P. Ferraboschi

发表

A comparative molecular modeling study of dydrogesterone with other progestational agents through theoretical calculations and nuclear magnetic resonance spectroscopy

D. Colombo, L. Toma, P. Ferraboschi, 2006, The Journal of Steroid Biochemistry and Molecular Biology.

A full conformational characterization of 13-ethylprogestogens through theoretical calculations and nuclear magnetic resonance spectroscopy

D. Colombo, L. Legnani, L. Toma, 2007, The Journal of Steroid Biochemistry and Molecular Biology.

Stereochemical analysis of the 3α‐ and 3β‐hydroxy metabolites of tibolone through NMR and quantum‐chemical investigations. An experimental test of GIAO calculations

D. Colombo, L. Toma, F. Ronchetti, 2002 .

Crystallographic and spectroscopic study on a known orally active progestin

F. Meneghetti, C. Castellano, P. Ferraboschi, 2015, Steroids.

Applications of Lysozyme, an Innate Immune Defense Factor, as an Alternative Antibiotic

P. Ferraboschi, S. Ciceri, P. Grisenti, 2021, Antibiotics.

Chemo-enzymatic approach to the synthesis of the antithrombotic clopidogrel

P. Ferraboschi, M. D. Mieri, Fiorella Galimberti, 2010 .

Synthesis of Antitumor Fluorinated Pyrimidine Nucleosides

P. Ferraboschi, S. Ciceri, P. Grisenti, 2017 .

A full conformational characterization of antiandrogen cortexolone-17α-propionate and related compounds through theoretical calculations and nuclear magnetic resonance spectroscopy

D. Colombo, L. Legnani, G. Celasco, 2014 .

A Simple Synthesis of Gestodene from 18-Methyl-4-estren-3,17-dione

P. Ferraboschi, Paolo Prestileo, A. Onofri, 2004 .

Control of androgen metabolism in the peripheral and central structures: physiological implications

M. Motta, L. Martini, P. Ferraboschi, 1981 .

Enhanced and reversed enantioselectivity of enzymic hydrolysis by simple substrate modifications: the case of 3-hydroxyglutarate diesters

M. Chiari, E. Santaniello, P. Ferraboschi, 1988 .

Vecuronium bromide and its advanced intermediates: A crystallographic and spectroscopic study

M. Mori, D. Colombo, F. Meneghetti, 2021, Steroids.

(S)-Pramipexole and Its Enantiomer, Dexpramipexole: A New Chemoenzymatic Synthesis and Crystallographic Investigation of Key Enantiomeric Intermediates

M. Mori, F. Meneghetti, C. Castellano, 2020 .

The Biocatalytic Approach to the Preparation of Enantiomerically Pure Chiral Building Blocks

E. Santaniello, P. Ferraboschi, P. Grisenti, 1992 .

Synthesis of the antitumoral nucleoside capecitabine through a chemo-enzymatic approach

P. Ferraboschi, P. Ciuffreda, S. Ciceri, 2015 .

Polyethylene Glycols as Solvents for Anionic Activation: Synthesis of Thioacetates by Means of Potassium Thioacetate in Polyethylene Glycol 400

E. Santaniello, P. Ferraboschi, A. Fiecchi, 1987 .

Estimation and characterisation of budesonide tablets impurities.

A. Venturini, R. Stradi, E. Pini, 2008, Journal of pharmaceutical and biomedical analysis.

Full spectroscopic characterization of two crystal pseudopolymorphic forms of the antiandrogen cortexolone 17α-propionate for topic application

M. Mori, F. Meneghetti, R. Stradi, 2017, Steroids.

Synthesis of the immunosuppressive agent 2-morpholinoethyl mycophenolate by a lipase-catalyzed transesterification

P. Ferraboschi, Paolo Prestileo, P. Grisenti, 2006 .

Crystallographic and NMR Investigation of Ergometrine and Methylergometrine, Two Alkaloids from Claviceps Purpurea

