Pravin S. Shirude

发表

BisPNA Targeting to DNA: Effect of Neutral Loop on DNA Duplex Strand Invasion by aepPNA‐N7G/aepPNA‐C Substituted Peptide Nucleic Acids

Krishna N. Ganesh, K. Ganesh, Vaijayanti A. Kumar, 2005 .

Isothermal Titration Calorimetry Studies on the Binding of Amino Acids to Gold Nanoparticles

Vipul Bansal, M. Sastry, V. Bansal, 2004 .

Single molecule conformational analysis of DNA G-quadruplexes

Shankar Balasubramanian, S. Balasubramanian, Pravin S. Shirude, 2008, Biochimie.

Formyl peptide receptor 2 and heart disease.

Pravin S. Shirude, J. Lupisella, Ricardo A. García, 2022, Seminars in immunology.

Ensemble and single molecule FRET analysis of the structure and unfolding kinetics of the c-kit promoter quadruplexes.

S. Balasubramanian, L. Ying, Pravin S. Shirude, 2010, Chemical communications.

G-quadruplex recognition by bis-indole carboxamides.

S. Balasubramanian, J. Dash, Pravin S. Shirude, 2008, Chemical communications.

Single molecule conformational analysis of the biologically relevant DNA G-quadruplex in the promoter of the proto-oncogene c-MYC.

S. Balasubramanian, L. Ying, Pravin S. Shirude, 2008, Chemical communications.

Quinolinyl Pyrimidines: Potent Inhibitors of NDH-2 as a Novel Class of Anti-TB Agents.

B. Paul, B. Ugarkar, Balachandra S Bandodkar, 2012, ACS medicinal chemistry letters.

Rigid cyanine dye nucleic acid labels.

S. Balasubramanian, Pravin S. Shirude, Adrian Fegan, 2008, Chemical communications.

Synthesis of bis-indole carboxamides as G-quadruplex stabilizing and inducing ligands.

S. Balasubramanian, R. Das, J. Dash, 2012, Chemistry.

Advancement of Cell Wall Inhibitors in Mycobacterium tuberculosis*Present address: Sai Life Sciences Ltd, Pune, India.

S. Narayanan, Pravin S. Shirude, P. Iyer, 2014 .

Single-molecule conformational analysis of G-quadruplex formation in the promoter DNA duplex of the proto-oncogene c-kit.

S. Balasubramanian, T. Ha, L. Ying, 2007, Journal of the American Chemical Society.

Macrocyclic and helical oligoamides as a new class of G-quadruplex ligands.

S. Balasubramanian, K. Shin‐ya, S. Ladame, 2007, Journal of the American Chemical Society.

Oxazole-based peptide macrocycles: a new class of G-quadruplex binding ligands.

S. Balasubramanian, S. Ladame, R. Rodriguez, 2006, Journal of the American Chemical Society.

(2S,5R/2R,5S)-Aminoethylpipecolyl aepip-aegPNA chimera: synthesis and duplex/triplex stability

K. Ganesh, Vaijayanti A. Kumar, Pravin S. Shirude, 2004 .

Chimeric peptide nucleic acids incorporating (2S,5R)-aminoethyl pipecolyl units: synthesis and DNA binding studies ☆

K. Ganesh, Vaijayanti A. Kumar, Pravin S. Shirude, 2004 .

Aminopyrazinamides: novel and specific GyrB inhibitors that kill replicating and nonreplicating Mycobacterium tuberculosis.

J. Tucker, T. Balganesh, V. Sambandamurthy, 2013, ACS chemical biology.

Diarylethynyl amides that recognize the parallel conformation of genomic promoter DNA G-quadruplexes.

S. Balasubramanian, S. Hsu, J. Dash, 2008, Journal of the American Chemical Society.

Trisubstituted isoalloxazines as a new class of G-quadruplex binding ligands: small molecule regulation of c-kit oncogene expression.

S. Balasubramanian, S. Sewitz, R. Rodriguez, 2007, Journal of the American Chemical Society.

Synthesis of aqueous Au core-Ag shell nanoparticles using tyrosine as a pH-dependent reducing agent and assembling phase-transferred silver nanoparticles at the air-water interface.

M. Sastry, R. Pasricha, P. Selvakannan, 2004, Langmuir : the ACS journal of surfaces and colloids.

Impact of CO2-solvent separators on the degradation of benzyl-2,3-dihydroxypiperidine-1-carboxylate during preparative supercritical fluid chromatographic (SFC) purification.

Pravin S. Shirude, Yingru Zhang, Dauh-Rurng Wu, 2017, Journal of chromatography. A.

G-Quadruplex DNA Bound by a Synthetic Ligand is Highly Dynamic

Prakrit V. Jena, S. Balasubramanian, T. Ha, 2009, Journal of the American Chemical Society.

Nonfluoroquinolone-Based Inhibitors of Mycobacterial Type II Topoisomerase as Potential Therapeutic Agents for TB

Pravin S. Shirude, S. Hameed, 2012 .

Discovery of pyrazolopyridones as a novel class of noncovalent DprE1 inhibitor with potent anti-mycobacterial activity.

A. Narayan, V. Ramachandran, V. Sambandamurthy, 2014, Journal of medicinal chemistry.

Azaindoles: noncovalent DprE1 inhibitors from scaffold morphing efforts, kill Mycobacterium tuberculosis and are efficacious in vivo.

Vijay T. Ahuja, A. Srivastava, A. Narayan, 2013, Journal of medicinal chemistry.

1,4-Azaindole, a Potential Drug Candidate for Treatment of Tuberculosis

Christopher B. Cooper, S. Narayanan, C. Cooper, 2014, Antimicrobial Agents and Chemotherapy.

Lead optimization of 1,4-azaindoles as antimycobacterial agents.

Christopher B. Cooper, S. Butler, A. Srivastava, 2014, Journal of medicinal chemistry.

Methyl-thiazoles: a novel mode of inhibition with the potential to develop novel inhibitors targeting InhA in Mycobacterium tuberculosis.

Shahul Hameed, Geoffrey Holdgate, V. Sambandamurthy, 2013, Journal of medicinal chemistry.

Scaffold Morphing To Identify Novel DprE1 Inhibitors with Antimycobacterial Activity.

Christopher B. Cooper, S. Butler, A. Narayan, 2019, ACS medicinal chemistry letters.

Challenges and opportunities in tuberculosis drug discovery: an industry perspective.

Pravin S. Shirude, V. Hosagrahara, Sreekanth A. Ramachandran, 2013, Future medicinal chemistry.

Challenges and opportunities in tuberculosis drug discovery: an industry perspective "Frequently, the hit rate for target-based screens, which deal with a single-gene target, is significantly lower compared with random whole cell-based screens."

Pravin S. Shirude, 2013 .

Alkylidene Oxapenem β-Lactamase Inhibitors Revisited: Potent Broad Spectrum Activity but New Stability Challenges.

Matthew D. Miller, S. Tentarelli, Minli Zhang, 2014, ACS medicinal chemistry letters.

Triarylpyridines: a versatile small molecule scaffold for G-quadruplex recognition.

S. Balasubramanian, Zoë A. E. Waller, R. Rodriguez, 2008, Chemical communications.

Impact of CO2-solvent separators on the degradation of benzyl-2,3-dihydroxypiperidine-1-carboxylate during preparative supercritical fluid chromatographic (SFC) purification.

Pravin S. Shirude, Yingru Zhang, R. Sarabu, 2017, Journal of chromatography. A.