A. Giannis

发表

Potent small molecule Hedgehog agonists induce VEGF expression in vitro.

K. Seifert, A. Büttner, S. Rigol, 2012, Bioorganic & medicinal chemistry.

Exo-cyclopamine--a stable and potent inhibitor of hedgehog-signaling.

B. Kirchner, S. Zahn, A. Büttner, 2011, Chemical communications.

Synthesis of cyclopamine using a biomimetic and diastereoselective approach.

A. Giannis, P. Heretsch, V. Sarli, 2009, Angewandte Chemie.

A scaffold-tree-merging strategy for prospective bioactivity annotation of gamma-pyrones.

Stefan Wetzel, Tudor I. Oprea, Herbert Waldmann, 2010, Angewandte Chemie.

Synthesis of the First Selective Irreversible Inhibitor of Neutral Sphingomyelinase

A. Giannis, C. Arenz, 2000 .

Peptidomimetics in Drug Design

Athanassios Giannis, A. Giannis, F. Rübsam, 1997 .

Integrin Antagonists and Other Low Molecular Weight Compounds as Inhibitors of Angiogenesis: New Drugs in Cancer Therapy

A. Giannis, F. Rübsam, 1997 .

Analogues of the Sialyl Lewisx Group and of the N‐Acetylneuraminic Acid in the Antiadhesion Therapy

A. Giannis, 2003 .

Inhibition of the Mitotic Kinesin Eg5 Up-regulates Hsp70 through the Phosphatidylinositol 3-Kinase/Akt Pathway in Multiple Myeloma Cells*

Min Liu, R. Aneja, Chunyong Liu, 2006, Journal of Biological Chemistry.

Barbier-type allylation of chiral α-aminoaldehydes: Dependence of the stereochemical outcome on metal and allylic halide

A. Giannis, F. Rübsam, S. Seck, 1997 .

Inhibition of N-acetylglucosamine kinase and N-acetylmannosamine kinase by 3-O-methyl-N-acetyl-D-glucosamine in vitro.

E. Henk, W. Reutter, K. Sandhoff, 1992, European journal of biochemistry.

Selectivity of commonly used pharmacological inhibitors for cystathionine β synthase (CBS) and cystathionine γ lyase (CSE)

Christos T. Chasapis, A. Papapetropoulos, Zongmin Zhou, 2013, British journal of pharmacology.

Increasing Muscle Mass Improves Vascular Function in Obese (db/db) Mice

Yunchao Su, J. Mintz, Christina Salet, 2014, Journal of the American Heart Association.

1-Methylthiodihydroceramide, a Novel Analog of Dihydroceramide, Stimulates Sphinganine Degradation Resulting in Decreased de Novo Sphingolipid Biosynthesis*

K. Sandhoff, A. Futerman, G. van Echten-Deckert, 1998, The Journal of Biological Chemistry.

Small molecules as inhibitors of cyclin-dependent kinases.

A. Huwe, Ralph Mazitschek, A. Giannis, 2003, Angewandte Chemie.

A sulindac analogue is effective against malignant pleural effusion in mice.

C. Roussos, I. Kalomenidis, S. Papiris, 2011, Lung cancer.

The role of soluble guanylyl cyclase in chronic obstructive pulmonary disease.

G. Joos, A. Papapetropoulos, P. Brouckaert, 2013, American journal of respiratory and critical care medicine.

A Novel Approach to Decrease Sialic Acid Expression in Cells by a C-3-modified N-Acetylmannosamine*

W. Reutter, S. Rigol, A. Giannis, 2014, The Journal of Biological Chemistry.

Use of costic acid, a natural extract from Dittrichia viscosa, for the control of Varroa destructor, a parasite of the European honey bee

H. Katerinopoulos, A. Büttner, A. Giannis, 2017, Beilstein journal of organic chemistry.

The soluble guanylyl cyclase inhibitor NS-2028 reduces vascular endothelial growth factor-induced angiogenesis and permeability.

C. Roussos, A. Papapetropoulos, A. Pyriochou, 2010, American journal of physiology. Regulatory, integrative and comparative physiology.

