J. Lancelot

发表

Synthesis, inhibition of NO production and antiproliferative activities of some indole derivatives

S. Rault, A. Caruso, M. Sinicropi, 2009, Journal of enzyme inhibition and medicinal chemistry.

Synthesis and evaluation of cytotoxic activities of new guanidines derived from carbazoles.

Aurélien Lesnard, S. Rault, T. Cresteil, 2014, Bioorganic & medicinal chemistry letters.

(6-bromo-1,4-dimethyl-9H-carbazol-3-yl-methylene)-hydrazine (carbhydraz) acts as a GPER agonist in breast cancer cells.

C. Rosano, S. Rault, M. Maggiolini, 2015, Current topics in medicinal chemistry.

First synthesis of 5,6‐dihydro‐4H‐furo[3,2‐f]pyrrolo‐ [1,2‐a][1,4]diazepines

S. Rault, J. Lancelot, Xiao Feng, 1998 .

First synthesis of 4H‐furo[3,2‐f]pyrrolo[1,2‐a][1,4]diazepines

S. Rault, J. Lancelot, Xiao Feng, 1996 .

9-Ethyl-1,4-dimethyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-9H-carbazole and 6-bromo-9-ethyl-1,4-dimethyl-9H-carbazole.

S. Rault, A. Caruso, J. Lancelot, 2008, Acta crystallographica. Section C, Crystal structure communications.

3D‐QSAR and Docking Studies of Selective GSK‐3β Inhibitors. Comparison with a Thieno[2,3‐b]pyrrolizinone Derivative, a New Potential Lead for GSK‐3β Ligands.

Jana Sopkova-de Oliveira Santos, S. Rault, V. Lisowski, 2005 .

Efficient and Simple Synthesis of 6-Aryl-1,4-dimethyl-9H-carbazoles

S. Rault, A. Garofalo, A. Caruso, 2008, Molecules.

Synthesis and evaluation of antileukemic activity of 5-thienyl- or 5-(2-furyl)-2,3-dihydro-6,7-bis(hydroxymethyl)-1H-pyrrolizine bis(alkylcarbamates) and derivatives.

G. Mathé, J. Lancelot, M. Robba, 1989, Journal of Medicinal Chemistry.

Synthesis of Trans-thienyl-3-ethoxycarbonyl-2,3-dihydro[1,5]benzothiazepin-4(5h)-ones

C. Saturnino, J. Lancelot, P. D. Caprariis, 1992 .

A novel synthesis of methyl cis-(3-thienyl)glycidate with 2-aminothiophenol and the synthesis of [1,5]benzothiazepine derivatives

S. Rault, C. Saturnino, J. Lancelot, 1992 .

A NOVEL SYNTHESIS OF 2,3-DIHYDRO[1,5]BENZOTHIAZEPIN-4(5H)-ONES

J. Lancelot, P. D. Caprariis, M. Robba, 1992 .

Synthesis and pharmacological activities of some 2,3,4,5-tetrahydro[1,5]benzo[f]thiazepines.

S. Rault, C. Saturnino, G. de Martino, 1997, Farmaco.

Preparation of 2,3-Dihydro [1,5] Benzothiazepines and 2,3-Dihydro [1,5] Benzodiazepines

C. Saturnino, J. Lancelot, M. Robba, 1991 .

Efficient synthesis of halohydroxypyridines by hydroxydeboronation

S. Rault, A. Voisin, A. Bouillon, 2005 .

Synthesis of novel halopyridinylboronic acids and esters. Part 2: 2,4, or 5-Halopyridin-3-yl-boronic acids and esters

S. Rault, A. Bouillon, J. Lancelot, 2002 .

Synthesis of novel halo-oxybispyridines, new building blocks in cholinergic medicinal chemistry

Aurélien Lesnard, S. Rault, A. Voisin, 2006 .

Synthesis of novel pyrazolopyrrolopyrazines, potential analogs of sildenafil

S. Rault, P. Dallemagne, J. Lancelot, 2001 .

Four Partners, Three‐Step, One‐Pot Reaction for a Library of New 2‐Alkyl(dialkyl)aminoquinazolin‐4(3H)‐ones

Aurélien Lesnard, S. Rault, Rémi Legay, 2014 .

Pyrido [2, 3-h] pyrrolo [1, 2-a] quinoxalines

S. Rault, J. Lancelot, M. Robba, 1983 .

Synthesis of 5-arylthiazoles. Comparative study between Suzuki cross-coupling reaction and direct arylation

S. Rault, A. Bouillon, J. Lancelot, 2009 .

Efficient synthesis of 6H-pyrido [3,2-b] carbazole derivatives from 3-amino-1,4-dimethyl carbazole

S. Rault, J. Lancelot, M. Robba, 1987 .

Synthesis of [1]benzothieno[2,3‐e]pyrrolo[1,2a]pyrazines and related compounds

S. Rault, J. Lancelot, H. El-Kashef, 1986 .

Original one-pot microwave-promoted Hunsdiecker–Suzuki strategy: straightforward access to trans-1,2-diarylethenes from cinnamic acids

S. Rault, J. Lancelot, L. Kihel, 2007 .

Synthesis of novel halopyridinylboronic acids and esters. Part 4: Halopyridin-2-yl-boronic acids and esters are stable, crystalline partners for classical Suzuki cross-coupling☆

Jana Sopkova-de Oliveira Santos, S. Rault, A. Bouillon, 2003 .

