Pot Synthesis of 8-Substituted Pyrazolo[1,5-a][1,3,5]triazines

Corinne Fruit, T. Besson, Jonathan Elie, 2021, Molecules.

Synthesis of 2-Mercapto-(2-Oxoindolin-3-Ylidene)Acetonitriles from 3-(4-Chloro-5H-1,2,3-Dithiazol-5-Ylidene)Indolin-2-ones

V. Thiéry, T. Besson, R. Delatouche, 2018, Molecules.

Suzuki cross-coupling of 5-bromothieno[2,3-b]pyridines for the convenient synthesis of 8-arylpyrido[3′,2′:4,5]thieno[3,2-d]pyrimidin-4-amines

T. Besson, V. Levacher, Yvonnick Loidreau, 2013 .

Novel synthesis of angular thiazolo[5,4-f] and [4,5-h]quinazolines, preparation of their linear thiazolo[4,5-g] and [5,4-g]quinazoline analogs

T. Besson, C. Logé, Rémi Guillon, 2013 .

Synthesis and kinase inhibitory activity of novel substituted indigoids.

L. Meijer, C. Guguen-Guillouzo, O. Lozach, 2009, Bioorganic & medicinal chemistry.

Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors

L. Meijer, O. Lozach, Mélina Blairvacq, 2005, Journal of enzyme inhibition and medicinal chemistry.

Synthesis of novel 2,3-substituted quinazolin-4-ones by condensation of alkyl or aromatic diamines with 5-(N-arylimino)-4-chloro-5H-1,2,3-dithiazoles

V. Thiéry, T. Besson, Maria de Fátima Pereira, 2007 .

Synthesis of polyfunctionalized benzo[d]thiazoles as novel anthranilic acid derivatives

Corinne Fruit, T. Besson, Damien Hédou, 2015 .

Efficient New Synthesis of N-Arylbenzo[b]furo[3,2-d]pyrimidin-4-amines and Their Benzo[b]thieno[3,2-d]pyrimidin-4-amine Analogues via a Microwave-Assisted Dimroth Rearrangement

C. Corbière, T. Besson, P. Marchand, 2013 .

Discovery of a novel broad-spectrum antifungal agent derived from albaconazole.

P. Le Pape, T. Besson, C. Logé, 2013, ACS medicinal chemistry letters.

First synthesis of 4-aminopyrido[2′,3′:4,5]furo[3,2-d]pyrimidines

T. Besson, P. Marchand, Yvonnick Loidreau, 2012 .

Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors.

L. Meijer, O. Lozach, N. Loaëc, 2012, European journal of medicinal chemistry.

Microwave-Assisted Synthesis of Sulfur and Nitrogen-Containing Heterocycles

T. Besson, 2006 .

Multistep synthesis of thiazoloquinazolines under microwave irradiation in solution

T. Besson, J. Guillard, C. Rees, 2000 .

Efficient synthesis of thiazoloquinazolinone derivatives

R. Wrigglesworth, T. Besson, F. Alexandre, 2003 .

Study of N1-alkylation of indoles from the reaction of 2(or 3)-aminoindole-3-(or 2)carbonitriles with DMF-dialkylacetals.

Sigismund T A G Melissen, T. Besson, C. Logé, 2012, Organic & biomolecular chemistry.

Design and Synthesis of Thiazolo[5,4-f]quinazolines as DYRK1A Inhibitors, Part II

T. Taverne, A. Casagrande, Angélique Girard, 2014, Molecules.

Microwave-Assisted Synthesis of Potential Bioactive Benzo-, Pyrido- or Pyrazino-thieno[3,2-d]pyrimidin-4-amine Analogs of MPC-6827

C. Corbière, Corinne Fruit, T. Besson, 2020, Pharmaceuticals.

Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

L. Meijer, P. Bonnet, Corinne Fruit, 2018, Molecules.

Kinase inhibitors and microwave-assisted chemistry, a nice story

T. Besson, 2015 .

Structure of N-(3,4-Dimethoxyphenyl)pyrido[3′,2′:4,5]-thieno[3,2-d]pyrimidin-4-amine, a New Inhibitor of CLK1 and DYRK1A Kinases

M. Marchivie, T. Besson, N. Pinaud, 2013 .

Convenient one-pot synthesis of N3-substituted pyrido[2,3-d]-, pyrido[3,4-d]-, pyrido[4,3-d]-pyrimidin-4(3H)-ones, and quinazolin-4(3H)-ones analogs

T. Besson, E. Chosson, V. Levacher, 2013 .

Rapid synthesis of 2,3-disubstituted-quinazolin-4-ones enhanced by microwave-assisted decomposition of formamide

E. Seguin, T. Besson, I. Kostakis, 2007 .

Microwave-assisted synthesis of bioactive quinazolines and quinazolinones.