Development and Biological Evaluation of a Novel Aurora A Kinase Inhibitor

J. Xu, Teresa Sardon, A. Giannis, 2009, Chembiochem : a European journal of chemical biology.

Identification of Gli-mediated transcription inhibitors through synthesis and evaluation of taepeenin D analogues

M. Chatzopoulou, A. Giannis, E. Pitsinos, 2016 .

Synthesis and biological evaluation of novel fumagillin and ovalicin analogues.

A. Huwe, Ralph Mazitschek, A. Giannis, 2005, Organic & biomolecular chemistry.

The Effect of Adjuvant Dimethylenastron, a Mitotic Kinesin Eg5 Inhibitor, in Experimental Glaucoma Filtration Surgery

H. Merz, S. Grisanti, A. Giannis, 2010, Current eye research.

Manumycin A and Its Analogues Are Irreversible Inhibitors of Neutral Sphingomyelinase

H. Waldmann, A. Giannis, C. Arenz, 2001, Chembiochem : a European journal of chemical biology.

Inhibitors of Mitotic Kinesins: Next‐Generation Antimitotics

A. Giannis, V. Sarli, 2006, ChemMedChem.

Synthesis and biological investigation of (+)-3-hydroxymethylartemisinin

M. Kaiser, A. Giannis, Xingzhao Tu, 2019, Beilstein journal of organic chemistry.

Total Synthesis and Biological Investigation of (-)-Artemisinin: The Antimalarial Activity of Artemisinin Is not Stereospecific.

T. Efferth, M. Kaiser, Ean-jeong Seo, 2018, Angewandte Chemie.

From Substrate to Transition State Analogues: The First Potent Inhibitor of Sialyltransferases.

A. Giannis, Peer Nils Schröder, 1999, Angewandte Chemie.

Aristoforin, a Novel Stable Derivative of Hyperforin, Is a Potent Anticancer Agent

J. Sleeman, J. Simon, T. Müller, 2005, Chembiochem : a European journal of chemical biology.

Synthesis and Εvaluation of Αnticancer Αctivity in Cells of Novel Stoichiometric Pegylated Fullerene-Doxorubicin Conjugates

C. Gialeli, N. Karamanos, K. Avgoustakis, 2015, Pharmaceutical Research.

Kinesin Motor Inhibitors as Effective Anticancer Drugs

A. Giannis, V. Sarli, 2008 .

NADPH Oxidase 4 Is Expressed in Pulmonary Artery Adventitia and Contributes to Hypertensive Vascular Remodeling

Yunchao Su, G. Kéri, S. Barman, 2014, Arteriosclerosis, thrombosis, and vascular biology.

Synthesis and evaluation of acyl protein thioesterase 1 (APT1) inhibitors.

H. Waldmann, A. Giannis, M. Biel, 2006, Chemistry.

Design and synthesis of novel platelet fibrinogen receptor antagonists with 2H-1,4-benzoxazine-3(4H)-one scaffold. A systematic study.

M. Anderluh, M. Dolenc, D. Kikelj, 2005, European journal of medicinal chemistry.

Synthesis and biological evaluation of new tetrahydro-beta-carbolines as inhibitors of the mitotic kinesin Eg5.

T. Surrey, Mathias Utz, T. Mayer, 2005, Bioorganic & medicinal chemistry.

Synthesis and Biological Evaluation of Novel Eg5 Inhibitors

T. Mayer, A. Giannis, V. Sarli, 2005, Chembiochem : a European journal of chemical biology.

Development and Biological Evaluation of Potent and Specific Inhibitors of Mitotic Kinesin Eg5

I. Vernos, T. Surrey, Mathias Utz, 2005, Chembiochem : a European journal of chemical biology.

The Veratrum and Solanum alkaloids.

A. Giannis, P. Heretsch, 2015, The Alkaloids. Chemistry and biology.

Thioglycine and L-thiovaline: biologically active H₂S-donors.

A. Papapetropoulos, Zongmin Zhou, C. Coletta, 2012, Bioorganic & medicinal chemistry.

Improved Isolation of Microbiologically Produced (2R,3S)-Isocitric Acid by Adsorption on Activated Carbon and Recovery with Methanol

S. Mauersberger, R. Gläser, R. Müller, 2017 .

Hünlich base: (re)discovery, synthesis, and structure elucidation after a century.

