P. Procopiou

发表

Pharmacological characterization of GSK3335103, an oral αvβ6 integrin small molecule RGD-mimetic inhibitor for the treatment of fibrotic disease.

R. Jenkins, L. Borthwick, S. Macdonald, 2021, European journal of pharmacology.

Ring-closing metathesis in the synthesis of biologically active peptidomimetics of apicidin A

R. Coombes, A. Barrett, P. Procopiou, 2007 .

P112 Discovery of a Novel, High Affinity, Small Molecule αvβ6 Inhibitor for the Treatment of Idiopathic Pulmonary Fibrosis

D. Flint, R. Chambers, S. Pyne, 2016 .

Catalytic 2,3,4-hexatriene formation by terminal alkyne coupling at calcium.

P. Hitchcock, A. Barrett, M. Hill, 2009, Chemical communications.

Heavier group 2 element-catalysed hydroamination of isocyanates.

A. Barrett, G. Kociok‐Köhn, M. Hill, 2008, Chemical communications.

Heavier Group‐2‐Element Catalyzed Hydroamination of Carbodiimides

A. Barrett, G. Kociok‐Köhn, M. Hill, 2008, European Journal of Inorganic Chemistry.

Triazenide complexes of the heavier alkaline earths: synthesis, characterization, and suitability for hydroamination catalysis.

P. Hitchcock, A. Barrett, G. Kociok‐Köhn, 2008, Inorganic chemistry.

Synthesis and structure-activity relationships of long-acting beta2 adrenergic receptor agonists incorporating metabolic inactivation: an antedrug approach.

I. McLay, Helen T Horsley, D. Coe, 2010, Journal of medicinal chemistry.

Selective plasma hydrolysis of glucocorticoid gamma-lactones and cyclic carbonates by the enzyme paraoxonase: an ideal plasma inactivation mechanism.

R. Angell, O. Singh, K. Biggadike, 2000, Journal of medicinal chemistry.

Determination of the absolute configuration of two αvβ6 integrin inhibitors for the treatment of idiopathic pulmonary fibrosis and investigations on the asymmetric 1,4-addition of arylboronic acids to crotonate esters bearing a C4-oxygen substituent

R. Copley, P. Procopiou, Tim N. Barrett, 2017 .

Lead optimisation of the N1 substituent of a novel series of indazole arylsulfonamides as CCR4 antagonists and identification of a candidate for clinical investigation.

S. Hodgson, D. Hall, P. Procopiou, 2012, Bioorganic & medicinal chemistry letters.

Thrombin inhibitors based on [5,5] trans-fused indane lactams.

N. Ramsden, H. Jhoti, H. Finch, 1999, Bioorganic & medicinal chemistry letters.

Modular Isoquinoline Synthesis Using Catalytic Enolate Arylation and in Situ Functionalization

Charlie T. McTernan, T. Donohoe, P. Procopiou, 2013, Organic letters.

Squalene synthase inhibitors: their potential as hypocholesterolaemic agents.

P. Procopiou, N. S. Watson, 1996, Progress in medicinal chemistry.

Semi-synthetic qualestatins: Squalene synthase inhibition and antifungal activity. The SAR of C6 and C7 modifications

J. Payne, A. H. Shingler, P. Procopiou, 1993 .

Carbodiimide insertion reactions of homoleptic heavier alkaline earth amides and phosphides.

P. Hitchcock, A. Barrett, M. Hill, 2010, Dalton transactions.

The discovery of quinoline based single-ligand human H1 and H3 receptor antagonists.

S. Hodgson, D. Holmes, P. Procopiou, 2016, Bioorganic & medicinal chemistry letters.

Short and Efficient Syntheses of Protoberberine Alkaloids using Palladium-Catalyzed Enolate Arylation**

T. Donohoe, P. Procopiou, B. S. Pilgrim, 2014, Angewandte Chemie.

The squalestatins: cleavage of the bicyclic core via the novel 6,8-dioxabicyclo[3.2.1]octane ring system

P. Sidebottom, P. Procopiou, G. Inglis, 1994 .

Structurally simplified squalestatins: monocyclic 1,3-dioxane analogues.

P. Procopiou, G. Inglis, N. S. Watson, 1994 .

The squalestatins: novel inhibitors of squalene synthase. The optimal C1 chain-length requirements.

P. Procopiou, B. E. Kirk, N. S. Watson, 1993 .

The squalestatins: potent inhibitors of squalene synthase. The role of the tricarboxylic acid moiety.

