A. Niewiadomy

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Differences in electrochemical response of prospective anticancer drugs IPBD and Cl-IPBD, doxorubicin and Vitamin C at plasmid modified glassy carbon.

P. Kulesza, A. Girstun, Dominika Janiszek, 2020, Bioelectrochemistry.

Spectroscopic Studies of Intramolecular Proton Transfer in 2-(4-Fluorophenylamino)-5-(2,4-Dihydroxybenzeno)-1,3,4-Thiadiazole

A. Niewiadomy, M. Gagoś, A. Matwijczuk, 2010, Journal of Fluorescence.

QSAR models of antiproliferative activity of imidazo[2,1-b][1,3,4]thiadiazoles in various cancer cell lines

A. Niewiadomy, J. Matysiak, 2016, Molecular Diversity.

EFFECT OF ORGANIC MODIFIER ON THE LIPOPHILICITY OF ANTIPROLIFERATIVE ACTIVE 4-(5-AMINO-1,3,4-THIADIAZOL-2-YL)BENZENE-1,3-DIOLS BY REVERSED-PHASE OVERPRESSURED LAYER CHROMATOGRAPHY

A. Niewiadomy, J. Matysiak, A. Skrzypek, 2010 .

Molecular organization of the antifungal and anticancer drug 2-(2,4-dihydroxyphenylo)-5,6-dichlorobenzothiazole in solution and in monolayers: an effect of pH.

W. Gruszecki, G. Menestrina, A. Niewiadomy, 2005, Journal of photochemistry and photobiology. B, Biology.

One‐Pot Synthesis of New (1,3‐Thiazolo[5,4‐b]pyridin‐2‐yl)benzenediols and Their Antiproliferative Activities against Human Cancer Cell Lines

J. Wietrzyk, M. Karpińska, A. Niewiadomy, 2012, Chemistry & biodiversity.

In Search of the Antimicrobial Potential of Benzimidazole Derivatives

M. Janeczko, Z. Kazimierczuk, A. Niewiadomy, 2016, Polish journal of microbiology.

Synthesis and biological activity of novel 4- and 6-(1-alkyl/aryl-1H-benzimidazol-2-yl)benzene-1,3-diols

J. Wietrzyk, M. Karpińska, A. Niewiadomy, 2012, Monatshefte für Chemie - Chemical Monthly.

Spectroscopic and theoretical studies of fluorescence effects in bio-active: 4-(5-(methyl-1,3,4-thiadiazol-2-yl))benzene-1,3-diol and 4-(5-(methylamino-1,3,4-thiadiazol-2-yl))benzene-1,3-diol compounds: Effect of molecular aggregation and amino group position

M. Makowski, M. Karpińska, A. Niewiadomy, 2018, Journal of Luminescence.

Spectroscopic and Theoretical Studies of Fluorescence Effects in 2-Methylamino-5-(2,4-dihydroxyphenyl)-1,3,4-thiadiazole Induced by Molecular Aggregation

M. Makowski, J. Wąs, A. Niewiadomy, 2017, Journal of Fluorescence.

Synthesis and antiproliferative activity of some N′-substituted 2,4-dihydroxybenzothiohydrazides

J. Wietrzyk, M. Karpińska, A. Niewiadomy, 2016, Journal of enzyme inhibition and medicinal chemistry.

Biological evaluation and molecular docking of novel 1,3,4-thiadiazole-resorcinol conjugates as multifunctional cholinesterases inhibitors.

M. Bajda, P. Szymański, M. Karpińska, 2021, Bioorganic chemistry.

Spectroscopic studies of the molecular organization of 4-([ 1,2,4 ] triazolo [ 4,3- a ] pyridin-3-yl)-6-methylbenzene-1,3-diol in selected solvents

W. Gruszecki, A. Niewiadomy, M. Gagoś, 2018 .

Influence of Solvent Polarizability on the Keto-Enol Equilibrium in 4-[5-(naphthalen-1-ylmethyl)-1,3,4-thiadiazol-2-yl]benzene-1,3-diol

B. Mysliwa-Kurdziel, A. Niewiadomy, M. Gagoś, 2015, Journal of Fluorescence.

New derivative of 2-(2,4-dihydroxyphenyl)thieno-1,3-thiazin-4-one (BChTT) elicits antiproliferative effect via p38-mediated cell cycle arrest in cancer cells.

