R. Volante

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Synthesis of a new generation reverse transcriptase inhibitor via the BCl3/GaCl3-induced condensation of anilines with nitriles (sugasawa reaction)

A. W. Douglas, I. Houpis, Audrey Molina, 1994 .

Preparation of enamides via palladium-catalyzed amidation of enol tosylates.

R. Volante, Cheng-yi Chen, A. Klapars, 2005, Organic letters.

A diastereospecific, non-racemic synthesis of a novel β-hydroxy-δ-lactone HMG-CoA reductase inhibitor

R. Volante, E. Corley, M. Sletzinger, 1985 .

An Efficient Chemoenzymatic Approach to (S)-γ-Fluoroleucine Ethyl Ester

Paul N. Devine, R. Volante, R. Reamer, 2005 .

A Concise Synthesis of ( S )-?-Fluoroleucine Ethyl Ester

I. Davies, F. Gosselin, R. Volante, 2006 .

AN EFFICIENT ASYMMETRIC HYDROGENATION APPROACH TO THE SYNTHESIS OF THE CRIXIVAN PIPERAZINE INTERMEDIATE

K. Rossen, R. Volante, P. Reider, 1998 .

Application of unreactive analogs of terpenoid pyrophosphates to studies of multistep biosynthesis. Demonstration that "presqualene pyrophosphate" is an essential intermediate on the path to squalene

E. Corey, R. Volante, 1976 .

Highly regioselective Friedländer annulations with unmodified ketones employing novel amine catalysts: syntheses of 2-substituted quinolines, 1,8-naphthyridines, and related heterocycles.

R. Volante, P. Reider, Roger N. Farr, 2003, The Journal of organic chemistry.

Preparation of a clinically investigated ras farnesyl transferase inhibitor

R. Volante, P. Reider, R. Reamer, 2003 .

An efficient synthesis of an alphavbeta3 antagonist.

L. Tan, M. Palucki, R. Volante, 2004, The Journal of organic chemistry.

A chemical synthesis of nicotinamide adenine dinucleotide (NAD

R. Volante, P. Reider, Woo-Baeg Choi, 1999 .

Crystallization-induced diastereoselection: asymmetric synthesis of substance P inhibitors.

K. Rossen, R. Ball, R. Volante, 2002, Chemistry.

Highly diastereoselective reaction of a chiral, non-racemic amide enolate with (S)-glycidyl tosylate. Synthesis of the orally active HIV-1 protease inhibitor L-735,524

K. Rossen, R. Volante, P. Reider, 1994 .

Chapter-12 – Total Synthesis of (–)FK506

R. Volante, 1991 .

A NOVEL SYNTHESIS OF DISUBSTITUTED UREAS USING TITANIUM(IV) ISOPROPOXIDE AND SODIUM BOROHYDRIDE

J. Armstrong, C. Wolfe, J. Lynch, 1997 .

Ullmann diaryl ether synthesis: rate acceleration by 2,2,6,6-tetramethylheptane-3,5-dione.

R. Volante, P. Reider, Z. Song, 2002, Organic letters.

Asymmetric hydrogenation of tetrahydropyrazines: Synthesis of (S)-piperazine-2-tert-butylcarboxamide, an intermediate in the preparation of the HIV protease inhibitor indinavir

K. Rossen, R. Volante, P. Reider, 1995 .

Stereocontrolled addition of propionate homoenolate equivalents to chiral α-amino aldehydes

R. Volante, I. Shinkai, A. DeCamp, 1991 .

Regioselective nucleophilic substitutions of fluorobenzene derivatives

R. Volante, P. Reider, G. Humphrey, 1996 .

Regioselective Nucleophilic Substitutions of Fluorobenzene Derivatives.

R. Volante, P. Reider, G. Humphrey, 1997 .

Practical synthesis of a neuropeptide Y antagonist via stereoselective addition to a ketene.

K. Maeda, R. Volante, Yuhei Yamamoto, 2005, The Journal of organic chemistry.

A practical enantioselective synthesis of odanacatib, a potent Cathepsin K inhibitor, via triflate displacement of an alpha-trifluoromethylbenzyl triflate.

