I. Kondratov

发表

Last of the gem-Difluorocycloalkanes: Synthesis and Characterization of 2,2-Difluorocyclobutyl-Substituted Building Blocks.

N. A. Tolmacheva, C. Daniliuc, O. Grygorenko, 2019, The Journal of organic chemistry.

4‐(Di‐/Trifluoromethyl)‐2‐heterabicyclo[2.1.1]hexanes: Advanced Fluorinated Phenyl Isosteres and Proline analogues

C. Daniliuc, Oleg M. Michurin, O. Grygorenko, 2021 .

Synthesis and Physicochemical Properties of 3‐Fluorocyclobutylamines

C. Daniliuc, G. Haufe, S. Zozulya, 2015 .

Straightforward hit identification approach in fragment-based discovery of bromodomain-containing protein 4 (BRD4) inhibitors.

Yurii S. Moroz, V. Hurmach, S. Zozulya, 2018, Bioorganic & Medicinal Chemistry.

Synthesis and reactions of ω-CF3O-substituted aliphatic sulfonyl chlorides

O. Grygorenko, I. Kondratov, Alexey V. Dobrydnev, 2021, Journal of Fluorine Chemistry.

GABA Analogues and Related Mono-/Bifunctional Building Blocks Derived from the Fluorocyclobutane Scaffold

G. Haufe, O. Grygorenko, I. Kondratov, 2020 .

Synthesis and Physical‐Chemical Properties of cis‐ and trans‐1‐Amino‐3‐fluoro‐3‐methylcyclobutanecarboxylic Acids

C. Daniliuc, G. Haufe, Anton V. Chernykh, 2016 .

Synthesis and physical chemical properties of CF3O-containg secondary amines – perspective building blocks for Drug Discovery

C. Mück‐Lichtenfeld, C. Daniliuc, G. Haufe, 2022, Journal of Fluorine Chemistry.

"Reported, but still unknown." A closer look into 3,4-bis- and 3,4,5-tris(trifluoromethyl)pyrazoles.

A. Tolmachev, O. Shishkin, I. Kondratov, 2012, The Journal of organic chemistry.

Large library docking for novel SARS-CoV-2 main protease non-covalent and covalent inhibitors

Yurii S. Moroz, J. Irwin, B. Shoichet, 2022, bioRxiv.

New synthetic approach to mevalonate and mevaldate fluoroanalogues

O. V. Manoilenko, I. Kondratov, I. Gerus, 2007 .

Synthesis and physical chemical properties of 2-amino-4-(trifluoromethoxy)butanoic acid - a CF3O-containing analogue of natural lipophilic amino acids.

C. Daniliuc, G. Haufe, M. Kliachyna, 2017, Organic & biomolecular chemistry.

Synthesis of Fused Pyridine Carboxylates by Reaction of β-Alkoxyvinyl Glyoxylates with Amino Heterocycles

A. Tolmachev, O. Grygorenko, I. Kondratov, 2020, Synthesis.

Synthesis and Properties of Polyfunctional Cyclic β-Alkoxy-α,β-Unsaturated Ketones Based on 4-Methylene-1,3-dioxolanes

I. Kondratov, I. Gerus, V. Kukhar, 2018, European Journal of Organic Chemistry.

Phenoxymethyl 1,3-oxazoles and 1,2,4-oxadiazoles as potent and selective agonists of free fatty acid receptor 1 (GPR40).

M. Platonov, S. Zozulya, I. Kondratov, 2015, Bioorganic & medicinal chemistry letters.

Synthesis, physico-chemical properties and microsomal stability of compounds bearing aliphatic trifluoromethoxy group

G. Haufe, M. Kliachyna, O. Grygorenko, 2020, Journal of Fluorine Chemistry.

Diels-Alder Reaction in the Synthesis of Fluorinated (Hetero)Aromatic Compounds

G. Haufe, I. Kondratov, Nataliya A. Tolmachova, 2018, European Journal of Organic Chemistry.

Synthesis of Trifluoromethyl-Containing Polysubstituted Aromatic Compounds by Diels–Alder Reaction of Ethyl 3-Benzamido-2-oxo-6-(trifluoromethyl)-2H-pyran-5-carboxylate

C. Daniliuc, G. Haufe, I. Kondratov, 2015 .

Diels–Alder Reaction of Ethyl 3-Benzamido-2-oxo-6-(trifluoromethyl)-2H-pyran-5-carboxylate with Alkoxyalkenes as an Effective Approach to Trifluoromethyl-Containing 3-Aminobenzoic Acid Derivatives

C. Daniliuc, G. Haufe, I. Kondratov, 2014 .

Reactions of β-alkoxyvinyl polyfluoroalkyl ketones with ethyl isocyanoacetate and its use for the synthesis of new polyfluoroalkyl pyrroles and pyrrolidines.

G. Haufe, I. Kondratov, K. Bergander, 2012, Organic & biomolecular chemistry.

Radical Reactions of Alkyl 2-Bromo-2,2-difluoroacetates with Vinyl Ethers: "Omitted" Examples and Application for the Synthesis of 3,3-Difluoro-GABA.

C. Daniliuc, G. Haufe, I. Kondratov, 2015, The Journal of organic chemistry.

Reaction of β-alkoxyvinyl α-ketoesters with acyclic NCN binucleophiles – Scalable approach to novel functionalized pyrimidines

A. Tolmachev, O. Grygorenko, I. Kondratov, 2019, Tetrahedron.

Conversions of 2-(2-Oxo Cyclohexylcarbonyl)Benzoic Acid Derivatives to Pyrazolo[ [5] , [1] , [2] , [3] , [4] , [5] , [6] , [7] , [8] , [9] , [10] ]Isoindole and Pyrimidine Rings

I. Kondratov, O. Pokholenko, Z. Voitenko, 2005 .

Synthesis of diverse pyrazole-4-sulfonyl chlorides starting from 2-(benzylthio)malonaldehyde

I. Kondratov, P. A. Sokolyuk, Olexiy V. Gavrylenko, 2015, Molecular Diversity.

Novel Synthetic Approaches to (Trifluoromethyl)triazoles

A. Tolmachev, I. Kondratov, Pavel K. Mykhailiuk, 2010 .

Synthesis, biological evaluation, and modeling studies of 1,3-disubstituted cyclobutane-containing analogs of combretastatin A4.

