Jeremy Green

发表

What do medicinal chemists actually make? A 50-year retrospective.

W Patrick Walters, Mark A Murcko, M. Murcko, 2011, Journal of medicinal chemistry.

Recent Advances in the Discovery of Dengue Virus Inhibitors

R. Rijnbrand, Jeremy Green, U. Bandarage, 2012 .

ROCK inhibitors 2. Improving potency, selectivity and solubility through the application of rationally designed solubilizing groups.

M. Jacobs, Jeremy Green, U. Bandarage, 2018, Bioorganic & medicinal chemistry letters.

Novel chemoenzymatic synthesis of peptide C-terminal amides from ester precursors

A. Margolin, Jeremy Green, 1992 .

Convenient synthesis of N-(4-(2-aminopyridin-4-yl)thiazol-2-yl)-2-phenylacetamides

Jeremy Green, U. Bandarage, J. Come, 2006 .

Application of the Photoredox Coupling of Trifluoroborates and Aryl Bromides to Analog Generation Using Continuous Flow.

Travis J. DeLano, Jeremy Green, U. Bandarage, 2016, The Journal of organic chemistry.

4-(Benzimidazol-2-yl)-1,2,5-oxadiazol-3-ylamine derivatives: potent and selective p70S6 kinase inhibitors.

G. Bemis, V. Savić, C. Moody, 2009, Bioorganic & medicinal chemistry letters.

NG-2,2,5,7,8-pentamethylchroman-6-sulphonyl-L-arginine: A new acid labile derivative for peptide synthesis

Jeremy Green, R. Ramage, 1987 .

Design , Synthesis , and Structure − Activity Relationships of Pyridine-Based Rho Kinase ( ROCK ) Inhibitors

D. Newsome, P. Taslimi, M. Jacobs, 2015 .

Design, synthesis and biological evaluation of potent NAD+-dependent DNA ligase inhibitors as potential antibacterial agents. Part I: aminoalkoxypyrimidine carboxamides.

F. Maltais, P. Charifson, Tiansheng Wang, 2012, Bioorganic & medicinal chemistry letters.

Novel phosphate ester-linked resins: The solid-phase generation of phenyl phosphate-containing compounds for SH2 inhibition

D. Holt, E. Laborde, Jeremy Green, 1998 .

Synthesis of β-Ketosulfonamides Derived from Amino Acids and Their Conversion to β-Keto-α,α-difluorosulfonamides via Electrophilic Fluorination.

Scott D. Taylor, J. Hein, Jeremy Green, 2017, The Journal of organic chemistry.

Structure-based design of 3-aryl-6-amino-triazolo[4,3-b]pyridazine inhibitors of Pim-1 kinase.

G. Bemis, A. Pierce, M. Jacobs, 2009, Bioorganic & medicinal chemistry letters.

3-Aryl-4-(arylhydrazono)-1H-pyrazol-5-ones: Highly ligand efficient and potent inhibitors of GSK3beta.

E. ter Haar, A. Pierce, Michael Arnost, 2010, Bioorganic & medicinal chemistry letters.

Mtb PKNA/PKNB Dual Inhibition Provides Selectivity Advantages for Inhibitor Design To Minimize Host Kinase Interactions.

G. Bemis, Tiansheng Wang, B. Hanzelka, 2017, ACS medicinal chemistry letters.

ROCK Inhibitors 4: Structure-Activity Relationship Studies of 7-Azaindole-Based Rho Kinase (ROCK) Inhibitors.

Jeremy Green, U. Bandarage, Huai Gao, 2020, Bioorganic & medicinal chemistry letters.

ROCK inhibitors 3: Design, synthesis and structure-activity relationships of 7-azaindole-based Rho kinase (ROCK) inhibitors.

M. Jacobs, Jeremy Green, U. Bandarage, 2018, Bioorganic & medicinal chemistry letters.

An acid labile arginine derivative for peptide synthesis: NG-2,2,5,7,8-pentamethylchroman-6-sulphonyl-L-arginine

A. J. Blake, A. Blake, Jeremy Green, 1991 .

Discovery of Novel Allosteric HCV NS5B Inhibitors. 2. Lactam-Containing Thiophene Carboxylates.

