D. Tape

发表

4-Phenyl-7-azaindoles as potent, selective and bioavailable IKK2 inhibitors demonstrating good in vivo efficacy.

P. Bamborough, W. Rumsey, C. Chung, 2012, Bioorganic & medicinal chemistry letters.

Strategies for the synthesis of spiropiperidines - a review of the last 10 years.

D. Tape, P. Clarke, Samuel D Griggs, 2018, Organic & biomolecular chemistry.

4-Phenyl-7-azaindoles as potent and selective IKK2 inhibitors.

P. Bamborough, J. Liddle, M. Morse, 2009, Bioorganic & medicinal chemistry letters.

Dissociated nonsteroidal glucocorticoid receptor modulators; discovery of the agonist trigger in a tetrahydronaphthalene-benzoxazine series.

H. T. Jones, I. McLay, I. Uings, 2006, Journal of medicinal chemistry.

Identification and Optimization of a Ligand-Efficient Benzoazepinone Bromodomain and Extra Terminal (BET) Family Acetyl-Lysine Mimetic into the Oral Candidate Quality Molecule I-BET432.

Darren L. Poole, I. Wall, P. Bamborough, 2022, Journal of medicinal chemistry.

Regioselective Synthesis of 3-Aminoimidazo[1,2-a]pyrimidines with Triflic Anhydride

E. Talbot, D. Tape, Sabri Ukuser, 2017, Synthesis.

Synthesis of highly substituted 2-spiropiperidines.

D. Tape, P. Clarke, Samuel D Griggs, 2018, Organic & biomolecular chemistry.

A Two-Step Synthesis of 2-Spiropiperidines.

D. Tape, P. Clarke, Samuel D Griggs, 2017, Chemistry.

Novel syntheses of the amino-1,2,4-triazine GW356194: identification of a synthesis amenable to scale up

D. Tape, M. Schilling, A. Burton, 2003 .