Chunhao Yang

发表

Direct Approach to 3-Fluoroindoles and 3,3-Difluoroindolines from 2,2-Difluoro-2-phenylethan-1-amines via C–H/N–H Coupling

Lanfei Zhang, Xiaofei Zhang, Yongmei Cui, 2021, Synthesis.

Synthesis of multisubstituted 2-aminopyrroles/pyridines via chemoselective Michael addition/intramolecular cyclization reaction.

Chunhao Yang, Haoyue Xiang, Xueyu Qi, 2014, Organic letters.

Regioselective synthesis of substituted thiazoles via cascade reactions from 3-chlorochromones and thioamides.

Chen Cui, Xiaofei Zhang, Chunhao Yang, 2020, Organic & biomolecular chemistry.

Copper(II)-catalyzed cascade approach for the synthesis of pyrrolo[2,1-f][1,2,4]triazine-fused isoquinolines

Chunhao Yang, Jianyang Chen, Qian He, 2014 .

Design, synthesis, and biological evaluations of substituted pyrazoles as pyrrolomycin analogues against staphylococcal biofilm.

L. Lan, Xiaofei Zhang, Chunhao Yang, 2022, European journal of medicinal chemistry.

Synthesis and Biological Evaluation of C-17-Amino-Substituted Pyrazole-Fused Betulinic Acid Derivatives as Novel Agents for Osteoarthritis Treatment.

Shi-qi Cao, Bintao Hu, Xiaofei Zhang, 2021, Journal of medicinal chemistry.

Visible-Light-Driven, Radical-Triggered Tandem Cyclization of o-Hydroxyaryl Enaminones: Facile Access to 3-CF2 /CF3-Containing Chromones.

Hua Yang, Chunhao Yang, Jun‐An Xiao, 2017, Organic letters.

Palladium-catalyzed direct approach to α-CF3 aryl ketones from arylboronic acids

Xiaofei Zhang, Chunhao Yang, Bo Jiang, 2018 .

C-H Trifluoromethylation of 2-Substituted/Unsubstituted Aminonaphthoquinones at Room Temperature with Bench-Stable (CF3SO2)2Zn: Synthesis and Antiproliferative Evaluation.

Jian Ding, Lin-jiang Tong, Xiaofei Zhang, 2017, The Journal of organic chemistry.

Alkylations of Arylboronic Acids including Difluoroethylation/Trifluoroethylation via Nickel‐Catalyzed Suzuki Cross‐Coupling Reaction

Xiaofei Zhang, Chunhao Yang, 2015 .

Synthesis and biological evaluation of rhein amides as inhibitors of osteoclast differentiation and bone resorption.

L. Deng, Changwei Li, Yufei Yan, 2016, European journal of medicinal chemistry.

Pd-Catalyzed intramolecular C–H activation and C–S formation to synthesize pyrazolo[5,1-b]benzothiazoles without an additional oxidant

Xiaofei Zhang, Chunhao Yang, Qian He, 2019, Organic Chemistry Frontiers.

Novel indole α-methylene-γ-lactones as potent inhibitors for AKT-mTOR signaling pathway kinases

Jian Ding, Xiongwen Zhang, Xihan Wu, 2005 .

Copper-mediated, palladium-catalyzed cross-coupling of 3-iodochromones, thiochromones, and quinolones with ethyl bromodifluoroacetate.

Xiaofei Zhang, Chunhao Yang, Zhizhou Yue, 2013, The Journal of organic chemistry.

A One‐Pot Copper(II)‐Catalyzed Tandem Synthesis of 2‐Substituted Pyrrolo[1,2‐b]pyridazin‐4(1H)‐ones

Chunhao Yang, Cun Tan, Qian He, 2015 .

A novel convenient approach towards pyrrolo[1,2-b]pyridazines through a domino coupling-isomerization-condensation reaction.

Chunhao Yang, Cun Tan, Qian He, 2013, Organic & biomolecular chemistry.

Synthesis and biological evaluation of novel bisphosphonates with dual activities on bone in vitro.

Chunhao Yang, Xueming Yan, Yuli Xie, 2005, Bioorganic & medicinal chemistry letters.

Efficient Pd-catalyzed domino synthesis of 1-phenyl-1H-indol-2-amine and 5-amino-indolo[1,2-a]quinazoline derivatives.

