A. Heim-Riether

发表

Fragment-based discovery of indole inhibitors of matrix metalloproteinase-13.

Xiang Li, Ingo Muegge, Hani S. Zaher, 2011, Journal of medicinal chemistry.

N-Arylsulfonyl-α-amino carboxamides are potent and selective inhibitors of the chemokine receptor CCR10 that show efficacy in the murine DNFB model of contact hypersensitivity.

D. Jeanfavre, N. Moss, Jiang-Ping Wu, 2016, Bioorganic & medicinal chemistry letters.

Lead optimization and structure-based design of potent and bioavailable deoxycytidine kinase inhibitors.

Alan G. E. Wilson, M. Shen, T. Stouch, 2009, Bioorganic & medicinal chemistry letters.

Exploration of cathepsin S inhibitors characterized by a triazole P1-P2 amide replacement.

E. Hickey, N. Moss, Yancey D. Ward, 2012, Bioorganic & medicinal chemistry letters.

SAR studies of non-zinc-chelating MMP-13 inhibitors: improving selectivity and metabolic stability.

J. Proudfoot, N. Moss, N. Farrow, 2010, Bioorganic & medicinal chemistry letters.

Tandem CH-Activation-Imine-Formation Reaction: A New Route to Imidazo[2,1-a]phthalazines

A. Heim-Riether, K. R. Gipson, 2009 .

A novel method for the synthesis of imidazo[5,1-f][1,2,4]triazin-4(3H)-ones.

A. Heim-Riether, J. Healy, 2005, The Journal of organic chemistry.

5-Fluorocytosine derivatives as inhibitors of deoxycytidine kinase.

Alan G. E. Wilson, M. Shen, D. Augeri, 2009, Bioorganic & medicinal chemistry letters.

Indole Inhibitors of MMP-13 for Arthritic Disorders

Qiang Zhang, I. Muegge, J. Proudfoot, 2021, ACS omega.

Improving potency and selectivity of a new class of non-Zn-chelating MMP-13 inhibitors.

Zhaoming Xiong, B. Farmer, Qiang Zhang, 2009, Bioorganic & medicinal chemistry letters.