P. Procopiou, B. E. Kirk, N. S. Watson, 1993 .

The squalestatins: C-3 Decarboxylation studies and rearrangement to the 6,8-dioxabicyclo[3.2.1]octane ring system

P. Procopiou, G. Inglis, N. S. Watson, 1993 .

Structurally simplified squalestatins: A convenient route to a 67-unsubstituted derivative

P. Procopiou, G. Inglis, G. Giblin, 1993 .

A synthetic approach to squalestatin 1

Joseph P. Adams, H. Abdel-Rahman, D. Slee, 1993 .

The squalestatins, novel inhibitors of squalene synthase produced by a species of Phoma. II. Structure elucidation.

P. Sidebottom, P. Procopiou, N. S. Watson, 1992, The Journal of antibiotics.

Rapid Entry into Mono-, Bi-, and Tricyclic β-Lactam Arrays via Alkene Metathesis

Andrew J. P. White, David J. Williams, A. Barrett, 1998 .

Synthesis of C-19-functionalized 1alpha-hydroxyvitamin D(2) analogues via ring-closing metathesis.

A. Barrett, P. Procopiou, Karine Malagu, 2003, Organic letters.

Heavier alkaline earth catalyzed ene-yne cyclizations: atom-efficient access to tetrahydroisoquinoline frameworks.

A. Barrett, M. Hill, P. Procopiou, 2014, Organic letters.

Synthesis and structure-activity relationships of indazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists.

A. Hill, D. Clapham, S. Hodgson, 2013, Journal of medicinal chemistry.

Identification of selective 8-(piperidin-4-yloxy)quinoline sulfone and sulfonamide histamine H1 receptor antagonists for use in allergic rhinitis.

K. Clark, S. Hodgson, D. Holmes, 2017, Bioorganic & medicinal chemistry letters.

Design of Phthalazinone Amide Histamine H1 Receptor Antagonists for Use in Rhinitis.

K. Clark, S. Hodgson, D. Holmes, 2017, ACS medicinal chemistry letters.

Synthesis and pharmacological investigation of azaphthalazinone human histamine H(1) receptor antagonists.

C. Browning, S. Lynn, P. Procopiou, 2012, Bioorganic & medicinal chemistry.

Lead identification and structure-activity relationships of heteroarylpyrazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists.

J. Percy, Afjal H. Miah, R. Copley, 2014, Organic & biomolecular chemistry.

Palladium-catalyzed enolate arylation as a key C-C bond-forming reaction for the synthesis of isoquinolines.

Charlie T. McTernan, T. Donohoe, P. Procopiou, 2016, Organic & biomolecular chemistry.

Heavier group 2 metals and intermolecular hydroamination: a computational and synthetic assessment.

A. Barrett, Christine Brinkmann, P. Hunt, 2009, Journal of the American Chemical Society.

Ring-closing metathesis: novel routes to aromatic heterocycles.

T. Donohoe, P. Procopiou, Lisa P. Fishlock, 2008, Chemistry.

Flexible metathesis-based approaches to highly functionalised furans and pyrroles

T. Donohoe, P. Procopiou, K. Wheelhouse, 2008 .

A RECYCLABLE 'BOOMERANG' POLYMER-SUPPORTED RUTHENIUM CATALYST FOR OLEFIN METATHESIS

S. Cramp, A. Barrett, P. Procopiou, 1999 .

An Extremely Powerful Acylation Reaction of Alcohols with Acid Anhydrides Catalyzed by Trimethylsilyl Trifluoromethanesulfonate

P. Procopiou, G. Inglis, S. Baugh, 1998 .

Ring-closing metathesis for the synthesis of heteroaromatics: evaluating routes to pyridines and pyridazines

T. Donohoe, J. Bower, P. Procopiou, 2009 .

A metathesis-based approach to the synthesis of furans.

T. Donohoe, P. Procopiou, A. R. Lacy, 2007, Organic letters.

Heavier alkaline earth catalysts for the intermolecular hydroamination of vinylarenes, dienes, and alkynes.

A. Barrett, Christine Brinkmann, M. Hill, 2012, Journal of the American Chemical Society.

Heterofunctionalization catalysis with organometallic complexes of calcium, strontium and barium

A. Barrett, M. Hill, Mark R. Crimmin, 2010, Proceedings of the Royal Society A: Mathematical, Physical and Engineering Sciences.

Intramolecular hydroamination of aminoalkenes by calcium and magnesium complexes: a synthetic and mechanistic study.

