E. Cauchon

发表

Discovery of MK-1439, an orally bioavailable non-nucleoside reverse transcriptase inhibitor potent against a wide range of resistant mutant HIV viruses.

Sébastien Gagné, Eric Langlois, Jean-François Truchon, 2014, Bioorganic & medicinal chemistry letters.

The discovery and synthesis of potent zwitterionic inhibitors of renin.

J. Falgueyret, M. Percival, S. Gagné, 2011, Bioorganic & medicinal chemistry letters.

A High-Throughput Continuous Assay for Screening and Characterization of Inhibitors of HIV Reverse-Transcriptase DNA Polymerase Activity

J. Falgueyret, R. Melnyk, E. Cauchon, 2011, Journal of biomolecular screening.

In Vitro Characterization of MK-1439, a Novel HIV-1 Nonnucleoside Reverse Transcriptase Inhibitor

Jason Burch, Yves Ducharme, Louis-Charles Campeau, 2013, Antimicrobial Agents and Chemotherapy.

Inhibition of human dermal fibroblast proliferation by removal of dermatan sulfate.

E. Denholm, E. Cauchon, P. Silver, 2000, European journal of pharmacology.

3,4-Diarylpiperidines as potent renin inhibitors.

J. Falgueyret, Yongxin Han, E. Cauchon, 2012, Bioorganic & medicinal chemistry letters.

Impact of Primer-induced Conformational Dynamics of HIV-1 Reverse Transcriptase on Polymerase Translocation and Inhibition*

J. Falgueyret, G. Beilhartz, R. Melnyk, 2011, The Journal of Biological Chemistry.

Design and synthesis of potent, isoxazole-containing renin inhibitors.

J. Falgueyret, M. Percival, Yongxin Han, 2012, Bioorganic & medicinal chemistry letters.

Renin inhibitors for the treatment of hypertension: design and optimization of a novel series of spirocyclic piperidines.

J. Falgueyret, Yongxin Han, S. Gagné, 2011, Bioorganic & medicinal chemistry letters.

Renin inhibitors for the treatment of hypertension: design and optimization of a novel series of tertiary alcohol-bearing piperidines.

J. Falgueyret, M. Percival, Yongxin Han, 2011, Bioorganic & medicinal chemistry letters.

Renin inhibitors for the treatment of hypertension: design and optimization of a novel series of pyridone-substituted piperidines.

J. Falgueyret, M. Percival, Yongxin Han, 2011, Bioorganic & medicinal chemistry letters.

Identification of an indole series of prostaglandin D2 receptor antagonists.

R. Young, D. Denis, C. Brideau, 2006, Bioorganic & medicinal chemistry letters.

Development of a homogeneous immunoassay for the detection of angiotensin I in plasma using AlphaLISA acceptor beads technology.

J. Falgueyret, M. Percival, Steve Rowland, 2009, Analytical biochemistry.

Molecular pharmacology of the human prostaglandin D2 receptor, CRTH2

G. O'neill, D. Nicholson, K. Metters, 2002, British journal of pharmacology.

An Automated Multistep High-Throughput Screening Assay for the Identification of Lead Inhibitors of the Inducible Enzyme mPGES-1

C. Brideau, D. Éthier, J. Guay, 2005, Journal of biomolecular screening.