A. Guarna

发表

New Evidence of Similarity between Human and Plant Steroid Metabolism: 5α-Reductase Activity in Solanum malacoxylon

M. Serio, G. Danza, F. Rosati, 2003 .

Neat reaction of carboxylic acid methyl esters and amines for efficient parallel synthesis of scaffold amide libraries

A. Guarna, F. Machetti, Ilaria Bucelli, 2003 .

Enantiodivergent Chemoenzymatic Synthesis of 4-Hydroxypiperidine Alkaloids

A. Guarna, D. Scarpi, E. Occhiato, 2010 .

Synthetic Approaches towards Peptidomimetic Design

A. Trabocchi, A. Guarna, 2014 .

A novel allergen-adjuvant conjugate suitable for specific immunotherapy of respiratory allergy.

L. Maggi, G. Petroni, F. Boscaro, 2013, The Journal of allergy and clinical immunology.

Diastereodivergent Synthesis of 4‐Hydroxy‐2,3‐methanopipecolic Acid Derivatives as Conformationally Constrained Homoserine Analogues

A. Guarna, D. Scarpi, E. Occhiato, 2011 .

A Systems Biology Approach to Dissection of the Effects of Small Bicyclic Peptidomimetics on a Panel of Saccharomyces cerevisiae Mutants*

D. Cavalieri, A. Trabocchi, A. Guarna, 2010, The Journal of Biological Chemistry.

Use of click-chemistry in the development of peptidomimetic enzyme inhibitors.

A. Trabocchi, A. Guarna, G. Menchi, 2014, Current medicinal chemistry.

The isoxazoline-5-spirocyclopropane route to (±)-Pumiliotoxin C

A. Brandi, F. M. Cordero, A. Guarna, 1992 .

Solvent‐Dependent Conformational Behaviour of Model Tetrapeptides Containing a Bicyclic Proline Mimetic

D. Potenza, A. Trabocchi, A. Guarna, 2004 .

Density functional studies on the Nazarov reaction involving cyclic systems.

A. Cavalli, M. Recanatini, Matteo Masetti, 2006, Chemistry.

Selective non-steroidal inhibitors of 5α-reductase type 1

M. Serio, G. Danza, A. Guarna, 2004, The Journal of Steroid Biochemistry and Molecular Biology.

Selective non-steroidal inhibitors of 5 alpha-reductase type 1.

M. Serio, G. Danza, A. Guarna, 2004, The Journal of steroid biochemistry and molecular biology.

Quantitative determination of 4-hydroxy-4-androstene-3,17-dione (4-OHA), a potent aromatase inhibitor, in human plasma, using isotope dilution mass spectrometry.

M. Serio, G. Moneti, R. Salerno, 1989, Journal of steroid biochemistry.

Measurement of testosterone and its 5-alfa-reduced metabolites in human prostatic tissue using isotope dilution mass spectrometry.

M. Serio, A. Natali, M. Pazzagli, 1986, Journal of steroid biochemistry.

Insight to the binding mode of triazole RGD-peptidomimetics to integrin-rich cancer cells by NMR and molecular modeling.

F. Vasile, D. Potenza, A. Trabocchi, 2016, Bioorganic & medicinal chemistry.

Role of Side‐Chain Bioisosteres in Determining the Binding Affinity of Click Chemistry Derived RGD Peptidomimetics to αvβ3 Integrin

A. Trabocchi, S. Raspanti, A. Guarna, 2014 .

Combination of click chemistry and sulfonamides to develop three-armed triazole compounds

F. Bianchini, A. Trabocchi, S. Raspanti, 2014 .

Case Study 2: Peptidomimetic Ligands for αvβ3 Integrin

A. Trabocchi, A. Guarna, 2014 .

Morpholine-based RGD-cyclopentapeptides as alphavbeta3/alphavbeta5 integrin ligands: role of configuration towards receptor binding affinity.