M. Mori, F. Meneghetti, P. Ferraboschi, 2020, Molecules.

Synthesis of thiomorpholino buffers for isoelectric focusing in immobilized pH gradients

P. Righetti, M. Chiari, P. Ferraboschi, 1990, Electrophoresis.

A-Ring nitration of estrone

E. Santaniello, P. Ferraboschi, M. Ravasi, 1983 .

An Insight into the Active Site of Pseudomonas Fluorecens (P. cepacia) Lipase to Define the Stereochemical Demand for the Transesterification in Organic Solvents

E. Santaniello, P. Ferraboschi, S. Casati, 1994 .

Further studies on sodium borohydride-polyethylene glycol 400 as a novel reducing system

E. Santaniello, P. Ferraboschi, A. Fiecchi, 1987 .

Reductions of esters, acyl halides, alkyl halides, and sulfonate esters with sodium borohydride in polyethylene glycols: scope and limitation of the reaction

E. Santaniello, P. Ferraboschi, A. Fiecchi, 1983 .

A chemoenzymatic synthesis of enantiomerically pure (R)- and (S)-2-methyldecan-1-ol

E. Santaniello, P. Ferraboschi, P. Grisenti, 1992 .

Recent Advances on Bioreductions Mediated by Baker’s Yeast and Other Microorganisms

E. Santaniello, P. Ferraboschi, A. Manzocchi, 2000 .

Biohydrogenation of unsaturated compounds by Saccharomyces cerevisiae. Part 1. Stereochemical aspects of the reaction and preparation of useful bifunctional chiral synthons

E. Santaniello, P. Ferraboschi, R. Casati, 1987 .

Studies on the regio- and enantioselectivity of the lipase-catalyzed transesterification of 1′- and 2′-naphthyl alcohols in organic solvent

E. Santaniello, P. Ferraboschi, S. Casati, 1995 .

Regio- and enantioselectivity of Pseudomonas cepacia lipase in the transesterification of 2-substituted-1,4-butanediols

E. Santaniello, P. Ferraboschi, P. Grisenti, 1994 .

A biocatalytic approach to the enantioselective synthesis of (R)- and (S)-malic acid

E. Santaniello, P. Ferraboschi, F. Aragozzini, 1991 .

A practical route for the synthesis of 17 substituted steroidal 3-thioxamides

P. Ferraboschi, P. Grisenti, A. Manzocchi, 1997, Steroids.

A chemoenzymatic approach to enantiomerically pure (R)- and (S)-2,3-epoxy-2-(4-pentenyl)-propanol, a chiral building block for the synthesis of (R)- and (S)-frontalin

E. Santaniello, P. Ferraboschi, S. Casati, 1993 .

A New Chemoenzymatic Synthesis of the Chiral Key Intermediate of the Antiepileptic Brivaracetam

P. Ferraboschi, S. Ciceri, P. Grisenti, 2018, Molecules.

Baker's yeast-mediated reduction of α-hydroxy ketones and derivatives: The steric course of the biotransformation

E. Santaniello, P. Ferraboschi, P. Grisenti, 1994 .

Baker′s Yeast Mediated Reduction of α‐Hydroxy Ketones and Derivatives: The Steric Course of the Biotransformation.

E. Santaniello, P. Ferraboschi, P. Grisenti, 1995 .

Baker's Yeast

E. Santaniello, P. Ferraboschi, P. Grisenti, 2001 .

Evaluation, synthesis and characterization of tacrolimus impurities

D. Colombo, P. Ferraboschi, P. Grisenti, 2012, The Journal of Antibiotics.

AN IMPROVED SYNTHESIS OF (S)-3-METHYL-γ-BUTYROLACTONE

E. Santaniello, P. Ferraboschi, A. Fiecchi, 1989 .

Biocatalysis as a new powerful tool for the synthesis of enantiomerically pure chiral building blocks

E. Santaniello, P. Ferraboschi, 1997 .

A novel versatile precursor suitable for 18 F-radiolabeling via "click chemistry".