F. Gosselin, G. Hughes, R. Volante, 2009, The Journal of organic chemistry.

Enantioselective syntheses of bicyclo[3.1.0]hexane carboxylic acid derivatives by intramolecular cyclopropanation

L. Tan, R. Volante, R. Tillyer, 2004 .

Facile synthesis of 2-bromo-3-fluorobenzonitrile: an application and study of the halodeboronation of aryl boronic acids.

Paul N. Devine, R. Volante, D. Gauthier, 2004, The Journal of organic chemistry.

Synthesis of functionalized furo[2,3-b]pyridines via the Pd-catalyzed coupling of acetylenes to iodopyridones. Preparation of a key intermediate to a new HIV protease inhibitor L-754,394

I. Houpis, Audrey Molina, J. Lynch, 1994 .

Methods for the Synthesis of 5,6,7,8-Tetrahydro-1,8-naphthyridine Fragments for αVβ3 Integrin Antagonists

L. Tan, D. Zewge, M. Palucki, 2004 .

Practical Asymmetric Synthesis of an Endothelin Receptor Antagonist

Paul N. Devine, R. Volante, P. Reider, 1999 .

Condensation of 2-methylbenzoxazole with aromatic aldehydes bearing acidic protons. A convenient coupling in the synthesis of the HIV-reverse transcriptase inhibitor L-696,229

I. Houpis, Audrey Molina, J. Lynch, 1993 .

Palladium-catalyzed amidation of enol triflates: a new synthesis of enamides.

David J. Klauber, R. Volante, Cheng-yi Chen, 2003, Organic letters.

A stereoselective synthesis of a key 1β-methylcarbapenem intermediate via a diastereoselective decarboxylation

R. Volante, P. Reider, A. Thompson, 1994 .

A Stereoselective Synthesis of a Key 1β‐Methylcarbapenem Intermediate via a Diastereoselective Decarboxylation.

R. Volante, P. Reider, A. Thompson, 1994 .

Highly Diastereoselective Alkylation of Chiral Amide Enolates: New Routes to Hydroxyethylene Dipeptide Isostere Inhibitors of HIV-1 Protease.

J. Vacca, R. Volante, R. Reamer, 1992 .

Highly diastereoselective alkylations of chiral amide enolates: new routes to hydroxyethylene dipeptide isostere inhibitors of HIV-1 protease

J. Vacca, R. Volante, R. Reamer, 1992 .

Asymmetric synthesis of α-amino acid derivatives via an electrophilic amination of chiral amide cuprates with Li t-butyl-N-tosyloxycarbamate

J. Armstrong, R. Volante, J. McWilliams, 1997 .

A practical synthesis of 5‐(chloromethyl)furo[2,3‐b]pyridine, a key intermediate for the HIV protease inhibitor, L‐754,394

K. Rossen, J. Hoffman, R. Volante, 1995 .

Synthesis of the orally active spiroindoline-based growth hormone secretagogue, MK-677

K. Rossen, I. Houpis, Audrey Molina, 1997 .

Synthesis of 5-pyridyl-2-furaldehydes via palladium-catalyzed cross-coupling with triorganozincates.

J. Armstrong, R. Volante, P. Reider, 2002, Organic letters.

An efficient enzyme-catalyzed kinetic resolution: large-scale preparation of an enantiomerically pure indole-ethyl ester derivative, a key component for the synthesis of a prostaglandin D2 receptor antagonist, an anti-allergic rhinitis drug candidate

R. Volante, E. Corley, E. Grabowski, 2005 .

Enantioselective preparation of ring-fused 1-fluorocyclopropane-1-carboxylate derivatives: en route to mGluR 2 receptor agonist MGS0028.

R. Volante, Z. Song, D. Tschaen, 2004, Organic letters.

Highly Regioselective Friedlaender Annulations with Unmodified Ketones Employing Novel Amine Catalysts: Syntheses of 2-Substituted Quinolines, 1,8-Naphthyridines, and Related Heterocycles.