A. Pupi, A. Trabocchi, S. Raspanti, 2009, Bioorganic & medicinal chemistry.

Modified Adenine (9-Benzyl-2-Butoxy-8-Hydroxyadenine) Redirects Th2-Mediated Murine Lung Inflammation by Triggering TLR71

D. Bani, S. Howie, F. Annunziato, 2009, The Journal of Immunology.

Carbonylative Suzuki–Miyaura Coupling Reaction of Lactam‐, Lactone‐, and Thiolactone‐Derived Enol Triflates for the Synthesis of Unsymmetrical Dienones

A. Guarna, E. Occhiato, L. Bartali, 2007 .

Suzuki reaction of vinyl triflates from six- and seven-membered N-alkoxycarbonyl lactams with boronic acids and esters.

A. Trabocchi, A. Guarna, E. Occhiato, 2001, The Journal of organic chemistry.

19-nor-10-azasteroids, a new class of steroid 5 alpha-reductase inhibitors. 2. X-ray structure, molecular modeling, conformational analysis of 19-nor-10-azasteroids and comparison with 4-azasteroids and 6-azasteroids.

M. Serio, P. Paoli, G. Danza, 1997, Journal of medicinal chemistry.

Inflammation by Triggering TLR7 Redirects Th2-Mediated Murine Lung (9-Benzyl-2-Butoxy-8-Hydroxyadenine) Modified Adenine

D. Bani, S. Howie, F. Annunziato, 2008 .

Low molecular weight, non-peptidic agonists of TrkA receptor with NGF-mimetic activity

A. Cavalli, G. Bottegoni, A. Palamara, 2012, Cell Death and Disease.

Low molecular weight, non-peptidic agonists of TrkA receptor with NGF-mimetic activity

A. Cavalli, G. Bottegoni, A. Palamara, 2012, Cell Death and Disease.

Synthesis and conformational analysis of small peptides containing 6-endo-BT(t)L scaffolds as reverse turn mimetics.

D. Potenza, A. Trabocchi, A. Guarna, 2002, The Journal of organic chemistry.

Peptidomimetics as protein arginine deiminase 4 (PAD4) inhibitors

C. Supuran, A. Scozzafava, F. Carta, 2015, Journal of enzyme inhibition and medicinal chemistry.

Synthesis of 8-chloro-benzo[c]quinolizin-3-ones as potent and selective inhibitors of human steroid 5alpha-reductase 1.

M. Serio, R. Mancina, G. Danza, 2000, Bioorganic & medicinal chemistry letters.

Synthesis of benzo[c]quinolizin-3-ones: selective non-steroidal inhibitors of steroid 5 alpha-reductase 1.

M. Serio, R. Mancina, G. Danza, 1998, Bioorganic & medicinal chemistry letters.

Synthesis of a chemiluminescent probe useful for the purification of steroid 5α-reductase

M. Serio, L. Martini, A. Poletti, 1996 .

Isotopic dilution GC-MS measurement of 4-hydroxyandrostenedione in postmenopausal breast cancer

M. Serio, G. Bartolucci, G. Danza, 1996 .

Pharmacokinetics of 4-hydroxyandrostenedione in man after intramuscular injection of different formulations and the effect of this drug on plasma aromatizable androgens and 17β-estradiol concentrations

M. Serio, M. Muratori, G. Danza, 1993, The Journal of Steroid Biochemistry and Molecular Biology.

Synthesis of 5,6,6-[2H3]finasteride and quantitative determination of finasteride in human plasma at picogram level by an isotope-dilution mass spectrometric method.

M. Serio, G. Bartolucci, G. Danza, 1995, Journal of chromatography. B, Biomedical applications.

Novel small molecules for the treatment of infections caused by Candida albicans: a patent review (2002 – 2010)

A. Trabocchi, A. Guarna, C. Calugi, 2011, Expert opinion on therapeutic patents.

Synthesis of γ‐ and δ‐Amino Acids

A. Trabocchi, A. Guarna, G. Menchi, 2010 .

The TLR7 Ligand 9-Benzyl-2-Butoxy-8-Hydroxy Adenine Inhibits IL-17 Response by Eliciting IL-10 and IL-10–Inducing Cytokines

F. Annunziato, L. Maggi, E. Maggi, 2011, The Journal of Immunology.

Synthesis and activity of 8-substituted benzo[c]quinolizin-3-ones as dual inhibitors of human 5α-reductases 1 and 2

M. Serio, R. Mancina, G. Danza, 2005 .

SC1 structure-activity relationship of inhibitors for steroid 5α-reductase

M. Serio, G. Danza, A. Guarna, 1994 .

Measurement of Steroids in Human Plasma and Tissues by Isotope Dilution Mass Spectrometry a

M. Serio, M. Pazzagli, G. Moneti, 1990, Annals of the New York Academy of Sciences.

Determination of testosterone and its tissue metabolites (DHT and 3 alpha-diol) in human plasma and prostatic tissue by isotopic dilution mass spectrometry.

