A. Messere

发表

Computer-Aided Identification and Lead Optimization of Dual Murine Double Minute 2 and 4 Binders: Structure-Activity Relationship Studies and Pharmacological Activity.

Ettore Novellino, Luciana Marinelli, Sandro Cosconati, 2017, Journal of medicinal chemistry.

Recent progress in chemically modified siRNAs.

M. Gaglione, A. Messere, M Gaglione, 2010, Mini reviews in medicinal chemistry.

Alternate PNA‐DNA chimeras (PNA‐DNA)n: Synthesis, binding properties and biological activity

R. Gambari, E. Fabbri, M. Borgatti, 2007, Biopolymers.

A novel synthetic strategy for monosubstituted cyclodextrin derivatives.

M. Gaglione, C. Isernia, G. Di Fabio, 2012, Chemical communications.

Synthesis, biophysical characterization and anti-HIV activity of d(TG3AG) Quadruplexes bearing hydrophobic tails at the 5'-end.

J. Balzarini, D. Milardi, C. La Rosa, 2014, Bioorganic & medicinal chemistry.

Cationic nucleopeptides as novel non-covalent carriers for the delivery of peptide nucleic acid (PNA) and RNA oligomers.

A. Chambery, E. Novellino, C. Ieranò, 2018, Bioorganic & medicinal chemistry.

Solid-phase synthesis of cyclic PNA and PNA-DNA chimeras.

G. Di Fabio, B. di Blasio, J. D’Onofrio, 2006, Organic letters.

Studies toward the synthesis of pinolidoxin, a phytotoxic nonenolide from the fungus Ascochyta pinodes. Determination of the configuration at the C-7, C-8, and C-9 chiral centers and stereoselective synthesis of the C(6)-C(18) fragment.

G. Piccialli, A. Evidente, L. de Napoli, 2000, The Journal of organic chemistry.

A Facile Solid‐Phase Strategy for the Synthesis of Oligonucleotide‐Tetraphenylporphyrin Conjugates

G. Piccialli, G. Morelli, D. Tesauro, 2000 .

Solid phase synthesis of DNA-3′-PNA chimeras by using Bhoc/Fmoc PNA monomers

G. Piccialli, M. Saviano, C. Pedone, 2001 .

Reaction of 3′,5′-di-O-acetyl-2′-deoxyinosine with the chlorinating agent PPh3–CCl4: synthesis of the 6-chloroderivative and of a new base linked dimer, useful intermediate to 15N-1-labelled 2′-deoxyinosine

G. Piccialli, D. Montesarchio, A. Messere, 1994 .

Tailoring the Structure of Cell Penetrating DNA and RNA Binding Nucleopeptides

A. Chambery, L. Portella, C. Ieranò, 2022, International journal of molecular sciences.

A new solid-phase synthesis of oligonucleotides 3'-conjugated with peptides.

G. Piccialli, E. Benedetti, E. Bucci, 1999, Bioorganic & medicinal chemistry.

Improved Synthesis of 2′,3′-Dideoxycytidine (d2C) and Its Correlated Nucleoside Analogues

G. Piccialli, D. Montesarchio, A. Messere, 1993 .

Allelopathic potential of alkylphenols from Dactylis glomerata subsp. hispanica (Roth) Nyman

M. Scognamiglio, V. Fiumano, A. Fiorentino, 2012 .

Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication.

E. Novellino, P. Grieco, S. Di Maro, 2019, Organic letters.

A new ferrocenemethyl-thymidine nucleoside: Synthesis, incorporation into oligonucleotides and optical spectroscopic studies on the resulting single strand, duplex and triplex structures

G. Piccialli, A. Romanelli, E. Bucci, 1999 .

Cyclic Uridine Diphosphate Glucose: A New Pyrimidine Analog of Cyclic ADP Ribose

G. Piccialli, G. Di Fabio, D. Montesarchio, 2003, Nucleosides, nucleotides & nucleic acids.

Synthetic studies on the glycosylation of the base residues of inosine and uridine

G. Piccialli, D. Montesarchio, A. Messere, 1999 .

1-Substituted 2′-deoxyinosine analogues

G. Piccialli, D. Montesarchio, A. Messere, 1997 .

Synthesis of [1-15N]-Labeled 2'-Deoxyinosine and 2'-Deoxyadenosine

G. Piccialli, D. Montesarchio, A. Messere, 1995 .

In-water reactivity of nucleosides and nucleotides: one-step preparation and biological evaluation of novel ferrocenyl-derivatives

G. Piccialli, M. Champdoré, R. Loddo, 2004 .

Antiproliferative activity of Pt(II) and Pd(II) phosphine complexes with thymine and thymidine.