R. Volante, P. Reider, Roger N. Farr, 2003 .

Mechanistic studies on the diastereoselective halohydroxylation of γ-δ unsaturated carboxamides

K. Rossen, R. Volante, P. Reider, 1996 .

Stereoelectronic effects in the DIBAL reduction of aryl-1,2-ethanediol benzylidene acetals

J. Armstrong, R. Volante, D. Gauthier, 2001 .

A highly enantioselective asymmetric hydrogenation route to β-(2R,3S)-methyltryptophan

R. Volante, P. Reider, D. Askin, 1998 .

Ni-catalyzed nucleophilic conjugate additions of Grignard and organozincate reagents to substituted 4-vinylpyridines. General synthesis of phosphodiesterase IV inhibitors

I. Houpis, Audrey Molina, R. Volante, 1998 .

An Efficient Procedure for the Synthesis of p-Anisidine Phenylglyoxal Imine from Acetophenone

R. Volante, S. Mills, Richard A Desmond, 1989 .

A New Planar Chiral Bisphosphine Ligand for Asymmetric Catalysis: Highly Enantioselective Hydrogenations under Mild Conditions.

K. Rossen, R. Volante, P. Reider, 1997 .

A New Planar Chiral Bisphosphine Ligand for Asymmetric Catalysis: Highly Enantioselective Hydrogenations under Mild Conditions

K. Rossen, R. Volante, P. Reider, 1997 .

An efficient synthesis of 4-benzoyloxyazetidinone: an important carbapenem intermediate

R. Volante, D. Tschaen, J. Lynch, 1988 .

Mechanism of an acid chloride-imine reaction by low-temperature FT-IR: .beta.-lactam formation occurs exclusively through a ketene intermediate

R. Volante, D. Tschaen, J. Lynch, 1989 .

Practical synthesis of α-amino acids using cis-aminoindanol derived hippuric acid amide as a glycine enolate equivalent

R. Volante, P. Reider, Woo-Baeg Choi, 1998 .

EFFICIENT SYNTHESIS OF N-ARYLPIPERAZINONES VIA A SELECTIVE INTRAMOLECULAR MITSUNOBU CYCLODEHYDRATION

R. Volante, P. Reider, D. Askin, 1998 .

Efficient and Practical Synthesis of a Potent Anti-MRSA β-Methylcarbapenem Containing a Releasable Side Chain.

K. Rossen, Ross A. Miller, R. Volante, 2000 .

Efficient and Practical Synthesis of a Potent Anti-MRSA β-Methylcarbapenem Containing a Releasable Side Chain

K. Rossen, Ross A. Miller, R. Volante, 1999 .

Cyclic imidate salts in acyclic stereochemistry: Diastereoselective syn-epoxidation of 2-alkyl-4-enamides to epoxyamides

K. Rossen, R. Volante, P. Reider, 1996 .

AN UNUSUAL STEREOSELECTIVE DECARBOXYLATION : A KEY REACTION TO AN IMPORTANT INTERMEDIATE FOR CARBAPENEM ANTIBIOTICS

D. Liotta, R. Volante, P. Reider, 1995 .

A Facially-Selective Protonation Controls the Stereochemistry of a Key Intermediate in the Synthesis of 1.beta.-Methylcarbapenems

D. Liotta, R. Volante, P. Reider, 1994 .

Photooxidative Cleavage of a Furanazetidinone Carbon-Carbon Bond: A Synthesis of 4-Acetoxyazetidinone.

R. Volante, R. Reamer, D. Tschaen, 1994 .

An efficient asymmetric synthesis of (R)-3-amino-2,3,4,5-tetrahydro-1H-[1]benzazepin-2-one

J. Armstrong, R. Volante, D. Askin, 1994 .

A Stereoselective Synthesis of a 2-Functionalized-methyl-1β-methylcarbapenem Key Intermediate via Decarboxylation.