M. Platonov, C. Daniliuc, V. Hurmach, 2020, Journal of molecular structure.

New Derivatives of Trifluoroacetyl Acetaldehyde and Trifluoroaldol.

I. Kondratov, I. Gerus, V. Kukhar, 2005 .

Synthesis of New Pyrazolo[1,5‐a]pyrimidines by Reaction of β,γ‐Unsaturated γ‐Alkoxy‐α‐keto Esters with N‐Unsubstituted 5‐Aminopyrazoles.

I. Kondratov, Andrei O. Tolmachev, Oleksandr O. Stepaniuk, 2013 .

Straightforward synthesis of fluorinated amino acids by Michael addition of ethyl bromodifluoroacetate to α,β-unsaturated α-amino acid derivatives

C. Daniliuc, G. Haufe, I. Kondratov, 2018, Journal of Fluorine Chemistry.

Synthesis of New Pyrazolo[1,5-a]pyrimidines by Reaction of β,γ-Unsaturated γ-Alkoxy-α-keto Esters with N-Unsubstituted 5-Aminopyrazoles

I. Kondratov, Andrei O. Tolmachev, Oleksandr O. Stepaniuk, 2013 .

Reactions of ethyl triphenylphosphoranylideneacetate with fluorinated β-ketoaldehyde derivatives

I. Kondratov, I. Gerus, S. Vdovenko, 2007 .

Cyclobutyl-Containing Rigid Analogues of Threonine: Synthesis and Physical Chemical Properties.

C. Daniliuc, G. Haufe, Anton V. Chernykh, 2017, The Journal of organic chemistry.

(Het)aryl Difluoromethyl-Substituted β-Alkoxyenones: Synthesis and Heterocyclizations

O. Grygorenko, I. Kondratov, B. Vashchenko, 2020 .

How Accurately Can We Predict the Melting Points of Drug-like Compounds?

Igor V. Tetko, Luc Patiny, Abdullah M. Asiri, 2014, J. Chem. Inf. Model..

Synthesis of 1,3-bifunctional cyclobutane derivatives with α-CHF2/CF3 group – advanced building blocks for medicinal chemistry

O. Grygorenko, I. Kondratov, Anton A. Homon, 2022, Journal of Fluorine Chemistry.

Synthesis of diverse pyrazole-4-sulfonyl chlorides starting from 2-(benzylthio)malonaldehyde

I. Kondratov, P. A. Sokolyuk, Olexiy V. Gavrylenko, 2016, Molecular Diversity.

Synthesis of New δ-(Polyfluoroalkyl)-δ-hydroxy-α-amino Acids

N. A. Tolmacheva, G. Haufe, I. Kondratov, 2009 .

New derivatives of trifluoroacetyl acetaldehyde and trifluoroaldol

R. Fröhlich, I. Kondratov, I. Gerus, 2005 .

Computationally driven discovery of SARS-CoV-2 Mpro inhibitors: from design to experimental validation

Pengyu Y. Ren, J. Ponder, M. Sturlese, 2021, Chemical science.

3-((Hetera)cyclobutyl)azetidines, "Stretched" Analogues of Piperidine, Piperazine, and Morpholine: Advanced Building Blocks for Drug Discovery.

C. Daniliuc, O. Grygorenko, Anton V. Chernykh, 2019, The Journal of organic chemistry.

Synthesis of new fluorinated proline analogues from polyfluoroalkyl β-ketoacetals and ethyl isocyanoacetate.

C. Daniliuc, Anton V. Chernykh, I. Kondratov, 2018, Chemical Communications.

Synthesis of Trifluoromethyl-Containing Polysubstituted Aromatic Compounds by Diels—Alder Reaction of Ethyl 3-Benzamido-2-oxo-6-(trifluoromethyl)-2H-pyran-5-carboxylate.

C. Daniliuc, I. Kondratov, I. Gerus, 2015 .

Synthesis and physical chemical properties of 2-amino-4-(trifluoromethoxy)butanoic acid - a CF3O-containing analogue of natural lipophilic amino acids.

C. Daniliuc, G. Haufe, M. Kliachyna, 2017, Organic & biomolecular chemistry.

Synthesis of new fluorinated proline analogues from polyfluoroalkyl β-ketoacetals and ethyl isocyanoacetate.

C. Daniliuc, Anton V. Chernykh, I. Kondratov, 2018, Chemical communications.

Reactions of β-alkoxyvinyl polyfluoroalkyl ketones with ethyl isocyanoacetate and its use for the synthesis of new polyfluoroalkyl pyrroles and pyrrolidines.

R. Fröhlich, G. Haufe, I. Kondratov, 2012, Organic & biomolecular chemistry.

Large library docking for novel SARS‐CoV‐2 main protease non‐covalent and covalent inhibitors

Yurii S. Moroz, J. Irwin, B. Shoichet, 2023, Protein science : a publication of the Protein Society.

Reactions of cyclic β-alkoxyvinyl α-keto esters with heteroaromatic NCC-binucleophiles

A. Tolmachev, O. Grygorenko, I. Kondratov, 2020, Chemistry of Heterocyclic Compounds.