J. Jakubík

发表

Direct product decompositions of bounded commutative residuated ℓ-monoids

J. Jakubík, 2008 .

On complete $MV$-algebras

Ján Jakubík, J. Jakubík, 1995 .

Towards predictive docking at aminergic G-protein coupled receptors

Jan Jakubík, Esam E. El-Fakahany, J. Jakubík, 2015, Journal of Molecular Modeling.

Projectability and weak homogeneity of pseudo effect algebras

Ján Jakubík, J. Jakubík, 2009 .

On the Schröder-Bernstein problem for carathéodory vector lattices

J. Jakubík, 2009 .

On Varieties of Pseudo MV-Algebras

Ján Jakubík, J. Jakubík, 2003 .

Constitutive activity of the M1–M4 subtypes of muscarinic receptors in transfected CHO cells and of muscarinic receptors in the heart cells revealed by negative antagonists

L. Bačáková, J. Jakubík, E. El-Fakahany, 1995, FEBS letters.

Mortality Due to Nosocomial Infection with Klebsiella pneumoniae ESBL.

J. Jakubík, K. Życińska, Katarzyna Starzyk-Łuszcz, 2017, Advances in experimental medicine and biology.

Unoriented graphs of modular lattices

Ján Jakubík, J. Jakubík, 1975 .

On lattices determined up to isomorphisms by their graphs

J. Jakubík, 1984 .

Role of membrane cholesterol in differential sensitivity of muscarinic receptor subtypes to persistently bound xanomeline

J. Jakubík, V. Rudajev, E. El-Fakahany, 2018, Neuropharmacology.

Novel long‐acting antagonists of muscarinic ACh receptors

J. Jakubík, V. Rudajev, V. Doležal, 2018, British journal of pharmacology.

ON K-RADICAL CLASSES OF LATTICE ORDERED GROUPS

J. Jakubík, 2020 .

K-Radical classes and product radical classes of MV-algebras

J. Jakubík, 2008 .

Radical classes and weak radical mappings of GMV-algebras

J. Jakubík, 2008 .

On Some Interpolation Rules for Lattice Ordered Groups

J. Jakubík, 2004 .

Torsion classes of generalized Boolean algebras

J. Jakubík, 2012 .

On slope factor of the operational model of agonism

J. Jakubík, 2021, bioRxiv.

Uncoupling of M1 muscarinic receptor/G-protein interaction by amyloid β1–42

H. Tanila, J. Jakubík, V. Rudajev, 2013, Neuropharmacology.

Impairment of muscarinic transmission in transgenic APPswe/PS1dE9 mice

H. Tanila, E. Machová, J. Jakubík, 2008, Neurobiology of Aging.

Differences in Kinetics of Xanomeline Binding and Selectivity of Activation of G Proteins at M1 and M2 Muscarinic Acetylcholine Receptors

J. Jakubík, E. El-Fakahany, V. Doležal, 2006, Molecular Pharmacology.

Molecular Mechanisms of Methoctramine Binding and Selectivity at Muscarinic Acetylcholine Receptors

J. Jakubík, E. El-Fakahany, V. Doležal, 2014, Molecular Pharmacology.

Asparagine, Valine, and Threonine in the Third Extracellular Loop of Muscarinic Receptor Have Essential Roles in the Positive Cooperativity of Strychnine-Like Allosteric Modulators

A. Krejci, J. Jakubík, V. Doležal, 2005, Journal of Pharmacology and Experimental Therapeutics.

Protection by Alcuronium of Muscarinic Receptors Against Chemical Inactivation and Location of the Allosteric Binding Site for Alcuronium

J. Jakubík, S. Tuček, 1994, Journal of neurochemistry.

Weak toxin WTX from Naja kaouthia cobra venom interacts with both nicotinic and muscarinic acetylcholine receptors

Ya. L. Polyak, Y. Utkin, V. Tsetlin, 2009, The FEBS journal.

Divergence of allosteric effects of rapacuronium on binding and function of muscarinic receptors

J. Jakubík, E. El-Fakahany, V. Doležal, 2009, BMC pharmacology.

Allosteric modulation by persistent binding of xanomeline of the interaction of competitive ligands with the M1 muscarinic acetylcholine receptor.