M. Giovannini, M. Serio, G. Forti, 1987, Journal of steroid biochemistry.

Synthesis and Conformational Analysis of Constrained β‐Turn Mimetics Incorporating a Bicyclic Turn Inducer by Use of the Petasis Three‐Component Reaction on Solid Phase

A. Trabocchi, A. Guarna, G. Menchi, 2007 .

Oxidation of 2-t-butyl-4-methoxyphenol (BHA) by horseradish and mammalian peroxidase systems.

P. Dolara, A. Guarna, L. Corte, 1980, Biochemical pharmacology.

Sugar Amino Acids

A. Trabocchi, A. Guarna, 2014 .

Oligomers of Enantiopure Bicyclic γ/δ-Amino Acids (BTAa). 1. Synthesis and Conformational Analysis of 3-Aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic Acid Oligomers (PolyBTG)

A. Guarna, F. Machetti, G. Menchi, 2000 .

N-Substituent effects on the diethylzinc addition to benzaldehyde catalysed by bicyclic 1,4-amino alcohols

A. Guarna, D. Scarpi, E. Occhiato, 2009 .

Enantioselective addition of diethylzinc to aldehydes using 1,4-aminoalcohols as chiral ligands

A. Guarna, D. Scarpi, E. Occhiato, 2004 .

The Basics of Peptidomimetics

A. Trabocchi, A. Guarna, 2014 .

5α-Reductase activity in Lycopersicon esculentum: Cloning and functional characterization of LeDET2 and evidence of the presence of two isoenzymes

M. Serio, G. Danza, F. Rosati, 2005, The Journal of Steroid Biochemistry and Molecular Biology.

Correlation Times measurements from Tin-Proton Dipolar interactions : A 1H NMR spin-lattice relaxation study

M. Rustici, M. Scarselli, N. Niccolai, 1990 .

Rearrangement of isoxazoline-5-spiro derivatives. 5. Diastereofacial selectivity in the cycloaddition of substituted five-membered cyclic nitrones and methylenecyclopropanes. Stereoselective synthesis of 3,5-substituted indolizidinones

A. Brandi, F. M. Cordero, A. Guarna, 1990 .

A new family of cinchona-derived amino phosphine precatalysts: application to the highly enantio- and diastereoselective silver-catalyzed isocyanoacetate aldol reaction.

D. Dixon, A. Trabocchi, A. Guarna, 2011, Journal of the American Chemical Society.

Effect of C-ring modifications in benzo[c]quinolizin-3-ones, new selective inhibitors of human 5 alpha-reductase 1.

M. Serio, R. Mancina, A. Trabocchi, 2001, Bioorganic & medicinal chemistry.

Stereoselective cyclopropanation of serine- and threonine-derived oxazines to access new morpholine-based scaffolds.

A. Trabocchi, A. Guarna, Filippo Sladojevich, 2008, Organic & biomolecular chemistry.

A new bicyclic proline-mimetic amino acid

A. Trabocchi, A. Guarna, N. Cini, 2003 .

Parallel synthesis of an amide library based on the 6,8-dioxa-3-azabicyclo[3.2.1]octane scaffold by direct aminolysis of methyl esters.