K. Walczak, W. Rzeski, M. Lemieszek, 2016, Bioorganic & medicinal chemistry.

On polymorphism of 2-(4-fluorophenylamino)-5-(2,4-dihydroxybenzeno)-1,3,4-thiadiazole (FABT) DMSO solvates

K. Woźniak, A. Niewiadomy, M. Gagoś, 2013 .

Design, synthesis and biological evaluation of novel 1,3,4-thiadiazole derivatives as anti-glioblastoma agents targeting the AKT pathway.

R. Rola, M. Karpińska, A. Niewiadomy, 2020, Bioorganic chemistry.

Spectroscopic Studies of Fluorescence Effects in Bioactive 4-(5-Heptyl-1,3,4-Thiadiazol-2-yl)Benzene-1,3-Diol and 4-(5-Methyl-1,3,4-Thiadiazol-2-yl)Benzene-1,3-Diol Molecules Induced by pH Changes in Aqueous Solutions

A. Niewiadomy, M. Gagoś, A. Matwijczuk, 2017, Journal of Fluorescence.

Synthesis and antimycotic activity of N-azolyl-2,4-dihydroxythiobenzamides.

A. Niewiadomy, J. Matysiak, 2003, Bioorganic & medicinal chemistry.

Antifungal effects of a 1,3,4-thiadiazole derivative determined by cytochemical and vibrational spectroscopic studies

A. Olender, A. Niewiadomy, M. Gagoś, 2019, PloS one.

In vitro antifungal activity of new thiatriazole derivative agents

W. Kułak, C. Łukaszuk, A. Niewiadomy, 2011 .

Effect of Solvent Polarizability on the Keto/Enol Equilibrium of Selected Bioactive Molecules from the 1,3,4-Thiadiazole Group with a 2,4-Hydroxyphenyl Function.

S. Wybraniec, A. Niewiadomy, M. Gagoś, 2017, The journal of physical chemistry. A.

Influence of Solvent Polarizability on the Keto-Enol Equilibrium in 4-[5-(naphthalen-1-ylmethyl)-1,3,4-thiadiazol-2-yl]benzene-1,3-diol

A. Niewiadomy, M. Gagoś, A. Matwijczuk, 2015, Journal of Fluorescence.

Synthesis and biological evaluation of 1,3,4-thiadiazole analogues as novel AChE and BuChE inhibitors.

Paweł Szymański, Marek Bajda, Joanna Matysiak, 2013, European journal of medicinal chemistry.

Synthesis of some 1-(2,4-dihydroxythiobenzoyl)imidazoles, -imidazolines and -tetrazoles and their potent activity against Candida species.

A. Niewiadomy, J. Matysiak, E. Krajewska-Kułak, 2003, Farmaco.

Application of Sulfinyl bis(2,4‐dihydroxythiobenzoyl) in the Synthesis of N‐Substituted 2‐Amino‐5‐(2,4‐dihydroxyphenyl)‐1,3,4‐thiadiazoles

A. Niewiadomy, J. Matysiak, 2006 .

Synthesis and Anticancer Activity of New 2‐Aryl‐4H‐3,1‐benzothiazines

M. Karpińska, A. Niewiadomy, J. Matysiak, 2011, Archiv der Pharmazie.

Synthesis and Antibacterial Activity of Novel Fused 1,3‐Thiazoles and 1,3‐Thiazines Incorporating a 2,4‐Dihydroxyphenyl Residue

M. Polz-Dacewicz, A. Malm, M. Karpińska, 2012, Archiv der Pharmazie.

2-Amino-1,3,4-thiadiazole derivative (FABT) inhibits the extracellular signal-regulated kinase pathway and induces cell cycle arrest in human non-small lung carcinoma cells.