R. Gambari, E. Fabbri, M. Borgatti, 2007, Journal of inorganic biochemistry.

Nitration of Cinnamic Acids Using Cerium (IV) Ammonium Nitrate Immobilized on Silica

A. Fiorentino, F. Temussi, B. di Blasio, 2004 .

Synthesis of platinum(II) complexes of thymidine and 1-methylthymine (1-MeThy); crystal structure of cis-[PtCl(1-MeThy)(PPh3)2]

G. Piccialli, M. Saviano, A. Romanelli, 1999 .

A new glucosylated cinnamoyl glycerol from aerial parts of Phleum subulatum

M. Scognamiglio, A. Fiorentino, B. D’Abrosca, 2012 .

Synthesis and Biological Properties of Caffeic Acid-PNA Dimers Containing Guanine

L. Russo, M. Gaglione, A. Fiorentino, 2013, Molecules.

Synthesis and Biological Properties of Caffeic Acid-PNA Dimers

L. Russo, M. Gaglione, A. Fiorentino, 2013 .

Automated solid phase synthesis of cyclic oligonucleotides: a further improvement.

G. Piccialli, L. Mayol, D. Montesarchio, 1995, Bioorganic & Medicinal Chemistry.

Facile preparation of cyclic oligoribonucleotides

G. Piccialli, L. Mayol, A. Messere, 1993 .

SOLID-PHASE SYNTHESIS OF CYCLIC OLIGODEOXYRIBONUCLEOTIDES : INTERMOLECULARVERSUS INTRAMOLECULAR COUPLING

G. Piccialli, D. Montesarchio, A. Messere, 1991 .

A Facile Solid‐Phase Synthesis of Oligonucleotides Containing a 3′−3′ Phosphodiester Bond for Alternate Strand Triple‐Helix Formation

G. Piccialli, D. Montesarchio, A. Messere, 1998 .

PEG-Supported Synthesis of Cyclic Oligodeoxyribonucleotides

G. Piccialli, D. Montesarchio, A. Messere, 1993 .

Synthesis of 4-Substituted Pyrimidine 2′,3′-Dideoxynucleosides

G. Piccialli, D. Montesarchio, A. Messere, 1991 .

Oligonucleotides containing a lysine residue as 3'-3' junction for alternate strand triple helix formation.

G. Piccialli, G. Barone, C. Giancola, 2001, Bioorganic & medicinal chemistry.

Synthesis and Triple Helix Formation by Alternate Strand Recognition of Oligonucleotides Containing 3‘-3‘ Phosphodiester Bonds

A. Pepe, D. Montesarchio, A. Messere, 1997 .

Synthesis and characterization of new 3′-3′ linked oligodeoxyribonucleotides for alternate strand triple helix formation

G. Piccialli, D. Musumeci, D. Montesarchio, 1999 .

New 3′-3′ Linkers for Alternate Strand Triplex Forming Oligonucleotides

G. Piccialli, D. Musumeci, D. Montesarchio, 1999 .

Studies on Alternate Strand Triple Helix Formation by Oligodeoxyribonucleotides Containing A 3′-3′ Phosphodiester Bond

G. Piccialli, L. Mayol, A. Pepe, 1998 .

Physico-chemical studies of a DNA triplex containing a new ferrocenemethyl-thymidine residue in the third strand.

G. Piccialli, G. Barone, C. Giancola, 2003, Biophysical chemistry.

6-Chloroxanthosine, a Useful Intermediate for the Efficient Syntheses of [6-15N]-Isoguanosine, Isoinosine and Other Purine Nucleoside Analogues

G. Piccialli, D. Montesarchio, A. Messere, 1997 .

Synthesis and Gene Silencing Properties of siRNAs Containing Terminal Amide Linkages

E. Novellino, S. Cosconati, M. Gaglione, 2014, BioMed research international.

PNA-based artificial nucleases as antisense and anti-miRNA oligonucleotide agents.

A. Chambery, A. Romanelli, M. Gaglione, 2011, Molecular bioSystems.

RNA Interference in Mammalia Cells by RNA-3’-PNA Chimeras

B. di Blasio, A. Messere, N. Potenza, 2008, International journal of molecular sciences.

Synthesis of 2′,3′-dideoxy-2′,3′-didehydronucleoside analogues as potential anti HIV agents

G. Piccialli, D. Montesarchio, A. Messere, 1992 .

6-Chloroxanthosine (I), a Useful Intermediate for Efficient Syntheses of (6-15N)-Isoguanosine (IV), Isoinosine (VII), and Other Purine Nucleoside Analogues (IX).

G. Piccialli, D. Montesarchio, A. Messere, 2010 .

A new synthesis of oxanosine and 2′-deoxyoxanosine

G. Piccialli, D. Montesarchio, A. Messere, 1998 .

Switchable Protecting Strategy for Solid Phase Synthesis of DNA and RNA Interacting Nucleopeptides.