L. Deng, M. Jiang, Xingzhu Xu, 2015, Organic & biomolecular chemistry.

One-pot syntheses of novel pyrazole-containing bisphosphonate esters at room temperature.

Chunhao Yang, Guangyu Xu, Xueyu Qi, 2012, Organic & biomolecular chemistry.

An efficient and practical approach to trifluoromethylthiolation of α-haloketones/α-haloarylmethanes.

L. Deng, M. Jiang, Xingzhu Xu, 2015, Organic & biomolecular chemistry.

A facile and general approach to 3-((trifluoromethyl)thio)-4H-chromen-4-one.

Chunhao Yang, H. Xiang, 2014, Organic letters.

Palladium-catalyzed oxidative C-H/C-H cross-coupling of benzothiazoles with thiophenes and thiazoles.

Chunhao Yang, Xuxing Chen, Qian He, 2014, Chemical communications.

Synthesis of Functionalized Chromeno[2,3-b]pyrrol-4(1H)-ones by Silver-Catalyzed Cascade Reactions of Chromones/Thiochromones and Isocyanoacetates.

Chunhao Yang, Xueyu Qi, H. Xiang, 2015, Organic letters.

Metal-Free Access to (E/Z )-α-Fluorovinyl Phosphorus Compounds from gem -Difluorostyrenes

Bin Zhang, Xiaofei Zhang, Chunhao Yang, 2019, European Journal of Organic Chemistry.

Syntheses of quinolone hydrochloride enantiomers from synthons (R)- and (S)-2-methylpiperazine.

J. Cui, Xihan Wu, Chunhao Yang, 2005, Bioorganic & medicinal chemistry.

Palladium-Catalyzed Direct Approach to α-Trifluoromethyl Alcohols by Selective Hydroxylfluorination of gem -Difluoroalkenes

Bin Zhang, Xiaofei Zhang, Chunhao Yang, 2018, European Journal of Organic Chemistry.

Direct Approach to N-Substituted-2-Fluoroindoles by Sequential Construction of C-N Bonds from gem-Difluorostyrenes.

Bin Zhang, Xiaofei Zhang, Chunhao Yang, 2017, Organic letters.

A Concise and Efficient Approach to 2,6-Disubstituted 4-Fluoropyrimidines from α-CF3 Aryl Ketones

Xiaofei Zhang, Chunhao Yang, Q. Qian, 2019, Synthesis.

SYNTHESIS OF 2-SUBSTITUTED PYRIMIDO[5,4-b]INDOLIZINE DERIVATIVES FROM ACETATES OF BAYLIS-HILLMAN ADDUCTS

M. Jiang, Chunhao Yang, Qian He, 2008 .

Convenient synthesis of 1,2,3,4-tetrahydroquinolines via direct intramolecular reductive ring closure

Chunhao Yang, Wuhong Chen, Bo Liu, 2006 .

One‐Pot Syntheses of Novel Pyrazole‐Containing Bisphosphonate Esters at Room Temperature.

Chunhao Yang, Guangyu Xu, Xueyu Qi, 2013 .

One-pot transition-metal-free cascade synthesis of thieno[2,3-c]coumarins from chromones

Yu-Hong Yang, Chunhao Yang, Xueyu Qi, 2016 .

Cascade synthesis of novel functionalized pyridine-fused coumarins in aqueous medium

Z. Miao, Chunhao Yang, Jianyang Chen, 2014 .

Rapid access to α-carbolines via a one-pot tandem reaction of α,β-unsaturated ketones with 2-nitrophenylacetonitrile and the anti-proliferative activities of the products.

Z. Miao, Xiaofei Zhang, Chunhao Yang, 2014, Organic & biomolecular chemistry.

Palladium(II)-catalyzed synthesis of functionalized indenones via oxidation and cyclization of 2-(2-arylethynylphenyl)acetonitriles.

Chunhao Yang, Xuxing Chen, Qian He, 2013, Organic & biomolecular chemistry.

Synthesis of Rigid Analogues of Flavone by Intramolecular Heck Reaction

L. Deng, M. Jiang, Xingzhu Xu, 2015 .

Silver-mediated synthesis of novel 3-CF3/CN/phosphonate-substituted pyrazoles as pyrrolomycin analogues from 3-formylchromones and diazo compounds

L. Lan, Xiaofei Zhang, Chunhao Yang, 2019, Organic Chemistry Frontiers.

Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2- c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones.