W. Rzeski, A. Niewiadomy, J. Albrecht, 2012, Bioorganic & medicinal chemistry letters.

Spectroscopic studies of dual fluorescence effects in a selected 1,3,4-thiadiazole derivative in organic solvents and aqueous solutions

S. Wybraniec, A. Niewiadomy, M. Gagoś, 2017 .

Solvent Effects on Molecular Aggregation in 4-(5-Heptyl-1,3,4-thiadiazol-2-yl)benzene-1,3-diol and 4-(5-Methyl-1,3,4-thiadiazol-2-yl)benzene-1,3-diol.

A. Niewiadomy, M. Gagoś, A. Matwijczuk, 2016, The journal of physical chemistry. B.

The activity of a new 2-amino-1,3,4-thiadiazole derivative 4ClABT in cancer and normal cells.

W. Rzeski, A. Niewiadomy, J. Matysiak, 2011, Folia histochemica et cytobiologica.

Solvatomorphism of 2-(4-Fluorophenylamino)-5- (2,4-dihydroxybenzeno)-1,3,4-thiadiazole Chloride

K. Woźniak, A. Niewiadomy, M. Gagoś, 2010 .

Synthesis, characterization, and pharmacological evaluation of novel azolo- and azinothiazinones containing 2,4-dihydroxyphenyl substituent as anticancer agents

K. Walczak, W. Rzeski, M. Lemieszek, 2015, Monatshefte für Chemie - Chemical Monthly.

A new approach to the synthesis of 2-aryl-substituted benzimidazoles, quinazolines, and other related compounds and their antibacterial activity

A. Malm, M. Karpińska, A. Niewiadomy, 2012 .

Synthesis, antifungal activity and SAR of N-substituted and N,N-disubstituted 2,4-dihydroxythiobenzamides

A. Niewiadomy, J. Matysiak, Z. Fekner, 2006 .

Synthesis and biological activity of novel benzoazoles, benzoazines and other analogs functionalized by 2,4-dihydroxyphenyl moiety

J. Wietrzyk, A. Niewiadomy, A. Matwijczuk, 2018, Research on Chemical Intermediates.

Synthesis of 4-(4-methylidene-4H-3,1-benzothiazin-2-yl)benzene1,3-diols and their antiproliferative activity against human cancer cell lines

J. Wietrzyk, M. Karpińska, A. Niewiadomy, 2016, Russian Journal of Bioorganic Chemistry.

Design, synthesis and antiproliferative activity against human cancer cell lines of novel benzo-, benzofuro-, azolo- and thieno-1,3-thiazinone resorcinol hybrids

W. Rzeski, J. Wietrzyk, M. Karpińska, 2015, Arabian Journal of Chemistry.

Synthesis of 2-(2,4-dihydroxyphenyl)thieno-1,3-thiazin-4-ones, their lipophilicity and anticancer activity in vitro

K. Walczak, W. Rzeski, M. Lemieszek, 2015, Molecular Diversity.

Synthesis of novel 4-(1H-benzimidazol-2-yl)benzene-1,3-diols and their cytotoxic activity against human cancer cell lines

A. Niewiadomy, J. Matysiak, Monika M Karpińka, 2011, Archives of pharmacal research.

Dynamic Method of Determination of Octanol‐Water Partition Coefficient of 2,4‐Dihydroxythiobenzanilides in QSAR Studies

B. Marczewska, A. Niewiadomy, J. Matysiak, 2004 .

N-heterocyclic derivatives of 2,4-dihydroxybenzcarbothioamide as antimycotic agents.

J. Karczewski, A. Niewiadomy, J. Matysiak, 2001, Journal of agricultural and food chemistry.

In vitro evaluation of 2,4-dihydroxythiobenzanilides against various moulds.

A. Niewiadomy, J. Matysiak, G. Macik-Niewiadomy, 2001, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

Synthesis and mycological activity of the compounds obtained in the reaction of N(3)-substituted amidrazones with sulphinyl-bis-2,4-dihydroxybenzenethioyl.

A. Niewiadomy, J. Matysiak, B. Modzelewska-Banachiewicz, 2001, European journal of medicinal chemistry.

In vitro inhibition properties of a new group of thiobenzanilides in relation to yeasts.

A. Niewiadomy, J. Matysiak, G. Macik-Niewiadomy, 2000, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

Dependence of fungistatic activity of 2, 4-dihydroxythiobenzanilideson the structure and lipophilic nature of the compounds.