C. Kappe, A. Guarna, F. Machetti, 2007, Journal of combinatorial chemistry.

1,3-Aminoalcohols by reductive cleavage of isoxazolidines with molybdenum hexacarbonyl

S. Cicchi, A. Brandi, A. Guarna, 1990 .

An Improved Synthesis of 1,3-Diphenyl-2-buten-1-ones (ß-Methylchalcones)

A. Guarna, L. J. Mazza, 1980 .

Skeletal diversity by sequential one-pot and stepwise routes using morpholine ester scaffolds

A. Trabocchi, A. Guarna, Filippo Sladojevich, 2010 .

A new synthesis of (2S)-4-oxopipecolic acid by thermal rearrangement of enantiopure spirocyclopropaneisoxazolidine

A. Brandi, F. M. Cordero, A. Guarna, 1996 .

Stereoselective Synthesis of (2S,4R)-4-Hydroxypipecolic Acid

A. Guarna, D. Scarpi, E. Occhiato, 2008 .

Bicyclic peptidomimetics targeting secreted aspartic protease 2 (SAP2) from Candida albicans reveal a constrained inhibitory chemotype.

P. Navarra, A. Cassone, F. De bernardis, 2012, Bioorganic & medicinal chemistry.

Identification of inhibitors of drug-resistant Candida albicans strains from a library of bicyclic peptidomimetic compounds.

A. Cassone, F. De bernardis, R. Cauda, 2010, Journal of medicinal chemistry.

Remote stereocontrol in the Nazarov reaction: a new approach to the core of roseophilin.

C. Prandi, A. Guarna, E. Occhiato, 2005, The Journal of organic chemistry.

Enantioselective synthesis of indolizine derivatives by rearrangement-cyclization of isoxazoline-5-spirocyclopropanes

A. Guarna, E. Occhiato, L. Spinetti, 1993 .

Rearrangement of isoxazoline-5-spiro derivatives. part 4. Synthesis of medium size benzofused azaheterocycles

A. Brandi, F. M. Cordero, A. Guarna, 1989 .

Rearrangement of isoxazoline-5-spiro derivatives. 2. Synthesis and rearrangement of tetrahydroisoxazole-5-spirocyclopropanes. Preparation of precursors of quinolizine, isoquinoline, and indole alkaloids

A. Brandi, F. M. Cordero, A. Guarna, 1988 .

Rearrangement of nitrone cycloadducts to methylene cyclopropane. Synthesis of indolizidine and quinolizidine derivatives.

A. Brandi, A. Guarna, A. Goti, 1986 .

One-pot sequential Ti-/Cu-catalysis for tandem amidation/Ullmann-type cyclization: synthesis of model benzodiazepine(di)ones promoted by microwave irradiation.

A. Trabocchi, A. Guarna, C. Lalli, 2012, Organic & biomolecular chemistry.

Diastereoselective Synthesis of Highly Constrained Spiro‐β‐Lactams by the Staudinger Reaction Using an Unsymmetrical Bicyclic Ketene

A. Trabocchi, A. Guarna, C. Lalli, 2007 .

A CONCISE ROUTE TO 19-NOR-10-AZASTEROIDS, A NEW CLASS OF STEROID 5ALPHA -REDUCTASE INHIBITORS. 3. SYNTHESIS OF (+)-19-NOR-10-AZATESTOSTERONE AND (+)-1 7BETA -(ACETYLOXY)-(5BETA )-10-AZAESTR-1-EN-3-ONE

A. Guarna, F. Machetti, D. Scarpi, 1998 .

Correction. N-Bridgehead Polycyclic Compounds by Sequential Rearrangement-Annulation of Isoxazoline-5-spirocyclopropanes. 6. A General Synthetic method for 5,6-Dihydro-7(8H)- and 2,3,5,6-Tetrahydro-7(1H)-indoliziones.

A. Brandi, A. Guarna, A. Goti, 1992 .

Preparation and Suzuki-Miyaura coupling reactions of tetrahydropyridine-2-boronic acid pinacol esters.

A. Guarna, E. Occhiato, Fabrizio Lo Galbo, 2005, The Journal of organic chemistry.

The Lewis acid-catalyzed nazarov reaction of 2-(n-methoxycarbonylamino)-1,4-pentadien-3-ones.