B. G. Rao, S. Das, D. Bilimoria, 2017, ACS medicinal chemistry letters.

Discovery of Novel Thiophene-Based, Thumb Pocket 2 Allosteric Inhibitors of the Hepatitis C NS5B Polymerase with Improved Potency and Physicochemical Profiles.

B. G. Rao, G. Iyer, L. Chan, 2016, Journal of medicinal chemistry.

Chapter 24. SH2 and SH3 Domains: Choreographers of Multiple Signaling Pathways

M. Botfield, Jeremy Green, 1995 .

Structure-guided design of potent and selective pyrimidylpyrrole inhibitors of extracellular signal-regulated kinase (ERK) using conformational control.

Xiaoling Xie, Jingrong Cao, Alex M Aronov, 2009, Journal of medicinal chemistry.

Flipped out: structure-guided design of selective pyrazolylpyrrole ERK inhibitors.

Xiaoling Xie, Jingrong Cao, Alex M Aronov, 2007, Journal of medicinal chemistry.

The Discovery of VX-745: A Novel and Selective p38α Kinase Inhibitor.

Huai Gao, Yow-Ming Wang, Yow-Ming C Wang, 2011, ACS medicinal chemistry letters.

Structure-based design and parallel synthesis of N-benzyl isatin oximes as JNK3 MAP kinase inhibitors.

G. Bemis, F. Salituro, Edmund M. Harrington, 2009, Bioorganic & medicinal chemistry letters.

Application of design of experiments (DoE) optimization to the one-pot synthesis of 4,6-dihydropteridinones.

Tiansheng Wang, Jeremy Green, W. Gu, 2015, Organic & biomolecular chemistry.

Solid Phase Synthesis of Lavendustin A and Analogs

Jeremy Green, 1995 .

Inhibitors of HIV protease based on modified peptide substrates

G. Marshall, S. Kent, L. Ratner, 1990 .

Studies on the acylation of hydroxy-functionalized resins using Fmoc amino acids activated using diisopropylcarbodiimide/HOBt or as acid fluorides

Jeremy Green, K. Bradley, 1993 .

Solid phase peptide synthesis of ubiquitin

Jeremy Green, O. M. Ogunjobi, R. Ramage, 1989 .

Synthesis of Cycloalkyl Substituted 7-Azaindoles via Photoredox Nickel Dual Catalytic Cross-Coupling in Batch and Continuous Flow.

Travis J DeLano, Jeremy Green, U. Bandarage, 2016, Organic letters.

Hydroxyethylamine analogues of the p17/p24 substrate cleavage site are tight-binding inhibitors of HIV protease.

G R Marshall, G. Marshall, S. Kent, 1990, Journal of medicinal chemistry.

Analogues of 4-[(7-Bromo-2-methyl-4-oxo-3H-quinazolin-6-yl)methylprop-2-ynylamino]-N-(3-pyridylmethyl)benzamide (CB-30865) as potent inhibitors of nicotinamide phosphoribosyltransferase (Nampt).

Brett R. Murphy, T. Fleischer, J. Boniface, 2010, Journal of medicinal chemistry.

Abstract LB-288: MPI-0486348: A novel inhibitor of nicotinamide phosphoribosyltransferase (Nampt) induces tumor regression in a preclinical model

V. Baichwal, T. Fleischer, Jeremy Green, 2010 .

Structure-based design and parallel synthesis of N-benzyl isatin oximes as JNK3 MAP kinase inhibitors.

G. Bemis, F. Salituro, Edmund M. Harrington, 2009, Bioorganic & Medicinal Chemistry Letters.

Development of methodology for arginine and N-alpha protection in peptide synthesis

Jeremy Green, R. Ramage, Michael R. Florence, 1988 .

Structure-guided design of potent and selective pyrimidylpyrrole inhibitors of extracellular signal-regulated kinase (ERK) using conformational control.

G. Bemis, F. Maltais, J. Janetka, 2009, Journal of medicinal chemistry.

Discovery of Novel Thiophene-Based, Thumb Pocket 2 Allosteric Inhibitors of the Hepatitis C NS5B Polymerase with Improved Potency and Physicochemical Profiles.

G. Iyer, L. Chan, C. Yannopoulos, 2016, Journal of medicinal chemistry.