A. Chambery, E. Novellino, S. Lama, 2016, The Journal of organic chemistry.

Long non-coding RNA containing ultraconserved genomic region 8 promotes bladder cancer tumorigenesis

Wei Zhang, E. Novellino, M. Fabbri, 2016, Oncotarget.

Structure-Activity Relationships and Biological Characterization of a Novel, Potent, and Serum Stable C-X-C Chemokine Receptor Type 4 (CXCR4) Antagonist.

E. Novellino, L. Portella, S. Scala, 2017, Journal of medicinal chemistry.

CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists.

V. Hruby, A. Mollica, M. Cai, 2022, Journal of medicinal chemistry.

New nucleoside based solid supports. Synthesis of 5′,3′-derivatized thymidine analogues

G. Piccialli, M. Champdoré, D. Montesarchio, 2001 .

Hairpin oligonucleotides forming G-quadruplexes: new aptamers with anti-HIV activity.

J. Balzarini, S. Noppen, S. Liekens, 2015, European journal of medicinal chemistry.

Disulfide bond replacement with 1,4- and 1,5-disubstituted [1,2,3]-triazole on C-X-C chemokine receptor type 4 (CXCR4) peptide ligands: small changes that make big differences.

E. Novellino, C. Ieranò, S. Scala, 2020, Chemistry.

Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO).

E. Novellino, F. Da Settimo, S. Taliani, 2017, Journal of medicinal chemistry.

Inhibition of net nitrification activity in a Mediterranean woodland: possible role of chemicals produced by Arbutus unedo

F. Miglietta, S. Castaldi, A. Fiorentino, 2009, Plant and Soil.

Ultrasound-assisted Peptide Nucleic Acids synthesis (US-PNAS)

A. Chambery, F. Merlino, S. Cosconati, 2023, Ultrasonics sonochemistry.

Dual MET and SMO Negative Modulators Overcome Resistance to EGFR Inhibitors in Human Nonsmall Cell Lung Cancer.

E. Novellino, S. Taliani, M. Trincavelli, 2017, Journal of medicinal chemistry.

An alternative strategy to synthesize PNA and DNA magnetic conjugates forming nanoparticle assembly based on PNA/DNA duplexes.

M. Gaglione, D. Musumeci, A. Messere, 2010, Molecular bioSystems.

Lead Discovery of SARS-CoV-2 Main Protease Inhibitors through Covalent Docking-Based Virtual Screening

T. Schirmeister, S. Cosconati, A. Messere, 2021, J. Chem. Inf. Model..

Chemical modifications in the seed region of miRNAs 221/222 increase the silencing performances in gastrointestinal stromal tumor cells.

E. Novellino, P. Grieco, A. Cimmino, 2016, European journal of medicinal chemistry.

Fully automated synthesis of peptide-oligonucleotide conjugates

G. Piccialli, C. Pedone, E. Benedetti, 2002 .

Targeting duplex DNA with DNA-PNA chimeras? Physico-chemical characterization of a triplex DNA-PNA/DNA/DNA.

G. Piccialli, G. Barone, C. Giancola, 2004, Biopolymers.

Glycosylations of Inosine and Uridine Nucleoside Bases and Synthesis of the New 1-(β-D-Glucopyranosyl)-Inosine-5′, 6″-diphosphate

G. Piccialli, D. Montesarchio, A. Messere, 2000, Nucleosides, nucleotides & nucleic acids.

Tuning RNA Interference by Enhancing siRNA/PAZ Recognition.

E. Novellino, S. Cosconati, M. Gaglione, 2013, ACS medicinal chemistry letters.

Long non-coding RNA containing ultraconserved genomic region 8 promotes bladder cancer tumorigenesis.

Wei Zhang, E. Novellino, M. Fabbri, 2016, Oncotarget.

Solid-Phase Synthesis of Glyco-Oligonucleotide Conjugates

G. Piccialli, M. Adinolfi, G. Di Fabio, 2001 .

Investigation of the Stereochemical-Dependent DNA and RNA Binding of Arginine-Based Nucleopeptides

Ettore Novellino, Stefano Tomassi, Francisco Franco Montalban, 2019, Symmetry.

Current Methods in Synthesis of Cyclic Oligonucleotides and Analogues

M. Gaglione, A. Messere, G. D. Fabio, 2012 .

PNA-DNA Chimeras Forming Quadruplex Structures

G. Piccialli, L. Mayol, A. Randazzo, 2003, Nucleosides, nucleotides & nucleic acids.

Polyphenols from the hydroalcoholic extract of Arbutus unedo living in a monospecific Mediterranean woodland

S. Castaldi, A. Fiorentino, B. D’Abrosca, 2007 .