T. Besson, E. Chosson, 2007, Combinatorial chemistry & high throughput screening.

Decomposition of formamide assisted by microwaves, a tool for synthesis of nitrogen-containing heterocycles

T. Besson, I. Kostakis, E. Chosson, 2008 .

Synthesis of novel 5a,10,14b,15-tetraaza-benzo[a]indeno[1,2-c]anthracen-5-one and benzimidazo[1,2-c]quinazoline derivatives under microwave irradiation

M. Soukri, E. Essassi, M. Akssira, 2000 .

Microwave-assisted thermal decomposition of formamide: a tool for coupling a pyrimidine ring with an aromatic partner

T. Besson, Yvonnick Loidreau, 2011 .

ChemInform Abstract: Microwave-Assisted Niementowski Reaction. Back to the Roots.

T. Besson, F. Alexandre, A. Berecibar, 2002 .

Microwave-accelerated Dimroth rearrangement for the synthesis of 4-anilino-6-nitroquinazolines. Application to an efficient synthesis of a microtubule destabilizing agent

C. Corbière, T. Besson, F. Marsais, 2010 .

Microwave-assisted regioselective N-alkylation of cyclic amidines

V. Thiéry, T. Besson, Maria de Fátima Pereira, 2007 .

Antimicrobial activity of novel N-quinolinyl and N-naphthylimino-1,2,3-dithiazoles

V. Thiéry, T. Besson, G. Cottenceau, 1998 .

Antimicrobial evaluation of 3,1-benzoxazin-4-ones, 3,1-benzothiazin-4-ones, 4-alkoxyquinazolin-2-carbonitriles and N-arylimino-1,2,3-dithiazoles

T. Besson, G. Cottenceau, A. Pons, 1996 .

DYRK 1 A controls the transition from proliferation to quiescence during lymphoid development by destabilizing Cyclin D 3

Daniel E. Cook, A. Casagrande, D. E. Cook, 2015 .

Diaryliodoniums Salts as Coupling Partners for Transition-Metal Catalyzed C- and N-Arylation of Heteroarenes

Corinne Fruit, T. Besson, Alexandra Pacheco-Benichou, 2020, Catalysts.

Fe and H2O2 distributions in the upper water column in the Indian sector of the Southern Ocean

C. Jeandel, O. Donard, D. Amouroux, 1997 .

Pharmacologic Inhibition of DYRK1A Results in MYC Hyperactivation and ERK Hyperphosphorylation rendering KMT2A-R ALL Cells Sensitive to BCL2 Inhibition

G. Wertheim, M. Carroll, X. Hua, 2022, bioRxiv.

Relieving DYRK1A repression of MKL1 confers an adult-like phenotype to human infantile megakaryocytes

Ashton T. Brock, P. Gadue, S. Morris, 2022, The Journal of clinical investigation.

Synthesis and Fluorescent Properties of New Heterobifunctional Fluorescent Probes

T. Besson, B. Joseph, P. Moreau, 1992 .

Microwave-assisted synthesis of 5-carboxymethoxy-N-acetyltryptamine derivatives

G. Guillaumet, T. Besson, S. Berteina‐Raboin, 2002 .

Microwave-assisted synthesis of novel N-(4-phenylthiazol-2-yl)-benzo[d]thiazole-, thiazolo[4,5-b]pyridine-, thiazolo[5,4-b]pyridine- and benzo[d]oxazole-2-carboximidamides inspired by marine topsentines and nortopsentines

T. Besson, V. Levacher, Carole Dubouilh-Benard, 2014 .

Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core

Florent Alix, T. Besson, Mihaela-Liliana Ţînţaş, 2022, Molecules.