A. Barrett, M. Hill, Mark R. Crimmin, 2009, Journal of the American Chemical Society.

Beta-diketiminato calcium and magnesium amides; model complexes for hydroamination catalysis.

A. Barrett, M. Hill, Mark R. Crimmin, 2009, Inorganic chemistry.

Insertion reactions of beta-diketiminate-stabilised calcium amides with 1,3-dialkylcarbodiimides.

P. Hitchcock, A. Barrett, M. Hill, 2008, Dalton transactions.

Synthesis of Functionalized Pyridines via a Regioselective Oxazoline Promoted C-H Amidation Reaction.

J. P. Harrity, P. Procopiou, S. Swanson, 2016, Organic letters.

Synthesis of substituted pyridines and pyridazines via ring closing metathesis.

T. Donohoe, J. Bower, P. Procopiou, 2009, Chemical communications.

Synthesis, Characterization, and Solution Lability of N-Heterocyclic Carbene Adducts of the Heavier Group 2 Bis(trimethylsilyl)amides

A. Barrett, G. Kociok‐Köhn, M. Hill, 2008 .

beta-Diketiminato Calcium Acetylides: Synthesis, Solution Dimerization, and Catalytic Carbon-Carbon Bond Formation

P. Hitchcock, A. Barrett, M. Hill, 2008 .

The discovery of phthalazinone-based human H1 and H3 single-ligand antagonists suitable for intranasal administration for the treatment of allergic rhinitis.

Kenneth L. Clark, Duncan S. Holmes, Michael Kranz, 2011, Journal of medicinal chemistry.

Inhibitors of cholesterol biosynthesis. 2. 3,5-Dihydroxy-7-(N-pyrrolyl)-6-heptenoates, a novel series of HMG-CoA reductase inhibitors.

P. Procopiou, G. Inglis, N. S. Watson, 1993, Journal of medicinal chemistry.

An extremely fast and efficient acylation reaction of alcohols with acid anhydrides in the presence of trimethylsilyl trifluoromethanesulfonate as catalyst

P. Procopiou, G. Inglis, S. Baugh, 1996 .

A mild and regioselective route to functionalized quinazolines.

J. P. Harrity, P. Procopiou, S. Swanson, 2015, Chemistry.

Heavier alkaline Earth amides as catalysts for the Tischenko reaction.

A. Barrett, M. Hill, Mark R. Crimmin, 2007, Organic letters.

Beta-diketiminate C-H activation with heavier group 2 alkyls.

A. Barrett, M. Hill, Mark R. Crimmin, 2009, Dalton transactions.

Alkaline Earth Catalysis of Alkynyl Alcohol Hydroalkoxylation/Cyclization

A. Barrett, Christine Brinkmann, M. Hill, 2012 .

Novel cyclodehydration reaction of hydroxyphenols. An alternative to the Mitsunobu reaction

M. Deal, P. Procopiou, Gary M. Smith, 1996 .

A novel cyclodehydration reaction of hydroxy-phenols using imidate esters as leaving groups

M. Deal, P. Procopiou, D. F. Hayman, 1993 .

Studies on the stereochemical assignment of 3-acylidene 2-oxindoles.

H. Adams, A. Meijer, J. P. Harrity, 2014, Organic & biomolecular chemistry.

Inhibitors of Cholesterol Biosynthesis. Part 2. 3,5-Dihydroxy-7-(N- pyrrolyl)-6-heptenoates, a Novel Series of HMG-CoA Reductase Inhibitors.

P. Procopiou, G. Inglis, N. S. Watson, 1994 .

A novel oxidatitive rearrangement of a pentasubstituted pyrrole to an unsaturated hydroxy γ-lactam

P. Procopiou, R. M. Highcock, 1994 .

Potassium trimethylsilanolate induced cleavage of 1,3-oxazolidin-2- and 5-ones, and application to the synthesis of (R)-salmeterol.

D. Coe, R. Perciaccante, P. Procopiou, 2003, Organic & biomolecular chemistry.

Synthesis and determination of absolute configuration of a non-peptidic αvβ6 integrin antagonist for the treatment of idiopathic pulmonary fibrosis.

S. Lynn, S. Macdonald, J. Pritchard, 2016, Organic & biomolecular chemistry.

Synthesis of diverse macrocyclic peptidomimetics utilizing ring-closing metathesis and solid-phase synthesis.

David J. Williams, A. Barrett, R. Upton, 2004, The Journal of organic chemistry.