J. Jakubík, E. El-Fakahany, S. Tuček, 2002, The Journal of pharmacology and experimental therapeutics.

On direct and subdirect product decompositions of partially ordered sets

J. Jakubík, 2002 .

Direct limits of cyclically ordered groups

J. Jakubík, Gabriela Pringerová, 1994 .

Synthesis of N-Substituted Piperidine Salts as Potential Muscarinic Ligands for Alzheimer's Applications

J. Jakubík, A. Randáková, John Boulos, 2013 .

The operational model of allosteric modulation of pharmacological agonism

J. Jakubík, E. El-Fakahany, V. Doležal, 2020, Scientific Reports.

Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators

J. Jakubík, E. El-Fakahany, V. Doležal, 2019, PloS one.

Applications and limitations of fitting of the operational model to determine relative efficacies of agonists

J. Jakubík, V. Rudajev, E. El-Fakahany, 2019, Scientific Reports.

Novel M 2 -selective, G i -biased agonists of muscarinic acetylcholine receptors

J. Jakubík, E. El-Fakahany, A. Randáková, 2020 .

Effects of an agonist, allosteric modulator, and antagonist on guanosine-gamma-[35S]thiotriphosphate binding to liposomes with varying muscarinic receptor/Go protein stoichiometry.

T. Haga, J. Jakubík, S. Tuček, 1998, Molecular pharmacology.

Two populations of muscarinic binding sites in the chick heart distinguished by affinities for ligands and selective inactivation

J. Jakubík, S. Tuček, 1994, British journal of pharmacology.

Classical and atypical agonists activate M1 muscarinic acetylcholine receptors through common mechanisms.

J. Jakubík, V. Rudajev, E. El-Fakahany, 2015, Pharmacological research.

Long-Term Activation upon Brief Exposure to Xanomleline Is Unique to M1 and M4 Subtypes of Muscarinic Acetylcholine Receptors

J. Jakubík, E. El-Fakahany, V. Doležal, 2014, PloS one.

Critical re-evaluation of the slope factor of the operational model of agonism

J. Jakubík, 2021 .

Allosteric Modulation of Muscarinic Receptors by Cholesterol, Neurosteroids and Neuroactive Steroids

J. Jakubík, A. Randáková, E. Kudova, 2022, International journal of molecular sciences.

Steroids as the novel class of high-affinity allosteric modulators of muscarinic receptors

J. Jakubík, V. Doležal, A. Randáková, 2021 .

Insights into the operational model of agonism of receptor dimers

J. Jakubík, A. Randáková, Alena Randáková, 2022, Expert opinion on drug discovery.

Lipid-Based Diets Improve Muscarinic Neurotransmission in the Hippocampus of Transgenic APPswe/PS1dE9 Mice.

H. Tanila, J. Jakubík, V. Rudajev, 2015, Current Alzheimer research.

Lateral completion of a projectable lattice ordered group

J. Jakubík, 2000 .

Radioligand Binding at Muscarinic Receptors

J. Jakubík, E. El-Fakahany, 2016 .

Graph Automorphisms and Cells of Lattices

J. Jakubík, 2003 .

Claire Kramsch, Language as Symbolic Power, Cambridge University Press, 2021, pp. 279

J. Jakubík, 2022, ANNALES UNIVERSITATIS PAEDAGOGICAE CRACOVIENSIS. STUDIA LINGUISTICA.

Modulation of Muscarinic Signalling in the Central Nervous System by Steroid Hormones and Neurosteroids

J. Jakubík, A. Randáková, E. Szczurowska, 2022, International journal of molecular sciences.

Finger tendon rupture following local application of triamcinolone-acetonide (Kenalog A-40).

J. Jakubík, 1981, Acta chirurgiae plasticae.

Comparative susceptibility of rabbits, rats, mice and pigs to infection with Aujeszky diseases virus (ADV) in the development of an efficacy test for ADV vaccines.

J. Jakubík, 2010, Zentralblatt fur Veterinarmedizin. Reihe B. Journal of veterinary medicine. Series B.

Muscarinic Receptor: From Structure to Animal Models

J. Jakubík, J. Myslivecek, 2016, Neuromethods.

On subgroups of a pseudo lattice ordered group

J. Jakubík, 1970 .

Allosteric Modulation of Muscarinic Acetylcholine Receptors

Jan Jakubík, Esam E. El-Fakahany, J. Jakubík, 2010, Pharmaceuticals.

Positive cooperativity of acetylcholine and other agonists with allosteric ligands on muscarinic acetylcholine receptors.

L. Bačáková, J. Jakubík, E. El-Fakahany, 1997, Molecular pharmacology.

Evidence for a Tandem Two-site Model of Ligand Binding to Muscarinic Acetylcholine Receptors*

J. Jakubík, E. El-Fakahany, S. Tuček, 2000, The Journal of Biological Chemistry.

Regulation of signal transduction at M2 muscarinic receptor.