C. Chinello, P. Ferraboschi, S. Todde, 2017, Journal of labelled compounds & radiopharmaceuticals.

Reduction of esters to alcohols by means of sodium borohydride in polyethylene glycols

P. Sozzani, E. Santaniello, P. Ferraboschi, 1981 .

Chemoenzymatic synthesis of the enantiomerically pure 1,2,3,4-tetrahydroquinoline moiety of the antithrombotic (21R)- and (21S)-argatroban

P. Ferraboschi, S. Ciceri, P. Grisenti, 2013 .

Diastereoselective synthesis of an argatroban intermediate, ethyl (2R,4R)-4-methylpipecolate, by means of a Mandyphos/rhodium complex-catalyzed hydrogenation

P. Ferraboschi, U. Nettekoven, P. Grisenti, 2011 .

Baker’s Yeast Mediated Biohydrogenation of 2-Substituted Allyl Alcohols: Synthesis of Enantiomerically Pure (2S)-3-Benzyloxy-2-methyl-1-propanol

E. Santaniello, P. Ferraboschi, E. Verza, 1996 .

Baker′s Yeast-Mediated Preparation of Optically Active Aryl Alcohols and Diols for the Synthesis of Chiral Hydroxy Acids.

E. Santaniello, P. Ferraboschi, P. Grisenti, 1990 .

Baker's yeast-mediated preparation of optically active aryl alcohols and diols for the synthesis of chiral hydroxy acids

E. Santaniello, P. Ferraboschi, P. Grisenti, 1990 .

First chemoenzymatic synthesis of immunomodulating macrolactam pimecrolimus

D. Colombo, P. Ferraboschi, P. Grisenti, 2009 .

Pseudomonas cepacia Lipase-Catalyzed Enantioselective Acylation of 2-Substituted-1-alkanols in Organic Solvents

E. Santaniello, P. Ferraboschi, 2001 .

Lipase-catalyzed resolution of stereogenic centers in steroid side chains by transesterification in organic solvents: the case of a 26-hydroxycholesterol

E. Santaniello, P. Ferraboschi, E. Verza, 1998 .

The first example of lipase-catalyzed resolution of a stereogenic center in steroid side chains by transesterification in organic solvent

E. Santaniello, P. Ferraboschi, E. Verza, 1996 .

Enantioselective transesterification of 2-methyl-1,3-propanediol derivatives catalyzed by pseudomonas fluorescens lipase in an organic solvent

E. Santaniello, P. Ferraboschi, P. Grisenti, 1992 .

Baker's yeast mediated biohydrogenation of unsaturated compounds containing a methylene group: enantioselective preparation of 2-methyl alkanols from 2-substituted acrolein acetals

E. Santaniello, P. Ferraboschi, E. Verza, 1999 .

Chemoenzymatic syntheses of (25R)- and (25S)-25-hydroxy-27-nor-cholesterol, a steroid bearing a secondary hydroxy group in the side chain

E. Santaniello, P. Ferraboschi, F. Pecora, 1999 .

Lipase-catalyzed transesterification in organic solvents: Applications to the preparation of enantiomerically pure compounds

E. Santaniello, P. Ferraboschi, P. Grisenti, 1993 .

The First Example of Lipase-Catalyzed Resolution of a Stereogenic Center in Steroid Side Chains by Transesterification in Organic Solvent.

E. Santaniello, P. Ferraboschi, E. Verza, 1996 .

Chiral Synthons by Enzymic Acylation and Esterification Reactions

E. Santaniello, P. Ferraboschi, Shahrzad Reza-Elahi, 2001 .

Enzyme recycling does not influence the enantioselectivity of the Pseudomonas cepacia lipase-catalyzed acylation of a racemic alcohol in organic solvents

E. Santaniello, P. Ferraboschi, S. Casati, 1997 .

Enantioselective Pseudomonas fluorescens (P. cepacia) lipase-catalyzed irreversible transesterification of 2-methyl-1,2-diols in an organic solvent