SYNTHESIS OF 3,1-BENZOXAZINES, 3,1-BENZOTHIAZINES AND 3,1-BENZOXAZEPINES VIA N-ARYLIMINO-1,2,3-DITHIAZOLES

G. Guillaumet, T. Besson, C. Rees, 1997 .

Synthesis of novel 1,3,4-benzotriazepine derivatives from 4-oxo-3,1-benzoxazine and 3,1-benzothiazine-2-carbonitriles

R. Wrigglesworth, J. Leger, V. Thiéry, 2005 .

Synthesis of novel 2-cyanothiazolocarbazoles analogues of ellipticine

G. Guillaumet, V. Thiéry, T. Besson, 2002 .

Expeditious synthesis and cytotoxic activity of new cyanoindolo[3,2-c]quinolines and benzimidazo[1,2-c]quinazolines.

P. Renard, B. Pfeiffer, G. Guillaumet, 2000, Bioorganic & medicinal chemistry letters.

Synthesis of 3,1‐Benzoxazines, 3,1‐Benzothiazines and 3,1‐ Benzoxazepines via N‐Arylimino‐1,2,3‐dithiazoles.

G. Guillaumet, T. Besson, C. Rees, 1997 .

Synthesis of latonduine derivatives via intramolecular Heck reaction

Lionel Joucla, T. Besson, B. Joseph, 2007 .

Microwave-induced by-products in the synthesis of 2-(4-methyl-2-phenylpiperazinyl)pyridine-3-carbonitrile

P. Carlier, T. Besson, R. T. Halle, 2009 .

First synthesis of 2-aminosubstituted-2-perfluoroalkyl-3,6-dihydro-2H-thiopyrans by hetero-Diels–Alder reactions of fluorinated thioamides under microwave heating

Yu. G. Shermolovich, T. Besson, J. Bouillon, 2010 .

Synthesis and antiproliferative activity of clausine E, mukonine, and koenoline bioisosteres.

C. Galmarini, F. Popowycz, T. Besson, 2007, Bioorganic & medicinal chemistry.

Influence of microwave radiation on free Candida antarctica lipase B activity and stability.

S. Lamare, T. Besson, M. Legoy, 2006, Organic & biomolecular chemistry.

Stability improvement of immobilized Candida antarctica lipase B in an organic medium under microwave radiation.

S. Lamare, T. Besson, M. Legoy, 2004, Organic & biomolecular chemistry.

Synthesis and evaluation of the antimicrobial activity of novel quinazolinones

Romain Chevrot, E. Rosenfeld, V. Thiéry, 2007, Journal of enzyme inhibition and medicinal chemistry.

Microwave-Assisted Niementowski Reaction. Back to the Roots.

T. Besson, F. Alexandre, A. Berecibar, 2002 .

Microwaves in drug discovery and multi-step synthesis

Stéphane Frère, V. Thiéry, T. Besson, 2004, Molecular Diversity.

Synthesis of novel 2,3-condensed thieno[2,3- d ]pyrimidin-4-ones via Appel's salt chemistry

V. Thiéry, T. Besson, Maria de Fatima Pereira, 2006 .

Efficient synthesis of novel pentacyclic 6,7-dihydro-5a,7a,13,14-tetraaza-pentaphene-5,8-diones

J. Leger, C. Jarry, V. Thiéry, 2005 .

Novel series of 8H-quinazolino[4,3-b]quinazolin-8-ones via two Niementowski condensations

R. Wrigglesworth, T. Besson, F. Alexandre, 2003 .

Cu/Pd-Catalyzed C-2–H Arylation of Quinazolin-4(3H)-ones with (Hetero)aryl Halides

Corinne Fruit, Sylvain Laclef, T. Besson, 2015 .

Synthesis and antitumoral activity of novel thiazolobenzotriazole, thiazoloindolo[3,2-c]quinoline and quinolinoquinoline derivatives.

C. Bailly, Anne Beauchard, V. Thiéry, 2009, European journal of medicinal chemistry.

Synthesis of original thiazoloindolo[3,2-c]quinoline and novel 8-N-substituted-11H-indolo[3,2-c]quinoline derivatives from benzotriazoles. Part I

P. Guenot, Anne Beauchard, V. Thiéry, 2006 .

Synthesis of novel 7-oxo and 7-hydroxy trifluoroallocolchicinoids with cytotoxic effect.

Jana Sopkova-de Oliveira Santos, Rémi Legay, T. Cresteil, 2012, Bioorganic & medicinal chemistry.