J. Sieler, S. Rigol, A. Giannis, 2013, Organic letters.

New Spiro-Lactam C-nor -D -homo Steroids

A. Giannis, Aybike Yektaoglu, Dimanthi Pliatsika, 2018, European Journal of Organic Chemistry.

Influence of the Scyphostatin Side Chain on the Mode of Inhibition of Neutral Sphingomyelinase

A. Giannis, E. Pitsinos, V. Wascholowski, 2006, ChemMedChem.

Lewis Acid Mediated Nazarov Cyclization as a Convergent and Enantioselective Entry to C-nor-D-homo-Steroids.

A. Giannis, Toni Smeilus, J. Krieger, 2017, Chemistry.

Synthesis and cytotoxic activity of new artemisinin hybrid molecules against human leukemia cells.

T. Efferth, Ean-jeong Seo, A. Giannis, 2017, Bioorganic & medicinal chemistry.

Synthesis of ¹³C-labeled and functionalized Hyaluronan derivatives for biophysical studies and surface modifications.

S. Rigol, A. Giannis, Liang Xia, 2013, Bioorganic & medicinal chemistry.

Selective inhibition of CBP/p300 HAT.

A. Giannis, V. Sarli, 2007, Chemistry & biology.

Hyperforin and aristoforin inhibit lymphatic endothelial cell proliferation in vitro and suppress tumor‐induced lymphangiogenesis in vivo

M. Rothley, A. Noël, J. Sleeman, 2009, International journal of cancer.

Guanylyl cyclase activation reverses resistive breathing-induced lung injury and inflammation.

A. Papapetropoulos, Zongmin Zhou, S. Theocharis, 2014, American journal of respiratory cell and molecular biology.

20-Aminosteroids as a novel class of selective and complete androgen receptor antagonists and inhibitors of prostate cancer cell growth.

Undine Schubert, A. Baniahmad, A. Giannis, 2010, Bioorganic & medicinal chemistry.

Inhibitors of Histone Acetyltransferases: Discovery and Biomedical Perspectives

A. Giannis, M. V. W. Rekowski, 2009 .

Immunological Alterations due to Hemodialysis Might Interfere with Early Complications in Renal Transplantation

U. Sack, A. Boldt, S. Schiekofer, 2019, Analytical cellular pathology.

Synthesis of phosphoramide analogues of sphinganine-1-phosphate

K. Sandhoff, T. Kolter, A. Giannis, 1996 .

Synthesis of potential inhibitors of the glycosphingolipid biosynthesis

K. Sandhoff, G. Brenner-Weiss, A. Giannis, 1992 .

Synthesis of 2-Carboxy-Substituted Sphingosine Derivatives

E. Henk, K. Sandhoff, T. Kolter, 1990 .

Synthesis of C-Nor-D-homo-steroidal Alkaloids and Their Derivatives

A. Giannis, D. Meyer, Farnoush Mousavizadeh, 2018, Synthesis.

A fast entry to furanoditerpenoid-based Hedgehog signaling inhibitors: identifying essential structural features.

M. Chatzopoulou, S. Haroutounian, A. Giannis, 2014, Organic letters.

Synthesis of a hexasaccharide partial sequence of hyaluronan for click chemistry and more

S. Rigol, A. Giannis, Marina Bantzi, 2015, Beilstein journal of organic chemistry.

Peptidomimetics for Receptor Ligands—Discovery, Development, and Medical Perspectives

Thomas Kolter, Athanassios Giannis, T. Kolter, 1993 .

Peptidomimetics in Drug Design

Athanassios Giannis, F. Ruebsam, A. Giannis, 1997 .

Development of new and efficient polymer-supported hypervalent iodine reagents

A. Giannis, M. Mülbaier, S. Ficht, 2001 .

Curare Alkaloids: Constituents of a Matis Dart Poison.

