T. Kogan

发表

Novel inhibitors of α4β1 integrin receptor interactions through library synthesis and screening

A. Souers, J. Ellman, W. Ankener, 1998 .

A Single Amino Acid Residue Can Determine the Ligand Specificity of E-selectin (*)

T. Kogan, B. M. Revelle, S. Tapp, 1995, The Journal of Biological Chemistry.

Structure-function analysis of P-selectin-sialyl LewisX binding interactions. Mutagenic alteration of ligand binding specificity.

T. Kogan, D. Scott, P. Beck, 1996, The Journal of biological chemistry.

State-of-the-Art Review: The Preclinical and Clinical Pharmacology of Novastan (Argatroban): A Small-Molecule, Direct Thrombin Inhibitor

J. Becker, T. Kogan, R. Schwarz, 1997 .

Glycomimetic selectin inhibitors: (α-D-mannopyranosyloxy)methylbiphenyls

T. Kogan, H. Bui, K. Keller, 1996 .

Rational design and synthesis of small molecule, non-oligosaccharide selectin inhibitors: (alpha-D-mannopyranosyloxy)biphenyl-substituted carboxylic acids.

T. Kogan, H. Bui, K. Keller, 1995, Journal of medicinal chemistry.

Selectin blockade prevents antigen-induced late bronchial responses and airway hyperresponsiveness in allergic sheep.

R. Dixon, E. Yeh, R. Bjercke, 1999, American journal of respiratory and critical care medicine.

Novastan® (Brand of Argatroban): A Small-Molecule, Direct Thrombin Inhibitor

Kenneth J. Alford, J. Becker, T. Kogan, 1997, Seminars in thrombosis and hemostasis.

Discovery of TBC11251, a potent, long acting, orally active endothelin receptor-A selective antagonist.

R. Dixon, I. Okun, T. Kogan, 1997, Journal of Medicinal Chemistry.

Small-molecule selectin inhibitor protects against liver inflammatory response after ischemia and reperfusion.

L. Toledo-Pereyra, R. Dixon, T. Kogan, 1997, Journal of the American College of Surgeons.

Modification of CD4 immunoadhesin with monomethoxypoly(ethylene glycol) aldehyde via reductive alkylation.

S. Shak, M. Venuti, A. Ashkenazi, 1994, Bioconjugate chemistry.

The synthesis of a phorbol 12,13-bis-lactone

T. Rawson, T. Kogan, 1992 .

A Regio- and stereocontrolled total synthesis of (-)-indolactam-V

M. Venuti, T. Somers, T. Kogan, 1990 .

Conjugation of soluble CD4 without loss of biological activity via a novel carbohydrate-directed cross-linking reagent.

A. Ashkenazi, S. Chamow, R. Byrn, 1992, The Journal of biological chemistry.

Use of halomethyl resins to immobilize amines: An efficient method for synthesis of sulfonamides and amides on a solid support

T. Kogan, B. Raju, 1997 .

A Highly Practical Route to 7-Hydroxy-1,3-dihydro-2H-1,4-benzodiazepin-2-one from p-Anisidine

T. Kogan, Chengde Wu, Ronald J. Biediger, 1999 .

The synthesis of chiral 3-oxo-6-[(phenylmethoxy)-carbonyl]-2-piperazineacetic acid esters designed for the presentation of an aspartic acid side chain. A subsequent novel Friedel Crafts reaction

T. Rawson, T. Kogan, 1992 .

Substituted (1,2-diarylethyl)amide acyl-CoA:cholesterol acyltransferase inhibitors: effect of polar groups on in vitro and in vivo activity.

R. Burrier, J. Clader, H. Davis, 1995, Journal of medicinal chemistry.

Separation of 21-(R)- and 21-(S)-argatroban: solubility and activity of the individual diastereoisomers.

T. Rawson, T. Kogan, J. Yang, 1993, Journal of pharmaceutical sciences.

Endothelin antagonists: substituted mesitylcarboxamides with high potency and selectivity for ET(A) receptors.

R. Dixon, T. Kogan, T. Brock, 1999, Journal of medicinal chemistry.

The Synthesis of Substituted Methoxy-Poly(Ethyleneglycol) Derivatives Suitable for Selective Protein Modification

T. Kogan, 1992 .

Novel synthetic inhibitors of selectin-mediated cell adhesion: synthesis of 1,6-bis[3-(3-carboxymethylphenyl)-4-(2-alpha-D- mannopyranosyloxy)phenyl]hexane (TBC1269).

R. Dixon, T. Kogan, P. Vanderslice, 1998, Journal of medicinal chemistry.

A 3D structure model of integrin alpha 4 beta 1 complex: I. Construction of a homology model of beta 1 and ligand binding analysis.

R. Dixon, T. You, J. Li, 2002, Biophysical journal.

A 3D Structure Model of Integrin α4β1 Complex: I. Construction of a Homology Model of β1 and Ligand Binding Analysis

Jian Li, Richard A. Dixon, Tony J. You, 2002 .

A cyclic hexapeptide is a potent antagonist of alpha 4 integrins.

E. Yeh, R. Bjercke, T. Kogan, 1997, Journal of immunology.

Solution-phase combinatorial synthesis of ureas using nitrophenylcarbamates.

T. Kogan, J. Kassir, B. Raju, 1998, Bioorganic & medicinal chemistry letters.

Novel Synthetic Inhibitors of Selectin‐Mediated Cell Adhesion: Synthesis of 1,6‐Bis[3‐(3‐carboxymethylphenyl)‐4‐ (2‐α‐D‐mannopyranosyloxy)phenyl]hexane (TBC1269).

R. Dixon, T. Kogan, P. Vanderslice, 1998 .

Role for heparin-binding growth factors in glucose-induced vascular dysfunction.

J. Williamson, R. Tilton, W. Lejeune, 1998, Diabetes.