Cytotoxic evaluation of sarcodifurines A and B, two novel dihydrofuroquinolines from Sarcomelicope follicularis (Rutaceae)

C. Guguen-Guillouzo, D. Glaise, E. Seguin, 2008 .

Regio- and Stereoselective Synthesis of (Z)-Vinylgermanes by Hydrogermylation of Alkynes

V. Thiéry, T. Besson, M. Abarbri, 2007 .

Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts

Corinne Fruit, T. Besson, 2021, Pharmaceuticals.

Microwave acceleration of the Pechmann reaction on graphite/montmorillonite K10: application to the preparation of 4-substituted 7-aminocoumarins

Stéphane Frère, V. Thiéry, T. Besson, 2001 .

Ligand-free Pd-catalyzed and copper-assisted C-H arylation of quinazolin-4-ones with aryl iodides under microwave heating.

Corinne Fruit, Sylvain Laclef, T. Besson, 2015, Organic letters.

New syntheses of aryl isothiocyanates

V. Thiéry, T. Besson, J. Guillard, 1998 .

Synthesis of Benzo-Fused 11H-Pyrido[2,1-b]quinazolin-11-ones by a Buchwald–Hartwig Coupling/Pyridine Dearomatization Sequence in Eucalyptol

Corinne Fruit, T. Besson, S. Berteina‐Raboin, 2020 .

Efficient modified von Niementowski synthesis of novel derivatives of 5a,14b,15-triazabenzo[a]indeno[1,2-c]anthracen-5-one from indolo[1,2-c]quinazoline

A. Grélard, V. Thiéry, T. Besson, 2001 .

Developments in Meyers' lactamization methodology: en route to bi(hetero)aryl structures with defined axial chirality.

M. Sabbah, T. Besson, S. Oudeyer, 2013, The Journal of organic chemistry.

Heterocyclic Chemistry Using Microwave‐Assisted Approaches

T. Besson, C. Brain, 2009 .

Microwave-assisted synthesis of galacto-oligosaccharides from lactose with immobilized β-galactosidase from Kluyveromyces lactis

T. Maugard, T. Besson, M. Legoy, 2003, Biotechnology Letters.

Microwave-assisted synthesis of a-ethoxycarbamates

A. Lumbroso, E. L. Grognec, T. Besson, 2009 .

Influence of microwave irradiation on enzymatic properties: applications in enzyme chemistry

S. Lamare, T. Besson, M. Legoy, 2007, Journal of enzyme inhibition and medicinal chemistry.

Microwave-assisted solid-phase synthesis of 5-carboxamido-N-acetyltryptamine derivatives.

G. Guillaumet, T. Besson, S. Berteina‐Raboin, 2002, Organic letters.

Synthesis of Bioactive 2-(Arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff Reaction or Cu- Catalyzed Intramolecular C-S Bond Formation

L. Meijer, N. Loaëc, Corinne Fruit, 2016, Molecules.

Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases

L. Meijer, N. Loaëc, Corinne Fruit, 2016, Molecules.

Design and Synthesis of Thiazolo[5,4-f]quinazolines as DYRK1A Inhibitors, Part I

L. Meijer, A. Casagrande, N. Loaëc, 2014, Molecules.

Novel 6-Substituted Benzothiazol-2-yl Indolo[1,2-c]quinazolines and Benzimidazo[1,2-c]quinazolines.

C. Bailly, Stéphane Frère, V. Thiéry, 2003 .

Synthesis and Cytotoxic Evaluation of Novel Thiazolocarbazoles. Part II1

P. Renard, B. Pfeiffer, G. Guillaumet, 2003, Journal of enzyme inhibition and medicinal chemistry.

Novel 6-substituted benzothiazol-2-yl indolo[1,2-c]quinazolines and benzimidazo[1,2-c]quinazolines

C. Bailly, Stéphane Frère, V. Thiéry, 2003 .

Synthesis and Cytotoxic Evaluation of Novel Thiazolocarbazoles

P. Renard, B. Pfeiffer, G. Guillaumet, 2002, Journal of enzyme inhibition and medicinal chemistry.

Efficient Modified von Niementowski Synthesis of Novel Derivatives of 5a,14b,15-Triazabenzo[a]indeno[1,2-c]anthracen-5-one from Indolo[1,2-c]quinazoline.

