G. Chevé

发表

A quantitative structure activity relationship approach to probe the influence of the functionalization on the drug encapsulation of porous metal-organic frameworks

C. Gaudin, C. Serre, G. Maurin, 2012 .

Insight into the selective inhibition of JNK family members through structure-based drug design

G. Chevé, A. Yasri, K. Bougrin, 2016 .

Structural Elucidation of the DFG-Asp in and DFG-Asp out States of TAM Kinases and Insight into the Selectivity of Their Inhibitors

G. Chevé, A. Yasri, K. Bougrin, 2014, Molecules.

Axl Kinase as a Key Target for Oncology: Focus on Small Molecule Inhibitors

G. Chevé, A. Yasri, Clémence Feneyrolles, 2014, Molecular Cancer Therapeutics.

Design, synthesis, and biological evaluation of bifunctional thyrointegrin inhibitors: new anti-angiogenesis analogs

S. Mousa, E. Dyskin, A. Bridoux, 2011, Journal of enzyme inhibition and medicinal chemistry.

Increased Susceptibility of Low-Density Lipoprotein to Ex Vivo Oxidation in Mice Transgenic for Human Apolipoprotein B Treated with 1 Melatonin-Related Compound Is Not Associated with Atherosclerosis Progression

R. Bordet, D. Lesieur, G. Torpier, 2005, Journal of cardiovascular pharmacology.

De novo design, synthesis and pharmacological evaluation of new azaindole derivatives as dual inhibitors of Abl and Src kinases

G. Chevé, A. Yasri, O. Loget, 2012 .

Anti-tumor Activity of Novel Compounds Targeting BCR-ABL, c-SRC and BCR-ABLT315I in Chronic Myelogenous Leukemia

P. Auberger, M. Coisy-Quivy, G. Chevé, 2013 .

Melatonin related compounds inhibit lipid peroxidation during copper or free radical‐induced LDL oxidation

D. Lesieur, J. Fruchart, D. Bonnefont-Rousselot, 2002, Journal of pineal research.

Antioxidant activity of pinoline analogues in the LDL oxidation model

J. Poupaert, D. Lesieur, J. Fruchart, 2002 .

Rational Design, Synthesis, and Biological Evaluation of 7-Azaindole Derivatives as Potent Focused Multi-Targeted Kinase Inhibitors.

A. Yasri, G. Chevé, F. Gassiot, 2016, Journal of medicinal chemistry.

Structure–activity relationship of phenytoinergic antiepileptic drugs related to ameltolide

J. Poupaert, C. McCurdy, G. Chevé, 2007, Medicinal Chemistry Research.

Structure–activity relationships of neuropeptide FF and related peptidic and non-peptidic derivatives

C. Mollereau, C. McCurdy, G. Chevé, 2006, Peptides.

Determination and validation of mTOR kinase-domain 3D structure by homology modeling

Gwénaël Chevé, Azeddine Ibrahimi, A. Yasri, 2015, OncoTargets and therapy.

Recent progress in the design, study, and development of c-Jun N-terminal kinase inhibitors as anticancer agents.

G. Chevé, A. Yasri, K. Bougrin, 2014, Chemistry & biology.

A combined ligand-based and target-based drug design approach for G-protein coupled receptors: application to salvinorin A, a selective kappa opioid receptor agonist

David M. Ferguson, Christopher R. McCurdy, Nidhi Singh, 2006, J. Comput. Aided Mol. Des..

Comparative Protein Modeling of 1-Deoxy-D-xylulose-5-phosphate Reductoisomerase Enzyme from Plasmodium falciparum: A Potential Target for Antimalarial Drug Discovery

Mitchell A. Avery, Christopher R. McCurdy, Nidhi Singh, 2006, J. Chem. Inf. Model..

Recent advances in drug design of epidermal growth factor receptor inhibitors.

M. Coisy-Quivy, R. Benhida, G. Chevé, 2013, Current medicinal chemistry.

Discovering novel 7-azaindole-based series as potent AXL kinase inhibitors.

A. Yasri, G. Chevé, Clémence Feneyrolles, 2017, Bioorganic & medicinal chemistry letters.