R. Badorrey

发表

Highly convergent stereoselective synthesis of chiral key intermediates in the synthesis of Palinavir from imines derived from l-glyceraldehyde

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2002 .

Vascular Reactivity Profile of Novel KCa3.1‐Selective Positive‐Gating Modulators in the Coronary Vascular Bed

H. Wulff, R. Köhler, L. Rivera, 2016, Basic & clinical pharmacology & toxicology.

tert-Butyl (7R)-7-[(4S)-2,2-dimethyl-[1,3]dioxolan-4-yl]-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxylate

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2002 .

A novel pan-negative-gating modulator of KCa 2 / 3 channels , the fluoro-di-benzoate , RA2 , inhibits EDH-type relaxation in coronary artery and produces bradycardia in vivo . ( RA2 , a negative-gating modulator of KCa 2 / 3 )

Brandon M. Brown, R. Badorrey, J. Gálvez, 2014 .

Efficient resolution of rac-2-cyano-2-methyl-3-phenylpropanoic acid. An appropriate starting material for the enantioconvergent synthesis of (S)-α-methylphenylalanine on a large laboratory scale

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2003 .

Recent advances in enantioselective organocatalyzed anhydride desymmetrization and its application to the synthesis of valuable enantiopure compounds.

R. Badorrey, J. Gálvez, Pablo Etayo, 2011, Chemical Society reviews.

Efficient stereodivergent synthesis of 1,4-dideoxy-1,4-iminohexitols from an (S)-glyceraldimine

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2004 .

Debenzylative cycloetherification as synthetic tool in the diastereoselective synthesis of 3,6-disubstituted hexahydro-2H-furo[3,2-b]pyrroles, PDE1 enzyme inhibitors with antiproliferative effect on melanoma cells.

J. Kehler, C. Christoffersen, R. Badorrey, 2020, The Journal of organic chemistry.

STEREOCONTROLLED SYNTHESIS OF ALL FOUR STEREOISOMERS OF FULLY PROTECTED 2-AMINO-3-HYDROXYPENTANOIC ACID FROM IMINES DERIVED FROM D-GLYCERALDEHYDE

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1999 .

Switch in regioselectivity of epoxide ring-opening by changing the organometallic reagent.

R. Badorrey, J. Gálvez, P. López‐Ram‐de‐Viu, 2011, Organic & biomolecular chemistry.

Stereoselective amination of chiral enolates: Synthesis of enantiomerically pure α,β-diamino acids, chiral key compounds in the synthesis of conformationally constrained peptido- and non-peptidomimetics

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1995 .

Asymmetric synthesis of (1R,5S)-2-methyl-6,7-benzomorphan via Aza-Prins reaction.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2021, Chirality.

Synthesis of (R)-quinuclidine-2-carboxylic acid in enantiomerically pure form

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2008 .

Diastereoselective reduction of ketimines derived from (R)-3,4-dihydroxybutan-2-one: an alternative route to key intermediates for the synthesis of anticancer agent ES-285

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2010 .

Highly Stereoselective Synthesis of Stereochemically Defined Polyhydroxylated Propargylamines by Alkynylation of N-Benzylimines Derived from (R)-Glyceraldehyde

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2007 .

On the mechanism of the copper-catalyzed enantioselective 1,4-addition of grignard reagents to alpha,beta-unsaturated carbonyl compounds.

B. Feringa, W. Browne, A. Minnaard, 2006, Journal of the American Chemical Society.

Organocatalysis in Enantioselective α-Functionalization of 2-Cyanoacetates

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2014 .

Diastereoselective Construction of the 6-Oxa-2-azabicyclo[3.2.1]octane Scaffold from Chiral α-Hydroxyaldehyde Derivatives by the Aza-Prins Reaction.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2017, The Journal of organic chemistry.

Organocatalyzed enantioselective desymmetrization of diols in the preparation of chiral building blocks.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2012, Chemistry.

Asymmetric Synthesis of ES-285, an Anticancer Agent Isolated from Marine Sources

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2009 .

Copper-catalyzed asymmetric conjugate addition of Grignard reagents to cyclic enones.

B. Feringa, A. Minnaard, S. Harutyunyan, 2004, Proceedings of the National Academy of Sciences of the United States of America.

Study of the Lewis acid-promoted addition of silylenol ethers to imines derived from glyceraldehyde

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2003 .

Asymmetric Hetero Diels-Alder Reaction of N-Benzylimines Derived from R-Glyceraldehyde: A New Approach to Homochiral Piperidine Building Blocks and its Application to the Synthesis of (2R)-4-Oxopipecolic Acid

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1997 .

Chiral Amino Diol Derivatives as New Modular Organocatalysts for the Enantioselective α-Chlorination of Cyclic β-Keto Esters

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2010 .