A. Grélard, V. Thiéry, T. Besson, 2001 .

Synthesis and in vitro antitumour evaluation of benzothiazole-2-carbonitrile derivatives

B. Pfeiffer, T. Besson, J. Guillard, 1999 .

Synthesis of novel dioxinobenzothiazole derivatives

T. Besson, J. Guillard, 1999 .

Expeditious Routes to 4‐Alkoxyquinazoline‐2‐carbonitriles and Thiocarbamates via N‐Arylimino‐1,2,3‐dithiazoles Using Microwave Irradiation.

T. Besson, J. Guillard, M. Legoy, 1998 .

Expeditious routes to 4-alkoxyquinazoline-2-carbonitriles and thiocarbamates via N-arylimino-1,2,3-dithiazoles using microwave irradiation

T. Besson, J. Guillard, M. Legoy, 1998 .

New route to 2-cyanobenzothiazoles via N -arylimino-1,2,3-dithiazoles†

T. Besson, J. Guillard, C. Rees, 1998 .

Rapid Synthesis of 2‐Cyanobenzothiazoles from N‐Aryliminodithiazoles under Microwave Irradiation.

T. Besson, C. Rees, V. Bénéteau, 1997 .

Rapid Synthesis of 2-Cyanobenzothiazoles from N-Aryliminodithiazoles Under Microwave Irradiation

T. Besson, C. Rees, V. Bénéteau, 1997 .

Some chemistry of 4,5-dichloro-1,2,3-dithiazolium chloride and its derivatives

T. Besson, C. Rees, 1995 .

Efficient solvent-free microwave phosphorylation of microcrystalline cellulose

Thierry Besson, Gabrielle Charlotte Chitanu, Adrian Carpov, 2002 .

Synthesis and Cytotoxic Activity of Thiazolofluorenone Derivatives

P. Renard, B. Pfeiffer, G. Guillaumet, 2004, Journal of enzyme inhibition and medicinal chemistry.

Microwave-assisted Synthesis of Novel Thiazolocarbazoles and Evaluation as Potential Anticancer Agents. Part III

V. Thiéry, T. Besson, Laurent Picot, 2004, Journal of enzyme inhibition and medicinal chemistry.

A rapid and convenient synthesis of novel 1-imino-2,3-dihydro-1H-pyrazino[2,1,-b]quinazolin-5-ones

V. Thiéry, T. Besson, F. Alexandre, 2004 .

Efficient Synthesis of Novel Pentacyclic 6,7‐Dihydro‐5a,7a,13,14‐tetraaza‐pentaphene‐5,8‐diones.

J. Leger, C. Jarry, V. Thiéry, 2005 .

Synthesis of novel pentacyclic pyrrolothiazolobenzoquinolinones, analogs of natural marine alkaloids

T. Besson, V. Bénéteau, 2001 .

Review on the Synthesis and Therapeutic Potential of Pyrido[2,3-d], [3,2-d], [3,4-d] and [4,3-d]pyrimidine Derivatives

T. Besson, S. Berteina‐Raboin, J. F. Campos, 2022, Pharmaceuticals.

Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: synthesis, biological evaluation and molecular modeling studies.

L. Meijer, O. Lozach, J. Robert, 2008, European journal of medicinal chemistry.

Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles

Stéphane Frère, V. Thiéry, T. Besson, 2003 .

Recent Developments in Microwave-Assisted Metal-Catalyzed C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications

Corinne Fruit, T. Besson, 2016 .

Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3.

L. Meijer, O. Lozach, J. Robert, 2006, Bioorganic & medicinal chemistry letters.

1,2,3-Dithiazoles and new routes to 3,1-benzoxazin-4-ones, 3,1-benzothiazin-4-ones and N-arylcyanothioformamides

K. Emayan, T. Besson, C. Rees, 1995 .

Copper-Catalyzed C–H Arylation of Fused-Pyrimidinone Derivatives Using Diaryliodonium Salts

Corinne Fruit, T. Besson, I. Kostakis, 2020, Catalysts.

Pd-Catalyzed and Copper Assisted Regioselective Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides.

Corinne Fruit, T. Besson, Marine Harari, 2016, Organic letters.

Cu/Pd‐Catalyzed C‐2—H Arylation of Quinazolin‐4(3H)‐ones with (Hetero)aryl Halides.

Corinne Fruit, Sylvain Laclef, T. Besson, 2016 .