E. Santaniello, P. Ferraboschi, S. Casati, 1994 .

ENZYMATIC RESOLUTION OF 2-SUBSTITUTED OXIRANEMETHANOLS, A CLASS OF SYNTHETICALLY USEFUL BUILDING-BLOCKS BEARING A CHIRAL QUATERNARY CENTER

E. Santaniello, P. Ferraboschi, P. Grisenti, 1991 .

New chemoenzymatic synthesis of (R)- and (S)-4-(phenylsulfonyl)-2-methyl-1-butanol : a chiral C5 isoprenoid synthon

E. Santaniello, P. Ferraboschi, P. Grisenti, 1990 .

Lipase‐Catalyzed Resolution of Stereogenic Centers in Steroid Side Chains by Transesterification in Organic Solvents: The Case of a 26‐Hydroxycholesterol.

E. Santaniello, P. Ferraboschi, E. Verza, 1998 .

Studies on the enantioselectivity of the transesterification of 2-methyl-1,4-butanediol and its derivatives catalyzed by Pseudomonas fluorescens lipase in organic solvents

E. Santaniello, P. Ferraboschi, S. Casati, 1993 .

Enantioselective Transesterification of 2-Methyl-1,3-propanediol Derivatives Catalyzed by Pseudomonas fluorescens Lipase in an Organic Solvent.

E. Santaniello, P. Ferraboschi, P. Grisenti, 1992 .

An efficient chemo-enzymatic approach to the enantioselective synthesis of 2-methyl-1,3-propamedical derivatives

E. Santaniello, P. Ferraboschi, P. Grisenti, 1990 .

Baker′s Yeast Mediated Biohydrogenation of Unsaturated Compounds Containing a Methylene Group: Enantioselective Preparation of 2-Methyl Alkanols from 2-Substituted Acrolein Acetals.

E. Santaniello, P. Ferraboschi, E. Verza, 1999 .

Baker′s Yeast Mediated Biohydrogenation of 2-Substituted Allyl Alcohols: Synthesis of Enantiomerically Pure (2S)-3-Benzyloxy-2-methyl- 1-propanol.

E. Santaniello, P. Ferraboschi, E. Verza, 1997 .

Baker's yeast-mediated hydrogenation of 2-substituted allyl alcohols: A biocatalytic route to a new highly enantioselective synthesis of (R)-2-methyl alkanols

E. Santaniello, P. Ferraboschi, S. Casati, 1994 .

A convenient synthesis of oxandrolone through a regioselective Candida antarctica lipase-catalyzed transformation

D. Colombo, P. Ferraboschi, Paolo Prestileo, 2003 .

A practical chemoenzymatic approach to the synthesis of 3-hydroxy metabolites of tibolone

D. Colombo, P. Ferraboschi, Shahrzad Reza-Elahi, 2002 .

Regio- and enantioselective properties of the lipase-catalyzed irreversible transesterification of some 2-substituted-1,4-butanediols in organic solvents

E. Santaniello, P. Ferraboschi, S. Casati, 1995 .

Selective enzymatic transformations of itaconic acid derivatives: An access to potentially useful building blocks

E. Santaniello, P. Ferraboschi, S. Casati, 1994 .

α-Substituted Primary Alcohols as Substrates for Enantioselective Lipase-Catalyzed Transesterification in Organic Solvents

E. Santaniello, P. Ferraboschi, P. Grisenti, 1992 .

Biohydrogenation of unsaturated compounds by Saccharomyces cerevisiae. Part 2: (S)-(–)-Ethyl 4-hydroxy-3-methylbutanoate as a chiral synthon for the preparation of (25S)-26-hydroxycholesterol

E. Santaniello, P. Ferraboschi, A. Fiecchi, 1987 .

A Convenient Synthesis of (S)-2-Methyl and (2S)-2,3-Dimethyl Butyl Phenylsulfones from (S)-(-)-3-Methyl-γ-butyrolactone

E. Santaniello, P. Ferraboschi, 1984 .

Enantioselective Pseudomonas fluorescens (P. cepacia) Lipase-Catalyzed Irreversible Transesterification of 2-Methyl-1,2-diols in an Organic Solvent.