In vitro anti-acanthamoeba action by thioureidic derivatives.

C. Saturnino, G. de Martino, Nicola Paesano, 2003, Farmaco.

A rapid and versatile synthesis of novel pyrimido[5,4-b]carbazoles

Aurélien Lesnard, S. Rault, Rémi Legay, 2009 .

13C Nmr study of 1,2,4-triazino[4,5-b]indazole derivatives

J. Lancelot, M. Robba, A. Rabaron, 1979 .

A new boronic-acid based strategy to synthesize 4(5)-(het)aryl-1H-imidazoles

Jana Sopkova-de Oliveira Santos, S. Rault, A. Bouillon, 2008 .

Pyrrolothienopyrimidines. Part 2. Synthesis of 4-Aminopyrrolo[1,2-a]thieno[3,2-e](and[2,3-e]) Pyrimidines.

S. Rault, J. Lancelot, M. Robba, 1986 .

PYRIDO(2,3-H)PYRROLO(1,2-A)QUINOXALINES

S. Rault, J. Lancelot, M. Robba, 1984 .

3-(Dipropylamino)-5-hydroxybenzofuro[2,3-f]quinazolin-1(2H)-one (DPA-HBFQ-1) plays an inhibitory role on breast cancer cell growth and progression.

S. Catalano, S. Andò, Aurélien Lesnard, 2016, European journal of medicinal chemistry.

Synthesis of 5‐Arylthiazoles. Comparative Study Between Suzuki Cross‐Coupling Reaction and Direct Arylation.

S. Rault, A. Bouillon, J. Lancelot, 2009 .

Synthesis of 2-TIPS-oxazol-5-ylboronic acid pinacol ester: efficient route to 5-(het)aryloxazoles via Suzuki cross-coupling reaction

S. Rault, A. Bouillon, J. Lancelot, 2009 .

Synthesis of novel triazolopyridylboronic acids and esters. Study of potential application to Suzuki-type reactions

S. Rault, A. Bouillon, J. Lancelot, 2004 .

A versatile synthesis of 2-amino-4H-pyrido[1,2-a][1,3,5]triazin-4-ones from 2-aminopyridines

S. Rault, J. Lancelot, Hugues Miel, 2002 .

Synthesis of new L-ascorbic ferulic acid hybrids.

S. Rault, J. Lancelot, M. Bazin, 2007, Molecules.

Novel oxybispyridylboronic acids: synthesis and study of their reactivity in Suzuki-type cross-coupling reactions

Aurélien Lesnard, S. Rault, A. Voisin, 2006 .

Novel Oxybispyridylboronic Acids: Synthesis and Study of Their Reactivity in Suzuki-Type Cross-Coupling Reactions.

Aurélien Lesnard, S. Rault, A. Voisin, 2007 .

2-bromo-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine, a new unexpected bifunctional building block for combinatorial chemistry.

S. Rault, A. Bouillon, J. Lancelot, 2003, Acta crystallographica. Section C, Crystal structure communications.

2-(6-bromopyridin-3-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane and (6-bromopyridin-3-yl)boronic acid, new bifunctional building blocks for combinatorial chemistry.

S. Rault, A. Bouillon, J. Lancelot, 2003, Acta crystallographica. Section C, Crystal structure communications.

Antiproliferative activity of some 1,4-dimethylcarbazoles on cells that express estrogen receptors: part I

S. Rault, C. Saturnino, A. Caruso, 2012, Journal of enzyme inhibition and medicinal chemistry.

Conformational Analysis and 3D QSAR Study on Novel Partial Agonists of 5‐HT3 Receptors

Ronan Bureau, S. Rault, R. Bureau, 1996 .

Synthesis of Some New Thieno[2,3-b][1,6]naphthyridines and Related Compounds

J. Lancelot, H. El-Kashef, A. Geies, 1993 .

Synthesis and preliminary biological evaluation of a new pyridocarbazole derivative covalently linked to a thymidine nucleoside as a potential targeted antitumoral agent. I.

O. Moltedo, C. Saturnino, D. Montesarchio, 2003, Chemical & pharmaceutical bulletin.

Synthesis and combinatorial approach of the reactivity of 6- and 7-arylthieno[3,2-d][1,3]oxazine-2,4-diones

S. Rault, J. Lancelot, Emmanuelle Braud, 2003 .

New Trimethoxybenzamides and Trimethoxyphenylureas Derived from Dimethylcarbazole as Cytotoxic Agents. Part I

Aurélien Lesnard, S. Rault, T. Cresteil, 2014 .

Synthesis and evaluation of cytotoxic activities of new guanidines derived from carbazoles.

Aurélien Lesnard, S. Rault, T. Cresteil, 2014, Bioorganic & medicinal chemistry letters.