Microwave-Assisted [3+2] Cycloaddition and Suzuki–Miyaura Cross-Coupling for a Concise Access to Polyaromatic Scaffolds†

T. Besson, E. Chosson, V. Levacher, 2013 .

Conception of DYRK1A kinase inhibitors via metal-catalyzed C–H arylation, inspired by fragment-growing studies

L. Meijer, P. Bonnet, Corinne Fruit, 2018, Proceedings of 4th International Electronic Conference on Medicinal Chemistry.

3,1-Benzoxazin-4-ones, 3,1-benzothiazin-4-ones and N-arylcyanothioformamides

K. Emayan, T. Besson, C. Rees, 1995 .

Synthesis of 2-Cyanobenzothiazoles via Pd-Catalyzed/Cu-Assisted C-H Functionalization/Intramolecular C-S Bond Formation from N-Arylcyanothioformamides

Corinne Fruit, T. Besson, Alexandra Pacheco-Benichou, 2022, Molecules.

Pictet–Spengler heterocyclizations via microwave-assisted degradation of DMSO

D. Lesieur, S. Yous, C. Mesangeau, 2005 .

Mitsunobu Thiofunctionalization-Part 2.1 an Expedient Synthesis of Aza-Heterocycle/Thiosugar Hybrids

T. Besson, P. Rollin, M. Viaud, 1990 .

4,5‐Dichloro‐1,2,3‐dithiazol‐1‐ium Chloride

T. Besson, E. Chosson, Alicia Foucourt, 2009 .

Microwave radiation can increase the rate of enzyme-catalysed reactions in organic media

S. Lamare, M. Parker, T. Besson, 1996 .

Biophysical and biological properties of newly synthesized dioxinocoumarin derivatives. II. Dark and photoinduced effects on T7 phage, yeast and HeLa cells.

D. Averbeck, S. Nocentini, G. Rontó, 1994, Journal of photochemistry and photobiology. B, Biology.

Biophysical and biological properties of newly synthesized dioxinocoumarin derivatives. Part I: Dark effects on T7 phage and HeLa cells.

S. Nocentini, G. Guillaumet, T. Besson, 1993, Journal of photochemistry and photobiology. B, Biology.

Synthesis of novel 7-substituted pyrido[2',3':4,5]furo[3,2-d]pyrimidin-4-amines and their N-aryl analogues and evaluation of their inhibitory activity against Ser/Thr kinases.

L. Meijer, N. Loaëc, T. Besson, 2013, Bioorganic & medicinal chemistry letters.

Synthesis and biological evaluation of N-aryl-7-methoxybenzo[b]furo[3,2-d]pyrimidin-4-amines and their N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amine analogues as dual inhibitors of CLK1 and DYRK1A kinases.

L. Meijer, N. Loaëc, T. Besson, 2013, European journal of medicinal chemistry.

A mild One-Step Procedure for the Synthesis of β-Iodo Epoxides from the Corresponding Epoxy-Alcohols

T. Besson, P. Rollin, 1990 .

Dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitors: a survey of recent patent literature

Y. Hérault, L. Meijer, Thu Lan Nguyen, 2017, Expert opinion on therapeutic patents.

Synthesis and molecular modelling studies of 8-arylpyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors.

L. Meijer, N. Loaëc, T. Besson, 2015, European journal of medicinal chemistry.

A novel DYRK1A (Dual specificity tyrosine phosphorylation‐regulated kinase 1A) inhibitor for the treatment of Alzheimer's disease: effect on Tau and amyloid pathologies in vitro

C. Oliveira, T. Taverne, M. Pando, 2015, Journal of neurochemistry.

DYRK1A regulates B cell acute lymphoblastic leukemia through phosphorylation of FOXO1 and STAT3.

Y. Goo, S. Izraeli, Q. Wen, 2021, The Journal of clinical investigation.

Biological Characterization of 8-Cyclopropyl-2-(pyridin-3-yl)thiazolo[5,4-f]quinazolin-9(8H)-one, a Promising Inhibitor of DYRK1A

L. Meijer, Corinne Fruit, J. Crispino, 2019, Pharmaceuticals.

DYRK1A controls the transition from proliferation to quiescence during lymphoid development by destabilizing Cyclin D3

Daniel E. Cook, A. Casagrande, D. E. Cook, 2015, The Journal of experimental medicine.

