S. Kudalkar

发表

A role for catalase-peroxidase large loop 2 revealed by deletion mutagenesis: control of active site water and ferric enzyme reactivity.

D. Goodwin, Ngolui René Fuanta, S. Kudalkar, 2015, Biochemistry.

Molecular and cellular studies evaluating a potent 2-cyanoindolizine catechol diether NNRTI targeting wildtype and Y181C mutant HIV-1 reverse transcriptase.

W. L. Jorgensen, K. Anderson, K. Frey, 2019, Bioorganic & medicinal chemistry letters.

Covalent inhibitors for eradication of drug-resistant HIV-1 reverse transcriptase: From design to protein crystallography

W. L. Jorgensen, K. Anderson, A. Chan, 2017, Proceedings of the National Academy of Sciences.

( R)- N-(1-Methyl-2-hydroxyethyl)-13-( S)-methyl-arachidonamide (AMG315): A Novel Chiral Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes.

K. Mackie, L. Marnett, A. Hohmann, 2018, Journal of medicinal chemistry.

Long‐acting and extended‐release implant and nanoformulations with a synergistic antiretroviral two‐drug combination controls HIV‐1 infection in a humanized mouse model

W. L. Jorgensen, K. Anderson, W. Saltzman, 2021, Bioengineering & translational medicine.

Reply to Pandey et al.: Understanding the efficacy of a potential antiretroviral drug candidate in humanized mouse model of HIV infection

W. L. Jorgensen, K. Anderson, W. Saltzman, 2018, Proceedings of the National Academy of Sciences.

Exploring ABOBEC3A and APOBEC3B substrate specificity and their role in HPV positive head and neck cancer

T. Schrank, N. Issaeva, W. Yarbrough, 2022, iScience.

APOBEC mutagenesis and selection for NFE2L2 contribute to the origin of lung squamous-cell carcinoma

J. Townsend, B. G. Rothberg, Vincent L. Cannataro, 2022, Lung cancer.

Substrate-selective activation of COX-2 by AM-8138

L. Marnett, C. Rouzer, S. Nikas, 2015 .

Potent Noncovalent Inhibitors of the Main Protease of SARS-CoV-2 from Molecular Sculpting of the Drug Perampanel Guided by Free Energy Perturbation Calculations

Farren J. Isaacs, Scott J. Miller, W. L. Jorgensen, 2021, ACS central science.

Enhancing the peroxidatic activity of KatG by deletion mutagenesis.

D. Goodwin, S. Kudalkar, Yongjiang Li, 2012, Journal of inorganic biochemistry.

Roles of Large Loops in Catalytic Versatility of Catalase-Peroxidases: Significance of Peripheral Structures in Improvising Enzyme Functions

S. Kudalkar, Shalley N. Kudalkar, 2012 .

From in silico hit to long-acting late-stage preclinical candidate to combat HIV-1 infection

W. L. Jorgensen, K. Anderson, W. Saltzman, 2017, Proceedings of the National Academy of Sciences.

Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV.

W. L. Jorgensen, K. Anderson, W. Saltzman, 2019, Antiviral research.

Structure-Guided Identification of DNMT3B Inhibitors.

Ana S. Newton, W. L. Jorgensen, K. Anderson, 2020, ACS medicinal chemistry letters.

Structural and Preclinical Studies of Computationally Designed Non-Nucleoside Reverse Transcriptase Inhibitors for Treating HIV infection

W. L. Jorgensen, K. Anderson, Priti Kumar, 2017, Molecular Pharmacology.

Assay of Endocannabinoid Oxidation by Cyclooxygenase-2.

L. Marnett, P. Kingsley, S. Kudalkar, 2016, Methods in molecular biology.

13-Methylarachidonic Acid Is a Positive Allosteric Modulator of Endocannabinoid Oxygenation by Cyclooxygenase*

Shu Xu, Lawrence J. Marnett, Alexandros Makriyannis, 2015, The Journal of Biological Chemistry.

DRONE: Direct Tracking of DNA Cytidine Deamination and Other DNA Modifying Activities.

K. Anderson, N. Bertoletti, S. Kudalkar, 2018, Analytical chemistry.

Action at a Distance

Anna L. Blobaum, L. Marnett, Shu Xu, 2015, The Journal of Biological Chemistry.