R. Bussmann, V. Tsetlin, I. Shelukhina, 2015, Journal of natural products.

LiBH4(NaBH4)/Me3SiCl, an Unusually Strong and Versatile Reducing Agent†

K. Sandhoff, A. Giannis, 1989 .

Fragmentation and wittig olefination of glucosamine derivatives-a simple route to open chain amino sugars and chiral glycerols

K. Sandhoff, A. Giannis, W. Steglich, 1988 .

Traceless solid-phase synthesis of 2-aminothiazoles: receptor tyrosine kinase inhibitors with dual selectivity for Tie-2 and VEGFR-2.

H. Waldmann, Ralph Mazitschek, F. Stieber, 2002, Angewandte Chemie.

A Mild and Effective Method for the Transesterification of Carboxylic Acid Esters P.B. and R.M. are grateful to the Land Baden-Württemberg for a scholarship from the Landesgraduiertenförderung.

Ralph Mazitschek, Patrick Baumhof, A. Giannis, 2001, Angewandte Chemie.

Diastereoselektive synthese von funktionalisierten C-α- und -β-glykosylderivaten der 2-acetamido-2-desoxy-d-glucose☆

K. Sandhoff, A. Giannis, 1987 .

Fragmentation and Wittig olefination of glucosamine derivatives: a simple toute to open chain amino sugars and chiral glycerols

K. Sandhoff, A. Giannis, W. Steglich, 1989 .

Natural product derived receptor tyrosine kinase inhibitors: identification of IGF1R, Tie-2, and VEGFR-3 inhibitors.

H. Waldmann, Ralph Mazitschek, A. Giannis, 2002, Angewandte Chemie.

Inhibitors of angiogenesis and cancer-related receptor tyrosine kinases.

Ralph Mazitschek, A. Giannis, 2004, Current opinion in chemical biology.

Enantioselective biocatalytic synthesis of (S)-monastrol.

Jürgen Wittmann, Athanassios Giannis, Harald Gröger, 2010, Bioorganic & medicinal chemistry letters.

Z-Selective olefination of base-sensitive chiral β-hydroxy-α-aminoaldehydes using a modified Horner-Wadsworth-Emmons reaction

A. Giannis, F. Rübsam, C. Michel, 1997 .

De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives

A. Giannis, M. Hartmann, Dimanthi Pliatsika, 2019, Journal of medicinal chemistry.

Multistep solid-phase synthesis of an antibiotic and receptor tyrosine kinase inhibitors using the traceless phenylhydrazide linker.

H. Waldmann, Ralph Mazitschek, U. Grether, 2003, Chemistry.

Sphingolactones: selective and irreversible inhibitors of neutral sphingomyelinase.

A. Giannis, V. Wascholowski, 2006, Angewandte Chemie.

Synthesis and Evaluation of Three Novel Scyphostatin Analogues as Neutral Sphingomyelinase Inhibitors

E. Couladouros, A. Giannis, E. Pitsinos, 2003, Chembiochem : a European journal of chemical biology.

On Artemisinin, Cyclopamine, D-Isocitric acid, Hyperforin, Epigenetics, Sialic Acid, and More

A. Giannis, Farnoush Mousavizadeh, 2019, Synlett.

A Mild and Effective Method for the Transesterification of Carboxylic Acid Esters.

Ralph Mazitschek, Patrick Baumhof, A. Giannis, 2002 .

Phloroglucinol derivatives guttiferone G, aristoforin, and hyperforin: inhibitors of human sirtuins SIRT1 and SIRT2.

S. Kyrylenko, C. Gey, A. Büttner, 2007, Angewandte Chemie.

N‐Sulfinyl benzenesulfonamide

A. Giannis, P. Heretsch, 2012 .

Oxone/Sodium Chloride: A Simple and Efficient Catalytic System for the Oxidation of Alcohols to Symmetric Esters and Ketones

A. Giannis, G. Pagona, A. Schulze, 2006 .

Synthesis and evaluation of caged Garcinia xanthones.

A. Batova, A. Yu, E. Theodorakis, 2007, Organic & biomolecular chemistry.

Design, synthesis, and biological evaluation of a small-molecule inhibitor of the histone acetyltransferase Gcn5.