Antimicrobial Activity of Novel N-Quinolinyl and N-Naphthylimino-1,2,3-dithiazoles.

V. Thiéry, T. Besson, G. Cottenceau, 1998 .

Antimicrobial Activity of Novel N-Arylimino-1, 2, 3-Dithiazoles

V. Thiéry, T. Besson, J. Guillard, 1998 .

Antibacterial evaluation of novel N-Arylimino-1,2,3-dithiazoles and N-arylcyanothioformamides

T. Besson, V. Gautier, G. Cottenceau, 1996 .

New syntheses of aryl isothiocyanates fromN-arylimino-1,2,3-dithiazoles

T. Besson, J. Guillard, M. Thérisod, 1997 .

Antibacterial Evaluation of Novel N-Arylimino-1,2,3-dithiazoles and N- Arylcyanothioformamides.

T. Besson, V. Gautier, G. Cottenceau, 1996 .

Synthesis and preliminary antiproliferative evaluation of 1,3,9-triazacyclopenta[b]fluorene derivatives

V. Thiéry, T. Besson, B. Joseph, 2005, Journal of enzyme inhibition and medicinal chemistry.

On the origin of some cubebene derivatives — Diels–Alder adducts and the diene structures of solidago compounds

André Pelletier, J. Bélanger, J. Paré, 2007 .

Gas-phase structure of a pi-allyl-palladium complex: efficient infrared spectroscopy in a 7 T Fourier transform mass spectrometer.

J. Lemaire, P. Maître, J. Bakker, 2007, The journal of physical chemistry. A.

Tautomerism of uracil probed via infrared spectroscopy of singly hydrated protonated uracil.

Rajeev Kumar Sinha, P. Maître, J. Bakker, 2008, The journal of physical chemistry. A.

Convenient synthesis of 5-substituted-6-methoxy or 6-hydroxy-2,3-dihydro-1,4-benzodioxins via lithiated intermediates

G. Guillaumet, T. Besson, G. Coudert, 1993 .

Synthesis of a benzodioxinic analog of 8-methoxypsoralen

G. Guillaumet, T. Besson, G. Coudert, 1995 .

Convenient Synthesis of 5-Substituted 6-Methoxy- or 6-Hydroxy-2,3- dihydro-1,4-benzodioxins via Lithiated Intermediates.

G. Guillaumet, T. Besson, G. Coudert, 1993 .

Synthesis of a Benzodioxinic Analogue of 8-Methoxypsoralen.

G. Guillaumet, T. Besson, G. Coudert, 1995 .

Expeditious Synthesis and Cytotoxic Activity of New Cyanoindolo[3,2‐c]quinolines and Benzimidazo[1,2‐c]quinazolines.

P. Renard, B. Pfeiffer, G. Guillaumet, 2000 .

Exploring Kinase Inhibition Properties of 9H-pyrimido[5,4-b]- and [4,5-b]indol-4-amine Derivatives

L. Meijer, N. Loaëc, T. Besson, 2020, Pharmaceuticals.

Microwave‐Accelerated Dimroth Rearrangement for the Synthesis of 4‐Anilino‐6‐nitroquinazolines. Application to an Efficient Synthesis of a Microtubule Destabilizing Agent.

C. Corbière, T. Besson, F. Marsais, 2010 .

An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases.

S. Knapp, A. Casagrande, P. Bonnet, 2016, Journal of medicinal chemistry.

Imidazoquinolinethiones from 8-aminoquinolines by a novel peri-participation

David G. Roe, V. Thiéry, T. Besson, 2000 .

Discovery of a novel broad-spectrum antifungal agent derived from albaconazole.

P. Le Pape, T. Besson, C. Logé, 2013, ACS medicinal chemistry letters.

Developments in Meyers' lactamization methodology: en route to bi(hetero)aryl structures with defined axial chirality.

M. Sabbah, T. Besson, S. Oudeyer, 2013, The Journal of organic chemistry.

Binaphthyl platform as starting materials for the preparation of electron rich benzo[g,h,i]perylenes. Application to molecular architectures based on amino benzo[g,h,i]perylenes and carborane combinations.

F. Teixidor, C. Viňas, M. Hursthouse, 2011, Chemical communications.

Dissociation reactions of free tetrapyridinium tetracations and of their catenanes.

D. Schröder, J. Roithová, Petr Milko, 2007, Journal of the American Chemical Society.