E. Merkul

发表

Discovery of novel 7-azaindoles as PDK1 inhibitors.

Dirk Finsinger, Margarita Wucherer-Plietker, Hans-Peter Buchstaller, 2016, Bioorganic & medicinal chemistry letters.

Concise syntheses of meridianins by carbonylative alkynylation and a four-component pyrimidine synthesis.

F. Rominger, E. Merkul, T. Müller, 2005, Angewandte Chemie.

Three-component synthesis of ynediones by a glyoxylation/Stephens-Castro coupling sequence.

F. Rominger, E. Merkul, T. Müller, 2011, Angewandte Chemie.

Consecutive three-component synthesis of ynones by decarbonylative Sonogashira coupling.

E. Merkul, T. Müller, T. Oeser, 2009, Chemistry.

A Novel Platinum(II)-Based Bifunctional ADC Linker Benchmarked Using 89Zr-Desferal and Auristatin F-Conjugated Trastuzumab.

G. V. van Dongen, G. Somsen, E. Merkul, 2017, Cancer research.

First platinum(II)-based metal-organic linker technology (Lx®) for a plug-and-play development of antibody-drug conjugates (ADCs)

G. V. van Dongen, E. Merkul, I. Aydin, 2019, Expert opinion on drug delivery.

In Vivo Characterization of Platinum(II)-Based Linker Technology for the Development of Antibody–Drug Conjugates: Taking Advantage of Dual Labeling with 195mPt and 89Zr

G. V. van Dongen, E. Merkul, J. Muns, 2018, The Journal of Nuclear Medicine.

Catalytic syntheses of N-heterocyclic ynones and ynediones by in situ activation of carboxylic acids with oxalyl chloride.

E. Merkul, T. Müller, Christina Boersch, 2011, Angewandte Chemie.

A new consecutive three-component oxazole synthesis by an amidation-coupling-cycloisomerization (ACCI) sequence.

E. Merkul, T. Müller, 2006, Chemical communications.

Rapid synthesis of bis(hetero)aryls by one-pot Masuda borylation-Suzuki coupling sequence and its application to concise total syntheses of meridianins A and G.

E. Schäfer, E. Merkul, T. Müller, 2011, Organic & biomolecular chemistry.

Synthesis of Pd Complexes Containing Tailed NHC Ligands and Their Use in a Semicontinuous Membrane-Assisted Suzuki Cross-Coupling Process

B. Maes, L. Eykens, E. Merkul, 2018, Organic Process Research & Development.

One‐Pot Synthesis of Diazine‐Bridged Bisindoles and Concise Synthesis of the Marine Alkaloid Hyrtinadine A

E. Merkul, T. Müller, Boris O. A. Tasch, 2011 .

Rapid preparation of triazolyl substituted NH-heterocyclic kinase inhibitors via one-pot Sonogashira coupling-TMS-deprotection-CuAAC sequence.

D. Dorsch, U. Grädler, E. Merkul, 2011, Organic & biomolecular chemistry.

One-pot three-component synthesis of 3-halofurans and 3-chloro-4-iodofurans

E. Merkul, T. Müller, Alexei S. Karpov, 2006 .

A novel one-pot three-component synthesis of 3-halofurans and sequential Suzuki coupling.

E. Merkul, T. Müller, Alexei S. Karpov, 2005, Chemical communications.

Consecutive One-Pot Sonogashira–Glaser Coupling Sequence – Direct Preparation of Symmetrical Diynes by Sequential Pd/Cu Catalysis†

E. Merkul, T. Müller, Dominik Urselmann, 2011 .

One-pot four-component synthesis of pyrimidyl and pyrazolyl substituted azulenes by glyoxylation–decarbonylative alkynylation–cyclocondensation sequences

E. Merkul, T. Müller, Charlotte F. Gers, 2011, Beilstein journal of organic chemistry.

Three-component synthesis of N-Boc-4-iodopyrroles and sequential one-pot alkynylation.

W. Frank, E. Merkul, T. Müller, 2009, Organic letters.

Catalytic one-pot synthesis of 4-(hetero)aryl substituted 5-(2-oxoethyl) oxazol-2(3H)-ones by coupling–isomerization–elimination (CIE) sequence

W. Frank, E. Merkul, T. Müller, 2016 .

Consecutive Three-Component Synthesis of 3-(Hetero)Aryl-1H-pyrazoles with Propynal Diethylacetal as a Three-Carbon Building Block

E. Merkul, T. Müller, Lucilla Levi, 2011, Molecules.

Catalysis and Multi-Component Reactions

O. V. Koryakova, M. Khorasani, D. Dorsch, 2011 .

One‐Pot Synthesis of Camalexins and 3,3′‐Biindoles by the Masuda Borylation–Suzuki Arylation (MBSA) Sequence

E. Merkul, T. Müller, Dragutin Antovic, 2013 .

One-Pot Synthesis of Camalexins and 3,3′-Biindoles by the Masuda Borylation—Suzuki Arylation (MBSA) Sequence.

T. Mueller, E. Merkul, Dragutin Antovic, 2013 .

A successful search for new, efficient, and silver-free manufacturing processes for key platinum(ii) intermediates applied in antibody–drug conjugate (ADC) production

G. V. van Dongen, E. Merkul, I. Aydin, 2020 .

Potential of Homogeneous Pd Catalyst Separation by Ceramic Membranes. Application to Downstream and Continuous Flow Processes

B. Maes, E. Merkul, S. Sergeyev, 2016 .

An Efficient Conjugation Approach for Coupling Drugs to Native Antibodies via the PtII Linker Lx for Improved Manufacturability of Antibody–Drug Conjugates

J. Reedijk, G. Dongen, E. Merkul, 2020, Angewandte Chemie.