M. Janssen

发表

Potent and selective inhibition of HIV-1 replication in vitro by a novel series of TIBO derivatives

Erik De Clercq, Jan Desmyter, Dominique Schols, 1990, Nature.

New tetrahydroimidazo[4,5,1-jk][1,4]-benzodiazepin-2(1H)-one and -thione derivatives are potent inhibitors of human immunodeficiency virus type 1 replication and are synergistic with 2',3'-dideoxynucleoside analogs

E. De Clercq, R. Pauwels, Z. Debyser, 1994, Antimicrobial Agents and Chemotherapy.

New [4,5,1-JK][1,4]benzodiazepin-2(1H)-one and -thione derivatives are potent inhibitors of human immunodeficiency virus type 1 and are synergistic with 2',3'-dideoxynucleoside analogs

R. Pauwels, E. Clercq, Z. Debyser, 1994 .

Comparative effects of the aromatase inhibitor R76713 and of its enantiomers R83839 and R83842 on steroid biosynthesis in vitro and in vivo

A. Raeymaekers, J. V. Gelder, M. Janssen, 1990, The Journal of Steroid Biochemistry and Molecular Biology.

New antihistaminic N-heterocyclic 4-piperidinamines. 3. Synthesis and antihistaminic activity of N-(4-piperidinyl)-3H-imidazo[4,5-b]pyridin-2-amines.

F. Janssens, M. Janssen, P. Janssen, 1985, Journal of medicinal chemistry.

New antihistaminic N-heterocyclic 4-piperidinamines. 2. Synthesis and antihistaminic activity of 1-[(4-fluorophenyl)methyl]-N-(4-piperidinyl)-1H-benzimidazol-2-a mines.

F. Janssens, M. Janssen, P. Janssen, 1985, Journal of medicinal chemistry.

Chemical development of astemizole‐like compounds

C. Niemegeers, F. Janssens, M. Janssen, 1986 .

New antihistaminic N-heterocyclic 4-piperidinamines. 1. Synthesis and antihistaminic activity of N-(4-piperidinyl)-1H-benzimidazol-2-amines.

F. Janssens, M. Janssen, P. Janssen, 1985, Journal of medicinal chemistry.

Levocabastine (R 50547): The prototype of a chemical series of compounds with specific H1‐antihistaminic activity

M. Janssen, J. V. Van Wauwe, M. Luyckx, 1986 .

Synthesis and screening of a new group of fungicides: 1‐(2‐phenyl‐1,3‐dioxolan‐2‐ylmethyl)‐1,2,4‐triazoles

J. Heeres, J. Gestel, M. Janssen, 1980 .

Synthesis and anti-HIV activity of 1,3,4,5-tetrahydro-2H-1,4-benzodiazepin-2-one (TBO) derivatives. truncated 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-ones (TIBO) analogues

Erik De Clercq, Koen Andries, Rudi Pauwels, 1999 .

New Antihistaminic N-Heterocyclic 4-Piperidinamines. Part 3. Synthesis and Antihistaminic Activity of N-(4-Piperidinyl)-3H-imidazo[4,5-b]pyridin-2-amines.

F. Janssens, M. Janssen, P. Janssen, 1986 .

Synthesis of 3H‐etomidate ano resolution into its enantiomers

M. Janssen, A. Knaeps, J. Heykants, 1975 .

The chemical development of selective and specific serotonin S2‐antagonists

M. Janssen, F. Awouters, L. Kennis, 1986 .

Synthesis of cisapride, a gastrointestinal stimulant derived from cis‐4‐amino‐3‐methoxypiperidine

F. Sommen, J. Leysen, C. Niemegeers, 1986 .

OXATOMIDE: THE PROTOTYPE OF A CHEMICAL SERIES OF COMPOUNDS INHIBITING BOTH THE RELEASE AND THE EFFECTS OF ALLERGIC MEDIATORS

C. Niemegeers, M. Janssen, F. Awouters, 1980 .

Lubeluzole protects sensorimotor function and reduces infarct size in a photochemical stroke model in rats.

G. Clincke, M. Janssen, M. De Ryck, 1996, The Journal of pharmacology and experimental therapeutics.