Kathy A Sarris

发表

SAR of amino pyrrolidines as potent and novel protein-protein interaction inhibitors of the PRC2 complex through EED binding.

Hongyu Zhao, Ying Wang, Zhiqin Ji, 2017, Bioorganic & medicinal chemistry letters.

Scaffold Oriented Synthesis. Part 1. Design, Preparation, and Biological Evaluation of Thienopyrazoles as Kinase Inhibitors.

J. R. Huth, D. Song, Eric F. Johnson, 2006 .

Discovery of a novel small molecule binding site of human survivin.

Jun Chen, Saul H Rosenberg, Kenneth M Comess, 2007, Bioorganic & medicinal chemistry letters.

Biochemical and biophysical characterization of unique switch pocket inhibitors of p38α.

P. Hajduk, S. Swann, Chaohong Sun, 2010, Bioorganic & medicinal chemistry letters.

Discovery of 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor.

C. Briggs, H. Ween, M. Gopalakrishnan, 2009, Journal of medicinal chemistry.

Discovery and pharmacological evaluation of growth hormone secretagogue receptor antagonists.

E. Bush, H. Sham, D. Beno, 2006, Journal of medicinal chemistry.

A simple and efficient automatable one step synthesis of triazolopyridines from carboxylic acids

D. Sauer, S. Djurić, Kathy A Sarris, 2007 .

A simple and efficient one step synthesis of benzoxazoles and benzimidazoles from carboxylic acids

D. Sauer, S. Djurić, Kathy A Sarris, 2006 .

SAR and characterization of non-substrate isoindoline urea inhibitors of nicotinamide phosphoribosyltransferase (NAMPT).

Ana L. Aguirre, Mikkel A. Algire, C. Tse, 2017, Bioorganic & medicinal chemistry letters.

The Chosen Few: Parallel Library Reaction Methodologies for Drug Discovery.

Ana L. Aguirre, A. Dombrowski, Ying Wang, 2021, The Journal of organic chemistry.

An expeditious and convenient synthesis of acylsulfonamides utilizing polymer-supported reagents

D. Sauer, S. Djurić, Kathy A Sarris, 2007 .

Isoindolinone ureas: a novel class of KDR kinase inhibitors.

K. Glaser, S. Davidsen, M. Michaelides, 2004, Bioorganic & medicinal chemistry letters.

An Expeditious and Convenient Synthesis of Acylsulfonamides Utilizing Polymer‐Supported Reagents.

D. Sauer, S. Djurić, Kathy A Sarris, 2007 .

An Automated Microwave-Assisted Synthesis Purification System for Rapid Generation of Compound Libraries

Noah P Tu, Philip A Searle, Kathy Sarris, 2016, Journal of laboratory automation.

Structure-activity relationship studies on N'-aryl carbohydrazide P2X7 antagonists.

D. Donnelly-roberts, P. Honore, M. Jarvis, 2008, Journal of medicinal chemistry.

Design and Development of Glucocorticoid Receptor Modulators as Immunology Antibody-Drug Conjugate Payloads.

A. Hobson, S. Mathieu, R. Stoffel, 2022, Journal of medicinal chemistry.

Tandem Click-Suzuki reactions in a novel flow reactor incorporating immobilized and exchangeable reagents

S. Djurić, Kathy A Sarris, N. Tu, 2015 .

Scaffold oriented synthesis. Part 1: Design, preparation, and biological evaluation of thienopyrazoles as kinase inhibitors.

J. R. Huth, D. Song, Eric F. Johnson, 2006, Bioorganic & medicinal chemistry letters.

SAR of amino pyrrolidines as potent and novel protein-protein interaction inhibitors of the PRC2 complex through EED binding.

Mikkel A. Algire, Justin D Dietrich, P. Richardson, 2017, Bioorganic & medicinal chemistry letters.