Athanassios Giannis, Joseph Papamatheakis, Markus Biel, 2004, Angewandte Chemie.

IBX‐Mediated Conversion of Primary Alcohols and Aldehydes to N‐Hydroxysuccinimide Esters

A. Giannis, A. Schulze, 2004 .

Synthesis of tetrahydrofurans by cyclization of homoallylic alcohols with iodine/iodine(III).

A. Giannis, L. F. Silva, R. S. Vasconcelos, 2011, The Journal of organic chemistry.

Synthesis of substituted chiral piperazinones as building blocks for peptidomimetics

T. Kolter, A. Giannis, Christina Dahl, 1995 .

Diastereoselective Synthesis of Functionalized C-α- and C-β-Glycosyl Derivatives of 2-Acetamido-2-deoxy-D-glucose.

K. Sandhoff, A. Giannis, 1988 .

STEREOSELECTIVE SYNTHESIS OF α-C-ALLYLGLYCOPYRANOSIDES

K. Sandhoff, A. Giannis, 1985 .

Indeno[1,2‐d]pyrido[1,2‐a]pyrimidines: A New Class of Receptor Tyrosine Kinase Inhibitors

A. Büttner, A. Giannis, V. Sarli, 2008, ChemMedChem.

LEWIS ACID MEDIATED α‐THIOALKYLATION OF KETONES

M. Reetz, A. Giannis, 1981 .

The Synthesis and Oxidative Properties of Polymer-Supported IBX.

A. Giannis, M. Mülbaier, 2001, Angewandte Chemie.

The Sialyl Lewisx Group and its Analogues as Ligands for Selectins: Chemoenzymatic Syntheses and Biological Functions

A. Giannis, 1994 .

Determination of the relative configuration of a five-membered lactone from residual dipolar couplings.

C. Thiele, R. Berger, A. Giannis, 2006, Angewandte Chemie.

Synthesis and Biological Investigation of Novel Tricyclic Benzodiazepinedione‐Based RGD Analogues

Ralph Mazitschek, A. Giannis, E. Addicks, 2002, Chembiochem : a European journal of chemical biology.

Curare alkaloids from Matis Dart Poison: Comparison with d-tubocurarine in interactions with nicotinic, 5-HT3 serotonin and GABAA receptors

S. Lummis, R. Bussmann, V. Tsetlin, 2019, PloS one.

Synthesis of novel C-9 carbon substituted derivatives of artemisinin.

A. Giannis, Dimanthi Pliatsika, D. Meyer, 2017, Bioorganic & medicinal chemistry.

Anthraquinone Content in Noni (Morinda citrifolia L.)

R. Bussmann, T. Kutchan, A. Giannis, 2013, Evidence-based complementary and alternative medicine : eCAM.

Transcriptional responses of zebrafish embryos exposed to potential sonic hedgehog pathway interfering compounds deviate from expression profiles of cyclopamine.

Wibke Busch, Stefan Scholz, Athanassios Giannis, 2012, Reproductive toxicology.

Histone acetylation modulation by small molecules: a chemical approach.

A. Giannis, M. V. W. Rekowski, Margarete von Wantoch Rekowski, 2010, Biochimica et biophysica acta.

Chirospecific synthesis of amino acids, amino aldehydes and amino alcohols from D-glucosamine hydrochloride. A multigram synthesis of N-boc-L-serinal

A. Giannis, T. Henk, Thomas Henk, 1990 .

Identification of azepinone fused tetracyclic heterocycles as new chemotypes with protein kinase inhibitory activities

A. Giannis, L. Hennig, M. Fousteris, 2016 .

Synthesis and biochemical properties of reversible inhibitors of UDP-N-acetylglucosamine 2-epimerase.

W. Reutter, S. Hinderlich, A. Giannis, 2004, Angewandte Chemie.

Chirospecific Synthesis of Amino Acids, Amino Aldehydes, and Amino Alcohols from D-Glucosamine Hydrochloride. A Multigram Synthesis of N-BOC-L-Serinal.