Qunyi Li, Xiaofei Zhang, Chunhao Yang, 2019, The Journal of organic chemistry.

Synthesis and activity of Combretastatin A-4 analogues: 1,2,3-thiadiazoles as potent antitumor agents.

Jian Ding, Li-ping Lin, Chunhao Yang, 2007, Bioorganic & medicinal chemistry letters.

Synthesis of substituted pyrroles using a silver-catalysed reaction between isocyanoacetates/benzyl isocyanides and chromones

Yu-Hong Yang, Chunhao Yang, Xueyu Qi, 2015 .

Pot, atom and step economic synthesis: a diversity-oriented approach to construct 2-substituted pyrrolo[2,1-f][1,2,4]triazin-4(3H)-ones

Chunhao Yang, Qian He, Yan-hong Chen, 2013 .

One Pot and Metal-Free Approach to 3-(2-Hydroxybenzoyl)-1-aza-anthraquinones

Z. Miao, Jiaqi Yuan, Xiaofei Zhang, 2019, Molecules.

Cascade Synthesis of Novel Functionalized Pyridine‐Fused Coumarins in Aqueous Medium.

Z. Miao, Chunhao Yang, Jianyang Chen, 2014 .

A Novel and Facile Method to Synthesize (R)‐ and (S)‐2‐methylpiperazine

Xihan Wu, Chunhao Yang, Guangyu Xu, 2004 .

A convenient synthesis of oxazolidinone derivatives linezolid and eperezolid from (S)-glyceraldehyde acetonide

Yi Zhou, Chunhao Yang, Guangyu Xu, 2008 .

Direct synthesis of diverse 2-aminobenzo[b]thiophenes via palladium-catalyzed carbon-sulfur bond formation using Na2S2O3 as the sulfur source.

Chunhao Yang, Qian He, Chuanwei Hou, 2014, Organic letters.

NOVEL PROCESS TO 4,4-DIALKYL-1,4-DIHYDRO-6-METHOXY-3-PHENYLCINNOLINES VIA GRIGNARD REACTION

Jian Ding, Chunhao Yang, Yuyuan Xie, 2009 .

Benzothieno[3,2-b]indole derivatives as potent selective estrogen receptor modulators.

Ming-Wei Wang, Xihan Wu, Chunhao Yang, 2005, Bioorganic & medicinal chemistry letters.

Benzothiophenes containing a piperazine side chain as selective ligands for the estrogen receptor alpha and their bioactivities in vivo.

Ming-Wei Wang, Xihan Wu, Chunhao Yang, 2005, Bioorganic & medicinal chemistry letters.

Facile Synthesis of 1,2,3,4‐Tetrahydrobenzo[b][1,8]‐naphthyridin‐2‐one via Baylis‐Hillman Adducts

Jing Xu, Chunhao Yang, Yuyuan Xie, 2009 .

Solvent-free synthesis of δ-carbolines/carbazoles from 3-nitro-2-phenylpyridines/2-nitrobiphenyl derivatives using DPPE as a reducing agent

X. L. Chen, Chunhao Yang, Qian He, 2011 .

Copper‐Assisted/Copper‐Free Synthesis of Functionalized Dibenzo[b,f]oxepins and Their Analogs via a One‐Pot Tandem Reaction

Chunhao Yang, Qian He, Yuqin Wang, 2013 .

Synthesis of 4-azachromeno〔2,3-b〕indol-11(6H)-one and its derivatives as analogues of ellipticine

Chunhao Yang, Yan-hong Chen, Yuyuan Xie, 2010 .

New Approach for the Synthesis of N‐Indolyl Ketones and Aldehydes

Chunhao Yang, Yuyuan Xie, Huasheng Ding, 2005 .

A NOVEL AND CONVENIENT METHOD FOR THE SYNTHESIS OF PHENSTATIN

Chunhao Yang, Qinggang Ji, Yuyuan Xie, 2005 .

Inhibition of hepatitis B virus replication by targeting ribonucleotide reductase M2 protein.

Weiliang Zhu, M. Wang, Zhijian Xu, 2016, Biochemical pharmacology.

