S. Demkowicz

发表

Development of Sulfamoylated 4-(1-Phenyl-1H-1,2,3-triazol-4-yl)phenol Derivatives as Potent Steroid Sulfatase Inhibitors for Efficient Treatment of Breast Cancer

C. Supuran, Karol Biernacki, Olga Ciupak, 2022, Journal of medicinal chemistry.

Synthesis of bicoumarin thiophosphate derivatives as steroid sulfatase inhibitors.

B. Gielniewski, Mateusz Daśko, J. Rachon, 2015, European journal of medicinal chemistry.

Synthesis and steroid sulfatase inhibitory activities of N-alkanoyl tyramine phosphates and thiophosphates†

A. Wołoś, Mateusz Daśko, J. Rachon, 2015 .

Synthesis and biological evaluation of N‐acylated tyramine sulfamates containing C–F bonds as steroid sulfatase inhibitors

Mateusz Daśko, J. Rachon, K. Kubiński, 2017, Chemical biology & drug design.

An efficient and convenient synthesis of unsymmetrical disulfides from thioacetates

Slawomir Lach, S. Demkowicz, D. Witt, 2013 .

Geometry optimization of steroid sulfatase inhibitors - the influence on the free binding energy with STS

A. Sosnowska, T. Puzyn, J. Leszczynski, 2017, Structural Chemistry.

Phosphate and Thiophosphate Biphenyl Analogs as Steroid Sulfatase Inhibitors

Mateusz Daśko, J. Rachon, W. Kozak, 2015, Drug development research.

Selected Methods for the Chemical Phosphorylation and Thiophosphorylation of Phenols

Mateusz Daśko, J. Rachon, W. Kozak, 2018 .

Convenient and efficient synthesis of functionalized unsymmetrical alkynyl sulfides

J. Rachon, S. Demkowicz, D. Witt, 2016 .

Steroid Sulfatase Inhibitors Based on Phosphate and Thiophosphate Flavone Analogs

Mateusz Daśko, J. Rachon, W. Kozak, 2015, Drug development research.

Novel 1,2,3-Triazole Derivatives as Mimics of Steroidal System—Synthesis, Crystal Structures Determination, Hirshfeld Surfaces Analysis and Molecular Docking

Karol Biernacki, Olga Ciupak, Mateusz Daśko, 2021, Molecules.

Synthesis and Biological Evaluation of Fluorinated 3‐Phenylcoumarin‐7‐O‐Sulfamate Derivatives as Steroid Sulfatase Inhibitors

Mateusz Daśko, J. Rachon, W. Kozak, 2016, Chemical biology & drug design.

Selected organophosphorus compounds with biological activity. Applications in medicine

Mateusz Daśko, J. Rachon, W. Kozak, 2016 .

Design, synthesis and biological evaluation of novel N-phosphorylated and O-phosphorylated tacrine derivatives as potential drugs against Alzheimer’s disease

Mateusz Daśko, S. Demkowicz, I. Inkielewicz-Stępniak, 2022, Journal of enzyme inhibition and medicinal chemistry.

Novel 1,2,4-Oxadiazole Derivatives in Drug Discovery

Karol Biernacki, Mateusz Daśko, Olga Ciupak, 2020, Pharmaceuticals.

Functionalization of Cysteine Derivatives by Unsymmetrical Disulfide Bond Formation

J. Rachon, S. Demkowicz, D. Witt, 2007 .

A Versatile and Convenient Preparation of Unsymmetrical Diaryl Disulfides

J. Rachon, S. Demkowicz, D. Witt, 2008 .

Taurine as a water structure breaker and protein stabilizer

S. Demkowicz, P. Bruździak, A. Panuszko, 2017, Amino Acids.

The Organophosphorus Sulfenyl Bromides as Versatile Reagents for Cysteine Derivatives Functionalization by Unsymmetrical Disulfide Bond Formation

J. Rachon, S. Demkowicz, D. Witt, 2008 .

Modifications at the C(5) position of pyrimidine nucleosides

J. Rak, Mateusz Daśko, J. Rachon, 2020, Russian Chemical Reviews.

Synthesis and biological evaluation of fluorinated N-benzoyl and N-phenylacetoyl derivatives of 3-(4-aminophenyl)-coumarin-7-O-sulfamate as steroid sulfatase inhibitors.

Mateusz Daśko, J. Rachon, K. Kubiński, 2017, European journal of medicinal chemistry.

Towards β-selectivity in functional estrogen receptor antagonists.

S. de Pascual-Teresa, M. Masłyk, S. Demkowicz, 2012, Organic & biomolecular chemistry.

Electron-Induced Decomposition of Uracil-5-yl O-(N,N-dimethylsulfamate): Role of Methylation in Molecular Stability

S. Denifl, J. Rak, Karol Biernacki, 2021, International journal of molecular sciences.

Recent progress in the development of steroid sulphatase inhibitors – examples of the novel and most promising compounds from the last decade

Karol Biernacki, Olga Ciupak, Mateusz Daśko, 2020, Journal of enzyme inhibition and medicinal chemistry.

Intramolecular Proton Transfer in the Radical Anion of Cytidine Monophosphate Sheds Light on the Sensitivities of Dry vs Wet DNA to Electron Attachment-Induced Damage

S. Denifl, Zhaoguo Zhu, Rachel M Harris, 2023, Journal of the American Chemical Society.

Phosphate tricyclic coumarin analogs as steroid sulfatase inhibitors: synthesis and biological activity

B. Gielniewski, Mateusz Daśko, J. Rachon, 2014 .

Hydration of Simple Model Peptides in Aqueous Osmolyte Solutions

Karol Biernacki, S. Demkowicz, A. Panuszko, 2021, International journal of molecular sciences.

Electron-Induced Decomposition of 5-Bromo-4-thiouracil and 5-Bromo-4-thio-2′-deoxyuridine: The Effect of the Deoxyribose Moiety on Dissociative Electron Attachment

S. Denifl, Olga Ciupak, Janusz Rak, 2023, International journal of molecular sciences.

New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives

Karol Biernacki, Olga Ciupak, Mateusz Daśko, 2020, Journal of enzyme inhibition and medicinal chemistry.