Chiral iminoesters derived from D-glyceraldehyde in [3 + 2] cycloaddition reactions. Asymmetric synthesis of a key intermediate in the synthesis of neuramidinase inhibitors.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2013, The Journal of organic chemistry.

Michael addition of carbonyl compounds to nitroolefins under the catalysis of new pyrrolidine-based bifunctional organocatalysts.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2018, Organic & biomolecular chemistry.

Asymmetric Synthesis of a Novel Conformationally Constrained D‐Lysine Analogue with a Piperidine Skeleton

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2008 .

Stereoselective Synthesis of Chiral 2,3‐Disubstituted 2,3‐Dihydro‐4(1H)‐pyridones

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2008 .

Asymmetric synthesis of (2R,3S)-4-halo-3-benzyloxy-2-(N-methoxycarbonyl-N-benzylamino)butyronitriles as precursors for the synthesis of β-hydroxy-α-amino acids

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2000 .

Reversal of the stereochemical course of the addition of phenylmagnesium bromide to N-benzylimines derived from R-glyceraldehyde depending on the O-protecting group and its application to the synthesis of both enantiomers of phenylglycine

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1997 .

Efficient enantioconvergent synthesis of (S)-α-benzyl-α-methyl-β-alanine from (R)- and (S)-2-cyano-2-methyl-3-phenylpropanoic acid

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2003 .

Synthesis of new pyrrolidine-based organocatalysts and study of their use in the asymmetric Michael addition of aldehydes to nitroolefins

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2017, Beilstein journal of organic chemistry.

Stereoselective synthesis and biological evaluation of D-fagomine, D-3-epi-fagomine and D-3,4-epi-fagomine analogs from D-glyceraldehyde acetonide as a common building block.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2012, Organic & biomolecular chemistry.

Study of the Reactions between Vinylmagnesium Bromide and Imines Derived from (R)‐Glyceraldehyde − The Key Step in the Stereodivergent Synthesis of Conveniently Protected, Enantiopure syn‐ and anti‐2‐Amino‐1,3,4‐butanetriol Derivatives

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2003 .

A Convenient Synthesis of L-α-Vinylglycine from D-Mannitol

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1997 .

Study of the Reactions Between Vinylmagnesium Bromide and Imines Derived from (R)-Glyceraldehyde — The Key Step in the Stereodivergent Synthesis of Conveniently Protected, Enantiopure syn- and anti-2-Amino-1,3,4-butanetriol Derivatives.

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2003 .

A Convenient Synthesis of L‐α‐Vinylglycine from D‐Mannitol.

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1997 .

Stereocontrolled synthesis of orthogonally protected 2-substituted 4-aminopiperidines.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2009, Organic & biomolecular chemistry.

Stereodivergent Addition of Allylmetal Reagents to Imines Derived from (R)‐2,3‐Di‐O‐benzylglyceraldehyde by Appropriate Selection of Metal and Double Stereodifferentiation

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 2002 .

A new approach to the stereoselective synthesis of conveniently protected α-allyl substituted amino acids; chiral key compounds in the synthesis of constrained peptide isostere constituents

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1997 .

A New Approach to the Stereoselective Synthesis of Conveniently Protected α-Allyl Substituted Amino Acids; Chiral Key Compounds in the Synthesis of Constrained Peptide Isostere Constituents.

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1997 .

First Stereoselective Synthesis of (1R,2R,4R)‐ and (1S,2R,4S)‐2‐Substituted‐1‐azabicyclo[2.2.1]heptanes

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2009 .

Study of the reaction of imines derived from (R)-glyceraldehyde with Danishefsky's diene

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1999 .

Efficient stereoselective synthesis of enantiopure cis-and trans-1,2,4-trisubstituted piperidines

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2007 .

Unexpected epimerization at C2 in the Horner-Wadsworth-Emmons reaction of chiral 2-substituted-4-oxopiperidines.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2006, Chemical communications.

Study of the Reaction of Imines Derived from (R)‐Glyceraldehyde with Danishefsky′s Diene.

C. Cativiela, R. Badorrey, M. D. Díaz-de-Villegas, 1999 .

Base-controlled diastereodivergent synthesis of (R)- and (S)-2-substituted-4-alkylidenepiperidines by the Wadsworth-Emmons reaction.

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2007, Journal of Organic Chemistry.

A Novel Pan-Negative-Gating Modulator of KCa2/3 Channels, Fluoro-Di-Benzoate, RA-2, Inhibits Endothelium-Derived Hyperpolarization–Type Relaxation in Coronary Artery and Produces Bradycardia In Vivo

Brandon M. Brown, H. Wulff, R. Köhler, 2015, Molecular Pharmacology.

Expedient asymmetric synthesis of (2S,3S)-Boc-phenylalanine epoxide, a key intermediate for the synthesis of biologically active compounds

R. Badorrey, M. D. Díaz-de-Villegas, J. Gálvez, 2009 .