Cation Charge Density and Precatalyst Selection in Group 2-Catalyzed Aminoalkene Hydroamination

A. Barrett, G. Kociok‐Köhn, M. Hill, 2011 .

Writing Your Next Medicinal Chemistry Article: Journal Bibliometrics and Guiding Principles for Industrial Authors.

N. Meanwell, W. R. Ewing, S. Macdonald, 2020, Journal of medicinal chemistry.

Synthesis and characterization of coronanes: multicyclopropane-fused macrocyclic arrays.

A. Barrett, D. J. Williams, P. Procopiou, 2001, The Journal of organic chemistry.

Calcium-Catalyzed Intermolecular Hydrophosphination

P. Hitchcock, A. Barrett, M. Hill, 2007 .

A convergent strategy towards febrifugine and related compounds.

J. P. Harrity, P. Procopiou, S. Swanson, 2018, Organic & biomolecular chemistry.

Oxazoline-Promoted Rh-Catalyzed C-H Amidation of Benzene Derivatives with Sulfonamides and Trifluoroacetamide. A Comparative Study.

J. P. Harrity, P. Procopiou, S. Swanson, 2016, The Journal of organic chemistry.

Synthesis of the beta 2 agonist (R)-salmeterol using a sequence of supported reagents and scavenging agents.

S. Ley, P. Procopiou, R. Bream, 2002, Organic letters.

Enantioselective synthesis of (S)-salmeterol via asymmetric reduction of azidoketone by Pichia angusta

G. Webb, P. Procopiou, Gillian E Morton, 2001 .

Tandem ireland-claisen rearrangement ring-closing alkene metathesis in the construction of bicyclic beta-lactam carboxylic esters.

A. Barrett, D. J. Williams, P. Procopiou, 2000, The Journal of organic chemistry.

Highly functionalised monocyclic and bicyclic β-lactamsvia alkene metathesis

A. Barrett, P. Procopiou, V. C. Gibson, 1997 .

Rapid Entry into Mono-, Bi-, and Tricyclic β-Lactam Arrays via Alkene Metathesis.

David J. Williams, A. Barrett, A. White, 1999 .

Synthetic Studies Towards the Core Structure of Nakadomarin A by a Thioamide-Based Strategy

S. Coles, P. Horton, P. Procopiou, 2013, European journal of organic chemistry.

A tripartite asymmetric allylboration — Silicon tethered alkene ring closing metathesis — in situ ring opening protocol for the regiospecific generation of functionalized (E)-disubstituted homoallylic alcohols

A. Barrett, P. Procopiou, D. C. Braddock, 1999 .

Nucleophilic substitution of (alkoxymethylene)dimethylammonium chloride with carboxylate salts: a convenient procedure for the synthesis of esters with inversion of configuration

A. Barrett, N. Koike, P. Procopiou, 1995 .

A mild, enantioselective synthesis of (R)-salmeterol via sodium borohydride–calcium chloride asymmetric reduction of a phenacyl phenylglycinol derivative

S. Ley, P. Procopiou, B. McDermott, 2002 .

Heavier group 2 element catalyzed hydrophosphination of carbodiimides

P. Hitchcock, A. Barrett, M. Hill, 2008 .

Bis(trimethylsilyl)methyl derivatives of calcium, strontium and barium: potentially useful dialkyls of the heavy alkaline earth elements.

A. Barrett, M. Hill, Mark R. Crimmin, 2008, Chemistry.

Trifluoromethyl coordination and C-F bond activation at calcium.

P. Hitchcock, A. Barrett, M. Hill, 2007, Angewandte Chemie.

Directed ring-closing metathesis of trienes by silyl substitution

A. Barrett, C. Schultz-Fademrecht, P. Procopiou, 2004 .

Lead identification of benzimidazolone and azabenzimidazolone arylsulfonamides as CC-chemokine receptor 4 (CCR4) antagonists.

J. Percy, Afjal H. Miah, P. Procopiou, 2014, Bioorganic & medicinal chemistry.

Ritter-type reactions of N-chlorosaccharin: a method for the electrophilic diamination of alkenes.

K. Booker‐Milburn, P. Procopiou, B. Cox, 2003, Organic letters.

Nucleophilic substitution of (alkoxymethylene)dimethylammonium chloride with potassium phthalimide; a convenient procedure for the synthesis of imides with inversion of configuration

A. Barrett, P. Procopiou, D. C. Braddock, 1997 .

Nucleophilic Substitution Reactions of (Alkoxymethylene)dimethylammonium Chloride.

