F Porreca

发表

Design of cyclic deltorphins and dermenkephalins with a disulfide bridge leads to analogues with high selectivity for delta-opioid receptors.

V J Hruby, R. Horváth, V. Hruby, 1994, Journal of medicinal chemistry.

Probes for narcotic receptor mediated phenomena. 19. Synthesis of (+)-4-[(alpha R)-alpha-((2S,5R)-4-allyl-2,5-dimethyl-1-piperazinyl)-3- methoxybenzyl]-N,N-diethylbenzamide (SNC 80): a highly selective, nonpeptide delta opioid receptor agonist.

J. Flippen-Anderson, K. Rice, R. Rothman, 1994, Journal of medicinal chemistry.

Development of a model for the delta opioid receptor pharmacophore. 1. Conformationally restricted Tyr1 replacements in the cyclic delta receptor selective tetrapeptide Tyr-c[D-Cys-Phe-D-Pen]OH (JOM-13).

A. Lomize, H. Mosberg, F. Porreca, 1994, Journal of medicinal chemistry.

Newly discovered stereochemical requirements in the side-chain conformation of delta opioid agonists for recognizing opioid delta receptors.

R. Horváth, B. Lou, A. Misicka, 1994, Journal of medicinal chemistry.

Statistical analysis of drug-drug and site-site interactions with isobolograms.

A Cowan, R. Tallarida, F. Porreca, 1989, Life sciences.

Synthesis, opioid receptor binding, and biological activities of naltrexone-derived pyrido- and pyrimidomorphinans.

S K Saini, K. Rice, R. Rothman, 1999, Journal of medicinal chemistry.

Glial cell line-derived neurotrophic factor normalizes neurochemical changes in injured dorsal root ganglion neurons and prevents the expression of experimental neuropathic pain

T. Vanderah, F. Porreca, M. Ossipov, 2003, Neuroscience.

Tramadol, M1 metabolite and enantiomer affinities for cloned human opioid receptors expressed in transfected HN9.10 neuroblastoma cells.

R. Raffa, F. Porreca, J. Lai, 1996, European journal of pharmacology.

Potent and nontoxic antisense oligonucleotides containing locked nucleic acids.

T. Hökfelt, C. Wahlestedt, J. Skouv, 2000, Proceedings of the National Academy of Sciences of the United States of America.

A comparison of the potential role of the tetrodotoxin-insensitive sodium channels, PN3/SNS and NaN/SNS2, in rat models of chronic pain.

R M Eglen, J C Hunter, R. Eglen, 1999, Proceedings of the National Academy of Sciences of the United States of America.

Antinociceptive actions of BW373U86 in the mouse.

T. Vanderah, F. Porreca, K D Wild, 1993, The Journal of pharmacology and experimental therapeutics.