Laurence Quéguiner

发表

Selection of a respiratory syncytial virus fusion inhibitor clinical candidate, part 1: improving the pharmacokinetic profile using the structure-property relationship.

K. Andries, P. Timmerman, E. Arnoult, 2007, Journal of medicinal chemistry.

Ion mobility-mass spectrometry analysis of diarylquinoline diastereomers: Drugs used for tuberculosis treatment

E. Arnoult, J. Guillemont, C. Afonso, 2018, European journal of mass spectrometry.

Discovery of pyrimidyl-5-hydroxamic acids as new potent histone deacetylase inhibitors.

M. Janicot, L. van Hijfte, H. De Winter, 2005, European journal of medicinal chemistry.

Identification of a series of substituted 2-piperazinyl-5-pyrimidylhydroxamic acids as potent histone deacetylase inhibitors.

M. Janicot, M. Noppe, L. van Hijfte, 2010, Bioorganic & medicinal chemistry letters.

Synthesis and biological evaluation of C-5 methyl substituted 4-arylthio and 4-aryloxy-3-Iodopyridin-2(1H)-one type anti-HIV agents.

K. Hertogs, C. Nguyen, K. Andries, 2009, Journal of medicinal chemistry.

Minisci-Photoredox-Mediated α-Heteroarylation of N-Protected Secondary Amines: Remarkable Selectivity of Azetidines.

J. Edwards, H. Beucher, L. Meerpoel, 2018, Organic letters.

Synthesis of novel diarylpyrimidine analogues of TMC278 and their antiviral activity against HIV-1 wild-type and mutant strains.

K. Hertogs, A. Peeters, J. Heeres, 2007, European journal of medicinal chemistry.

Selection of a respiratory syncytial virus fusion inhibitor clinical candidate. 2. Discovery of a morpholinopropylaminobenzimidazole derivative (TMC353121).

K. Andries, C. Meyer, P. Timmerman, 2008, Journal of medicinal chemistry.

Synthesis and evaluation of analogues of the tuberculosis drug bedaquiline containing heterocyclic B-ring units

Christopher B. Cooper, W. Denny, B. Palmer, 2017, Bioorganic & medicinal chemistry letters.

Short Communication Discovery of pyrimidyl-5-hydroxamic acids as new potent histone deacetylase inhibitors

M. Janicot, Laurence Quéguiner, L. Hijfte, 2005 .