Design, synthesis, and preliminary biological evaluation of novel ketone derivatives of shikimic acid

M. Jiang, Yu-mei Shen, B. Xiong, 2013 .

Discovery and bioactivity of 4-(2-arylpyrido[3',2':3,4]pyrrolo[1,2-f][1,2,4]triazin-4-yl) morpholine derivatives as novel PI3K inhibitors.

Jian Ding, Lin-jiang Tong, Linghua Meng, 2012, Bioorganic & medicinal chemistry letters.

Synthesis of isoquinolinone-based tricycles as novel poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors.

Z. Miao, Chunhao Yang, Jin-Xue He, 2014, Bioorganic & medicinal chemistry letters.

Design and synthesis of 2-(4,5,6,7-tetrahydrothienopyridin-2-yl)-benzoimidazole carboxamides as novel orally efficacious Poly(ADP-ribose)polymerase (PARP) inhibitors.

Xuxing Chen, Qian He, Qiufeng Liu, 2018, European journal of medicinal chemistry.

Catalyst-free synthesis of benzofuran-fused pyrido[4,3-d]pyrimidines from 2-(2-hydroxyaryl)acetonitrile and 4,6-dichloropyrimidine-5-carbaldehyde through domino condensation reactions

Z. Miao, Chunhao Yang, Zhizhou Yue, 2014 .

Convenient Synthesis of 6,7,12,13-Tetrahydro-5H-Cyclohepta[2,1-b:3,4-b’]diindole Derivatives Mediated by Hypervalent Iodine (III) Reagent

Xiaofei Zhang, Chunhao Yang, Lei Peng, 2019, Molecules.

Synthesis of 2-C-substituted benzothiazoles via a copper-promoted domino condensation/S-arylation/heterocyclization process.

L. Deng, M. Jiang, Chunhao Yang, 2014, Organic & biomolecular chemistry.

Ru-Catalyzed Defluorinative Alkylation or Catalyst-Free Hydroalkylation of gem-Difluoroalkenes Enabled by Visible Light.

Xiaofei Zhang, Chunhao Yang, Q. Qian, 2022, Journal of Organic Chemistry.

Synthesis of new potential chelating agents: Catechol–bisphosphonate conjugates for metal intoxication therapy

Xihan Wu, Chunhao Yang, Guangyu Xu, 2004 .

Synthesis of New Potential Chelating Agents: Catechol—Bisphosphonate Conjugates for Metal Intoxication Therapy.

Xihan Wu, Chunhao Yang, Guangyu Xu, 2004 .

Synthesis and biological evaluation of pyrazole-fused oleanolic acid derivatives as novel inhibitors of inflammatory and osteoclast differentiation.

Xiaofei Zhang, Chunhao Yang, Shijun He, 2023, Bioorganic & medicinal chemistry.

Regioselective Pd-catalyzed α-alkylation of furans using alkyl iodides

Jiaqi Yuan, Xiaofei Zhang, Chunhao Yang, 2021, RSC advances.

Aza analogues of equol: novel ligands for estrogen receptor beta.

Xu Shen, Ming-Wei Wang, Chunhao Yang, 2007, Bioorganic & medicinal chemistry.

Synthesis of Functionalized Chromeno[2,3-b]pyrrol-4(1H)-ones by Silver-Catalyzed Cascade Reactions of Chromones/Thiochromones and Isocyanoacetates.

Chunhao Yang, Xueyu Qi, H. Xiang, 2015, Organic Letters.

Synthesis of 2-alkyl-chroman-4-ones via cascade alkylation-dechlorination of 3-chlorochromones.

Lanfei Zhang, Xiaofei Zhang, Chunhao Yang, 2021, Organic & biomolecular chemistry.

Direct synthesis of diverse 2-aminobenzo[b]thiophenes via palladium-catalyzed carbon-sulfur bond formation using Na2S2O3 as the sulfur source.

Chunhao Yang, Qian He, Chuanwei Hou, 2014, Organic letters.

Rapid access to α-carbolines via a one-pot tandem reaction of α,β-unsaturated ketones with 2-nitrophenylacetonitrile and the anti-proliferative activities of the products.

Z. Miao, Xiaofei Zhang, Chunhao Yang, 2014, Organic & biomolecular chemistry.