A. Krejci, J. Říčný, J. Jakubík, 2004, Physiological research.

Subtype‐selective inhibition of [methyl‐3H]‐N‐methylscopolamine binding to muscarinic receptors by α‐truxillic acid esters

J. Jakubík, S. Tuček, T. Elbert, 1999, British journal of pharmacology.

Current Advances in Allosteric Modulation of Muscarinic Receptors

J. Jakubík, E. El-Fakahany, 2020, Biomolecules.

Microsoft Word-22167934-file00

J. Jakubík, E. El-Fakahany, V. Doležal, 2014 .

Outline of therapeutic interventions with muscarinic receptor-mediated transmission.

J. Jakubík, V. Rudajev, E. El-Fakahany, 2014, Physiological research.

Importance and prospects for design of selective muscarinic agonists.

E. Machová, J. Jakubík, V. Doležal, 2008, Physiological research.

Roles of external loops of muscarinic receptors in interactions between N-methylscopolamine and allosteric modulators

J. Jakubík, M. Lysíková, Stanislav Tuek, 2004 .

Use of a Sandwich Enzyme-linked Immunosorbent Assay Strategy to Study Mechanisms of G Protein-coupled Receptor Assembly*

J. Wess, J. Jakubík, 1999, The Journal of Biological Chemistry.

Positive allosteric interactions on cardiac muscarinic receptors: effects of chemical modifications of disulphide and carboxyl groups.

J. Jakubík, S. Tuček, 1995, European journal of pharmacology.

Neurosteroids and steroid hormones are allosteric modulators of muscarinic receptors

J. Jakubík, V. Doležal, A. Randáková, 2021, Neuropharmacology.

Functionally selective and biased agonists of muscarinic receptors.

J. Jakubík, A. Randáková, Alena Randáková, 2021, Pharmacological research.

Colostral immunity in piglets from sows vaccinated with inactivated Aujeszky disease virus vaccine

J. Jakubík, G. Wittmann, 2005, Archives of Virology.

Cell-mediated immunity in Aujeszky disease virus infected pigs

J. Jakubík, G. Wittmann, G. Bartenbach, 1976, Archives of Virology.

Neutralizing antibody titres in pig serum after revaccination with an inactivated Aujeszky disease virus (ADV) vaccine.

J. Jakubík, G. Wittmann, 2010, Zentralblatt fur Veterinarmedizin. Reihe B. Journal of veterinary medicine. Series B.

[Early stages of immunity following vaccination of piglets with an inactivated Aujezsky's virus vaccine].

J. Jakubík, G. Wittmann, 2010, Zentralblatt fur Veterinarmedizin. Reihe B. Journal of veterinary medicine. Series B.

Vaccination experiments in cattle with a live and with an inactivated Aujeszky's disease virus vaccine.

P. Rondhuis, J. Jakubík, J. Akkermans, 2010, Zentralblatt fur Veterinarmedizin. Reihe B. Journal of veterinary medicine. Series B.

Challenge experiments with the virus of Aujeszky's disease in non-vaccinated and vaccinated sheep.

P. Rondhuis, J. Jakubík, J. Akkermans, 2010, Zentralblatt fur Veterinarmedizin. Reihe B. Journal of veterinary medicine. Series B.

Fusion with Promiscuous Gα16 Subunit Reveals Signaling Bias at Muscarinic Receptors

J. Jakubík, A. Randáková, P. Zimčík, 2021, International journal of molecular sciences.

Multiplication and distribution of Aujeszky's disease (pseudorabies) virus in vaccinated and non-vaccinated pigs after intranasal infection

J. Jakubík, R. Ahl, G. Wittmann, 1980, Archives of Virology.

On homology modeling of the M2 muscarinic acetylcholine receptor subtype

Jan Jakubik, Alena Randáková, Vladimír Dolezal, 2013, Journal of Computer-Aided Molecular Design.

[Early occurrence of Dupuytren's contracture].

J. Jakubík, 1965, Acta chirurgiae orthopaedicae et traumatologiae Cechoslovaca.

On archimedean MV-algebras

Ján Jakubík, J. Jakubík, 1998 .

Allosteric Modulation of GPCRs of Class A by Cholesterol

J. Jakubík, E. El-Fakahany, 2021, International journal of molecular sciences.

Activation of muscarinic acetylcholine receptors via their allosteric binding sites.