A. Niewiadomy, J. Matysiak, G. Macik-Niewiadomy, 2000, European journal of medicinal chemistry.

Use of reversed-phase high-performance liquid chromatography in QSAR analysis of 2,4-dihydroxythiobenzanilide analogues.

A. Niewiadomy, K. Jóźwiak, H. Szumiło, 1999, SAR and QSAR in environmental research.

Molecular organization of the antifungal and anticancer drug 2-(2,4-dihydroxyphenylo)-5,6-dichlorobenzothiazole (dHBBT) in solution and in lipid membranes studied by means of electronic absorption spectroscopy.

W. Gruszecki, A. Niewiadomy, M. Gagoś, 2004, Journal of photochemistry and photobiology. B, Biology.

Determination of the Lipophilicity of Bioactive 2-Phenylbenzothiazoles by RPTLC

A. Niewiadomy, J. Matysiak, A. Żabińska, 2002, JPC – Journal of Planar Chromatography – Modern TLC.

Molecular Organization of Dipalmitoylphosphatidylcholine Bilayers Containing Bioactive Compounds 4-(5-Heptyl-1,3,4-thiadiazol-2-yl) Benzene-1,3-diol and 4-(5-Methyl-1,3,4-thiadiazol-2-yl) Benzene-1,3-diols.

M. Szymanek, M. Karpińska, A. Niewiadomy, 2016, The journal of physical chemistry. B.

Evaluation of the effect of 2-(2,4-dihydroxyphenyl)-4H-benzofuro[3,2-d][1,3]thiazin-4-one on colon cells and its anticancer potential

W. Rzeski, M. Lemieszek, M. Karpińska, 2018, Medicinal Chemistry Research.

OPLC and HPTLC methods in physicochemical studies of a new group of antimycotic compounds.

A. Niewiadomy, J. Matysiak, A. Żabińska, 2002, Journal of chromatographic science.

Evaluation of N-Substituted 2,4-Dihydroxyphenylthioamide Fungicide Lipophilicity Using the Chromatographic Techniques HPLC and HPTLC

A. Niewiadomy, M. Kostecka, R. Czeczko, 2005 .

In vivo and in silico pharmacological studies on some new 4-(1,3,4-thiadiazol-2-yl)benzene-1,3-diol analogues

A. Niewiadomy, E. Jagiełło-wójtowicz, A. Chodkowska, 2014, Russian Journal of Bioorganic Chemistry.

Synergistic antifungal interactions of amphotericin B with 4-(5-methyl-1,3,4-thiadiazole-2-yl) benzene-1,3-diol

A. Olender, A. Niewiadomy, M. Gagoś, 2019, Scientific Reports.

In vitro antifungal activity of 2,5 disubstituted amino-oksometyloso-arylo-thiadiazole derivatives.

A. Niewiadomy, E. Krajewska-Kułak, U. Głaszcz, 2007, Advances in medical sciences.

In vitro antifungal activity of N-3-( 1 , 2 , 4-dithiazole-5-thione )-- -

A. Niewiadomy, Krajewska-Kułak, Kostecka, 2022 .

Spectroscopic Studies of Dual Fluorescence in 2-(4-Fluorophenylamino)-5-(2,4-dihydroxybenzeno)-1,3,4-thiadiazole: Effect of Molecular Aggregation in a Micellar System

A. Szcześ, G. Gładyszewski, A. Niewiadomy, 2018, Molecules.

Spectroscopic Studies of Dual Fluorescence in 2-((4-Fluorophenyl)amino)-5-(2,4-dihydroxybenzeno)-1,3,4-thiadiazole.

A. Niewiadomy, M. Gagoś, A. Matwijczuk, 2015, The journal of physical chemistry. A.

Effect of 2-(4-fluorophenylamino)-5-(2,4-dihydroxyphenyl)-1,3,4-thiadiazole on the molecular organisation and structural properties of the DPPC lipid multibilayers.

