E. Morelli

发表

Characterization of the 1H-cyclopentapyrimidine-2,4(1H,3H)-dione derivative (S)-CPW399 as a novel, potent, and subtype-selective AMPA receptor full agonist with partial desensitization properties.

E. Novellino, T. Liljefors, A. Schousboe, 2001, Journal of medicinal chemistry.

1H-cyclopentapyrimidine-2,4(1H,3H)-dione-related ionotropic glutamate receptors ligands. structure-activity relationships and identification of potent and Selective iGluR5 modulators.

E. Novellino, A. Schousboe, S. Gemma, 2008, Journal of medicinal chemistry.

Development and Validation of an Analytical Method for Total Polyphenols Quantification in Extra Virgin Olive Oils

S. Seccia, E. Morelli, I. Dini, 2019, Food Analytical Methods.

Specific targeting of peripheral serotonin 5-HT(3) receptors. Synthesis, biological investigation, and structure-activity relationships.

E. Novellino, M. Hamon, R. Budriesi, 2009, Journal of medicinal chemistry.

Effects of Drug Resistance Mutations L100I and V106A on the Binding of Pyrrolobenzoxazepinone Nonnucleoside Inhibitors to the Human Immunodeficiency Virus Type 1 Reverse Transcriptase Catalytic Complex

G. Maga, S. Gemma, G. Campiani, 2004, Antimicrobial Agents and Chemotherapy.

Antagonizing S1P3 Receptor with Cell-Penetrating Pepducins in Skeletal Muscle Fibrosis

A. Lavecchia, G. Caliendo, V. Santagada, 2021, International journal of molecular sciences.

Focus on renal blood flow in mechanically ventilated patients with SARS-CoV-2: a prospective pilot study

L. Gesualdo, S. Grasso, S. Spadaro, 2020, Journal of Clinical Monitoring and Computing.

Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity.

A. Bergamini, E. Novellino, G. Greco, 1999, Journal of medicinal chemistry.

Pyrrolo[1,3]benzothiazepine-based serotonin and dopamine receptor antagonists. Molecular modeling, further structure-activity relationship studies, and identification of novel atypical antipsychotic agents.

Caterina Fattorusso, Giuseppe Campiani, Alfredo Cagnotto, 2004, Journal of medicinal chemistry.

Synthesis of new molecular probes for investigation of steroid biosynthesis induced by selective interaction with peripheral type benzodiazepine receptors (PBR).

E. Novellino, G. Campiani, D. Zisterer, 2002, Journal of medicinal chemistry.

Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT(3) receptor agonists: synthesis, further structure-activity relationships, and biological studies.

E. Novellino, G. Greco, M. Hamon, 1999, Journal of medicinal chemistry.

Polycondensed heterocycles. Part 12: An approach to the synthesis of 2-acetyl-1′-methyl-1,2,3,4-tetrahydrospiro[isoquinoline-1,4′-pyrrolidine]-2′-one

S. Gemma, G. Campiani, S. Butini, 2002 .

Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent.

E Novellino, A. Bergamini, E. Novellino, 2001, Journal of medicinal chemistry.

Novel, potent, and selective quinoxaline-based 5-HT(3) receptor ligands. 1. Further structure-activity relationships and pharmacological characterization.

E. Novellino, M. Hamon, R. Budriesi, 2009, Journal of medicinal chemistry.

Inherent desensitisation-preventing properties of a novel, subtype-selective AMPA receptor agonist, (S)-CPW 399, as a possible explanation for its excitotoxic action in cultured cerebellar granule cells

E. Novellino, A. Schousboe, G. Campiani, 2003, Neurochemistry International.

Non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors: past, present, and future perspectives.

Ettore Novellino, Caterina Fattorusso, Giuseppe Campiani, 2002, Current pharmaceutical design.

Investigating the role of T7 and T12 residues on the biological properties of thrombin-binding aptamer: enhancement of anticoagulant activity by a single nucleobase modification.

Gennaro Piccialli, Nicola Borbone, Marco Persico, 2012, Journal of medicinal chemistry.

Exploring the Photodynamic Properties of Two Antiproliferative Benzodiazopyrrole Derivatives

C. Altucci, C. Dell’Aversano, L. Tartaglione, 2020, International journal of molecular sciences.

Outstanding effects on antithrombin activity of modified TBA diastereomers containing an optically pure acyclic nucleotide analogue.

E. Novellino, G. Piccialli, L. Mayol, 2014, Organic & biomolecular chemistry.

Synthesis, structural studies and biological properties of new TBA analogues containing an acyclic nucleotide.

Nicola Borbone, Giuseppe Cirino, Giorgia Oliviero, 2008, Bioorganic & medicinal chemistry.

D-galactose as a vector for prodrug design.

M. G. Rimoli, Elvira Luongo, E. Morelli, 2011, Current topics in medicinal chemistry.

Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis and Biological Evaluation of Novel Quinoxalinylethylpyridylthioureas as Potent Antiviral Agents

A. Bergamini, E. Novellino, G. Greco, 2000, Antiviral chemistry & chemotherapy.