A. Barrett, N. Koike, P. Procopiou, 1998, The Journal of organic chemistry.

Nucleophilic Substitution Reactions of (Alkoxymethylene)dimethylammonium Chloride.

A. Barrett, N. Koike, P. Procopiou, 1998, The Journal of organic chemistry.

Reactions of β-Diketiminate-Stabilized Calcium Amides with 9-Borabicyclo[3.3.1]nonane (9-BBN)

P. Hitchcock, A. Barrett, M. Hill, 2007 .

Total synthesis of antifungal natural products.

A. Barrett, D. Williams, P. Procopiou, 2000, Ernst Schering Research Foundation workshop.

An Extremely Powerful Acylation Reaction of Alcohols with Acid Anhydrides Catalyzed by Trimethylsilyl Trifluoromethanesulfonate.

P. Procopiou, G. Inglis, S. Baugh, 1998 .

Novel Glucocorticoid Antedrugs Possessing a 17β-(γ-Lactone) Ring

C. Tralau-Stewart, G. N. Hagger, K. Biggadike, 2001 .

Rearrangement of a 16α,17α-Epoxy-16β-methylandrostane-17β-carbothioic Acid to a 17β-Mercapto-16β-methylandrostane-17α,16α-carbolactone

R. Upton, P. Procopiou, G. H. Phillipps, 1998 .

Imino sulfinamidines: synthesis and coordination chemistry of a novel class of chiral bidentate ligands.

P. Hitchcock, A. Barrett, M. Hill, 2006, Inorganic Chemistry.

Profile of a Highly Selective Quaternized Pyrrolidine Betaine αvβ6 Integrin Inhibitor-(3S)-3-(3-(3,5-Dimethyl-1H-pyrazol-1-yl)phenyl)-4-((1S and 1R,3R)-1-methyl-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-ium-1-yl)butanoate Synthesized by Stereoselective Methylation.

Joelle Le, S. Lynn, S. Macdonald, 2019, Journal of medicinal chemistry.

Second Generation Recyclable `Boomerang' Polymer Supported Catalysts for Olefin Metathesis: Application of Arduengo Carbene Complexes

A. Barrett, P. Procopiou, D. C. Braddock, 2000 .

Novel squalestatin derivatives arising from reactions at the allylic centre of the C1-side chain

B. Dymock, P. Sidebottom, P. Procopiou, 1998 .

Investigation of a Late‐Stage Derivatization Approach to Isatogens: Discovery of New Reaction Pathways

J. P. Harrity, P. Procopiou, S. Swanson, 2016 .

2-Iodoisatogens: versatile intermediates for the synthesis of nitrogen heterocycles.

J. P. Harrity, P. Procopiou, S. Swanson, 2015, Organic letters.

4-acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a novel class of non-brain-penetrant histamine H3 receptor antagonists.

Christopher Browning, Helen Connor, David M. Wilson, 2007, Journal of medicinal chemistry.

Alkene metathesis in the synthesis of novel β-lactams

A. Barrett, P. Procopiou, V. C. Gibson, 1996 .

Discovery of ( S)-3-(3-(3,5-Dimethyl-1 H-pyrazol-1-yl)phenyl)-4-(( R)-3-(2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl)pyrrolidin-1-yl)butanoic Acid, a Nonpeptidic αvβ6 Integrin Inhibitor for the Inhaled Treatment of Idiopathic Pulmonary Fibrosis.

Joelle Le, S. Macdonald, J. Pritchard, 2018, Journal of medicinal chemistry.

Semi‐Synthetic Squalestatins: Squalene Synthase Inhibition and Antifungal Activity. The SAR of C6 and C7 Modifications.

J. Payne, A. H. Shingler, P. Procopiou, 1994 .

Oxazole synthesis with minimal purification: synthesis and application of a ROMPgel Tosmic reagent.

S. Cramp, A. Barrett, P. Procopiou, 2001, Organic letters.

A reinvestigation of the synthesis of trans-(±)-1,2,3,4,4a,10a-hexahydro [1,4] benzodioxino[2,3-c]pyridine

M. Deal, P. Procopiou, P. C. Cherry, 1994 .

The squalestatins: decarboxy and 4-deoxy analogues as potent squalene synthase inhibitors.

C. Chan, B. Dymock, J. Scicinski, 1996, Journal of medicinal chemistry.

Discovery of a rapidly metabolized, long-acting β(2) adrenergic receptor agonist with a short onset time incorporating a sulfone group suitable for once-daily dosing.

K. Biggadike, D. Holmes, P. Procopiou, 2014, Journal of medicinal chemistry.

Solid-phase synthesis of isoxazoles using vinyl ethers as chameleon catches.