E. Santaniello, P. Ferraboschi, S. Casati, 1995 .

Enzymatic Resolution of 2-Substituted Oxiranemethanols, a Class of Synthetically Useful Building Blocks Bearing a Chiral Quaternary Center.

E. Santaniello, P. Ferraboschi, P. Grisenti, 1992 .

New Chemoenzymatic Synthesis of (R)‐ and (S)‐4‐(Phenylsulfonyl)‐2‐ methyl‐1‐butanol: A Chiral C5 Isoprenoid Synthon.

E. Santaniello, P. Ferraboschi, P. Grisenti, 1991 .

Studies on the Enantioselectivity of the Transesterification of 2- Methyl-1,4-butanediol and Its Derivatives Catalyzed by Pseudomonas fluorescens Lipase in Organic Solvents.

E. Santaniello, P. Ferraboschi, S. Casati, 2010 .

Synthesis of 3-methyl-1,3,5-pentanetriol and its mono- and diesters

E. Santaniello, P. Ferraboschi, P. Grisenti, 1988 .

An Efficient Chemoenzymatic Approach to the Enantioselective Synthesis of 2‐Methyl‐1,3‐propanediol Derivatives.

E. Santaniello, P. Ferraboschi, P. Grisenti, 1991 .

Microbial reduction of 2-keto acetals as a biocatalytic approach to the enantioselective synthesis of optically active 2-hydroxy acetals

F. Molinari, E. Santaniello, P. Ferraboschi, 1993 .

Biocatalytic, enantioselective preparations of (R)- and (S)-ethyl 4-chloro-3-hydroxybutanoate, a useful chiral synthon

E. Santaniello, P. Ferraboschi, F. Aragozzini, 1992 .

Lipase‐Catalyzed Transesterification in Organic Solvents: Applications to the Preparation of Enantiomerically Pure Compounds

E. Santaniello, P. Ferraboschi, P. Grisenti, 1993 .

Complete 1H and 13C assignments of (21R) and (21S) diastereomers of argatroban

D. Colombo, L. Legnani, P. Ferraboschi, 2008, Magnetic resonance in chemistry : MRC.

Synthesis of Isosteric Analogues of Acylglycosylglycerols Active as Chemoprevention Agents

D. Colombo, F. Compostella, L. Toma, 2002 .

Crystallographic, spectroscopic, and theoretical investigation of the efficiently separated 21R and 21S-diastereoisomers of argatroban.

G. Vistoli, D. Colombo, F. Meneghetti, 2013, Chirality.

Biological Profile of Cortexolone 17a-Propionate (CB-03-01), a New Topical and Peripherally Selective Androgen Antagonist

G. Celasco, L. Moro, C. Quattrocchi, 2004, Arzneimittelforschung.

Regioselective synthesis of 2-chloromercurio-estradiol and -estrone derivatives: a novel approach to A-ring substituted estrogens

E. Santaniello, P. Ferraboschi, A. Fiecchi, 1983 .

New routes to a-ring substituted estrogens.

E. Santaniello, P. Ferraboschi, 1983, Journal of steroid biochemistry.

Reactions of Periodate Under Homogeneous and Phase-Transfer Conditions: Examples of New Oxidations of Unusual Groups

E. Santaniello, P. Ferraboschi, Morteza Nasr Azadani, 1986 .

Effects of 6- and 7-hydroxy metabolites of 3β,17β-dihydroxy-5α-androstane on gonadotrophin and prolactin secretion and on sex accessories weight of male rats

M. Motta, E. Santaniello, P. Ferraboschi, 1983 .

Pharmacological Profile of 9,11-Dehydrocortexolone 17α-Butyrate (CB-03-04), a New Androgen Antagonist with Antigonadotropic Activity

F. Nicoletti, R. Marco, G. Celasco, 2005, Arzneimittelforschung.

Corticosteroids 21-glucuronides: Synthesis and complete characterization by 1H and 13C NMR

P. Ferraboschi, P. Ciuffreda, S. Casati, 2009, Steroids.

Pharmacological control of the mevalonate pathway: effect on arterial smooth muscle cell proliferation.