R. Volante, P. Reider, R. Reamer, 1998 .

Nickel catalyzed addition of organozincates to optically pure vinylic sulfoxides. Synthesis of the phosphodiesterase IV inhibitor L-765,527 (CDP-840)

I. Houpis, Audrey Molina, R. Volante, 1997 .

Practical and efficient synthesis of N-halo compounds

Hua Zhou, R. Volante, D. Gauthier, 2005 .

Synthesis of a muscarinic receptor antagonist via a diastereoselective Michael reaction, selective deoxyfluorination and aromatic metal-halogen exchange reaction.

J. Song, D. Zewge, I. Houpis, 2001, The Journal of organic chemistry.

Practical synthesis of a potent indolocarbazole-based, DNA topoisomerase inhibitor

K. Rossen, T. Nemoto, A. Kamatani, 2001 .

Unprecedented catalytic asymmetric reduction of N-H imines.

F. Gosselin, R. Volante, Cheng-yi Chen, 2005, Organic letters.

A stereoselective aldol reaction via diisopinocampheyl boron-enolate in preparation of chromane carboxylate with quaternary carbon

D. Zewge, R. Volante, P. Reider, 2003 .

Synthesis of an HMG-COA reductase inhibitor; A diastereoselective aldol approach

R. Volante, J. Lynch, I. Shinkai, 1987 .

[2.2]PHANEPHOS-Ruthenium(II) complexes: Highly active asymmetric catalysts for the hydrogenation of β-ketoesters

K. Rossen, R. Volante, P. Reider, 1998 .

Kinetic Resolution of rac-4,12-Dibromo[2.2]paracyclophane in a Palladium [2.2]PHANEPHOS Catalyzed Amination

K. Rossen, R. Volante, P. Pye, 1997 .

Diastereoselective syn-epoxidation of 2-alkyl-4-enamides to epoxyamides: Synthesis of the Merck HIV-1 protease inhibitor epoxide intermediate

K. Rossen, R. Volante, P. Reider, 1995 .

Stereocontrolled addition of chiral, non-racemic amide homoenolates to t-Boc-(S)-phenylalaninal

J. Armstrong, R. Volante, F. W. Hartner, 1992 .

Approaches to installing a N-gem-dimethylmethylene-2-oxazolyl group and application to the synthesis of a second generation HIV protease inhibitor

J. Armstrong, Ross A. Miller, F. Fleitz, 2005 .

Diastereoselective Reductive Amination of Aryl Trifluoromethyl Ketones and α‐Amino Esters

Paul N. Devine, J. R. Naber, G. Hughes, 2007 .

Synthesis of benzofuroquinolizine for α-2 adrenoceptor antagonist MK-912: an O-analogue of the Pictet-Spengler reaction

K. Rossen, R. Volante, P. Reider, 1999 .

Alkylation of chiral prolinol propionamide enolates with epoxides: Complete reversal of predicted facial selectivity

R. Volante, R. Reamer, D. Askin, 1988 .

Towards the synthesis of HIV-protease inhibitors. Synthesis optically pure 3-carboxyl-decahydroisoquinolines.

I. Houpis, Audrey Molina, R. Volante, 1993 .

Tandem asymmetric transformations: An asymmetric 1,2-migration from a higher order zincate coupled with a stereoselective homoaldol reaction

J. Armstrong, R. Volante, P. Reider, 1996 .

Total synthesis of a second generation HIV protease inhibitor

J. Armstrong, F. Fleitz, R. Volante, 2003 .

The enantioselective synthesis of LTD4 antagonist L-708,738

D. Sidler, R. Volante, M. Bhupathy, 1997 .

Oxazolidine Ring Opening and Isomerization to (E)-Imines. Asymmetric Synthesis of Aryl-α-fluoroalkyl Amino Alcohols.

F. Gosselin, R. Volante, Cheng-yi Chen, 2004 .

Oxazolidine ring opening and isomerization to (E)-imines. Asymmetric synthesis of aryl-alpha-fluoroalkyl amino alcohols.