A. Barrett, P. Procopiou, U. Voigtmann, 2001, Organic letters.

The discovery of long-acting saligenin β₂ adrenergic receptor agonists incorporating a urea group.

P. Procopiou, V. Barrett, G. Somers, 2011, Bioorganic & medicinal chemistry.

The discovery of long-acting saligenin β₂ adrenergic receptor agonists incorporating hydantoin or uracil rings.

R. Perciaccante, Valerie S. Morrison, P. Procopiou, 2011, Bioorganic & medicinal chemistry.

Synthesis and structure-activity relationships of long-acting beta2 adrenergic receptor agonists incorporating arylsulfonamide groups.

I. McLay, D. Coe, K. Biggadike, 2009, Journal of medicinal chemistry.

Identification of pyrazolopyrimidine arylsulfonamides as CC-chemokine receptor 4 (CCR4) antagonists.

S. Hodgson, J. Percy, Afjal H. Miah, 2017, Bioorganic & medicinal chemistry.

2,8-Diazaspiro[4.5]decan-8-yl)pyrimidin-4-amine potent CCR4 antagonists capable of inducing receptor endocytosis.

S. Hodgson, J. Percy, Lena Shukla, 2016, European journal of medicinal chemistry.

Medicinal chemistry in drug discovery in big pharma: past, present and future.

Simon J F Macdonald, S. Macdonald, P. Procopiou, 2017, Drug discovery today.

Second Generation Recyclable “Boomerang” Polymer‐Supported Catalysts for Olefin Metathesis: Application of Arduengo Carbene Complexes.

A. Barrett, P. Procopiou, D. C. Braddock, 2000 .

Synthesis of Benzodioxinopyrroles as selective α2-adrenoceptor antagonists

P. Procopiou, P. C. Cherry, A. Pipe, 1995 .

Novel Glucocorticoid Antedrugs Possessing a 21-(γ-Lactone) Ring.

R. Angell, S. Lynn, K. Biggadike, 2010 .

Novel glucocorticoid antedrugs possessing a 21-(?-lactone) ring

R. Angell, S. Lynn, K. Biggadike, 2002 .

Lead Optimization of the N1 Substituent of a Novel Series of Indazole Arylsulfonamides as CCR4 Antagonists and Identification of a Candidate for Clinical Investigation.

S. Hodgson, D. Hall, P. Procopiou, 2012 .

Synthesis of (R)-alpha-benzylmethionine: a novel rearrangement during alkylation of the Seebach (R)-methionine oxazolidinone.

R. Perciaccante, P. Procopiou, Mahmood Ahmed, 2003, Organic & biomolecular chemistry.

Enyne metathesis for the facile synthesis of highly functionalisednovel bicyclic β-lactams

A. Barrett, P. Procopiou, D. C. Braddock, 1997 .

A metathesis-based approach to the synthesis of 2-pyridones and pyridines.

T. Donohoe, P. Procopiou, Lisa P. Fishlock, 2008, Organic letters.

Novel glucocorticoid antedrugs possessing a C16,17-fused γ-lactone ring

S. Lynn, K. Biggadike, P. Procopiou, 2000 .

Base catalysed rearrangement of fluocinolone acetonide to a 17α-pregnane-21,16α-carbolactone

S. Lynn, P. Procopiou, S. A. Richards, 2000 .

The squalestatins: inhibitors of squalene synthase. Enzyme inhibitory activities and in vivo evaluation of C3-modified analogues.

B. Dymock, P. Procopiou, A. Craven, 1994, Journal of medicinal chemistry.

Synthesis and Structure−Activity Relationships of Long-acting β2 Adrenergic Receptor Agonists Incorporating Arylsulfonamide Groups

I. McLay, D. Coe, K. Biggadike, 2009 .

A re-investigation of the Fries rearrangement of 3-chlorophenyl acetate and synthesis of 2-azido-1-(4-(benzyloxy)-2-chlorophenyl)ethanone from 4-bromo-3-chlorophenol

D. Coe, P. Procopiou, George Procopiou, 2017 .

Heavier group 2 metals and intermolecular hydroamination: a computational and synthetic assessment.

A. Barrett, Christine Brinkmann, P. Hunt, 2009, Journal of the American Chemical Society.

Novel secosteroids arising from acid catalysed rearrangement of fluocinonide acetonide in the presence of Tf2O and TMSOTf

S. Lynn, P. Procopiou, A. D. Roberts, 1999 .