L. Bačáková, V. Lisa, J. Jakubík, 1996, Proceedings of the National Academy of Sciences of the United States of America.

Role of Receptor Protein and Membrane Lipids in Xanomeline Wash-Resistant Binding to Muscarinic M1 Receptors

J. Jakubík, E. El-Fakahany, S. Tuček, 2004, Journal of Pharmacology and Experimental Therapeutics.

Subtype selectivity of the positive allosteric action of alcuronium at cloned M1-M5 muscarinic acetylcholine receptors.

L. Bačáková, J. Jakubík, E. El-Fakahany, 1995, The Journal of pharmacology and experimental therapeutics.

Positive effects of allosteric modulators on the binding properties and the function of muscarinic acetylcholine receptors

J. Jakubík, E. El-Fakahany, S. Tuček, 1998, Journal of Physiology-Paris.

Radical classes of generalized Boolean algebras

J. Jakubík, 1998 .

On some types of radical classes

J. Jakubík, 2008 .

Generalized Cardinal Properties of Lattices and Lattice Ordered Groups

J. Jakubík, 2004 .

Torsion classes of Specker lattice ordered groups

J. Jakubík, 2002 .

RADICAL CLASSES OF DISTRIBUTIVE LATTICES HAVING THE LEAST ELEMENT

J. Jakubík, 2002 .

Radical classes of MV-algebras

J. Jakubík, 1999 .

On K -radicals classes of lattice ordered groups

J. Jakubík, 1983 .

Agonist-Specific Conformations of the M2 Muscarinic Acetylcholine Receptor Assessed by Molecular Dynamics

Alena Randaková, Dominik Nelic, Vladimír Doležal, 2020, J. Chem. Inf. Model..

Subtype Differences in Pre-Coupling of Muscarinic Acetylcholine Receptors

Jan Jakubík, Alena Randáková, Esam E. El-Fakahany, 2011, PloS one.

Guanidine Derivatives: How Simple Structural Modification of Histamine H3R Antagonists Has Led to the Discovery of Potent Muscarinic M2R/M4R Antagonists

H. Stark, M. Bajda, J. Jakubík, 2021, ACS chemical neuroscience.

Negative cooperativity in binding of muscarinic receptor agonists and GDP as a measure of agonist efficacy

J. Jakubík, E. El-Fakahany, V. Doležal, 2011, British journal of pharmacology.

Synthesis of novel and functionally selective non‐competitive muscarinic antagonists as chemical probes

J. Jakubík, A. Randáková, John Boulos, 2018, Chemical biology & drug design.

Critical re-evaluation of the slope factor of the operational model of agonism: Do not exponentiate operational efficacy

J. Jakubík, 2021, bioRxiv.

Applications and limitations of fitting of the operational model to determine relative efficacies of agonists

J. Jakubík, V. Rudajev, E. El-Fakahany, 2019, Scientific Reports.

Novel M2‐selective, Gi‐biased agonists of muscarinic acetylcholine receptors

J. Jakubík, E. El-Fakahany, V. Doležal, 2020, British journal of pharmacology.

Wash-Resistantly Bound Xanomeline Inhibits Acetylcholine Release by Persistent Activation of Presynaptic M2 and M4 Muscarinic Receptors in Rat Brain

E. Machová, J. Jakubík, E. El-Fakahany, 2007, Journal of Pharmacology and Experimental Therapeutics.

Allosteric Modulation of Muscarinic Receptors

J. Jakubík, E. El-Fakahany, 2016 .

On the theory of partially ordered groups

J. Jakubík, 1961 .

Dataset Enhancement in Hair Follicle Detection: ESENSEI Challenge

Jan Jakubik, J. Jakubík, 2018, FedCSIS.

On a type of distributivity of lattice ordered groups

J. Jakubík, 2014 .

Generalized Specker lattice-ordered groups and two types of distributivity

J. Jakubík, J. Lihová, 2013 .

Higher degrees of distributivity in complete generalized MV-algebras

J. Jakubík, 2011 .

On the distributive radical of an Archimedean lattice-ordered group

J. Jakubík, 2009 .

Weak homogeneity of lattice ordered groups

J. Jakubík, 2007 .

Weak homogeneity and Pierce’s theorem for MV-algebras

J. Jakubík, 2006 .

Weak % MathType!Translator!2!1!AMS LaTeX.tdl!TeX -- AMS-LaTeX! % MathType!MTEF!2!1!+- % feaafeart1ev1aqatCvAUfeBSjuyZL2yd9gzLbvyNv2CaerbuLwBLn % hiov2DGi1BTfMBaeXatLxBI9gBaerbd9wDYLwzYbItLDharqqtubsr % 4rNCHbGeaGqiVu0Je9sqqrpepC0xbbL8F4rqqrFfpeea0xe9Lq-Jc9 % vqaqpepm0xbba9pwe9Q8fs0-yqaqpepae9pg0Firp

Ján Jakubík, J. Jakubík, 2005 .