NOVEL AND EFFICIENT SYNTHESIS OF 5,8-DIMETHYL-9H- CARBAZOL-3-OL VIA A HYDROXYDEBORONATION REACTION

S. Rault, A. Garofalo, A. Caruso, 2007 .

First tricyclic oximino derivatives as 5-HT3 ligands.

P Delagrange, P. Renard, B. Pfeiffer, 2001, Bioorganic & medicinal chemistry letters.

Solution-phase parallel synthesis of a 1140-member ureidothiophene carboxylic acid library.

S. Rault, J. Lancelot, Emmanuelle Braud, 2005, Journal of combinatorial chemistry.

Novel fused triheterocyclic systems. Synthesis of 6H-pyrido[2,3-c]pyrrolo[1,2-e]-1,2,5-triazepines

J. Lancelot, M. Robba, D. Ladurée, 1985 .

Pyrrolo [1', 2' : 1, 2] pyrazino [6, 5-b] carbazoles

S. Rault, J. Lancelot, M. Robba, 1983 .

NOVEL AND EFFICIENT ACCESS TO THIENO[3,4-c]CINNOLINES

S. Rault, J. Lancelot, H. El-Kashef, 2008 .

A New Boronic‐Acid Based Strategy to Synthesize 4(5)‐(Het)aryl‐1H‐imidazoles.

Jana Sopkova-de Oliveira Santos, S. Rault, A. Bouillon, 2008 .

Pyridazino [4,5-b] carbazole : Synthese et Etude des Spectres de Resonance Magnetique Nucleaire

J. Lancelot, M. Robba, H. Landelle, 1984 .

An efficient two-step total synthesis of the quaterpyridine nemertelline.

S. Rault, A. Voisin, A. Bouillon, 2003, The Journal of organic chemistry.

Molecular Modeling Studies Focused on 5-HT7 versus 5-HT1A Selectivity. Discovery of Novel Phenylpyrrole Derivatives with High Affinity for 5-HT7 Receptors

Aurélien Lesnard, Frédéric Fabis, Ronan Bureau, 2005, J. Chem. Inf. Model..

New fused pyrazines. Synthesis of pyrido[3′,2′:4,5]-thieno[2,3-e]pyrrolo[1,2-a]pyrazine derivatives

S. Rault, A. El-Dean, P. Dallemagne, 2000 .

Pyrrolothienopyrazines. IV. Synthese de derives de 1′amino-5 pyrrolo[1,2-a]thieno[2,3-e]pyrazine

S. Rault, J. Lancelot, M. Robba, 1987 .

New Fused Pyrazines. Synthesis of Pyrido[3′,2′:4,5]thieno[2,3‐e]pyrrolo[1,2‐a]pyrazine Derivatives.

S. Rault, A. El-Dean, P. Dallemagne, 2010 .

Pyrrolothienopyrazines. Part 4. Synthesis of Derivatives of 5-Aminopyrrolo(1,2-a)thieno(2,3-e)pyrazine.

S. Rault, J. Lancelot, M. Robba, 1987 .

ChemInform Abstract: Synthesis of Novel Halopyridinylboronic Acids and Esters. Part 2. 2,4, or 5-Halopyridin-3-yl-boronic Acids and Esters.

S. Rault, A. Bouillon, J. Lancelot, 2002 .

Synthesis of New Avenalumic Carboxamide Derivatives in the Ferulic Series

S. Rault, M. Jouanne, J. Lancelot, 2008 .

Molecular Design Based on 3D-Pharmacophore. Application to 5-HT4 Receptor

Ronan Bureau, Sylvain Rault, Cyril Daveu, 2002, J. Chem. Inf. Comput. Sci..

Molecular Design Based on 3D-Pharmacophore. Application to 5-HT Subtypes Receptors

Ronan Bureau, Sylvain Rault, Cyril Daveu, 2002, J. Chem. Inf. Comput. Sci..

Association of Two 3D QSAR Analyses. Application to the Study of Partial Agonist Serotonin-3 Ligands

Jana Sopkova-de Oliveira Santos, Ronan Bureau, Sylvain Rault, 2001, J. Chem. Inf. Comput. Sci..

Definition of a Pharmacophore for Partial Agonists of Serotonin 5-HT3 Receptors

Ronan Bureau, Sylvain Rault, Cyril Daveu, 1999, J. Chem. Inf. Comput. Sci..

Unusual behaviour of pyridinylboronic acids in the Petasis boronic Mannich reaction

Aurélien Lesnard, S. Rault, A. Voisin, 2006 .

2-(6-Bromopyridin-2-yl)-6-methyl-[1,3,6,2]dioxazaborocane, a new stable (pyridin-2-yl)boronic acid derivative.

S. Rault, A. Bouillon, J. Lancelot, 2004, Acta crystallographica. Section C, Crystal structure communications.

Design, synthesis and antiproliferative activity of tripentones: a new series of antitubulin agents.

P. Renard, S. Rault, V. Lisowski, 2001, Bioorganic & medicinal chemistry letters.

Pharmacophores of 5-HT4 Receptor Ligands: Experience of CERMN and Implications for Drug Design

Aurélien Lesnard, S. Rault, F. Dauphin, 2008 .