A. Guarna, E. Occhiato, Paolo Larini, 2006, Organic letters.

Cyclic α‐Amino Acids as Proline Mimetics

A. Trabocchi, A. Guarna, 2014 .

Structural diversity of bicyclic amino acids

A. Trabocchi, A. Guarna, D. Scarpi, 2007, Amino Acids.

Solid‐Phase Synthesis and Combinatorial Approaches to Peptidomimetics

A. Trabocchi, A. Guarna, 2014 .

Synthesis of a new enantiopure bicyclic γ/δ-amino acid (BTKa) derived from tartaric acid and α-amino acetophenone

A. Trabocchi, A. Guarna, F. Machetti, 2002 .

Synthesis and conformational studies of a hybrid β-alanine–morpholine tetramer

A. Trabocchi, A. Guarna, G. Menchi, 2012 .

¹²⁵I-radiolabeled morpholine-containing arginine-glycine-aspartate (RGD) ligand of αvβ₃ integrin as a molecular imaging probe for angiogenesis.

Alberto Pupi, Andrea Trabocchi, Eleonora Vanzi, 2012, Journal of medicinal chemistry.

Diversity-oriented synthesis of morpholine-containing molecular scaffolds.

A. Trabocchi, A. Guarna, C. Lalli, 2009, Chemistry.

Synthesis of a new 1,4-aminoalcohol and its use as catalyst in the enantioselective addition of organozinc to aldehydes

A. Guarna, D. Scarpi, Fabrizio Lo Galbo, 2006 .

β‐Turn Peptidomimetics

A. Trabocchi, A. Guarna, 2014 .

Synthesis of a bicyclic δ-amino acid as a constrained Gly-Asn dipeptide isostere

A. Trabocchi, A. Guarna, G. Menchi, 2008, Amino Acids.

Synthesis of bicyclic molecular scaffolds (BTAa): an investigation towards new selective MMP-12 inhibitors.

Vito Calderone, Marco Nievo, Athanasios Papakyriakou, 2006, Bioorganic & medicinal chemistry.

3-Aza-6,8-dioxabicyclo[3.2.1]octanes as new enantiopure heteroatom-rich tropane-like ligands of human dopamine transporter.

A. Pupi, A. Trabocchi, S. Raspanti, 2006, Bioorganic & medicinal chemistry.

3-Aza-8,10-dioxa-bicyclo[5.2.1]decane (9-exo BTKa) carboxylic acid as a new reverse turn inducer: synthesis and conformational analysis of a model peptide

A. Trabocchi, A. Guarna, D. Stranges, 2006 .

Synthesis of a constrained tricyclic scaffold based on trans-4-hydroxy-l-proline

A. Trabocchi, A. Guarna, G. Menchi, 2005 .

Synthesis of Glycidol‐ and Sugar‐Derived Bicyclic β‐ and γ/δ‐Amino Acids for Peptidomimetic Design

A. Trabocchi, A. Guarna, G. Menchi, 2005 .

Introduction of the new dipeptide isostere 7-endo-BtA as reverse turn inducer in a Bowman-Birk proteinase inhibitor: synthesis and conformational analysis.

R. Leatherbarrow, A. Trabocchi, A. Guarna, 2001, Bioorganic & medicinal chemistry.

Synthesis and Reactivity of Bicycles Derived from Tartaric Acid and α-Amino Acids: A Novel Class of Conformationally Constrained Dipeptide Isosteres Based upon Enantiopure 3-Aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic Acid

A. Trabocchi, A. Guarna, F. Machetti, 1999 .

Evaluation of efficacy, pharmacokinetics and tolerability of peptidomimetic aspartic proteinase inhibitors as cream formulation in experimental vaginal candidiasis

P. Navarra, A. Cassone, F. De bernardis, 2014, The Journal of pharmacy and pharmacology.

Preparation of cyclopenta-fused N-, O-, and s-heterocycles by Lewis acid catalyzed Nazarov reaction

A. Guarna, E. Occhiato, L. Bartali, 2007 .

New synthetic approach to cyclopenta-fused heterocycles based upon a mild nazarov reaction. 2. Further studies on the torquoselectivity.

P. Venturello, C. Prandi, A. Guarna, 2004, The Journal of organic chemistry.

New synthetic approach to cyclopenta-fused heterocycles based upon a mild Nazarov reaction.

