Angus M MacLeod

Pharmacokinetics and metabolism studies on (3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy) pyrazolo[1,5-d][1,2,4]triazine, a functionally selective GABA(A) alpha5 inverse agonist for cognitive dysfunction.

Desmond O'Connor, Robert Maxey, J. Atack, 2006, Bioorganic & medicinal chemistry letters.

Selective, orally active gamma-aminobutyric acidA alpha5 receptor inverse agonists as cognition enhancers.

Desmond O'Connor, Gerard R Dawson, John R Atack, 2004, Journal of medicinal chemistry.

4-(Phenylsulfonyl)piperidines: novel, selective, and bioavailable 5-HT(2A) receptor antagonists.

Desmond O'Connor, Peter Blurton, Robert Clarkson, 2002, Journal of medicinal chemistry.

4-Fluorosulfonylpiperidines: selective 5-HT2A ligands for the treatment of insomnia.

Desmond O'Connor, Angus M MacLeod, Smita Patel, 2005, Bioorganic & medicinal chemistry letters.