M. Gelb, P. McGeady, R. Paoletti, 1997, The Journal of pharmacology and experimental therapeutics.

Ovotransferrin Supplementation Improves the Iron Absorption: An In Vitro Gastro-Intestinal Model

P. Ferraboschi, F. Uberti, P. Grisenti, 2021, Biomedicines.

Preliminary studies on the sponge-oxygenator; an improved simple method for extracorporeal blood oxygenation.

G. Tiberio, P. Ferraboschi, A. Bencini, 1957, Surgery.

Baker’s yeast catalyzed preparation of a new enantiomerically pure synthon of (S)-pramipexole and its enantiomer (dexpramipexole)

P. Ferraboschi, P. Ciuffreda, D. Romano, 2014 .

Reduction of esters to alcohols by means of sodium borohydride in polyethylene glycols

P. Sozzani, E. Santaniello, P. Ferraboschi, 1981 .

An Outline of the Latest Crystallographic Studies on Inhibitor-Enzyme Complexes for the Design and Development of New Therapeutics against Tuberculosis

M. Mori, D. Colombo, F. Meneghetti, 2021, Molecules.

Synthesis of C-2 and C-4 deuterium-labeled estradiol-17β

E. Santaniello, P. Ferraboschi, M. Ravasi, 1983, Steroids.

Anti-Tumor-Promoting Activity of Tibolone and its Metabolites

D. Colombo, H. Nishino, H. Tokuda, 2008, Arzneimittel-Forschung (Drug Research).

Testosterone metabolites do not participate in the control of hypothalamic LH-releasing hormone.

M. Motta, P. Ferraboschi, F. Celotti, 1986, The Journal of endocrinology.

Preparation of an A-ring building block for the total synthesis of 1α,25-dihydroxy vitamin D3 and structurally related congeners: lipase-catalyzed stereoselective esterification of a suitable epoxyalcohol

E. Santaniello, P. Ferraboschi, L. Scotti, 2000 .

A new flexible synthesis of (R,S)-mevalonolactone

R. Canevotti, E. Santaniello, P. Ferraboschi, 1987 .

Selective Enzymatic Transformations of Itaconic Acid Derivatives: An Access to Potentially Useful Building Blocks.

E. Santaniello, P. Ferraboschi, S. Casati, 1994 .

Substrate interaction with 5α-reductase enzyme: influence of the 17β-chain chirality in the mechanism of action of 4-azasteroid inhibitors

P. Ferraboschi, V. Villani, F. Celotti, 2001, Steroids.

Interactions between type 1 astrocytes and LHRH-secreting neurons (GT1-1 cells): modification of steroid metabolism and possible role of TGFβ1

R. Melcangi, L. Martini, P. Ferraboschi, 1999, The Journal of Steroid Biochemistry and Molecular Biology.

Heat-Treated Lysozyme Hydrochloride: A Study on Its Structural Modifications and Anti-SARS-CoV-2 Activity

E. Pariani, S. Parapini, S. Delbue, 2023, Molecules.

Total assignment of 1H and 13C NMR spectra of 13α‐ and 13β‐estrone methyl ethers

P. Ferraboschi, P. Ciuffreda, E. Verza, 2001 .

Reduction of Ozonides by Means of Polymeric Triphenylphosphine: Simplified Synthesis of Carbonyl Compounds from Alkenes

E. Santaniello, P. Ferraboschi, Morteza Nasr Azadani, 1986 .

Synthesis of one diastereomeric couple of the mucolytic drug domiodol [(4S, 2R,S)‐2‐iodomethyl‐4‐hydroxymethyl‐1,3‐dioxolane] from D‐mannitol as chiral starting material

E. Santaniello, P. Ferraboschi, P. Grisenti, 1995 .

Seawater‐Based Biocatalytic Strategy: Stereoselective Reductions of Ketones with Marine Yeasts

F. Molinari, G. Burgaud, A. Pinto, 2016 .