P. Venturello, C. Prandi, A. Guarna, 2003, The Journal of organic chemistry.

Synthesis of α-acyl-functionalized azacycles by Pd-catalyzed cross-coupling reactions of α-alkoxyboronates with lactam-derived vinyl triflates

P. Venturello, C. Prandi, A. Guarna, 2002 .

Stereoselective Meisenheimer rearrangement using BTAa's as chiral auxiliaries

A. Guarna, D. Scarpi, E. Occhiato, 2000 .

A solid-phase approach towards the development of 3-aza-6,8-dioxabicyclo[3.2.1]octane scaffolds

A. Trabocchi, A. Guarna, G. Menchi, 2004, Molecular Diversity.

Peptidomimetics in Organic and Medicinal Chemistry: The Art of Transforming Peptides in Drugs

A. Trabocchi, A. Guarna, 2014 .

Organocatalytic diastereo- and enantioselective Michael addition reactions of 5-aryl-1,3-dioxolan-4-ones.

D. Dixon, A. Guarna, D. Stranges, 2007, Organic letters.

Preparation and cycloaddition reactions of enantiopure 2-(N-acylamino)-1,3-dienes for the synthesis of octahydroquinoline derivatives.

A. Guarna, C. Faggi, E. Occhiato, 2003, The Journal of organic chemistry.

Bicyclic Compounds Derived from Tartaric Acid and α‐Amino Acids (BTAas): Synthesis of New Molecular Scaffolds Derived from the Combination of (R,R)‐Tartaric Acid and L‐Serine

A. Guarna, N. Cini, F. Machetti, 2002 .

Condensation Product between (R,R)‐Tartaric Acid and a L‐Phenylalanine Derivative as a New Molecular Scaffold

A. Guarna, G. Menchi, A. Giolitti, 1997 .

Cleavage of Isoxazolines with Tricarbonyltris(acetonitrile)molybdenum and Silica Gel. Synthesis of 1-(2-Oxoalkyl)cyclopropanols from lsoxazoline-5-spirocyclopropanes

A. Brandi, A. Guarna, A. Goti, 1989 .

Chemical genetics approach to identify new small molecule modulators of cell growth by phenotypic screening of Saccharomyces cerevisiae strains with a library of morpholine-derived compounds.

D. Cavalieri, A. Trabocchi, A. Guarna, 2010, Organic & biomolecular chemistry.

Evaluation of stereochemically dense morpholine-based scaffolds as proline surrogates in beta-turn peptides.

A. Trabocchi, A. Guarna, Filippo Sladojevich, 2010, Organic & biomolecular chemistry.

Configurationally driven folding of model tetrapeptides containing L- or D-morpholine-3-carboxylic acids as beta-turn nucleators.

A. Trabocchi, A. Guarna, Filippo Sladojevich, 2009, Chirality.

Convenient route to enantiopure fmoc-protected morpholine-3-carboxylic acid.

A. Trabocchi, A. Guarna, Filippo Sladojevich, 2007, The Journal of organic chemistry.

Skeletal diversity from carbohydrates: use of mannose for the diversity-oriented synthesis of polyhydroxylated compounds.

Elena Lenci, Andrea Trabocchi, A. Trabocchi, 2015, The Journal of organic chemistry.

Enantiospecific synthesis of 3-aza-6,8-dioxa-bicyclo[3.2.1]octane carboxylic acids from erythrose

A. Trabocchi, A. Guarna, F. Machetti, 2003 .

New Synthesis of Azaheterocycles by Rearrangement of Isoxazoline-5-spirocycloalkane Compounds

A. Brandi, F. M. Cordero, A. Guarna, 1993 .

Cyclopropane pipecolic acids as templates for linear and cyclic peptidomimetics: application in the synthesis of an Arg-Gly-Asp (RGD)-containing peptide as an αvβ3 integrin ligand.

F. Bianchini, A. Trabocchi, A. Guarna, 2014, Chemistry.

1,3‐Amino Alcohols by Reductive Cleavage of Isoxazolidines with Molybdenum Hexacarbonyl.