F. Gosselin, R. Volante, Cheng-yi Chen, 2004, Organic letters.

Asymmetric synthesis of (2S,3S)-3-hydroxy-2-phenylpiperidine via ring expansion

R. Volante, P. Reider, D. Askin, 2001 .

Practical synthesis of a potent hepatitis C virus RNA replication inhibitor.

R. Volante, E. Grabowski, Feng Xu, 2004, The Journal of organic chemistry.

A Practical Synthesis of the 5‐Chloromethyl‐furo(2,3‐b)pyridine Pharmacophore.

I. Houpis, Audrey Molina, R. Volante, 1995 .

Efficient degradation of FK-506 to a versatile synthetic intermediate

R. Volante, R. Reamer, D. Askin, 1990 .

Diastereospecific, non-racemic synthesis of the C.20–C.34 segment of the novel immunosuppressant FK-506

R. Volante, R. Reamer, S. Mills, 1988 .

A convergent asymmetric synthesis of a growth hormone secretagogue

J. Armstrong, J. Lynch, R. Volante, 2003 .

An efficient asymmetric synthesis of the mercaptopyrrolidine side chain of an important β-methyl carbapenem antibiotic

J. Armstrong, J. Lynch, R. Volante, 1997 .

ASYMMETRIC SYNTHESIS OF CDP840 BY JACOBSEN EPOXIDATION. AN UNUSUAL SYN SELECTIVE REDUCTION OF AN EPOXIDE

R. Ball, R. Volante, Woo-Baeg Choi, 1997 .

A regioselective approach to 5-substituted-3-amino-1,2,4-triazines.

Paul N. Devine, R. Volante, R. Reamer, 2003, Organic letters.

Total synthesis of immunosuppressant (-)-FK-506

R. Volante, R. Reamer, S. Mills, 1989 .

Total Synthesis of the Immunosuppressant (‐)‐FK‐506.

R. Volante, R. Reamer, S. Mills, 1989 .

A mechanistic study of the FK-506 tricarbonyl system rearrangement: Synthesis of C.9 Labeled FK-506

R. Volante, R. Reamer, D. Askin, 1989 .

Practical asymmetric synthesis of a selective endothelin A receptor (ETA) antagonist.

H. Satō, T. Nemoto, R. Volante, 2001, Organic Letters.

The enantioselective synthesis of LTD 4 antagonist L-708,738

D. Sidler, R. Volante, J. Bergan, 1997 .

Michael Additions of 3,3‐Dimethylacrylamides and ‐amines: Synthesis of the Growth Hormone Secretagogue L‐692,585.

K. Rossen, R. Volante, P. Reider, 1995 .

Kilogram Scale Synthesis of the Pyrazinone Acetic Acid Core of an Orally Efficacious Thrombin Inhibitor

J. Armstrong, F. Fleitz, R. Volante, 2000 .

Highly Diastereoselective Reaction of a Chiral, Non‐Racemic Amide Enolate with (S)‐Glycidyl Tosylate. Synthesis of the Orally Active HIV‐ 1 Protease Inhibitor L‐735,524

K. Rossen, R. Volante, P. Reider, 1994 .

Amination of aryl halides using copper catalysis

D. Zewge, I. Houpis, R. Volante, 2001 .

Palladium-Catalyzed Synthesis of Aryl Sulfides from Aryl Triflates

R. Volante, J. McWilliams, N. Zheng, 1998 .

Synthesis of a New Generation Reverse Transcriptase Inhibitor via the BCl3/GaCl3‐Induced Condensation of Anilines with Nitriles (Sugasawa Reaction).

A. W. Douglas, I. Houpis, Audrey Molina, 1995 .

A Highly Selective Method for the Synthesis of E‐α‐Methyl‐α,β‐Unsaturated Aldehydes.

R. Volante, S. Mills, Richard A Desmond, 1989 .

An efficient asymmetric synthesis of an estrogen receptor modulator by sulfoxide-directed borane reduction.

D. Zewge, D. Mathre, R. Volante, 2004, Proceedings of the National Academy of Sciences of the United States of America.