S. Kaldor

发表

Antiviral and resistance studies of AG1343, an orally bioavailable inhibitor of human immunodeficiency virus protease

D. Ho, M. Markowitz, H. Mo, 1996, Antimicrobial agents and chemotherapy.

Synthesis of 2′,3′-dideoxy-3′-hydroxymethylcytidine; a unique antiviral nucleoside

M. Faul, L. L. Winneroski, M. Staszak, 1997 .

Design and synthesis of pyrimidinone and pyrimidinedione inhibitors of dipeptidyl peptidase IV.

D. Kassel, S. L. Gwaltney, K. Aertgeerts, 2011, Journal of medicinal chemistry.

Viracept (nelfinavir mesylate, AG1343): a potent, orally bioavailable inhibitor of HIV-1 protease.

N. Chirgadze, D. Clawson, K. Appelt, 1997, Journal of medicinal chemistry.

Total Synthesis of the Macrolide Antibiotic Cytovaricin.

J. Clardy, Davidr . Evans, S. Kaldor, 1990 .

A CONVENIENT, LARGE SCALE SYNTHESIS OF N-CBZ-(S-PHENYL)-L-CYSTEINE

A. Trippe, S. Kaldor, B. Shamblin, 1995 .

Design, synthesis and biological evaluation of novel 4-phenylisoquinolinone BET bromodomain inhibitors.

J. Veal, D. Hosfield, Jiangchun Xu, 2018, Bioorganic & medicinal chemistry letters.

Glutamine-derived aldehydes for the inhibition of human rhinovirus 3C protease

B. Heinz, A. D. Kline, S. Kaldor, 1995 .

Azetidinones as vasopressin V1a antagonists.

C. Ferris, M. Brownstein, M. Clay, 2007, Bioorganic & medicinal chemistry.

Discovery of CC-90011: A Potent and Selective Reversible Inhibitor of Lysine Specific Demethylase 1 (LSD1).

J. Veal, D. Hosfield, L. Lawton, 2020, Journal of medicinal chemistry.

Simple in vitro translation assay to analyze inhibitors of rhinovirus proteases

B. Heinz, S. Kaldor, J. Labus, 1996, Antimicrobial agents and chemotherapy.

Discovery of TAK-960: an orally available small molecule inhibitor of polo-like kinase 1 (PLK1).

V. Feher, D. Hosfield, T. Kawamoto, 2013, Bioorganic & medicinal chemistry letters.

Solid phase synthesis of hydantoins using a carbamate linker and a novel cyclization / cleavage step

S. Kaldor, L. A. Spangle, B. Dressman, 1996 .

Rapid purification of small molecule libraries by ion exchange chromatography

M. Siegel, J. Grunwell, S. Kaldor, 1997 .

Use of solid supported nucleophiles and electrophiles for the purification of non-peptide small molecule libraries

Miles G. Siegel, M. Siegel, S. Kaldor, 1996 .

Assignment of stereochemistry in the oligomycin/rutamycin/cytovaricin family of antibiotics. Asymmetric synthesis of the rutamycin spiroketal synthon

Davidr . Evans, S. Kaldor, T. K. Jones, 1990 .

Combinatorial chemistry using polymer-supported reagents.

M. Siegel, S. Kaldor, 1997, Current opinion in chemical biology.

The stereoselective osmylation of 1,1-disubstituted olefins. Effect of allylic substituents on reaction diastereoselectivity

Davidr . Evans, S. Kaldor, 1990 .

N-[3-(2-Dimethylaminoethyl)-2-methyl-1H- indol-5-yl]-4-fluorobenzamide: a potent, selective, and orally active 5-HT(1F) receptor agonist potentially useful for migraine therapy.

J. Zgombick, D. Nelson, J. Audia, 2001, Journal of medicinal chemistry.

Synthesis of 2′,3′-dideoxy-3′-hydroxymethylcytidine: A novel hydroformylation route

S. Kaldor, J. Ward, J. E. Fritz, 1997 .

A mild, osmium tetraoxide-catalyzed method for the oxidation of sulfides to sulfones

S. Kaldor, M. Hammond, 1991 .

The synthesis of ethanolamine libraries from olefin scaffolds

D. Parks, M. Siegel, S. Kaldor, 2000 .

Solution phase synthesis of libraries of variably substituted olefin scaffolds: a library of allylic amines.

M. Siegel, J. Cooper, S. Kaldor, 2001, Journal of combinatorial chemistry.

Isophthalic acid derivatives: amino acid surrogates for the inhibition of HIV-1 protease

K. Appelt, M. Muesing, S. Kaldor, 1995 .

Solid phase synthesis of urea libraries using a diversifiable thiophenoxy carbonyl linker

S. Kaldor, B. Dressman, Bruce A. Dressman, 1998 .

Discovery of antirhinoviral leads by screening a combinatorial library of ureas prepared using covalent scavengers

S. Kaldor, Stephen W. Kaldor, James E. Fritz, 1996 .

Structure-based drug design of nonpeptidic P2 substituents for HIV-1 protease inhibitors

K. Appelt, V. Kalish, J. Davies, 1995 .

ITERATIVE PROTEIN STRUCTURE-BASED DRUG DESIGN AND SYNTHESIS OF HIV PROTEASE INHIBITORS

K. Appelt, V. Kalish, J. Davies, 1995, European Journal of Medicinal Chemistry.

New dipeptide isosteres useful for the inhibition of HIV-1 protease

S. Kaldor, B. Dressman, Bruce A. Dressman, 1994 .

Discovery of alogliptin: a potent, selective, bioavailable, and efficacious inhibitor of dipeptidyl peptidase IV.

D. Kassel, S. L. Gwaltney, K. Takeuchi, 2007, Journal of medicinal chemistry.

Rapid Purification of Small Molecule Libraries by Ion Exchange Chromatography.

M. Siegel, J. Grunwell, S. Kaldor, 1997 .

5‐HT1F receptor agonists inhibit neurogenic dural inflammation in guinea pigs

Kirk W. Johnson, T. Branchek, J. Zgombick, 1997, Neuroreport.

A systematic study of P1–P3 spanning sidechains for the inhibition of HIV-1 protease

K. Appelt, M. Muesing, S. Kaldor, 1995 .

The Discovery of Exarafenib (KIN-2787): Overcoming the Challenges of Pan-RAF Kinase Inhibition.

S. Kaldor, J. Tyhonas, Toufike Kanouni, 2024, Journal of medicinal chemistry.