S. Cicchi, A. Brandi, A. Guarna, 1991 .

New synthesis of azepin-4-ones by flash vacuum thermolysis of dihydro and tetrahydroisoxazole-5-spirocyclobutane derivatives

A. Brandi, A. Guarna, A. Goti, 1986 .

Cyclic DGR-peptidomimetic containing a bicyclic reverse turn inducer as a selective αvβ5 integrin ligand

A. Pupi, D. Potenza, A. Trabocchi, 2009, Amino Acids.

γ- and δ-Amino Acids: Synthetic Strategies and Relevant Applications

A. Trabocchi, A. Guarna, F. Guarna, 2005 .

Click Chemistry: The Triazole Ring as a Privileged Peptidomimetic Scaffold

A. Trabocchi, A. Guarna, 2014 .

Case Study 1: Peptidomimetic HIV Protease Inhibitors

A. Trabocchi, A. Guarna, 2014 .

Asymmetric hydrogenation of prochiral γ-nitroketones by ruthenium complexes

A. Guarna, G. Menchi, D. Scarpi, 1996 .

γ‐ and δ‐Amino Acids: Synthetic Strategies and Relevant Applications

A. Trabocchi, A. Guarna, F. Guarna, 2006 .

Deciphering the mechanism of action of 089, a compound impairing the fungal cell cycle

S. Heath, M. Gut, I. Gut, 2018, Scientific Reports.

Synthesis and preliminary biological characterization of a new potential (125)I-radioligand for dopamine and serotonin receptors.

A. Pupi, G. Berti, S. Raspanti, 2001, Bioorganic & medicinal chemistry.

Diversity-Oriented Synthesis as a Tool for Chemical Genetics

A. Trabocchi, E. Lenci, A. Guarna, 2014, Molecules.

Identification of constrained peptidomimetic chemotypes as HIV protease inhibitors.

A. Trabocchi, A. Guarna, C. Calugi, 2014, European journal of medicinal chemistry.

Microbial biotransformations in water/organic solvent system. Enantioselective reduction of aromatic β- and γ-nitroketones

F. Molinari, A. Guarna, F. Aragozzini, 1998 .

Selectivity of Daucus carota roots and baker’s yeast in the enantioselective reduction of γ-nitroketones

A. Guarna, D. Scarpi, E. Occhiato, 2005 .

2,2'-dihydroxy-3,3'-di-t-butyl-5,5'-dimethoxydiphenyl, a new metabolite of 2-t-butyl-4-methoxyphenol in the rat.

L. Della Corte, M. Giovannini, A. Guarna, 1983, Drug metabolism and disposition: the biological fate of chemicals.

Synthesis of 17β-N-Substituted 19-Nor-10-azasteroids as Inhibitors of Human 5α-Reductases I and II

M. Serio, G. Danza, A. Guarna, 2002 .

Novel inhibitors of 5α-reductase

A. Guarna, F. Machetti, 2002 .

Behaviour of nitrile oxides towards nucleophiles. Part III. Dimerisation of aromatic nitrile oxides catalysed by trimethylamine

A. Guarna, F. Sarlo, 1976 .

Synthesis of new molecular scaffolds: 3-aza-7,9-dioxa-bicyclo[4.2.1]nonane (8-exo BTKa) and 3-aza-8,10-dioxa-bicyclo[5.2.1]decane (9-exo BTKa) carboxylic acids

A. Guarna, D. Stranges, D. Scarpi, 2004 .

Reactivity in the gas phase. Behaviour of isoxazoles under negative ion chemical ionization conditions

G. Moneti, A. Guarna, 1989 .

The chemistry of fulminic acid revised

A. Brandi, A. Guarna, A. Goti, 1985 .

Low molecular weight, non-peptidic agonists of TrkA receptor with NGF-mimetic activity

A. Cavalli, G. Bottegoni, A. Palamara, 2012, Cell Death and Disease.

Low molecular weight, non-peptidic agonists of TrkA receptor with NGF-mimetic activity

A. Cavalli, G. Bottegoni, A. Palamara, 2012, Cell Death and Disease.

Click-chemistry-derived triazole ligands of arginine-glycine-aspartate (RGD) integrins with a broad capacity to inhibit adhesion of melanoma cells and both in vitro and in vivo angiogenesis.

A. Pupi, F. Bianchini, A. Trabocchi, 2010, Journal of medicinal chemistry.

Erratum: Low molecular weight, non-peptidic agonists of TrkA receptor with NGF-mimetic activity (Cell Death and Disease (2012) 3 (e339) Doi: 10.1038/cddis.2012.80)

A. Cavalli, G. Bottegoni, A. Palamara, 2012 .

Redirection of allergen-specific TH2 responses by a modified adenine through Toll-like receptor 7 interaction and IL-12/IFN release.

