A. Fivush

发表

Identification of a nonsteroidal liver X receptor agonist through parallel array synthesis of tertiary amines.

Timothy M Willson, L. Moore, T. Willson, 2002, Journal of medicinal chemistry.

Discovery of (1R,2R)-N-(4-(6-isopropylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide, a potent and orally efficacious mGlu5 receptor negative allosteric modulator.

D. McKinzie, S. Iyengar, B. Clark, 2013, Bioorganic & medicinal chemistry letters.

Novel selective small molecule agonists for peroxisome proliferator-activated receptor delta (PPARdelta)--synthesis and biological activity.

T. Willson, M. Lambert, H. Xu, 2003, Bioorganic & medicinal chemistry letters.

Novel bicyclo[3.1.0]hexane analogs as antagonists of metabotropic glutamate 2/3 receptors for the treatment of depression.

J. F. Soriano, P. Ornstein, M. Blanco, 2016, Bioorganic & medicinal chemistry letters.

AMEBA: An acid sensitive aldehyde resin for solid phase synthesis

T. Willson, A. Fivush, 1997 .

Metabotropic Glutamate Receptor

J. F. Soriano, P. Ornstein, S. Atwell, 2016 .

Rearrangement of a-Phenylselenenylketones

D. Liotta, M. Saindane, A. Fivush, 1986 .

Novel selective small molecule agonists for peroxisome proliferator-activated receptor δ (PPARδ)—synthesis and biological activity

T. Willson, M. Lambert, H. Xu, 2003 .

In vitro characterisation of the novel positive allosteric modulators of the mGlu5 receptor, LSN2463359 and LSN2814617, and their effects on sleep architecture and operant responding in the rat

Janice W. Smith, M. Tricklebank, F. Gastambide, 2013, Neuropharmacology.

Discovery of (1S,2R,3S,4S,5R,6R)-2-Amino-3-[(3,4-difluorophenyl)sulfanylmethyl]-4-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid Hydrochloride (LY3020371·HCl): A Potent, Metabotropic Glutamate 2/3 Receptor Antagonist with Antidepressant-Like Activity.

J. F. Soriano, P. Ornstein, S. Atwell, 2016, Journal of medicinal chemistry.

Identification of a chemical tool for the orphan nuclear receptor FXR.

L. Moore, T. Willson, K. Plunket, 2000, Journal of medicinal chemistry.

Identification of peroxisome proliferator-activated receptor ligands from a biased chemical library.

J. Lehmann, T. Smith-Oliver, T. Willson, 1997, Chemistry & biology.

A Unique and Convenient One-Step Preparation of Spiro[4.5]deca-6,9-diene-2,8-dione

A. Fivush, Sanford R. Strunk, 1996 .