S. Jaroch

发表

New Approaches to Drug Discovery

U. Nielsch, U. Fuhrmann, S. Jaroch, 2016, Handbook of Experimental Pharmacology.

Putting small molecules in the lead

H. Weinmann, S. Jaroch, 2005, Nature chemical biology.

SEGRAs: a novel class of anti-inflammatory compounds.

K. Asadullah, A. Schottelius, H. Schäcke, 2002, Ernst Schering Research Foundation workshop.

Discovery of the potent non-steroidal glucocorticoid receptor modulator BAY 1003803 as clinical candidate.

A. Rottmann, T. Zollner, H. Schäcke, 2020, Bioorganic & medicinal chemistry letters.

Characterization of ZK 245186, a novel, selective glucocorticoid receptor agonist for the topical treatment of inflammatory skin diseases

K. Asadullah, W. Döcke, H. Schäcke, 2009, British journal of pharmacology.

THEMED SECTION: MEDIATORS AND RECEPTORS IN THE RESOLUTION OF INFLAMMATION RESEARCH PAPER Characterization of ZK 245186, a novel, selective glucocorticoid receptor agonist for the topical treatment of inflammatory skin diseases

K. Asadullah, T. Zollner, S. Jaroch, 2009 .

CCR5 receptor antagonists: discovery and SAR of novel 4-hydroxypiperidine derivatives.

D. Davey, G. Phillips, J. Onuffer, 2007, Bioorganic & medicinal chemistry letters.

Discovery of new selective glucocorticoid receptor agonist leads.

A. Reichel, H. Schäcke, S. Jaroch, 2017, Bioorganic & medicinal chemistry letters.

Inhibition of neuronal nitric oxide synthase in ovine model of acute lung injury*

D. Herndon, C. Szabó, L. Traber, 2009, Critical care medicine.

Fluorinated dihydroquinolines as potent n-NOS inhibitors.

D. Sülzle, S. Jaroch, H. Rehwinkel, 2004, Bioorganic & medicinal chemistry letters.

Asymmetric Organocatalysis

H. Weinmann, K. Zeitler, S. Jaroch, 2007, ChemMedChem.

Synthesis and Reactivity of α,α-Dichloroglycyl Peptides†‡

S. Jaroch, W. Steglich, T. Schwarz, 1993 .

Studies towards a total synthesis of sarains A-C. Stereospecific condensation of α,β-unsaturated esters with the phenyl oxazoline derivative of threonine

L. Overman, R. Matsuoka, S. Jaroch, 1999 .

Generation of α-acetoxyglycine residues within peptide chains: a new strategy for the modification of oligopeptides

S. Jaroch, W. Steglich, M. Kratzel, 1993 .

Dissociation of transactivation from transrepression by a selective glucocorticoid receptor agonist leads to separation of therapeutic effects from side effects

K. Asadullah, A. Schottelius, W. Döcke, 2003, Proceedings of the National Academy of Sciences of the United States of America.

Methyl 2‐Bromo‐N‐(t‐butoxycarbonyl)glycinate

S. Jaroch, W. Steglich, 2001 .

Comprar Organocatalysis | Reetz, Manfred T. | 9783540734949 | Springer

H. Weinmann, M. Reetz, B. List, 2008 .

Dihydroquinolines with amine-containing side chains as potent n-NOS inhibitors.

D. Sülzle, S. Jaroch, H. Rehwinkel, 2003, Bioorganic & medicinal chemistry letters.

Application of α-chloroglycine residues for the modification of oligopeptides

S. Jaroch, W. Steglich, Peter Zistler, 1994 .

Dihydroquinolines as novel n-NOS inhibitors.

D. Sülzle, S. Jaroch, H. Rehwinkel, 2002, Bioorganic & medicinal chemistry letters.

Total synthesis of (+)-sarain A.

L. Overman, C. Douglas, R. Matsuoka, 2006, Journal of the American Chemical Society.

Discovery of quinolines as selective glucocorticoid receptor agonists.

Markus Berger, Werner Skuballa, Stefan Jaroch, 2010, Bioorganic & medicinal chemistry letters.

ROLE OF NEURONAL NITRIC OXIDE SYNTHASE IN OVINE SEPSIS MODEL

D. Herndon, L. Traber, D. Traber, 2009, Shock.

IMI European Lead Factory — democratizing access to high-throughput screening

Stuart P. McElroy, Philip S. Jones, H. V. van Vlijmen, 2021, Nature reviews. Drug discovery.

Differential Inhibition of Inducible T Cell Cytokine Secretion by Potent Iron Chelators

Hong-tao Lu, M. Berger, D. Schilling, 2005, Journal of biomolecular screening.

A Soluble Amyloid Fibril Segment to Study Aggregate Formation

S. Jaroch, 2007, ChemMedChem.

The European lead factory—an experiment in collaborative drug discovery

Fabrizio Giordanetto, Dimitrios Tzalis, Hugh Laverty, 2016, Journal of Medicines Development Sciences.

Total synthesis of (+)-sarain A.

L. Overman, C. Douglas, R. Matsuoka, 2007, Journal of the American Chemical Society.