On vector lattices of elementary Carathéodory functions

J. Jakubík, 2005 .

On the Schröder-Bernstein problem for abelian lattice ordered groups and for MV-algebras

Jan Jakubik, J. Jakubík, 2004, Soft Comput..

Higher Degrees of Distributivity in MV-Algebras

J. Jakubík, 2003 .

Complete Distributivity of Lattice Ordered Groups and of Vector Lattices

J. Jakubík, 2001 .

Sequential Convergences on Boolean Algebras Defined by Systems of Maximal Filters

J. Jakubík, R. Fric, 2001 .

Cantor-Bernstein theorem for MV-algebras

J. Jakubík, 1999 .

Conditionally orthogonally complete l-groups

J. Jakubík, 1975 .

Binding of N-methylscopolamine to the extracellular domain of muscarinic acetylcholine receptors

J. Jakubík, E. El-Fakahany, V. Doležal, 2017, Scientific Reports.

Good and Bad Infinitesimals, and States on Pseudo MV-algebras

Anatolij Dvurecenskij, Antonio di Nola, Jan Jakubik, 2004, Order.

Relatively uniform convergences in archimedean lattice ordered groups

J. Jakubík, Stefan Cernák, 2010 .

Affine completeness and wreath product decompositions of lattice ordered group

J. Jakubík, 2008 .

Isometries of generalized MV-algebras

J. Jakubík, 2007 .

Subdirect decompositions and the radical of a generalized Boolean algebra extension of a lattice ordered group

J. Jakubík, 2006 .

Strong Projectability of Lattice Ordered Groups

J. Jakubík, 2005 .

On Free MV-Algebras

J. Jakubík, 2003 .

Convex Chains in a Pseudo MV-Algebra

J. Jakubík, 2003 .

On Product MV-Algebras

Ján Jakubík, J. Jakubík, 2002 .

On intervals and isometries of MV-algebras

J. Jakubík, 2002 .

Distinguished Completion of a Direct Product of Lattice Ordered Groups

J. Jakubík, 2001 .

State-Homomorphisms on MV-Algebras

J. Jakubík, 2001 .

On cut completions of abelian lattice ordered groups

J. Jakubík, 2000 .

Affine completness of projectable lattice ordered groups

J. Jakubík, Mária Csontóová, 1998 .

Isomorphisms of direct products of lattice-ordered groups

J. Jakubík, 2004 .

On absolute retracts and absolute convex retracts in some classes of l-groups

J. Jakubík, 2003 .

Affine completeness of complete lattice ordered groups

J. Jakubík, 1995 .

Closure operators on the lattice of radical classes of lattice ordered groups

J. Jakubík, 1988 .

Radical subgroups of lattice ordered groups

J. Jakubík, 1986 .

On value selectors and torsion classes of lattice ordered groups

J. Jakubík, 1981 .

Prime selectors and torsion classes of lattice ordered groups

J. Jakubík, 1981 .

Isometries of lattice ordered groups

J. Jakubík, 1980 .

MAXIMAL COMPLETION OF A PSEUDO MV – ALGEBRA

J. Jakubík, 2022 .

Graph automorphisms of a finite modular lattice

J. Jakubík, 1999 .

Convex isomorphisms of directed multilattices

J. Jakubík, Mária Csontóová, 1993 .

On some types of kernels of a convergence $l$-group

J. Jakubík, 1989 .

Convergences and complete distributivity of lattice ordered groups

J. Jakubík, 1988 .

Sequential convergences in Boolean algebras

J. Jakubík, 1988 .

Graph isomorphisms of semimodular lattices

J. Jakubík, 1985 .

On the lattice of additive hereditary properties of finite graphs

J. Jakubík, Ján Jakub́ık, 2002 .

Complete generators and maximal completions of MV-algebras

J. Jakubík, 1998 .

Projectability and Splitting Property of Lattice Ordered Groups

J. Jakubík, 2003 .

On σ-complete lattice ordered groups

J. Jakubík, 2016 .

Formations of lattice ordered groups and of GMV-algebras

J. Jakubík, 2008 .