A. Giannis, T. Henk, 1990 .

Determination of the relative configuration of a five-membered ring compound using RDCs

C. Thiele, R. Berger, A. Giannis, 2006 .

SYNTHESIS OF PHOSPHONATE ANALOGUES OF SPHINGANINE-1-PHOSPHATE AND SPHINGOSINE-1-PHOSPHATE

K. Sandhoff, T. Kolter, A. Giannis, 1995 .

Epigenetics--an epicenter of gene regulation: histones and histone-modifying enzymes.

A. Giannis, V. Wascholowski, M. Biel, 2005, Angewandte Chemie.

Synthesis and biological evaluation of SANT-2 and analogues as inhibitors of the hedgehog signaling pathway.

S. Scholz, K. Seifert, A. Büttner, 2009, Bioorganic & medicinal chemistry.

Oxidation of Alcohols with Catalytic Amounts of IBX

A. Giannis, A. Schulze, 2006 .

Tripolin A, a Novel Small-Molecule Inhibitor of Aurora A Kinase, Reveals New Regulation of HURP's Distribution on Microtubules

B. Agianian, Joe D. Lewis, A. Giannis, 2013, PloS one.

MAZ51, an indolinone that inhibits endothelial cell and tumor cell growth in vitro, suppresses tumor growth in vivo

J. Sleeman, J. Waltenberger, Ralph Mazitschek, 2004, International journal of cancer.

Targeting the Kinesin Spindle Protein: Basic Principles and Clinical Implications

A. Giannis, V. Sarli, 2008, Clinical Cancer Research.

Current aspects of targeted therapy in head and neck tumors

Andreas Dietz, Gunnar Wichmann, Athanassios Giannis, 2008, European Archives of Oto-Rhino-Laryngology.

Synthesis of novel derivatives of 5-hydroxymethylcytosine and 5-formylcytosine as tools for epigenetics

A. Giannis, A. Chentsova, E. Kapourani, 2014, Beilstein journal of organic chemistry.

De Novo Peptide Design and Experimental Validation of Histone Methyltransferase Inhibitors

Christodoulos A. Floudas, Benjamin A. Garcia, Athanassios Giannis, 2014, PloS one.

C–H-Functionalization logic guides the synthesis of a carbacyclopamine analog

A. Giannis, P. Heretsch, Sebastian Rabe, 2014, Beilstein journal of organic chemistry.

Cyclopamine and Congeners

A. Giannis, P. Heretsch, 2014 .

Cyclopamine analogs bearing exocyclic methylenes are highly potent and acid-stable inhibitors of hedgehog signaling

Nicole Eilert, A. Giannis, P. Heretsch, 2013, Beilstein journal of organic chemistry.

Configuratively Stable Dipeptide Aldehydes from D‐Glucosamine Hydrochloride

T. Kolter, A. Giannis, A. Klein, 1992 .

A novel approach to indoloditerpenes by Nazarov photocyclization: synthesis and biological investigations of terpendole E analogues.

Y. Ishikawa, T. Surrey, A. Giannis, 2010, Organic letters.

Inhibition of Angiogenesis‐Relevant Receptor Tyrosine Kinases by Sulindac Analogues

H. Waldmann, Patrick Baumhof, E. Gourzoulidou, 2005, Chembiochem : a European journal of chemical biology.

Peptidomimetics: Modern Approaches and Medical Perspectives

Athanassios Giannis, A. Giannis, 2003 .

Local injection of receptor tyrosine kinase inhibitor MAE 87 reduces retinal neovascularization in mice.

Ralph Mazitschek, H. Agostini, L. Hansen, 2004, Molecular vision.

Synthesis and biological evaluation of an indomethacin library reveals a new class of angiogenesis-related kinase inhibitors.

H. Waldmann, Patrick Baumhof, C. Rosenbaum, 2004, Angewandte Chemie.

Indoloquinolizidine Derivatives as Novel and Potent Apoptosis Inducers and Cell‐Cycle Blockers

H. Waldmann, F. Wehner, A. Nören-Müller, 2008, ChemBioChem.

Modulators of the hedgehog signaling pathway.