L. Cosmi, F. Annunziato, F. Liotta, 2006, The Journal of allergy and clinical immunology.

Multinuclear magnetic resonance study of organomercury fulminates. The structure of mercury fulminate in solution

N. Niccolai, A. Brandi, A. Guarna, 1984 .

Radiosynthesis and micro-SPECT analysis of triazole-based RGD integrin ligands as non-peptide molecular imaging probes for angiogenesis.

A. Pupi, A. Passeri, F. Bianchini, 2015, Bioorganic & medicinal chemistry.

Chemical genetics approach to drug discovery by diversity-oriented synthesis (DOS) of peptidomimetics

D. Cavalieri, A. Trabocchi, A. Guarna, 2011 .

A study of a D-proline peptidomimetic inhibitor of melanoma and endothelial cell invasion through activity towards MMP-2 and MMP-9

F. Bianchini, Jessica Ruzzolini, A. Trabocchi, 2015 .

5α-Reductase Inhibitors, Chemical and Clinical Models

M. Serio, G. Danza, A. Guarna, 1998, Steroids.

5 alpha-reductase inhibitors, chemical and clinical models.

M. Serio, G. Danza, A. Guarna, 1998, Steroids.

Heterocyclic HIV-protease inhibitors.

A. Trabocchi, A. Guarna, C. Calugi, 2013, Current medicinal chemistry.

Stereoselectivity in the TiCl4-catalysed reaction of Danishefsky's diene with a N-(acyloxy)iminium ion: Synthesis of 5α versus 5β Δ1(2)-19-Nor-10-azasteroids. 4

A. Guarna, F. Machetti, D. Scarpi, 1998 .

Simple in situ preparation of fulmimic acid

S. Corezzi, A. Brandi, A. Guarna, 1983 .

A multinuclear magnetic resonance study of nitrile oxides

Neri Niccolai, N. Niccolai, A. Brandi, 1982 .

Baker's yeast reduction of prochiral γ-nitroketones: Enantioselective synthesis of (S)-4-nitroalcohols

A. Guarna, D. Scarpi, E. Occhiato, 1995 .

Insight into the structural similarity between HIV protease and secreted aspartic protease-2 and binding mode analysis of HIV-Candida albicans inhibitors

A. Trabocchi, A. Guarna, C. Calugi, 2013, Journal of enzyme inhibition and medicinal chemistry.

A lactam-derived vinyl boronate as a stable and crystalline reagent for the synthesis of 2-substituted piperidines by Pd-catalyzed coupling reactions

A. Guarna, E. Occhiato, Alessandro Ferrali, 2004 .

Deciphering the mechanism of action of 089, a compound impairing the fungal cell cycle

S. Heath, M. Gut, I. Gut, 2018, Scientific Reports.

A Short and Efficient Route to Enantiopure 3,5-Diarylpyrrolizidines.

A. Guarna, D. Scarpi, E. Occhiato, 1999, The Journal of organic chemistry.

Gas chromatographic analysis of trans- and cis-dypnone

A. Guarna, N. Gelsomini, L. J. Mazza, 1974 .

Interaction between aromatic residues. Molecular dynamics and ab initio exploration of the potential energy surface of the tryptophan-histidine pair

Schettino, F. Gervasio, P. Procacci, 2000 .

D-proline-based peptidomimetic inhibitors of anthrax lethal factor.

A. Trabocchi, A. Guarna, C. Lalli, 2012, European journal of medicinal chemistry.

Behaviour of nitrile oxides towards nucleophiles. Part II. Substituent effect on the rate of dimerisation of aromatic nitrile oxides to 3,6-diaryl-1,4,2,5-dioxadiazines

A. Guarna, F. Sarlo, 1976 .

Rearrangement of isoxazoline-5-spiro derivatives. Part 7 : Thermal rearrangement of 4,5-dihydro and tetrahydroisoxazole-5-spirocyclobutanes to azepin-4-one derivatives

A. Brandi, A. Guarna, A. Goti, 1992 .