Krzysztof Szafrański

发表

Target-based drug discovery through inversion of quantitative structure-drug-property relationships and molecular simulation: CA IX-sulphonamide complexes

C. Supuran, Petar Žuvela, T. Bączek, 2018, Journal of enzyme inhibition and medicinal chemistry.

Novel 5-Substituted 2-(Aylmethylthio)-4-chloro-N-(5-aryl-1,2,4-triazin-3-yl)benzenesulfonamides: Synthesis, Molecular Structure, Anticancer Activity, Apoptosis-Inducing Activity and Metabolic Stability

T. Bączek, Szymon Ulenberg, Mariusz Belka, 2016, Molecules.

Novel 2-benzylthio-5-(1,3,4-oxadiazol-2-yl)benzenesulfonamides with anticancer activity: Synthesis, QSAR study, and metabolic stability.

T. Bączek, Katarzyna Macur, Mariusz Belka, 2017, European journal of medicinal chemistry.

Novel 2-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)-1-(1,3,5-triazin-2-ylamino)guanidine derivatives: Inhibition of human carbonic anhydrase cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII, anticancer activity, and molecular modeling studies.

C. Supuran, T. Bączek, A. Angeli, 2018, European journal of medicinal chemistry.

New 2-[(4-Amino-6-N-substituted-1,3,5-triazin-2-yl)methylthio]-N-(imidazolidin-2-ylidene)-4-chloro-5-methylbenzenesulfonamide Derivatives, Design, Synthesis and Anticancer Evaluation

E. Grzybowska, A. Kawiak, Krzysztof Szafrański, 2022, International journal of molecular sciences.

Synthesis, QSAR studies, and metabolic stability of novel 2‐alkylthio‐4‐chloro‐N‐(5‐oxo‐4,5‐dihydro‐1,2,4‐triazin‐3‐yl)benzenesulfonamide derivatives as potential anticancer and apoptosis‐inducing agents

T. Bączek, Mariusz Belka, A. Kawiak, 2017, Chemical biology & drug design.

Syntheses of Novel 4-Substituted N-(5-amino-1H-1,2,4-triazol-3-yl)pyridine-3-sulfonamide Derivatives with Potential Antifungal Activity

Krzysztof Szafrański, J. Sławiński, A. Kędzia, 2017, Molecules.

Carbonic anhydrase inhibitors. Synthesis of heterocyclic 4-substituted pyridine-3-sulfonamide derivatives and their inhibition of the human cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII.

C. Supuran, D. Vullo, Krzysztof Szafrański, 2013, European journal of medicinal chemistry.

Synthesis of a new series of N⁴-substituted 4-(2-aminoethyl)benzenesulfonamides and their inhibitory effect on human carbonic anhydrase cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII.

C. Supuran, D. Vullo, Krzysztof Szafrański, 2014, European journal of medicinal chemistry.

Inhibition studies of Brucella suis β-carbonic anhydrases with a series of 4-substituted pyridine-3-sulphonamides

C. Supuran, Angela Meccariello, M. Ceruso, 2017, Journal of enzyme inhibition and medicinal chemistry.

Comparison of the Sulfonamide Inhibition Profiles of the b- and c-Carbonic Anhydrases from the Pathogenic Bacterium Burkholderia pseudomallei

C. Supuran, Angela Meccariello, M. Ceruso, 2022 .

Synthesis of 2-alkylthio-N-(quinazolin-2-yl)benzenesulfonamide derivatives: anticancer activity, QSAR studies, and metabolic stability

T. Bączek, Mariusz Belka, A. Kawiak, 2018, Monatshefte für Chemie - Chemical Monthly.

Synthesis of Novel 1-(4-Substituted pyridine-3-sulfonyl)-3-phenylureas with Potential Anticancer Activity

Krzysztof Szafrański, J. Sławiński, 2015, Molecules.

Synthesis, Antitumor Evaluation, Molecular Modeling and Quantitative Structure–Activity Relationship (QSAR) of Novel 2-[(4-Amino-6-N-substituted-1,3,5-triazin-2-yl)methylthio]-4-chloro-5-methyl-N-(1H-benzo[d]imidazol-2(3H)-ylidene)Benzenesulfonamides

A. Kawiak, Krzysztof Szafrański, B. Żołnowska, 2020, International journal of molecular sciences.

Synthesis, Molecular Structure, Metabolic Stability and QSAR Studies of a Novel Series of Anticancer N-Acylbenzenesulfonamides

T. Bączek, Mariusz Belka, A. Kawiak, 2015, Molecules.

Novel 2-(2-alkylthiobenzenesulfonyl)-3-(phenylprop-2-ynylideneamino)guanidine derivatives as potent anticancer agents - Synthesis, molecular structure, QSAR studies and metabolic stability.

Jarosław Chojnacki, Szymon Ulenberg, Tomasz Bączek, 2017, European journal of medicinal chemistry.

Synthesis, molecular structure, and metabolic stability of new series of N'-(2-alkylthio-4-chloro-5-methylbenzenesulfonyl)-1-(5-phenyl-1H-pyrazol-1-yl)amidine as potential anti-cancer agents.

T. Bączek, Szymon Ulenberg, A. Kawiak, 2018, European journal of medicinal chemistry.

Novel 5-Substituted 2-(Aylmethylthio)-4-chloro-N-(5-aryl-1,2,4-triazin-3-yl)benzenesulfonamides: Synthesis, Molecular Structure, Anticancer Activity, Apoptosis-Inducing Activity and Metabolic Stability

T. Bączek, Szymon Ulenberg, Mariusz Belka, 2016, Molecules.