D. Pociecha, E. Górecka, A. Niewiadomy, 2012, Biochimica et biophysica acta.

RPHPLC as a tool for determining the congenericity of a set of 2,4-dihydroxythiobenzanilide derivatives

A. Niewiadomy, K. Jóźwiak, H. Szumiło, 2000 .

Evaluation of the Antiproliferative Activity of 2-(Monohalogenophenylamino)-5-(2,4-dihydroxyphenyl)-1,3,4-thiadiazoles

W. Rzeski, A. Niewiadomy, J. Matysiak, 2008, Arzneimittel-Forschung (Drug Research).

A. Oniszczuk, A. Niewiadomy, M. Gagoś, 2020, Molecules.

Interplay of Inter- and Intramolecular Interactions in Crystal Structures of 1,3,4-Thiadiazole Resorcinol Derivatives

K. Woźniak, A. Niewiadomy, M. Gagoś, 2018, Crystal Growth & Design.

Isolation and spectroscopic characterization of Zn(II), Cu(II), and Pd(II) complexes of 1,3,4-thiadiazole-derived ligand

B. Creaven, A. Niewiadomy, M. Gagoś, 2017 .

Phase Transition Detection in Accumulation of a Potential Anticancer Drug Cl-IPBD with DNA: Supercoiled and Linear pUC19 Plasmids

P. Kulesza, A. Girstun, M. Maj-Zurawska, 2016 .

Synthesis and anticholinesterase activities of novel 1,3,4-thiadiazole based compounds

M. Karpińska, A. Niewiadomy, J. Matysiak, 2013, Journal of enzyme inhibition and medicinal chemistry.

Biological Evaluation, Molecular Docking, and SAR Studies of Novel 2-(2,4-Dihydroxyphenyl)-1H- Benzimidazole Analogues

M. Bajda, P. Szymański, M. Karpińska, 2019, Biomolecules.

Relationships between LC retention, octanol-water partition coefficient, and fungistatic properties of 2-(2,4-dihydroxyphenyl)benzothiazoles.

A. Niewiadomy, J. Matysiak, B. Senczyna, 2004, Journal of AOAC International.

Structure and retention of 2,4-dihydroxythiobenzanilides in a reversed-phase system

A. Niewiadomy, J. Matysiak, A. Żabińska, 1999 .

Reversed-phase high-performance liquid chromatography in quantitative structure–activity relationship studies of new fungicides

A. Niewiadomy, J. Matysiak, K. Jóźwiak, 1998 .

Synthesis of 4-(4-methylidene-4H-3,1-benzothiazin-2-yl)benzene1,3-diols and their antiproliferative activity against human cancer cell lines

J. Wietrzyk, M. Karpińska, A. Niewiadomy, 2016, Russian journal of bioorganic chemistry.

2-Amino-1,3,4-thiadiazole derivative (FABT) inhibits the extracellular signal-regulated kinase pathway and induces cell cycle arrest in human non-small lung carcinoma cells.

W. Rzeski, J. Albrecht, A. Niewiadomy, 2012, Bioorganic & Medicinal Chemistry Letters.

Spectroscopic studies of dual fluorescence effects in a selected 1,3,4-thiadiazole derivative in organic solvents and aqueous solutions

S. Wybraniec, A. Niewiadomy, M. Gagoś, 2017 .

New derivative of 2-(2,4-dihydroxyphenyl)thieno-1,3-thiazin-4-one (BChTT) elicits antiproliferative effect via p38-mediated cell cycle arrest in cancer cells.

K. Walczak, W. Rzeski, M. Lemieszek, 2016, Bioorganic & medicinal chemistry.

Characterization and preliminary anticonvulsant assessment of some 1,3,4-thiadiazole derivatives

J. Luszczki, M. Karpińska, A. Niewiadomy, 2015, Pharmacological reports : PR.

A simple HPLC method for determining 2-(3-chlorophenyloamino)-5-(2,4-dihydroxyphenyl)-1,3,4-thiadiazole in brain and plasma of animals: Application to a pharmacokinetic study

G. Raszewski, W. Rzeski, M. Lemieszek, 2014 .

In vitro Antifungal Activity of N,N-Phenyl-1,2,3,4-thiatriazole-5-yl-2,4-ßresorcylcarbothioamide

C. Łukaszuk, A. Niewiadomy, J. Matysiak, 2003, Arzneimittelforschung.