A. Giannis, P. Heretsch, Lito Tzagkaroulaki, 2010, Bioorganic & medicinal chemistry.

Abstracts from the 8th International Conference on cGMP Generators, Effectors and Therapeutic Implications

Jordi Villà-Freixa, Peter Sandner, Bernd J. Pichler, 2017, BMC Pharmacology and Toxicology.

Cyclopamine and Hedgehog Signaling: Chemistry, Biology, Medical Perspectives

A. Giannis, P. Heretsch, Lito Tzagkaroulaki, 2010 .

In Vitro and In Silico Antimalarial Evaluation of FM-AZ, a New Artemisinin Derivative

A. Pantaleo, Ioannis Tsamesidis, F. Benoit‐Vical, 2022, Medicines.

Cyclopamine and hedgehog signaling: chemistry, biology, medical perspectives.

A. Giannis, P. Heretsch, Lito Tzagkaroulaki, 2010, Angewandte Chemie.

Microbiologically produced carboxylic acids used as building blocks in organic synthesis.

G. Barth, Christina Otto, R. Müller, 2012, Sub-cellular biochemistry.

Syntheses with a chiral building block from the citric acid cycle: (2R,3S)-isocitric acid by fermentation of sunflower oil.

H. Krautscheid, A. Giannis, P. Heretsch, 2008, Angewandte Chemie.

Small Molecules as Inhibitors of Cyclin-Dependent Kinases

A. Huwe, Ralph Mazitschek, A. Giannis, 2003 .

Inhibitors of kinesin Eg5: antiproliferative activity of monastrol analogues against human glioblastoma cells

Christin Müller, A. Buschauer, G. Bernhardt, 2006, Cancer Chemotherapy and Pharmacology.

Small molecules, big plans--can low-molecular-weight compounds control human regeneration?

C. Gey, A. Giannis, 2004, Angewandte Chemie.

Small Molecules, Big Plans — Can Low‐Molecular‐Weight Compounds Control Human Regeneration?

C. Gey, A. Giannis, 2004 .

Synthesis and biological evaluation of oxadiazole derivatives as inhibitors of soluble guanylyl cyclase.

A. Papapetropoulos, A. Pyriochou, A. Giannis, 2010, Bioorganic & medicinal chemistry.

Synthesis of all diastereomers of the piperidine--alkaloid substructure of cyclopamine.

A. Giannis, P. Heretsch, Sebastian Rabe, 2009, Organic letters.

A biomimetic approach to C-nor-D-homo-steroids.

A. Giannis, P. Heretsch, Sebastian Rabe, 2010, Journal of the American Chemical Society.

Synthesis and Εvaluation of Αnticancer Αctivity in Cells of Novel Stoichiometric Pegylated Fullerene-Doxorubicin Conjugates

C. Gialeli, K. Avgoustakis, A. Giannis, 2015, Pharmaceutical Research.

Novel Activators of the Tumour Suppressor p53

A. Giannis, Nils Sunder-Plassmann, 2004, Chembiochem : a European journal of chemical biology.

Oxidation of Alcohols with Catalytic Amounts of IBX.

A. Giannis, A. Schulze, 2006 .

Insights into soluble guanylyl cyclase activation derived from improved heme-mimetics.

A. Papapetropoulos, Zongmin Zhou, V. Kumar, 2013, Journal of medicinal chemistry.

Epigenetics — An Epicenter of Gene Regulation: Histones and Histone‐Modifying Enzymes

A. Giannis, V. Wascholowski, M. Biel, 2005 .

Sensitive and site-specific identification of carboxymethylated and carboxyethylated peptides in tryptic digests of proteins and human plasma.

R. Hoffmann, A. Frolov, Uta Greifenhagen, 2015, Journal of proteome research.

Abstracts from the 8th International Conference on cGMP Generators, Effectors and Therapeutic Implications

James C. Campbell, Dong I. Lee, M. Zaccolo, 2017, BMC Pharmacology and Toxicology.

Backbone and side chain NMR assignments of the H-NOX domain from Nostoc sp. in complex with BAY58-2667 (cinaciguat)

Georgios A. Dalkas, Garyfallia I. Makrynitsa, A. Papapetropoulos, 2020, Biomolecular NMR Assignments.